SCHEMBL4940237

SCHEMBL4940237

Cc1ccc(S(=O)(=O)N2CCC(O)CC2)cc1

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.64
PKM P14618 3/20 0.64
POLB P06746 1/20 0.64
HTT P42858 1/20 0.64
KDM4E B2RXH2 1/20 0.63
HSD11B1 P28845 1/20 0.62
NPC1 O15118 1/20 0.62
RAB9A P51151 1/20 0.62
LMNA P02545 2/20 0.61
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
EBP Q15125 1/20 0.57
DHCR7 Q9UBM7 1/20 0.57
USP2 O75604 1/20 0.57
GAA P10253 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535608 0.95 LMNA (0.60) ALDH1A1PKMPOLBHTTKDM4E
SCHEMBL3235046 0.90 PKM (0.57) ALDH1A1PKMPOLBHTTKDM4E
SCHEMBL4516709 0.90 PKM (0.57) ALDH1A1PKMPOLBHTTKDM4E
SCHEMBL3235054 0.90 PKM (0.57) ALDH1A1PKMPOLBHTTKDM4E
SCHEMBL10360133 0.90 HSD11B1 (0.67) ALDH1A1PKMPOLBHTTKDM4E
SCHEMBL28882522 0.84 ALDH1A1 (0.66) ALDH1A1PKMPOLBHTTKDM4E
SCHEMBL12793343 0.84 USP2 (0.71) ALDH1A1POLBHTTKDM4EHSD11B1
SCHEMBL266466 0.84 MEN1 (0.77) ALDH1A1PKMPOLBHTTKDM4E
SCHEMBL2474562 0.83 ALDH1A1 (0.62) ALDH1A1PKMPOLBHTTKDM4E
SCHEMBL565301 0.83 PKM (0.88) ALDH1A1PKMPOLBHTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4413012-A1 PROCESS FOR C-H INSERTION BY GEM-HYDROGENATION OF AN INTERNAL ALKYNE Studiengesellschaft Kohle gGmbH (DE) 2024-08-14 EP disclosed
CN-117164505-A Method for synthesizing organic sulfate by dialkyl sulfate or pyrosulfate 湖南大学 2023-12-05 CN disclosed
US-20230321016-A1 COMBINATION THERAPY FOR TREATING CANCER GONGWIN BIOPHARM CO., LTD (TW) 2023-10-12 US disclosed
US-11752118-B2 Method for treating melanoma GONGWIN BIOPHARM CO., LTD (TW) 2023-09-12 US disclosed
US-11752160-B2 Method for reducing fat by administering benzenesulfonamide compositions GONGWIN BIOPHARM CO., LTD (TW) 2023-09-12 US disclosed
WO-2023110394-A1 PROCESS FOR C-H INSERTION BY GEM-HYDROGENATION OF AN INTERNAL ALKYNE STUDIENGESELLSCHAFT KOHLE GGMBH (DE) 2023-06-22 WO disclosed
US-20220168248-A1 METHOD FOR TREATING MELANOMA GONGWIN BIOPHARM CO., LTD (TW) 2022-06-02 US disclosed
US-20200338028-A1 BENZENESULFONAMIDE DERIVATIVES AND METHOD FOR MODULATING LIPID RAFT GONGWIN BIOPHARM CO., LTD. (TW) 2020-10-29 US disclosed
US-10548862-B2 Topical formulation and method for preventing or treating acne Wu, Lester J. (US) 2020-02-04 US disclosed
US-20190321313-A1 BENZENESULFONAMIDE DERIVATIVES AND METHOD FOR TREATING CANCER Gongwin Biopharm Holdings Co., Ltd. 2019-10-24 US disclosed
WO-2007056075-A2 SIX MEMBERED HETEROAROMATIC INHIBITORS TARGETING RESISTANT KINASE MUTATIONS TARGEGEN, INC. (US) 2007-05-18 WO disclosed
WO-2006008260-A1 DIMERIC PIPERIDINE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 2006-01-26 WO disclosed
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-5070087-A Aryl(alkyland alkylene)-N-((phenoxy and phenylthio)alkyl) aminoheterocyclics as cardiovascular, anthihistaminic, antisecretory and antiallergy agents A. H. ROBINS COMPANY, INCORPORATED (US) 1991-12-03 US disclosed
US-4950674-A Arylalkylheterocyclic amines,N-substituted by aryloxyalkyl group in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1990-08-21 US disclosed
US-4839374-A TREATING ALLERGIES JANSSEN PHARMACEUTICA, N.V. (BE) 1989-06-13 US disclosed
US-4810713-A Arylalkyl-heterocyclic amines, n-substituted by aryloxyalkyl groups used in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1989-03-07 US disclosed
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed
EP-0235463-A2 N-substituted-arylalkyl and arylalkylene piperidines as cardiovascular antihistaminic and antisecretory agents A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1987-09-09 EP disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190321313-A1 BENZENESULFONAMIDE DERIVATIVES AND METHOD FOR TREATING CANCER ARSA, ABCB1, ABCG2 ALDH1A1 689/4885PKM 1749/4885POLB 1930/4885
US-10548862-B2 Topical formulation and method for preventing or treating acne CUTA, STS, ALAD ALDH1A1 669/4885PKM 2529/4885POLB 2365/4885
US-11752160-B2 Method for reducing fat by administering benzenesulfonamide compositions LIPE, FABP4, LIPA ALDH1A1 728/4885PKM 521/4885POLB 1703/4885
US-20220168248-A1 METHOD FOR TREATING MELANOMA TYR, MITF, BRAF ALDH1A1 528/4885PKM 1050/4885POLB 1410/4885
US-20230321016-A1 COMBINATION THERAPY FOR TREATING CANCER TP53, MCL1, TOP2B ALDH1A1 381/4885PKM 2022/4885POLB 907/4885
US-11752118-B2 Method for treating melanoma TYR, MITF, BRAF ALDH1A1 528/4885PKM 1050/4885POLB 1410/4885
US-20200338028-A1 BENZENESULFONAMIDE DERIVATIVES AND METHOD FOR MODULATING LIPID RAFT ABCB4, SPTSSB, SMPD2 ALDH1A1 1604/4885PKM 2929/4885POLB 3145/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.