Casokefamide

Casokefamide

SCHEMBL1373200

C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 5/20 0.69
OPRM1 P35372 4/20 0.69
OPRK1 P41145 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29440670 1.00 OPRD1 (0.69) OPRD1OPRM1OPRK1
Frakefamide SCHEMBL29388146 0.95 OPRD1 (0.63) OPRD1OPRM1OPRK1
SCHEMBL30661444 0.92 OPRD1 (0.70) OPRD1OPRM1OPRK1
SCHEMBL31140206 0.92 OPRD1 (0.80) OPRD1OPRM1OPRK1
SCHEMBL27755089 0.91 ACE (0.60)
SCHEMBL29437738 0.91 ACE (0.60)
SCHEMBL30786035 0.90 OPRD1 (0.69) OPRD1OPRM1OPRK1
SCHEMBL29789555 0.90 OPRD1 (0.69) OPRD1OPRM1OPRK1
SCHEMBL29365670 0.89 NPY4R (0.62) OPRD1OPRM1OPRK1
SCHEMBL7900841 0.88 OPRD1 (0.74) OPRD1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12624002-B2 Dimers for use in synthesis of peptidomimetics THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2026-05-12 US disclosed
US-12600699-B2 Thiosemicarbazates and uses thereof THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2026-04-14 US disclosed
US-12595233-B2 Thiosemicarbazates and uses thereof THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2026-04-07 US disclosed
US-20260070894-A1 COMPOUNDS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2026-03-12 US disclosed
US-12351573-B2 Compounds for use in synthesis of peptidomimetics THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2025-07-08 US disclosed
US-20230159450-A1 DIMERS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH 2023-05-25 US disclosed
US-20230111252-A1 THIOSEMICARBAZATES AND USES THEREOF THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2023-04-13 US disclosed
EP-4146629-A1 DIMERS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS The Feinstein Institutes for Medical Research (US) 2023-03-15 EP disclosed
CN-115515937-A Dimers for the synthesis of peptidomimetics 范因斯坦医学研究院 2022-12-23 CN disclosed
US-20220372022-A1 COMPOUNDS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2022-11-24 US disclosed
US-20150051371-A1 CARBOHYDRATE-BASED DRUG DELIVERY POLYMERS AND CONJUGATES THEREOF NEKTAR THERAPEUTICS (US) 2015-02-19 US disclosed
US-20130281657-A1 MACROCYCLES AND MACROCYCLE STABILIZED PEPTIDES BRISTOL-MYERS SQUIBB COMPANY (US) 2013-10-24 US disclosed
US-20130281657-A1 MACROCYCLES AND MACROCYCLE STABILIZED PEPTIDES BRISTOL-MYERS SQUIBB COMPANY (US) 2013-10-24 US disclosed
EP-2627662-A1 METHODS FOR PREPARING MACROCYCLES AND MACROCYCLE STABILIZED PEPTIDES Bristol-Myers Squibb Company (US) 2013-08-21 EP disclosed
WO-2012051405-A1 METHODS FOR PREPARING MACROCYCLES AND MACROCYCLE STABILIZED PEPTIDES BRISTOL-MYERS SQUIBB COMPANY (US) 2012-04-19 WO disclosed
US-20110288011-A1 PEPTIDE THERAPEUTIC CONJUGATES AND USES THEREOF ANGIOCHEM INC. (CA) 2011-11-24 US disclosed
US-20110171312-A1 MODIFIED THERAPEUTIC PEPTIDES, METHODS OF THEIR PREPARATION AND USE NEKTAR THERAPEUTICS (US) 2011-07-14 US disclosed
EP-2341942-A1 POLYMER CONJUGATES OF THERAPEUTIC PEPTIDES Nektar Therapeutics (US) 2011-07-13 EP disclosed
US-20110166063-A1 POLYMER CONJUGATES OF THERAPEUTIC PEPTIDES NEKTAR THERAPEUTICS (US) 2011-07-07 US disclosed
WO-2010033207-A1 POLYMER CONJUGATES OF THERAPEUTIC PEPTIDES NEKTAR THERAPEUTICS (US) 2010-03-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12351573-B2 Compounds for use in synthesis of peptidomimetics DNPEP, NPEPPS, PAM OPRD1 2574/4885OPRM1 1752/4885OPRK1 2628/4885
US-12624002-B2 Dimers for use in synthesis of peptidomimetics GLUL, ARGLU1, ASNS OPRD1 905/4885OPRM1 1215/4885OPRK1 2463/4885
US-20150051371-A1 CARBOHYDRATE-BASED DRUG DELIVERY POLYMERS AND CONJUGATES THEREOF STT3B, STT3A, DDOST OPRD1 3859/4885OPRM1 3352/4885OPRK1 3229/4885
US-20260070894-A1 COMPOUNDS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS NPR1, NGLY1, DDAH1 OPRD1 1029/4885OPRM1 453/4885OPRK1 1473/4885
US-12595233-B2 Thiosemicarbazates and uses thereof TST, THRB, HSPB1 OPRD1 2834/4885OPRM1 1506/4885OPRK1 3659/4885
US-20230111252-A1 THIOSEMICARBAZATES AND USES THEREOF TST, ABAT, AADAC OPRD1 4147/4885OPRM1 3052/4885OPRK1 4194/4885
US-20220372022-A1 COMPOUNDS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS DNPEP, NPEPPS, PAM OPRD1 2574/4885OPRM1 1752/4885OPRK1 2628/4885
US-20110166063-A1 POLYMER CONJUGATES OF THERAPEUTIC PEPTIDES NGLY1, CD44, IAPP OPRD1 3100/4885OPRM1 2317/4885OPRK1 2737/4885
US-20130281657-A1 MACROCYCLES AND MACROCYCLE STABILIZED PEPTIDES PTMS, VIP, MTPN OPRD1 4530/4885OPRM1 4478/4885OPRK1 4371/4885
US-20230159450-A1 DIMERS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS DNPEP, DAP3, ANPEP OPRD1 4010/4885OPRM1 2471/4885OPRK1 3891/4885
US-20110171312-A1 MODIFIED THERAPEUTIC PEPTIDES, METHODS OF THEIR PREPARATION AND USE DNPEP, VIP, PTMS OPRD1 2871/4885OPRM1 1535/4885OPRK1 2169/4885
US-12600699-B2 Thiosemicarbazates and uses thereof MET, THRB, ABAT OPRD1 2236/4885OPRM1 780/4885OPRK1 2051/4885
US-20110288011-A1 PEPTIDE THERAPEUTIC CONJUGATES AND USES THEREOF VIP, SLC1A5, SLC47A1 OPRD1 4036/4885OPRM1 3822/4885OPRK1 3911/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.