SCHEMBL409080

SCHEMBL409080

CCC(C)(C)C(=O)NCCN(C)C

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DNM1 Q05193 2/20 0.44
RIPK1 Q13546 3/20 0.43
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
ALDH1A1 P00352 1/20 0.38
DRD2 P14416 2/20 0.38
DRD4 P21917 2/20 0.38
USP2 O75604 1/20 0.37
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPK1 P28482 1/20 0.36
PRMT3 O60678 1/20 0.34
CARM1 Q86X55 1/20 0.34
PRMT6 Q96LA8 1/20 0.34
PRMT1 Q99873 1/20 0.34
PRMT8 Q9NR22 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8279451 0.89 DNM1 (0.49) DNM1RIPK1ALDH1A1DRD2DRD4
SCHEMBL14153995 0.88 RIPK1 (0.43) DNM1RIPK1ALDH1A1DRD2DRD4
SCHEMBL16316500 0.83 RIPK1 (0.40) DNM1RIPK1DRD2DRD4
SCHEMBL14153992 0.83 RIPK1 (0.52) RIPK1ALDH1A1DRD2DRD4USP2
SCHEMBL24406352 0.82 DNM1 (0.40) DNM1CA1CA2CA12CA9
SCHEMBL21018349 0.82 ALDH1A1 (0.42) RIPK1ALDH1A1SMN1; SMN2MAPK1KMT2A
SCHEMBL2878101 0.82 DNM1 (0.40) DNM1CA1CA2CA12CA9
SCHEMBL22317342 0.82 DNM1 (0.51) DNM1CA1CA2CA12CA9
SCHEMBL10201790 0.81 DNM1 (0.44) DNM1CA1CA2CA12CA9
SCHEMBL14153988 0.81 RIPK1 (0.41) DNM1RIPK1ALDH1A1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230338415-A1 SUBSTITUTED PHENYL BORONIC ACID CONTAINING POLYMERS AND METHODS OF USE GLYSCEND, INC. 2023-10-26 US disclosed
US-10961202-B2 Bis-benzimidazole compounds and methods of using the same THE SCRIPPS RESEARCH INSTITUTE (US) 2021-03-30 US disclosed
US-20190152924-A1 BIS-BENZIMIDAZOLE COMPOUNDS AND METHODS OF USING THE SAME UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED 2019-05-23 US disclosed
US-20170273893-A1 AGENT FOR TEMPORARY SHAPING OF KERATIN-CONTAINING FIBERS HAVING A MIXTURE OF CONDITIONING POLYMERS HENKEL AG & CO. KGAA (DE) 2017-09-28 US disclosed
EP-2490659-B1 COMPOSITION FOR THE TEMPORARY SHAPING OF KERATINIC FIBRES COMPRISING A NONIONIC PROPYLENEOXIDE-MODIFIED STARCH AND A CHITOSAN HENKEL AG & CO KGAA (DE) 2017-03-01 EP disclosed
US-20150352032-A1 ARTIFICIAL NAIL COMPOSITION, ARTIFICIAL NAIL, METHOD FOR FORMING ARTIFICIAL NAIL, AND NAIL ART KIT FUJIFILM CORPORATION (JP) 2015-12-10 US disclosed
US-20140305462-A1 Powdery Hair Cosmetics HENKEL AG & CO. KGAA (DE) 2014-10-16 US disclosed
US-8785917-B2 Actinic ray-sensitive or radiation-sensitive resin composition, and actinic ray-sensitive or radiation-sensitive film and pattern forming method using the same FUJIFILM CORPORATION (JP) 2014-07-22 US disclosed
US-8785917-B2 Actinic ray-sensitive or radiation-sensitive resin composition, and actinic ray-sensitive or radiation-sensitive film and pattern forming method using the same FUJIFILM CORPORATION (JP) 2014-07-22 US disclosed
WO-2014095166-A2 COMPOSITIONS FOR SHAPING KERATIN FIBERS HENKEL AG & CO. KGAA (DE) 2014-06-26 WO disclosed
US-20130001751-A1 ACTINIC RAY-SENSITIVE OR RADIATION-SENSITIVE RESIN COMPOSITION, AND ACTINIC RAY-SENSITIVE OR RADIATION-SENSITIVE FILM AND PATTERN FORMING METHOD USING THE SAME FUJIFILM CORPORATION (JP) 2013-01-03 US disclosed
US-8329384-B2 Resist-modifying composition and pattern forming process SHIN-ETSU CHEMICAL CO., LTD. (JP) 2012-12-11 US disclosed
US-20120207693-A1 AGENT FOR KERATIN-CONTAINING FIBERS, COMPRISING AT LEAST ONE NON-IONIC STARCH MODIFIED BY PROPYLENE OXIDE AND AT LEAST ONE ADDITIONAL FILM-FORMING CATIONIC AND/OR STABILIZING POLYMER MUELLER BURKHARD (DE) 2012-08-16 US disclosed
US-20120064023-A1 AGENTS FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIAL CROSS-LINKED AMPHIPHILIC, ANIONIC POLYMER AND AT LEAST ONE FURTHER SPECIAL NON-CROSS-LINKED AMPHIPHILIC ANIONIC POLYMER HENKEL AG & CO. KGAA (DE) 2012-03-15 US disclosed
US-20110135590-A1 PRODUCT FOR KERATIN-CONTAINING FIBERS COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC, CATIONIC POLYMER, AND AT LEAST ONE POLYOL KNAPPE THORSTEN 2011-06-09 US disclosed
US-20110135591-A1 AGENT FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE ADDITIONAL FILM-FORMING CATIONIC AND/OR STABILIZING POLYMER HENKEL AG & CO. KGAA (DE) 2011-06-09 US disclosed
US-20100297563-A1 RESIST-MODIFYING COMPOSITION AND PATTERN FORMING PROCESS SHIN-ETSU CHEMICAL CO., LTD. (JP) 2010-11-25 US disclosed
US-20070225285-A1 5-LIPOXYGENASE-ACTIVATING PROTEIN (FLAP) INHIBITORS AMIRA PHARMACEUTICALS, INC. (US) 2007-09-27 US disclosed
US-7186786-B2 Chain transfer agents for RAFT polymerization in aqueous media UNIVERSITY OF SOUTHERN MISSISSIPPI (US) 2007-03-06 US disclosed
US-7179872-B2 Chain transfer agents for RAFT polymerization in aqueous media UNIVERSITY OF SOUTHERN MISSISSIPPI (US) 2007-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120207693-A1 AGENT FOR KERATIN-CONTAINING FIBERS, COMPRISING AT LEAST ONE NON-IONIC STARCH MODIFIED BY PROPYLENE OXIDE AND AT LEAST ONE ADDITIONAL FILM-FORMING CATIONIC AND/OR STABILIZING POLYMER KRT18, FLNA, CUTA DNM1 2895/4885RIPK1 3831/4885CA1 3140/4885
US-20110135590-A1 PRODUCT FOR KERATIN-CONTAINING FIBERS COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC, CATIONIC POLYMER, AND AT LEAST ONE POLYOL KRT18, F12, H1-10 DNM1 2550/4885RIPK1 4220/4885CA1 2482/4885
US-10961202-B2 Bis-benzimidazole compounds and methods of using the same HNRNPH1, HNRNPH3, HNRNPUL2 DNM1 1376/4885RIPK1 3980/4885CA1 4481/4885
US-20120064023-A1 AGENTS FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIAL CROSS-LINKED AMPHIPHILIC, ANIONIC POLYMER AND AT LEAST ONE FURTHER SPECIAL NON-CROSS-LINKED AMPHIPHILIC ANIONIC POLYMER KRT18, DSG1, CUTA DNM1 3463/4885RIPK1 4244/4885CA1 1954/4885
US-20070225285-A1 5-LIPOXYGENASE-ACTIVATING PROTEIN (FLAP) INHIBITORS ALOX5, ALOX15B, ALOX15 DNM1 2877/4885RIPK1 469/4885CA1 4787/4885
US-20110135591-A1 AGENT FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE ADDITIONAL FILM-FORMING CATIONIC AND/OR STABILIZING POLYMER KRT18, POLR1C, F12 DNM1 1185/4885RIPK1 3734/4885CA1 2531/4885
US-20150352032-A1 ARTIFICIAL NAIL COMPOSITION, ARTIFICIAL NAIL, METHOD FOR FORMING ARTIFICIAL NAIL, AND NAIL ART KIT NACA, PIK3C3, POLR1C DNM1 2872/4885RIPK1 2840/4885CA1 2668/4885
US-20140305462-A1 Powdery Hair Cosmetics CUTA, SHH, H1-0 DNM1 2903/4885RIPK1 4721/4885CA1 3362/4885
US-20230338415-A1 SUBSTITUTED PHENYL BORONIC ACID CONTAINING POLYMERS AND METHODS OF USE SLC10A2, PYGL, SLC10A1 DNM1 3976/4885RIPK1 3307/4885CA1 1553/4885
US-20190152924-A1 BIS-BENZIMIDAZOLE COMPOUNDS AND METHODS OF USING THE SAME HNRNPH1, HNRNPH3, HNRNPUL2 DNM1 1376/4885RIPK1 3980/4885CA1 4481/4885
US-20170273893-A1 AGENT FOR TEMPORARY SHAPING OF KERATIN-CONTAINING FIBERS HAVING A MIXTURE OF CONDITIONING POLYMERS KRT18, DSG1, CD69 DNM1 4572/4885RIPK1 3409/4885CA1 1244/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.