SCHEMBL6358704

SCHEMBL6358704

CC(=O)c1ccc(NC(N)=O)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.60
NPC1 O15118 4/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
RAB9A P51151 2/20 0.60
TAAR1 Q96RJ0 1/20 0.60
PEPD P12955 1/20 0.59
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
HTT P42858 1/20 0.58
NLRP1 Q9C000 1/20 0.58
ALDH1A1 P00352 6/20 0.57
KIF11 P52732 3/20 0.57
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
GAA P10253 1/20 0.53
GFER P55789 1/20 0.53
LMNA P02545 2/20 0.52
GLA P06280 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5062623 0.83 PEPD (0.80) MAPTNPC1RAB9APEPDMEN1
SCHEMBL6931409 0.83 MAPT (0.56) MAPTNPC1SMN1; SMN2RAB9ATAAR1
SCHEMBL1880013 0.83 RAB9A (0.57) MAPTNPC1SMN1; SMN2RAB9ATAAR1
Benzenesulfonamide SCHEMBL28177870 0.82 CA1 (0.68) MAPTNPC1SMN1; SMN2RAB9ATAAR1
SCHEMBL14047972 0.82 PEPD (0.64) MAPTNPC1SMN1; SMN2RAB9APEPD
SCHEMBL11925383 0.82 SMN1; SMN2 (0.67) MAPTNPC1SMN1; SMN2RAB9ATAAR1
SCHEMBL3633396 0.82 NPC1 (0.84) MAPTNPC1SMN1; SMN2RAB9ATAAR1
SCHEMBL474757 0.82 ALDH1A1 (0.70) MAPTNPC1SMN1; SMN2RAB9ATAAR1
SCHEMBL10456830 0.80 PEPD (0.52) MAPTNPC1PEPDMEN1KMT2A
SCHEMBL10456829 0.80 PEPD (0.52) MAPTNPC1PEPDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103221388-A Novel sulfonamide compounds for inhibition of metastatic tumor growth METASIGNAL THERAPEUTICS INC 2013-07-24 CN claimed
US-20050113450-A1 Antibacterial agents PHARMACIA & UPJOHN COMPANY 2005-05-26 US claimed
US-20040142981-A1 Antibacterial benzoic acid derivatives PHARMACIA & UPJOHN COMPANY 2004-07-22 US claimed
US-20040110802-A1 Antibacterial benzoic acid derivatives PHARMACIA & UPJOHN COMPANY 2004-06-10 US claimed
WO-2004018461-A2 ANTIBACTERIAL BENZOIC ACID DERIVATIVES PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-04 WO claimed
US-20230357165-A1 QUINAZOLINONES DERIVATIVES FOR TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE, PREPARATION AND USE THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2023-11-09 US disclosed
WO-2022003712-A1 QUINAZOLINONES DERIVATIVES FOR TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE, PREPARATION AND USE THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2022-01-06 WO disclosed
US-10202388-B2 Fused-ring compounds, pharmaceutical composition and uses thereof Shanghai De Novo Pharmatech Co., Ltd. (CN) 2019-02-12 US disclosed
US-20180022752-A1 FUSED-RING COMPOUNDS, PHARMACEUTICAL COMPOSITION AND USES THEREOF Shanghai De Novo Pharmatech Co., Ltd. (CN) 2018-01-25 US disclosed
EP-3075726-A1 UREA DERIVATIVE OR PHARMACOLOGICALLY ACCEPTABLE SALT THEREOF Kyorin Pharmaceutical Co., Ltd. (JP) 2016-10-05 EP disclosed
CN-103221388-B For the novel sulfonamide compounds suppressing metastatic tumo(u)r to grow 维理生物技术公司 2016-09-28 CN disclosed
CN-102800816-B There is the OLED device of fluoranthene electron transport materials GLOBAL OLED TECHNOLOGY LLC (US) 2016-05-18 CN disclosed
CN-1304060-A Photographic component, compound and its preparing method EASTMAN KODAK CO (US) 2001-07-18 CN disclosed
CN-1288176-A Tensile strength and durable fibrous photosensitive base materials EASTMAN KODAK CO (US) 2001-03-21 CN disclosed
CN-1284660-A Flexible imaging element using microporous polyester piece EASTMAN KODAK CO (US) 2001-02-21 CN disclosed
CN-1260514-A Colour photography element comprising compound for increasing light sensitivity EASTMAN KODAK CO (US) 2000-07-19 CN disclosed
CN-1260513-A Pyrazolopyrrodiazole colour coupling component for photography EASTMAN KODAK CO (US) 2000-07-19 CN disclosed
CN-1258861-A Photographic element containing high dye productivity colour former EASTMAN KODAK CO (US) 2000-07-05 CN disclosed
CN-1258021-A Photographic material EASTMAN KODAK CO (US) 2000-06-28 CN disclosed
CN-1235280-A Photographic element containing yellow dye-forming photographic coupler EASTMAN KODAK CO (US) 1999-11-17 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050113450-A1 Antibacterial agents CLPP, SPOUT1, SAMHD1 MAPT 4753/4885NPC1 3512/4885SMN1; SMN2 3015/4885
US-20230357165-A1 QUINAZOLINONES DERIVATIVES FOR TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE, PREPARATION AND USE THEREOF ATG7, GOT1, LIPC MAPT 2243/4885NPC1 268/4885SMN1; SMN2 3760/4885
US-10202388-B2 Fused-ring compounds, pharmaceutical composition and uses thereof IDO1, IDO2, TDO2 MAPT 1811/4885NPC1 2820/4885SMN1; SMN2 3655/4885
US-20180022752-A1 FUSED-RING COMPOUNDS, PHARMACEUTICAL COMPOSITION AND USES THEREOF IDO1, IDO2, TDO2 MAPT 1811/4885NPC1 2820/4885SMN1; SMN2 3655/4885
US-20040142981-A1 Antibacterial benzoic acid derivatives GABRD, PHB1, GABBR1 MAPT 4754/4885NPC1 3891/4885SMN1; SMN2 2635/4885
US-20040110802-A1 Antibacterial benzoic acid derivatives GABRD, GABBR1, GABRA1 MAPT 4759/4885NPC1 3778/4885SMN1; SMN2 2022/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.