SCHEMBL872200

SCHEMBL872200

CCCCCCCCCC(CCCCCCC[C@H]1C[C@H]1CCCCCCCC)CCN(C)C

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.44
DNM1 Q05193 3/20 0.41
LMNA P02545 1/20 0.37
LYPLA1 O75608 2/20 0.33
LYPLA2 O95372 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
PLA2G1B P04054 1/20 0.33
PLA2G2A P14555 1/20 0.33
ALDH1A1 P00352 1/20 0.32
SPHK2 Q9NRA0 3/20 0.32
SPHK1 Q9NYA1 3/20 0.32
TBXA2R P21731 1/20 0.31
PTGFR P43088 1/20 0.31
PTGER2 P43116 1/20 0.31
EPHX1 P07099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10084617 1.00 ALOX5 (0.44) ALOX5DNM1LMNALYPLA1LYPLA2
SCHEMBL23282462 1.00 ALOX5 (0.44) ALOX5DNM1LMNALYPLA1LYPLA2
SCHEMBL23437455 1.00 ALOX5 (0.44) ALOX5DNM1LMNALYPLA1LYPLA2
SCHEMBL23923252 0.93 ALOX5 (0.39) ALOX5DNM1LMNA
SCHEMBL15155771 0.88 ALOX5 (0.62) ALOX5ALDH1A1TBXA2RPTGFRPTGER2
SCHEMBL15155996 0.88 ALOX5 (0.62) ALOX5ALDH1A1TBXA2RPTGFRPTGER2
SCHEMBL15156129 0.88 ALOX5 (0.62) ALOX5ALDH1A1TBXA2RPTGFRPTGER2
SCHEMBL15155744 0.88 ALOX5 (0.62) ALOX5ALDH1A1TBXA2RPTGFRPTGER2
SCHEMBL31700901 0.88 ALOX5 (0.53) ALOX5DNM1LMNAALDH1A1SPHK2
SCHEMBL23390582 0.86 ALOX5 (0.39) ALOX5DNM1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 686 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240123047-A1 LIPID NANOPARTICLE ADJUVANT COMPOSITION FOR PNEUMOCOCCAL CONJUGATE VACCINES MERCK SHARP & DOHME LLC (US) 2024-04-18 US claimed
US-11566051-B2 Stabilized RSV F proteins and uses thereof MERCK SHARP & DOHME LLC (US) 2023-01-31 US claimed
EP-3939604-A2 INFLUENZA HEMAGGLUTININ PROTEIN VACCINES Merck Sharp & Dohme Corp. (US) 2022-01-19 EP claimed
US-20210300971-A1 STABILIZED RSV F PROTEINS AND USES THEREOF MERCK SHARP & DOHME LLC 2021-09-30 US claimed
CN-111655715-A Stabilized RSV F proteins and uses thereof 默沙东公司 2020-09-11 CN claimed
US-10576155-B2 Low molecular weight cationic lipids for oligonucleotide delivery SIRNA THEREAPEUTICS, INC. (US) 2020-03-03 US claimed
EP-3556353-A2 LIPID NANOPARTICLE VACCINE ADJUVANTS AND ANTIGEN DELIVERY SYSTEMS MERCK SHARP & DOHME CORP. (US) 2019-10-23 EP claimed
US-20190167811-A1 LIPID COMPOSITIONS AND THEIR USES FOR INTRATUMORAL POLYNUCLEOTIDE DELIVERY MODERNATX, INC. 2019-06-06 US claimed
US-20180311176-A1 NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACID COMPLEXES TRANSLATE BIO MA, INC. (US) 2018-11-01 US claimed
EP-3368089-A1 NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACID COMPLEXES TRANSLATE BIO MA, INC. (US) 2018-09-05 EP claimed
US-20180000939-A1 NOVEL LOW MOLECULAR WEIGHT CATIONIC LIPIDS FOR OLIGONUCLEOTIDE DELIVERY SIRNA THERAPEUTICS, INC. (US) 2018-01-04 US claimed
WO-2017192470-A1 COMBINATION THERAPY OF ANTI-IL-10 ANTIBODY AND COMPOSITIONS COMPRISING LIPID NANOPARTICLES AND TLR9 AGONIST CPG OLIGONUCLEOTIDES MERCK SHARP & DOHME CORP. (US) 2017-11-09 WO claimed
WO-2017075038-A1 NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACID COMPLEXES RANA THERAPEUTICS, INC. (US) 2017-05-04 WO claimed
US-20160361411-A1 LIPID NANOPARTICLE VACCINE ADJUVANTS AND ANTIGEN DELIVERY SYSTEMS MERCK SHARP & DOHME CORP (US) 2016-12-15 US claimed
EP-2618847-A2 NOVEL LOW MOLECULAR WEIGHT CATIONIC LIPIDS FOR OLIGONUCLEOTIDE DELIVERY Merck Sharp & Dohme Corp. (US) 2013-07-31 EP claimed
US-20130178541-A1 NOVEL LOW MOLECULAR WEIGHT CATIONIC LIPIDS FOR OLIGONUCLEOTIDE DELIVERY BANK OF AMERICA, N.A. 2013-07-11 US claimed
WO-2012040184-A2 NOVEL LOW MOLECULAR WEIGHT CATIONIC LIPIDS FOR OLIGONUCLEOTIDE DELIVERY MERCK SHARP & DOHME CORP. (US) 2012-03-29 WO claimed
US-12629412-B2 Betacoronavirus mRNA vaccines MODERNATX, INC. (US) 2026-05-19 US disclosed
US-20130156849-A1 MODIFIED NUCLEOSIDE, NUCLEOTIDE, AND NUCLEIC ACID COMPOSITIONS modeRNA Therapeutics (US) 2013-06-20 US disclosed
WO-2012040184-A2 NOVEL LOW MOLECULAR WEIGHT CATIONIC LIPIDS FOR OLIGONUCLEOTIDE DELIVERY MERCK SHARP & DOHME CORP. (US) 2012-03-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180311176-A1 NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACID COMPLEXES DIS3, SYNCRIP, EXOSC5 ALOX5 4111/4885DNM1 1458/4885LMNA 291/4885
US-12629412-B2 Betacoronavirus mRNA vaccines RNMT, RNGTT, METTL16 ALOX5 2873/4885DNM1 2514/4885LMNA 616/4885
US-20180000939-A1 NOVEL LOW MOLECULAR WEIGHT CATIONIC LIPIDS FOR OLIGONUCLEOTIDE DELIVERY LDLR, APOB, CETP ALOX5 1273/4885DNM1 624/4885LMNA 1763/4885
US-10576155-B2 Low molecular weight cationic lipids for oligonucleotide delivery LDLR, APOB, CETP ALOX5 1243/4885DNM1 486/4885LMNA 1800/4885
US-20130156849-A1 MODIFIED NUCLEOSIDE, NUCLEOTIDE, AND NUCLEIC ACID COMPOSITIONS NSUN2, RNMT, NSUN3 ALOX5 4052/4885DNM1 1918/4885LMNA 122/4885
US-20160361411-A1 LIPID NANOPARTICLE VACCINE ADJUVANTS AND ANTIGEN DELIVERY SYSTEMS TLR3, TLR5, TLR1 ALOX5 167/4885DNM1 3095/4885LMNA 1798/4885
US-20190167811-A1 LIPID COMPOSITIONS AND THEIR USES FOR INTRATUMORAL POLYNUCLEOTIDE DELIVERY RNMT, PHOSPHO1, POLM ALOX5 1911/4885DNM1 1045/4885LMNA 2115/4885
US-20240123047-A1 LIPID NANOPARTICLE ADJUVANT COMPOSITION FOR PNEUMOCOCCAL CONJUGATE VACCINES PLTP, NAPEPLD, PHOSPHO1 ALOX5 65/4885DNM1 2136/4885LMNA 1355/4885
US-20130178541-A1 NOVEL LOW MOLECULAR WEIGHT CATIONIC LIPIDS FOR OLIGONUCLEOTIDE DELIVERY LDLR, LIPC, CETP ALOX5 859/4885DNM1 627/4885LMNA 870/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.