Dihydrolipoic Acid

Dihydrolipoic Acid

SCHEMBL1659440

O=C([O-])CCCCC(S)CCS.[K+]

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

AGTR1DHFRGABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTNR3C2PBP2XPTGS1PTGS2VKORC1blablaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAftsImrcAmrcBmrdApbp1apbp1bpbp2apbp2bpbp3polthyA

The experimentally established mechanism targets of Dihydrolipoic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.39
CA1 P00915 3/20 0.35
FABP3 P05413 7/20 0.35
GSTK1 Q9Y2Q3 2/20 0.34
GPR84 Q9NQS5 1/20 0.34
ENPEP Q07075 1/20 0.33
BBOX1 O75936 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dihydrolipoic Acid SCHEMBL5827361 0.96 NFKB1 (0.39) NFKB1CA1FABP3GSTK1GPR84
Dihydrolipoic Acid SCHEMBL718014 0.96 NFKB1 (0.43) NFKB1CA1FABP3GSTK1GPR84
Dihydrolipoic Acid SCHEMBL2582100 0.96 NFKB1 (0.39) NFKB1CA1FABP3GSTK1GPR84
Dihydrolipoic Acid SCHEMBL4761909 0.94 NFKB1 (0.38) NFKB1CA1FABP3GSTK1GPR84
Dihydrolipoic Acid SCHEMBL4094129 0.89 GSTK1 (0.46) NFKB1GSTK1ENPEP
Zinc Ion SCHEMBL3337795 0.82 HDAC3 (0.36) NFKB1
SCHEMBL3276879 0.82 HDAC3 (0.36) NFKB1
Tetrabuthylammonium SCHEMBL7185399 0.82 NFKB1 (0.47) NFKB1CA1FABP3GPR84BBOX1
SCHEMBL3276632 0.81 HDAC3 (0.41)
Zinc Ion SCHEMBL2580314 0.81 HDAC3 (0.35) NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100335037-C Free-flowing powder composition comprising alpha-lipoic acid (derivatives) DEGUSSA (DE) 2007-09-05 CN claimed
CN-1662222-A Free-flowing powder composition comprising alpha-lipoic acid (derivatives) DEGUSSA (DE) 2005-08-31 CN claimed
US-8541465-B2 Docetaxel formulations with lipoic acid and/or dihydrolipoic acid SCIDOSE, LLC (US) 2013-09-24 US disclosed
US-20110092580-A1 Docetaxel formulations with lipoic acid and/or dihydrolipoic acid SCIDOSE LLC (US) 2011-04-21 US disclosed
US-20110092579-A1 Solubilized formulation of docetaxel SCIDOSE LLC (US) 2011-04-21 US disclosed
CN-100335037-C Free-flowing powder composition comprising alpha-lipoic acid (derivatives) DEGUSSA (DE) 2007-09-05 CN disclosed
CN-1662222-A Free-flowing powder composition comprising alpha-lipoic acid (derivatives) DEGUSSA (DE) 2005-08-31 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110092580-A1 Docetaxel formulations with lipoic acid and/or dihydrolipoic acid DLST, TTPA, LIPA NFKB1 413/4885CA1 3748/4885FABP3 818/4885
US-20110092579-A1 Solubilized formulation of docetaxel DSG1, TTPA, TPSG1 NFKB1 940/4885CA1 3192/4885FABP3 3157/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.