SCHEMBL916360

SCHEMBL916360

O=Nc1ccc(O)c(=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.59
TDP1 Q9NUW8 2/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
HSP90AA1 P07900 2/20 0.59
KDM4E B2RXH2 1/20 0.59
MAPT P10636 1/20 0.59
TYR P14679 1/20 0.46
ALDH1A1 P00352 3/20 0.44
HSD17B10 Q99714 3/20 0.44
DBH P09172 3/20 0.44
MMP2 P08253 1/20 0.44
TSHR P16473 2/20 0.39
TP53 P04637 1/20 0.39
HIF1A Q16665 1/20 0.39
HTT P42858 2/20 0.37
CYP3A4 P08684 1/20 0.37
PDE4A P27815 1/20 0.34
BLVRB P30043 1/20 0.34
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10616379 0.75 MEN1 (1.00) MAPK1TDP1MEN1KMT2AHSP90AA1
SCHEMBL234461 0.74 ALDH1A1 (0.58) MAPK1TDP1MEN1KMT2AHSP90AA1
SCHEMBL31217749 0.73 ALDH1A1 (0.38) MAPK1TDP1MEN1KMT2AHSP90AA1
SCHEMBL10339603 0.73 TYR (0.54) MAPK1TDP1MEN1KMT2AHSP90AA1
SCHEMBL107699 0.73
SCHEMBL3316934 0.72 PTGS2 (0.48) MAPK1TDP1MEN1KMT2AHSP90AA1
SCHEMBL24265884 0.70 KDM4E (0.42) MAPK1TDP1MEN1KMT2AHSP90AA1
SCHEMBL31493923 0.70 ALDH1A1 (0.50) MAPK1TDP1MEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL28416859 0.70 CA2 (0.50) MAPK1TDP1MEN1KMT2AKDM4E
SCHEMBL3673256 0.70 ALDH1A1 (0.50) MAPK1TDP1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240018105-A1 TROPOLONE DERIVATIVES AND TAUTOMERS THEREOF FOR IRON REGULATION IN ANIMALS KINESID THERAPEUTICS, INC. (US) 2024-01-18 US disclosed
WO-2021076938-A1 TROPOLONE DERIVATIVES AND TAUTOMERS THEREOF FOR IRON REGULATION IN ANIMALS Ambys Medicines, Inc. (US) 2021-04-22 WO disclosed
WO-2021076945-A1 TROPOLONE DERIVATIVES AND TAUTOMERS THEREOF FOR IRON REGULATION IN ANIMALS Ambys Medicines, Inc. (US) 2021-04-22 WO disclosed
US-10980754-B2 Anti-fungal compounds SAINT LOUIS UNIVERSITY (US) 2021-04-20 US disclosed
US-10980754-B2 Anti-fungal compounds SAINT LOUIS UNIVERSITY (US) 2021-04-20 US disclosed
WO-2020138265-A1 METHOD, APPARATUS AND PROGRAM FOR ASSESSING AMYLOID FORMATION 国立大学法人室蘭工業大学 2020-07-02 WO disclosed
US-10463664-B2 Inhibitors of HSV nucleotidyl transferases and uses therefor SAINT LOUIS UNIVERSITY (US) 2019-11-05 US disclosed
US-10329542-B2 HBV RNAse H purification and enzyme inhibitors SAINT LOUIS UNIVERSITY (US) 2019-06-25 US disclosed
US-10329542-B2 HBV RNAse H purification and enzyme inhibitors SAINT LOUIS UNIVERSITY (US) 2019-06-25 US disclosed
US-20190099385-A1 ANTI-FUNGAL COMPOUNDS SAINT LOUIS UNIVERSITY (US) 2019-04-04 US disclosed
US-7259187-B2 Tropolone derivatives RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2007-08-21 US disclosed
US-7259187-B2 Tropolone derivatives RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2007-08-21 US disclosed
EP-1802973-A2 METHODS FOR ALTERING SURFACE CHARACTERISTICS OF MICROSPHERES Luminex Corporation (US) 2007-07-04 EP disclosed
WO-2006044275-A2 METHODS FOR ALTERING SURFACE CHARACTERISTICS OF MICROSPHERES LUMINEX CORPORATION (US) 2006-04-27 WO disclosed
US-20060078997-A1 Methods for altering surface characteristics of microspheres LUMINEX CORPORATION 2006-04-13 US disclosed
US-4754041-A 3-acylamino-2-oxo-1-azetidinesulfonic acids E. R. SQUIBB & SONS, INC. (US) 1988-06-28 US disclosed
US-4638062-A 3-acylamino-2-oxo-1-azetidinesulfonic acids E. R. SQUIBB & SONS, INC. (US) 1987-01-20 US disclosed
US-4183955-A Troponyl-oxamic acid derivatives for treating allergic conditions Ayerst. McKenna & Harrison Limited (CA) 1980-01-15 US disclosed
US-4125625-A ANTIALLERGENS AYERST, MCKENNA & HARRISON LIMITED (CA) 1978-11-14 US disclosed
US-4057556-A ANTIALLERGENS AYERST, MCKENNA & HARRISON LTD. (CA) 1977-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240018105-A1 TROPOLONE DERIVATIVES AND TAUTOMERS THEREOF FOR IRON REGULATION IN ANIMALS TXNRD2, TXNRD1, SDHB MAPK1 2798/4885TDP1 503/4885MEN1 2972/4885
US-20190099385-A1 ANTI-FUNGAL COMPOUNDS ERG28, NANS, DPM1 MAPK1 1371/4885TDP1 3088/4885MEN1 1879/4885
US-10980754-B2 Anti-fungal compounds ERG28, NANS, DPM1 MAPK1 1371/4885TDP1 3088/4885MEN1 1879/4885
US-10463664-B2 Inhibitors of HSV nucleotidyl transferases and uses therefor TYMP, TYMS, NAMPT MAPK1 3786/4885TDP1 218/4885MEN1 2603/4885
US-10329542-B2 HBV RNAse H purification and enzyme inhibitors RNASEH1, RNASE1, RNASEL MAPK1 3951/4885TDP1 1014/4885MEN1 2978/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.