SCHEMBL507839

SCHEMBL507839

OCc1ccc(Br)cc1F

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 1/20 0.46
DGAT1 O75907 1/20 0.44
PDPK1 O15530 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.41
KDM1A O60341 1/20 0.41
AKR1B1 P15121 4/20 0.40
HSD17B10 Q99714 2/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
KMT2A Q03164 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
NAAA Q02083 1/20 0.39
MAPK1 P28482 1/20 0.38
CHRM5 P08912 1/20 0.38
USP28 Q96RU2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20465747 1.00 PYCR1 (0.46) PYCR1DGAT1PDPK1PTGDR2KDM1A
SCHEMBL5826 0.83 PDPK1 (0.48) PYCR1DGAT1PDPK1KDM1AAKR1B1
SCHEMBL135165 0.82 PTGDR2 (0.49) DGAT1PTGDR2HSD17B10MEN1KMT2A
SCHEMBL8828 0.79 CA2 (0.54) PYCR1DGAT1PDPK1KDM1AAKR1B1
SCHEMBL20465750 0.79 PYCR1 (0.47) PYCR1DGAT1PDPK1KDM1AAKR1B1
SCHEMBL308050 0.79 PYCR1 (0.47) PYCR1DGAT1PDPK1KDM1AAKR1B1
SCHEMBL11918441 0.79 ALOX15 (0.46) PTGDR2CYP1A2CYP2C9
SCHEMBL15806743 0.79 PYCR1 (0.47) PYCR1DGAT1PDPK1KDM1AAKR1B1
SCHEMBL31448605 0.79 PYCR1 (0.47) PYCR1DGAT1PDPK1KDM1AAKR1B1
SCHEMBL30380405 0.79 ALOX15 (0.46) PTGDR2CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 368 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260049092-A1 ANTIBACTERIAL COMPOUNDS BLACKSMITH MEDICINES INC (US) 2026-02-19 US disclosed
US-20260035362-A1 GLP-1R AGONISTS AND USES THEREOF QILU REGOR THERAPEUTICS INC (CN) 2026-02-05 US disclosed
US-12509423-B2 Compound, aldehyde dehydrogenase 2 activating agent, pharmaceutical composition, and therapeutic and/or prophylactic drug ALCHEMEDICINE, INC. (JP) 2025-12-30 US disclosed
US-12503452-B2 Antimicrobial compounds and methods CURZA GLOBAL, LLC (US) 2025-12-23 US disclosed
US-20250361210-A1 3,4-DIHYDROQUINOLIN-2(1H)-ONE COMPOUND KISSEI PHARMACEUTICAL CO., LTD. (JP) 2025-11-27 US disclosed
US-20250333429-A1 MODULATORS OF TNF-ALPHA ACTIVITY FORWARD THERAPEUTICS INC (US) 2025-10-30 US disclosed
EP-4638436-A1 PRMT5 INHIBITORS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2025-10-29 EP disclosed
EP-4622981-A1 MODULATORS OF TNF-ALPHA ACTIVITY Forward Therapeutics, Inc. (US) 2025-10-01 EP disclosed
US-20250263402-A1 BENZIMIDAZOLONE GLP-1 RECEPTOR AGONIST AND USE THEREOF HANGZHOU ZHONGMEIHUADONG PHARMACEUTICAL CO., LTD. (CN) 2025-08-21 US disclosed
US-12384808-B2 Modulators of TNF-α activity FORWARD THERAPEUTICS, INC. (US) 2025-08-12 US disclosed
EP-1343775-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-09-17 EP disclosed
WO-2003002118-A1 SUBSTITUTED 8-ARYLQUINOLINE PDE4 INHIBITORS MERCK FROSST CANADA & CO. (CA) 2003-01-09 WO disclosed
US-20020143020-A1 Novel piperazine derivatives VERNALIS RESEARCH LIMITED (GB) 2002-10-03 US disclosed
US-6452056-B1 REDUCING FLUORINATED BENZONITRILE TO A BENZYLAMINE WHICH IS REPLACED WITH A HYDROXYL GROUP ASAHI GLASS COMPANY, LIMITED (JP) 2002-09-17 US disclosed
WO-2002048124-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-20 WO disclosed
CN-1349963-A Direct method of reducing sodium bisuflite affixture of adhehyde or methyl ketone into correspondent alcohol SHANGHAI INST ORGANIC CHEM (CN) 2002-05-22 CN disclosed
CN-1077095-C Preparation method of p-fluorophenol BROMINE COMPOUNDS LTD (IL) 2002-01-02 CN disclosed
CN-1312783-A Process for preparing fluorobenzyl derivatives ASASHI GLASS CO (JP) 2001-09-12 CN disclosed
EP-1114809-A1 PROCESS FOR THE PREPARATION OF FLUOROBENZYL DERIVATIVES Asahi Glass Co., Ltd. (JP) 2001-07-11 EP disclosed
CN-1208398-A Preparation method of p-fluorophenol BROMINE COMPOUNDS LTD (IL) 1999-02-17 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260035362-A1 GLP-1R AGONISTS AND USES THEREOF GLP1R, GPR119, IAPP PYCR1 1128/4885DGAT1 1327/4885PDPK1 334/4885
US-12509423-B2 Compound, aldehyde dehydrogenase 2 activating agent, pharmaceutical composition, and therapeutic and/or prophylactic drug ALDH2, ALDH1A1, ADH1A PYCR1 1612/4885DGAT1 352/4885PDPK1 1231/4885
US-20250263402-A1 BENZIMIDAZOLONE GLP-1 RECEPTOR AGONIST AND USE THEREOF GLP1R, GIPR, GCGR PYCR1 1671/4885DGAT1 1377/4885PDPK1 371/4885
US-20260049092-A1 ANTIBACTERIAL COMPOUNDS H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CBR1, FPR1 PYCR1 64/4885DGAT1 948/4885PDPK1 3421/4885
US-20020143020-A1 Novel piperazine derivatives CYP4B1, UGT1A1, CYP1B1 PYCR1 1188/4885DGAT1 2449/4885PDPK1 2550/4885
US-12384808-B2 Modulators of TNF-α activity TNF, NFKBIA, TNFRSF1A PYCR1 3790/4885DGAT1 1528/4885PDPK1 1059/4885
US-20250333429-A1 MODULATORS OF TNF-ALPHA ACTIVITY TNF, NFKBIA, TNFRSF1A PYCR1 3654/4885DGAT1 1768/4885PDPK1 1155/4885
US-20250361210-A1 3,4-DIHYDROQUINOLIN-2(1H)-ONE COMPOUND TSHR, TRHR, GHSR PYCR1 2651/4885DGAT1 2748/4885PDPK1 816/4885
US-12503452-B2 Antimicrobial compounds and methods MPO, NISCH, RPN2 PYCR1 2907/4885DGAT1 598/4885PDPK1 2714/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.