SCHEMBL4594149

SCHEMBL4594149

CC(C)(C)[C@@](CO)(Cc1ccncc1)NC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.43
GAA P10253 4/20 0.42
FDPS P14324 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 3/20 0.37
POLB P06746 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
KDM4E B2RXH2 1/20 0.37
PTPRB P23467 1/20 0.36
TSHR P16473 1/20 0.36
NPC1 O15118 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MEN1 O00255 1/20 0.35
CYP17A1 P05093 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4073210 0.86 CYP3A4 (0.46) RAB9AALDH1A1MAPTTSHRNPC1
SCHEMBL1273081 0.86 CYP3A4 (0.46) RAB9AALDH1A1MAPTTSHRNPC1
SCHEMBL4379160 0.83 FDPS (0.46) FDPSALDH1A1MAPTKDM4E
SCHEMBL4773478 0.82 LMNA (0.41) RAB9AALDH1A1POLBNPC1KMT2A
SCHEMBL4583741 0.79 MMP1 (0.43) RAB9APOLBKDM4EPTPRBNPC1
SCHEMBL1932047 0.79 RAB9A (0.49) RAB9AGAAFDPSALDH1A1MAPT
SCHEMBL3958834 0.77 OPRM1 (0.41) RAB9APOLBTDP1NPC1KMT2A
SCHEMBL3722221 0.75 RIPK1 (0.40) ALDH1A1MAPTPOLBTDP1KDM4E
SCHEMBL1539491 0.74 VNN1 (0.42) RAB9APOLBKMT2AMEN1
SCHEMBL3960044 0.74 RIPK1 (0.41) RAB9AALDH1A1NPC1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874768-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113837-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed