SCHEMBL2107628

SCHEMBL2107628

Fc1ccc(-c2noc(CCl)n2)cc1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.64
HTT P42858 1/20 0.64
RAB9A P51151 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
SIRT2 Q8IXJ6 4/20 0.62
NOTUM Q6P988 3/20 0.51
HDAC8 Q9BY41 3/20 0.50
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
MAPT P10636 2/20 0.50
S1PR1 P21453 1/20 0.49
TNKS2 Q9H2K2 2/20 0.47
THRB P10828 1/20 0.47
FFAR1 O14842 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL507782 0.84 NOTUM (0.72) NPC1HTTRAB9ASMN1; SMN2SIRT2
SCHEMBL201423 0.82 NOTUM (0.56) NPC1HTTRAB9ASMN1; SMN2SIRT2
SCHEMBL26232436 0.82 NPC1 (0.73) NPC1HTTRAB9ASMN1; SMN2SIRT2
SCHEMBL26009685 0.82 NOTUM (0.56) NPC1HTTRAB9ASMN1; SMN2SIRT2
SCHEMBL14948949 0.82 NOTUM (0.70) NPC1HTTRAB9ASMN1; SMN2SIRT2
SCHEMBL12617891 0.82 NOTUM (0.64) NPC1RAB9ASMN1; SMN2NOTUMMAPT
SCHEMBL28912728 0.82 SIRT2 (0.71) NPC1HTTRAB9ASMN1; SMN2SIRT2
SCHEMBL10937283 0.82 SIRT2 (0.71) NPC1HTTRAB9ASMN1; SMN2SIRT2
SCHEMBL10904042 0.82 SMN1; SMN2 (0.59) NPC1HTTRAB9ASMN1; SMN2MAPT
SCHEMBL25916014 0.82 NOTUM (0.51) NPC1HTTRAB9ASMN1; SMN2SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093377-B Haloalkyl-containing 1,2, 4-oxadiazole derivative and preparation method and application thereof 贵州大学 2023-04-07 CN claimed
CN-115093377-A Haloalkyl-containing 1,2, 4-oxadiazole derivative and preparation method and application thereof 贵州大学 2022-09-23 CN claimed
US-20250223278-A1 PYRIDAZINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. 2025-07-10 US disclosed
US-12240831-B2 Pyridazinone compounds and uses thereof EDGEWISE THERAPEUTICS, INC. (US) 2025-03-04 US disclosed
US-12012395-B2 Pyridazinone compounds and uses thereof EDGEWISE THERAPEUTICS, INC. (US) 2024-06-18 US disclosed
US-11970470-B1 {5-chloro-2-(2-(3-(substitutedphenyl)-1,2,4-oxadiazol-5-yl)ethyl)phenyl}(phenyl)methanones as larvicidal agents King Faisal University (SA) 2024-04-30 US disclosed
US-20240025879-A1 PYRIDAZINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. 2024-01-25 US disclosed
US-11873290-B2 2024-01-16 US disclosed
US-20230348476-A1 CBP/CATENIN SIGNALING PATHWAY INHIBITORS AND USES THEREOF 3 2 PHARMA LLC (US) 2023-11-02 US disclosed
US-20230348476-A1 CBP/CATENIN SIGNALING PATHWAY INHIBITORS AND USES THEREOF 3 2 PHARMA LLC (US) 2023-11-02 US disclosed
US-20230321091-A1 SUBSTITUTED PYRIDAZINONES FOR USE IN THE TREATMENT OF NEUROMUSCULAR DISEASES EDGEWISE THERAPEUTICS, INC. 2023-10-12 US disclosed
WO-2009139709-A1 QUINUCLIDINE DERIVATIVES AND THEIR USE AS MUSCARINIC RECEPTOR ANTAGONISTS FOR THE TREATMENT OF ASTHMA AND CHRONIC OBSTRUCTIVE PULMONARY DISEASE (COPD) ASTRAZENECA AB (SE) 2009-11-19 WO disclosed
US-20090209533-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION AMYGDALA NEUROSCIENCES, INC. 2009-08-20 US disclosed
WO-2009094028-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION CV THERAPEUTICS, INC. (US) 2009-07-30 WO disclosed
WO-2009061924-A2 ALDH-2 INHIBITORS IN THE TREATMENT OF PSYCHIATRIC DISORDERS CV THERAPEUTICS, INC. (US) 2009-05-14 WO disclosed
US-20090124672-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF PSYCHIATRIC DISORDERS AMYGDALA NEUROSCIENCES, INC. 2009-05-14 US disclosed
EP-2046769-A2 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION CV THERAPEUTICS, INC. (US) 2009-04-15 EP disclosed
US-20080207610-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION AMYGDALA NEUROSCIENCES, INC. 2008-08-28 US disclosed
US-20080032995-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF DRUG ADDICTION AMYGDALA NEUROSCIENCES, INC. 2008-02-07 US disclosed
WO-2008014497-A2 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION CV THERAPEUTICS, INC. (US) 2008-01-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230348476-A1 CBP/CATENIN SIGNALING PATHWAY INHIBITORS AND USES THEREOF CREBBP, CREB1, EP300 NPC1 1730/4885HTT 2537/4885RAB9A 2899/4885
US-20230321091-A1 SUBSTITUTED PYRIDAZINONES FOR USE IN THE TREATMENT OF NEUROMUSCULAR DISEASES IL6, MUSK, SMN1; SMN2 NPC1 4135/4885HTT 2529/4885RAB9A 2744/4885
US-12012395-B2 Pyridazinone compounds and uses thereof IL6, IL1B, IL1A NPC1 4205/4885HTT 3021/4885RAB9A 3148/4885
US-20080207610-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION ALDH1A1, ADH1A, ALDH3A1 NPC1 2592/4885HTT 3807/4885RAB9A 2946/4885
US-12240831-B2 Pyridazinone compounds and uses thereof IL6, IL1B, IL1A NPC1 4205/4885HTT 3021/4885RAB9A 3148/4885
US-11970470-B1 {5-chloro-2-(2-(3-(substitutedphenyl)-1,2,4-oxadiazol-5-yl)ethyl)phenyl}(phenyl)methanones as larvicidal agents CASP3, CASP2, CASP7 NPC1 1200/4885HTT 4304/4885RAB9A 3675/4885
US-11873290-B2 IL6, MUSK, IL6ST NPC1 4167/4885HTT 2657/4885RAB9A 3240/4885
US-20090209533-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION ALDH1A1, ADH1A, ALDH3A1 NPC1 2592/4885HTT 3807/4885RAB9A 2946/4885
US-20250223278-A1 PYRIDAZINONE COMPOUNDS AND USES THEREOF IL6, IL1B, IL1A NPC1 4205/4885HTT 3021/4885RAB9A 3148/4885
US-20080032995-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF DRUG ADDICTION ALDH1A1, ADH1A, ALDH3A1 NPC1 2682/4885HTT 3853/4885RAB9A 2475/4885
US-20090124672-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF PSYCHIATRIC DISORDERS ALDH2, ALDH1A2, ALDH1A1 NPC1 1978/4885HTT 3900/4885RAB9A 2092/4885
US-20240025879-A1 PYRIDAZINONE COMPOUNDS AND USES THEREOF IL6, IL1B, IL1A NPC1 4205/4885HTT 3021/4885RAB9A 3148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.