SCHEMBL20143947

SCHEMBL20143947

O=C(NC(=O)c1ccc(S(=O)(=O)NC(=O)c2ccccc2)cc1)OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BCL2L1 Q07817 11/20 0.59
MCL1 Q07820 11/20 0.59
FLT1 P17948 2/20 0.56
FLT4 P35916 2/20 0.56
KDR P35968 2/20 0.56
MEN1 O00255 1/20 0.56
LMNA P02545 1/20 0.56
KMT2A Q03164 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA9 Q16790 2/20 0.53
PTGES O14684 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8815917 0.84 SLC6A2 (0.61) LMNAKMT2ACA12CA1CA2
SCHEMBL3829119 0.82 CA1 (0.57) BCL2L1MCL1MEN1KMT2ACA12
SCHEMBL27643285 0.80 CA1 (0.55) BCL2L1MCL1CA12CA1CA2
SCHEMBL11862063 0.80 CA1 (0.65) LMNACA12CA1CA2CA9
SCHEMBL3819564 0.79 CA1 (0.53) BCL2L1MCL1MEN1LMNAKMT2A
SCHEMBL9967798 0.77 FLT1 (0.69) BCL2L1MCL1FLT1FLT4KDR
SCHEMBL9177535 0.77 CA1 (0.63) MEN1LMNAKMT2AL3MBTL1CA12
SCHEMBL8424044 0.77 FLT1 (0.73) BCL2L1MCL1FLT1FLT4KDR
SCHEMBL30278496 0.76 CA1 (0.57) MEN1KMT2AL3MBTL1CA12CA1
SCHEMBL5931288 0.76 FLT1 (0.71) BCL2L1MCL1FLT1FLT4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11219209-B2 Method of reducing crop damage BAYER AKTIENGESELLSCHAFT (DE) 2022-01-11 US disclosed
US-11197477-B2 Aqueous capsule suspension concentrates based on 2-[(2,4-dichlorophenyl)methyl]-4,4′-dimethyl-3-isoxazolidinone BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2021-12-14 US disclosed
US-11191265-B2 Method of reducing crop damage BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2021-12-07 US disclosed
US-20210307322-A1 CONTROLLED RELEASE FORMULATIONS WITH LIGNIN FOR AGROCHEMICALS DSM IP ASSETS B.V. (NL) 2021-10-07 US disclosed
US-20210289777-A1 METHOD OF REDUCING CROP DAMAGE FMC CORPORATION 2021-09-23 US disclosed
US-20210289781-A1 HERBICIDAL MIXTURES BAYER AKTIENGESELLSCHAFT (DE) 2021-09-23 US disclosed
US-20210276974-A1 SUBSTITUTED 2-HETEROARYLOXYPYRIDINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2021-09-09 US disclosed
US-20210227824-A1 METHOD OF REDUCING CROP DAMAGE BAYER AKTIENGESELLSCHAFT (DE) 2021-07-29 US disclosed
US-20210137117-A1 HERBICIDAL MIXTURES FMC CORPORATION 2021-05-13 US disclosed
US-20210127667-A1 METHOD OF REDUCING CROP DAMAGE BAYER AKTIENGESELLSCHAFT (DE) 2021-05-06 US disclosed
US-20200196601-A1 HERBICIDE SAFENER COMPOSITIONS CONTAINING QUINAZOLINEDIONE-6CARBONYL DERIVATIVES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2020-06-25 US disclosed
US-20200181117-A1 SUBSTITUTED 3-HETEROARYLOXY-1H-PYRAZOLES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2020-06-11 US disclosed
US-20200172491-A1 SUBSTITUTED 5-(HET-)ARYLPYRAZOLAMIDES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2020-06-04 US disclosed
US-20200085055-A1 New uses of 2-(2,4-dichlorophenyl)methyl-4,4-dimethyl-3-isoxazolidone as foliar herbicide FMC CORPORATION 2020-03-19 US disclosed
US-20190330192-A1 SUBSTITUTED AZOLYLPYRROLONES AND AZOLYLHYDANTOINS AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2019-10-31 US disclosed
US-20190320656-A1 HERBICIDE COMBINATIONS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-10-24 US disclosed
US-20190200614-A1 AQUEOUS CAPSULE SUSPENSION CONCENTRATES BASED ON 2-[(2,4-DICHLOROPHENYL)METHYL]-4,4'-DIMETHYL-3-ISOXAZOLIDINONE FMC CORPORATION 2019-07-04 US disclosed
US-20190166840-A1 SUBSTITUTED PYRAZOLINYL DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND/OR PLANT GROWTH REGULATORS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-06-06 US disclosed
US-20190053484-A1 SOLVENT-FREE FORMULATIONS OF LOW-MELTING ACTIVE INGREDIENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-02-21 US disclosed
US-9968090-B2 Herbicide-safener compositions containing N-(1,3,4-oxadiazol-2-yl)aryl carboxylic acid amides BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-05-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (19 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190200614-A1 AQUEOUS CAPSULE SUSPENSION CONCENTRATES BASED ON 2-[(2,4-DICHLOROPHENYL)METHYL]-4,4'-DIMETHYL-3-ISOXAZOLIDINONE ACMSD, DDT, CCND2 BCL2L1 2108/4885MCL1 3862/4885FLT1 4757/4885
US-20200172491-A1 SUBSTITUTED 5-(HET-)ARYLPYRAZOLAMIDES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES CYP4Z1, CYP3A5, CYP4X1 BCL2L1 2697/4885MCL1 4361/4885FLT1 1782/4885
US-20210289781-A1 HERBICIDAL MIXTURES ATL3, DDT, CLSPN BCL2L1 1466/4885MCL1 1501/4885FLT1 3547/4885
US-20190053484-A1 SOLVENT-FREE FORMULATIONS OF LOW-MELTING ACTIVE INGREDIENTS CYP51A1, ABCG2, FASTKD5 BCL2L1 909/4885MCL1 1908/4885FLT1 4518/4885
US-20200181117-A1 SUBSTITUTED 3-HETEROARYLOXY-1H-PYRAZOLES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES GLRX3, CYP4F3, AGXT BCL2L1 1607/4885MCL1 3660/4885FLT1 1355/4885
US-11197477-B2 Aqueous capsule suspension concentrates based on 2-[(2,4-dichlorophenyl)methyl]-4,4′-dimethyl-3-isoxazolidinone ACMSD, DDT, CCND2 BCL2L1 2113/4885MCL1 3878/4885FLT1 4755/4885
US-11191265-B2 Method of reducing crop damage DDT, GAP43, GSS BCL2L1 413/4885MCL1 3402/4885FLT1 3144/4885
US-20210307322-A1 CONTROLLED RELEASE FORMULATIONS WITH LIGNIN FOR AGROCHEMICALS LCT, LSS, PGLS BCL2L1 901/4885MCL1 2757/4885FLT1 2594/4885
US-20210137117-A1 HERBICIDAL MIXTURES DDT, MTX2, ATL3 BCL2L1 1406/4885MCL1 2478/4885FLT1 4592/4885
US-20190320656-A1 HERBICIDE COMBINATIONS DDT, MTHFD2, DHFR BCL2L1 1371/4885MCL1 4398/4885FLT1 580/4885
US-20210276974-A1 SUBSTITUTED 2-HETEROARYLOXYPYRIDINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS DDT, AGPS, GMDS BCL2L1 875/4885MCL1 3541/4885FLT1 1013/4885
US-20210227824-A1 METHOD OF REDUCING CROP DAMAGE DDT, GAP43, GSS BCL2L1 413/4885MCL1 3402/4885FLT1 3144/4885
US-11219209-B2 Method of reducing crop damage DDT, GAP43, GSS BCL2L1 413/4885MCL1 3402/4885FLT1 3144/4885
US-20210289777-A1 METHOD OF REDUCING CROP DAMAGE DDT, GAP43, GSS BCL2L1 413/4885MCL1 3402/4885FLT1 3144/4885
US-20210127667-A1 METHOD OF REDUCING CROP DAMAGE DDT, GAP43, GSS BCL2L1 413/4885MCL1 3402/4885FLT1 3144/4885
US-20190166840-A1 SUBSTITUTED PYRAZOLINYL DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND/OR PLANT GROWTH REGULATORS HPD, GMDS, WEE1 BCL2L1 1282/4885MCL1 3488/4885FLT1 501/4885
US-20200085055-A1 New uses of 2-(2,4-dichlorophenyl)methyl-4,4-dimethyl-3-isoxazolidone as foliar herbicide DDT, DAO, CYP4X1 BCL2L1 1329/4885MCL1 3742/4885FLT1 3621/4885
US-20200196601-A1 HERBICIDE SAFENER COMPOSITIONS CONTAINING QUINAZOLINEDIONE-6CARBONYL DERIVATIVES CYP2F1, CYP2W1, CYP4F12 BCL2L1 923/4885MCL1 3462/4885FLT1 2471/4885
US-20190330192-A1 SUBSTITUTED AZOLYLPYRROLONES AND AZOLYLHYDANTOINS AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES AGPS, AASDHPPT, HPD BCL2L1 2320/4885MCL1 4466/4885FLT1 1308/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.