SCHEMBL437306

SCHEMBL437306

CNC(=O)CN1C(=O)C=CC1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.50
GSK3B P49841 1/20 0.50
POLB P06746 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MGLL Q99685 4/20 0.44
ALDH1A1 P00352 3/20 0.44
BLM P54132 2/20 0.44
LMNA P02545 2/20 0.44
MAPT P10636 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
GMNN O75496 1/20 0.44
THPO P40225 1/20 0.44
PMP22 Q01453 1/20 0.44
HPGD P15428 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
WRN Q14191 1/20 0.42
HIF1A Q16665 1/20 0.42
PLK1 P53350 1/20 0.41
GAA P10253 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19545832 0.83 GSK3A (0.47) GSK3AGSK3BKDM4EMGLLALDH1A1
SCHEMBL29995038 0.82 GSK3A (0.48) GSK3AGSK3BKDM4EMGLLALDH1A1
SCHEMBL22281365 0.80 GSK3A (0.47) GSK3AGSK3BMGLLALDH1A1BLM
SCHEMBL836019 0.79 PTGS1 (0.47) GSK3AGSK3BPOLBMGLLALDH1A1
SCHEMBL3665093 0.79 GSK3A (0.52) GSK3AGSK3BKDM4EMGLLALDH1A1
SCHEMBL8738193 0.78 GSK3A (0.46) GSK3AGSK3BKDM4EMGLLALDH1A1
SCHEMBL7049984 0.78 GSK3A (0.50) GSK3AGSK3BKDM4EMGLLALDH1A1
SCHEMBL15386866 0.78 KMT2A (0.56) GSK3AGSK3BPOLBKDM4EMGLL
SCHEMBL25699409 0.77 GSK3A (0.42) GSK3AGSK3BMGLLALDH1A1BLM
SCHEMBL20287639 0.76 GSK3A (0.44) GSK3AGSK3BPOLBMGLLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12036285-B2 Immunogenic conjugates and use thereof GLAXOSMITHKLINE BIOLOGICALS SA (BE) 2024-07-16 US disclosed
US-11795195-B2 Antibody-drug conjugates including hemiasterlin derivative Sumitomo Pharma Co., Ltd. (JP) 2023-10-24 US disclosed
US-20230137914-A1 nOMV-ANTIGEN CONJUGATED COMPOUNDS AND USE THEREOF GLAXOSMITHKLINE BIOLOGICALS, S.A. (BE) 2023-05-04 US disclosed
US-20230137821-A1 IMMUNOGENIC CONJUGATES AND USE THEREOF GLAXOSMITHKLINE BIOLOGICALS, S.A. (BE) 2023-05-04 US disclosed
US-11092594-B2 Haptens, hapten conjugates, compositions thereof and method for their preparation and use VENTANA MEDICAL SYSTEMS, INC. (US) 2021-08-17 US disclosed
US-10561739-B2 Targeted pyrrolobenzodiazapine conjugates SEATTLE GENETICS INC. (US) 2020-02-18 US disclosed
US-10016512-B2 Immobilised biological entities CARMEDA AB (SE) 2018-07-10 US disclosed
US-20180140713-A1 IMMOBILISED BIOLOGICAL ENTITIES CARMEDA AB (SE) 2018-05-24 US disclosed
US-20180120306-A1 HAPTENS, HAPTEN CONJUGATES, COMPOSITIONS THEREOF AND METHOD FOR THEIR PREPARATION AND USE VENTANA MED SYST INC (US) 2018-05-03 US disclosed
US-20170368237-A1 IMMOBILISED BIOLOGICAL ENTITIES GORE & ASS (US) 2017-12-28 US disclosed
EP-2143736-A1 Hydroxyalkyl starch derivatives Fresenius Kabi Deutschland GmbH (DE) 2010-01-13 EP disclosed
US-20090317328-A1 TRICYCLIC OXAZEPINES AS IN VIVO IMAGING COMPOUNDS ARSTAD ERIK 2009-12-24 US disclosed
US-7601332-B2 Minimized toxicity; eliminating pathogenic cell populations; synthesis; claimed intermediates ENDOCYTE, INC. (US) 2009-10-13 US disclosed
US-20090181398-A1 Nanoparticle conjugates VENTANA MEDICAL SYSTEMS, INC. 2009-07-16 US disclosed
US-20090176253-A1 Antibody conjugates VENTANA MEDICAL SYSTEMS, INC. 2009-07-09 US disclosed
EP-2017287-A2 Method of producing hydroxyalkyl starch derivatives Fresenius Kabi Deutschland GmbH (DE) 2009-01-21 EP disclosed
US-20080292547-A1 Novel Imaging Agents for Fibrosis TOLLESHAUG HELGE 2008-11-27 US disclosed
US-20080279765-A1 Novel Imaging Agents for Fibrosis CHETTIBI SALAH 2008-11-13 US disclosed
US-20080268462-A1 Derivatives containing oxazole, pyrazole, thiazole, nitroaryl compound, benzofurazan, triterpene, urea, thiourea, rotenoid, coumarin or cyclolignan such as 4-(2-hydroxyphenyl)-1H-benzo[b][1,4]diazepine-2(3H)-one; multiplexed diagnostic assay for multiple targets in sample; antibodies; kits VENTANA MEDICAL SYSTEMS, INC. 2008-10-30 US disclosed
EP-1398327-B1 Method of producing hydroxyalkyl starch derivatives FRESENIUS KABI DE GMBH (DE) 2008-08-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080268462-A1 Derivatives containing oxazole, pyrazole, thiazole, nitroaryl compound, benzofurazan, triterpene, urea, thiourea, rotenoid, coumarin or cyclolignan such as 4-(2-hydroxyphenyl)-1H-benzo[b][1,4]diazepine-2(3H)-one; multiplexed diagnostic assay for multiple targets in sample; antibodies; kits HRH4, CRBN, NCDN GSK3A 2940/4885GSK3B 2797/4885POLB 3693/4885
US-20180120306-A1 HAPTENS, HAPTEN CONJUGATES, COMPOSITIONS THEREOF AND METHOD FOR THEIR PREPARATION AND USE CRBN, AHR, RORB GSK3A 1917/4885GSK3B 1866/4885POLB 3921/4885
US-20230137821-A1 IMMUNOGENIC CONJUGATES AND USE THEREOF VAPB, CHMP4B, CD14 GSK3A 4767/4885GSK3B 4699/4885POLB 3969/4885
US-20080279765-A1 Novel Imaging Agents for Fibrosis M6PR, IGF2R, MPI GSK3A 2676/4885GSK3B 2386/4885POLB 4784/4885
US-20230137914-A1 nOMV-ANTIGEN CONJUGATED COMPOUNDS AND USE THEREOF VAPB, CD14, CHMP4B GSK3A 4820/4885GSK3B 4759/4885POLB 3999/4885
US-10561739-B2 Targeted pyrrolobenzodiazapine conjugates QDPR, SBDS, DNPEP GSK3A 4103/4885GSK3B 3939/4885POLB 2322/4885
US-20180140713-A1 IMMOBILISED BIOLOGICAL ENTITIES FGB, SELE, EPCAM GSK3A 3514/4885GSK3B 3847/4885POLB 4441/4885
US-11795195-B2 Antibody-drug conjugates including hemiasterlin derivative HSD3B2, HSD3B1, HSD11B2 GSK3A 333/4885GSK3B 229/4885POLB 4594/4885
US-20090317328-A1 TRICYCLIC OXAZEPINES AS IN VIVO IMAGING COMPOUNDS CNR2, CNR1, OPRL1 GSK3A 784/4885GSK3B 485/4885POLB 967/4885
US-12036285-B2 Immunogenic conjugates and use thereof VAPB, CHMP4B, CD14 GSK3A 4767/4885GSK3B 4699/4885POLB 3969/4885
US-10016512-B2 Immobilised biological entities FGB, SELE, EPCAM GSK3A 3514/4885GSK3B 3847/4885POLB 4441/4885
US-20080292547-A1 Novel Imaging Agents for Fibrosis LOXL1, LOXL2, LOXL3 GSK3A 2451/4885GSK3B 2018/4885POLB 4032/4885
US-11092594-B2 Haptens, hapten conjugates, compositions thereof and method for their preparation and use CRBN, AHR, RORB GSK3A 1917/4885GSK3B 1866/4885POLB 3921/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.