SCHEMBL6580109

SCHEMBL6580109

NCCN(C(C(=O)[O-])c1ccccc1O)C(C(=O)O)c1ccccc1O.NCCN(C(C(=O)[O-])c1ccccc1O)C(C(=O)O)c1ccccc1O.NCCN(C(C(=O)[O-])c1ccccc1O)C(C(=O)O)c1ccccc1O.NCCN(C(C(=O)[O-])c1ccccc1O)C(C(=O)O)c1ccccc1O.[Fe+3].[Na+]

nearest known ligand 0.34

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 known ✓ P14867 1/20 0.30
GABRB2 known ✓ P47870 1/20 0.30
PTGS1 known ✓ P23219 1/20 0.30
PTGS2 known ✓ P35354 1/20 0.30
PTPN9 P43378 1/20 0.34
ALPL P05186 1/20 0.33
POLB P06746 1/20 0.33
ALPG P10696 1/20 0.33
ALOX15 P16050 1/20 0.32
HPGD P15428 2/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.31
ADRB2 P07550 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
HRH1 P35367 1/20 0.31
CX3CR1 P49238 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19362158 0.99 POLB (0.34) PTPN9ALPLPOLBALPGALOX15
SCHEMBL10615720 0.93 PTPN9 (0.35) PTPN9ALPLPOLBALPGALOX15
SCHEMBL157144 0.90 TSHR (0.37) POLBALOX15HPGDKDM4EALDH1A1
SCHEMBL4729408 0.74 TSHR (0.37) PTPN9POLBALOX15ALDH1A1TSHR
SCHEMBL4663927 0.73 KMT2A (0.35) HPGDALDH1A1TDP1PTGS1
SCHEMBL2797912 0.71 KDM4E (0.42) POLBHPGDKDM4EALDH1A1TSHR
SCHEMBL487951 0.71 LMNA (0.43) POLBALOX15HPGDKDM4EALDH1A1
SCHEMBL2799841 0.71 ALDH1A1 (0.44) POLBHPGDKDM4EALDH1A1ADRB2
Ethylenediamine SCHEMBL5159409 0.70 TSHR (0.40) PTPN9ALPLPOLBALPGHPGD
Ethylenediamine SCHEMBL7181567 0.69 HPGD (0.40) PTPN9ALPLPOLBALPGHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1413197-A2 Method of preparation of a stomach-action molluscicides Young, Colin Leslie (AU) 2004-04-28 EP disclosed
US-6447794-B2 INCLUDING A METAL COMPLEXONE AS AN ACTIVE INGREDIENT; SUCH AS IRON AND CALCIUM WITH ETHYLENEDIAMINETETRAACETIC ACID (EDTA) Young, Colin Leslie (AU) 2002-09-10 US disclosed
US-20020006426-A1 Stomach-action molluscicides YOUNG, COLIN LESLIE (AU) 2002-01-17 US disclosed
US-6093416-A COMPRISING AN IRON COMPLEXES OF ETHYLENEDIAMINETETRAACETIC ACID YOUNG, COLIN LESLIE (AU) 2000-07-25 US disclosed
EP-0921726-A4 STOMACH-ACTION MOLLUSCICIDES YOUNG COLIN LESLIE (AU) 2000-06-21 EP disclosed
EP-0921726-A1 STOMACH-ACTION MOLLUSCICIDES Young, Colin Leslie (AU) 1999-06-16 EP disclosed
WO-1997026789-A1 STOMACH-ACTION MOLLUSCICIDES YOUNG COLIN LESLIE (AU) 1997-07-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020006426-A1 Stomach-action molluscicides HRH2, MDH1, OGDH GABRA1 2954/4885GABRB2 1933/4885PTGS1 1167/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.