SCHEMBL2556418

SCHEMBL2556418

COc1ccc(C[C@@H](C)N)c(OC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.75
HTR1A P08908 1/20 0.59
HTR2C P28335 1/20 0.59
HTR2B P41595 1/20 0.59
TAAR1 Q96RJ0 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968339 1.00 HTR2A (0.75) HTR2AHTR1AHTR2CHTR2BTAAR1
SCHEMBL266899 1.00 HTR2A (0.75) HTR2AHTR1AHTR2CHTR2BTAAR1
SCHEMBL1740902 0.86 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BTAAR1
SCHEMBL31545209 0.86 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BTAAR1
SCHEMBL1740903 0.86 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BTAAR1
SCHEMBL3460220 0.86 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BTAAR1
SCHEMBL3027061 0.85 APLNR (0.59) HTR2A
Hydrochloric Acid SCHEMBL29542459 0.84 HTR2A (0.97) HTR2AHTR1AHTR2CHTR2BTAAR1
Hydrochloric Acid SCHEMBL3486527 0.84 HTR2A (0.97) HTR2AHTR1AHTR2CHTR2BTAAR1
Hydrochloric Acid SCHEMBL30861235 0.84 HTR2A (0.97) HTR2AHTR1AHTR2CHTR2BTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260108544-A1 TRYPTAMINE COMPOSITIONS FOR ENHANCING NEURITE OUTGROWTH TURTLE BEAR HOLDINGS LLC (US) 2026-04-23 US disclosed
US-12599578-B2 Compositions comprising enzyme-cleavable prodrugs and controlled release nafamostat and methods of use thereof Ensysce Biosciences Inc. (US) 2026-04-14 US disclosed
EP-4704806-A1 INJECTABLE PHARMACEUTICAL FORMULATIONS Cybin IRL Limited (IE) 2026-03-11 EP disclosed
EP-4673127-A1 DEUTERATED AND FLUORINATED EMPATHOGENS Alexander Shulgin Research Institute, Inc. (US) 2026-01-07 EP disclosed
EP-4673430-A2 PHENYLALKYLAMINE PRODRUGS Alexander Shulgin Research Institute, Inc. (US) 2026-01-07 EP disclosed
US-20250388529-A1 N-Substituted Phenylalkylamines and Their Use as Therapeutic Agents ALEXANDER SHULGIN RES INSTITUTE INC (US) 2025-12-25 US disclosed
US-12465578-B2 Substituted alpha-ethyl phenylalkylamines ALEXANDER SHULGIN RESEARCH INSTITUTE, INC. (US) 2025-11-11 US disclosed
US-20250195471-A1 ASYMMETRIC ALLYL TRYPTAMINES ALEXANDER SHULGIN RES INSTITUTE INC (US) 2025-06-19 US disclosed
US-12239632-B2 Asymmetric allyl tryptamines ALEXANDER SHULGIN RESEARCH INSTITUTE, INC. (US) 2025-03-04 US disclosed
US-20240408038-A1 SUBSTITUTED PHENYLALKYLAMINES ALEXANDER SHULGIN RESEARCH INSTITUTE, INC. 2024-12-12 US disclosed
US-20150025063-A1 Antiparkinsonian Action of Phenylisopropylamines UNIV DUKE (US) 2015-01-22 US disclosed
US-8877802-B2 Antiparkinsonian action of phenylisopropylamines Duke Univerity (US) 2014-11-04 US disclosed
US-20130059914-A1 Compositions Comprising Enzyme-Cleavable Amphetamine Prodrugs and Inhibitors Thereof SIGNATURE THERAPEUTICS, INC. (US) 2013-03-07 US disclosed
EP-2560486-A1 COMPOSITIONS COMPRISING ENZYME-CLEAVABLE AMPHETAMINE PRODRUGS AND INHIBITORS THEREOF Signature Therapeutics, Inc. (US) 2013-02-27 EP disclosed
WO-2012122412-A2 COMPOSITIONS FOR REDUCING RISK OF ADVERSE EVENTS CAUSED BY DRUG-DRUG INTERACTIONS SIGNATURE THERAPEUTICS, INC. (US) 2012-09-13 WO disclosed
US-20120232066-A1 COMPOSITIONS FOR REDUCING RISK OF ADVERSE EVENTS CAUSED BY DRUG-DRUG INTERACTIONS SIGNATURE THERAPEUTICS, INC. 2012-09-13 US disclosed
WO-2011133348-A1 COMPOSITIONS COMPRISING ENZYME-CLEAVABLE AMPHETAMINE PRODRUGS AND INHIBITORS THEREOF PHARMACOFORE, INC. (US) 2011-10-27 WO disclosed
WO-2011133347-A1 COMPOSITIONS COMPRISING TRYPSIN-CLEAVABLE AMPHETAMINE PRODRUGS AND INHIBITORS THEREOF PHARMACOFORE, INC. (US) 2011-10-27 WO disclosed
WO-2007016190-A2 ANTIPARKINSONIAN ACTION OF PHENYLISOPROPYLAMINES DUKE UNIVERSITY (US) 2007-02-08 WO disclosed
US-20070027208-A1 Antiparkinsonian Action of Phenylisopropylamines NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2007-02-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12239632-B2 Asymmetric allyl tryptamines TPH2, TPH1, HTR2A HTR2A 3/4885HTR1A 4/4885HTR2C 6/4885
US-20250388529-A1 N-Substituted Phenylalkylamines and Their Use as Therapeutic Agents CNR2, CNR1, HCN3 HTR2A 25/4885HTR1A 37/4885HTR2C 6/4885
US-20070027208-A1 Antiparkinsonian Action of Phenylisopropylamines PNMT, SNCA, COMT HTR2A 18/4885HTR1A 29/4885HTR2C 44/4885
US-20250195471-A1 ASYMMETRIC ALLYL TRYPTAMINES TPH2, TPH1, HTR2A HTR2A 3/4885HTR1A 4/4885HTR2C 6/4885
US-12465578-B2 Substituted alpha-ethyl phenylalkylamines PNMT, SLC18A2, SLC1A2 HTR2A 4/4885HTR1A 5/4885HTR2C 15/4885
US-20240408038-A1 SUBSTITUTED PHENYLALKYLAMINES PNMT, HTR2A, SLC18A2 HTR2A 2/4885HTR1A 4/4885HTR2C 8/4885
US-20150025063-A1 Antiparkinsonian Action of Phenylisopropylamines PNMT, SNCA, COMT HTR2A 18/4885HTR1A 29/4885HTR2C 44/4885
US-20120232066-A1 COMPOSITIONS FOR REDUCING RISK OF ADVERSE EVENTS CAUSED BY DRUG-DRUG INTERACTIONS CYP2C19, CYP3A5, CYP3A4 HTR2A 823/4885HTR1A 727/4885HTR2C 673/4885
US-12599578-B2 Compositions comprising enzyme-cleavable prodrugs and controlled release nafamostat and methods of use thereof OPRK1, OPRL1, OPRM1 HTR2A 2491/4885HTR1A 1360/4885HTR2C 1619/4885
US-20130059914-A1 Compositions Comprising Enzyme-Cleavable Amphetamine Prodrugs and Inhibitors Thereof ACHE, COMT, CES2 HTR2A 375/4885HTR1A 293/4885HTR2C 227/4885
US-20260108544-A1 TRYPTAMINE COMPOSITIONS FOR ENHANCING NEURITE OUTGROWTH HTR1B, HTR6, BDNF HTR2A 9/4885HTR1A 11/4885HTR2C 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.