SCHEMBL945677

SCHEMBL945677

CCCCC/C=C\C/C=C\C/C=C\CCCCCOC(C)C(OCCCCC/C=C\C/C=C\C/C=C\CCCCC)N(C)C

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
CNR1 P21554 1/20 0.54
CNR2 P34972 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL170865 1.00 ALDH1A1 (0.54) ALDH1A1CNR1CNR2
SCHEMBL251553 0.95 CNR1 (0.46) ALDH1A1CNR1CNR2
SCHEMBL251555 0.95 CNR1 (0.46) ALDH1A1CNR1CNR2
SCHEMBL27320 0.91 ALDH1A1 (0.43) ALDH1A1CNR1CNR2
SCHEMBL1921025 0.87 ALDH1A1 (0.56) ALDH1A1CNR1CNR2
SCHEMBL5561906 0.86 SPHK1 (0.43)
SCHEMBL251629 0.86 SPHK1 (0.43)
SCHEMBL30290989 0.82 ALDH1A1 (0.50) ALDH1A1CNR1CNR2
SCHEMBL15018073 0.81 ALDH1A1 (0.55) ALDH1A1CNR1CNR2
SCHEMBL15018493 0.81 ALDH1A1 (0.55) ALDH1A1CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 189 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122094668-A Preparation method and application of lipid nanoparticle 2026-05-26 CN claimed
EP-3201338-B1 COMPOSITIONS AND METHODS FOR SILENCING HEPATITIS B VIRUS GENE EXPRESSION ARBUTUS BIOPHARMA CORP (CA) 2021-11-03 EP claimed
US-20210284733-A1 ANTI-PD-1 ANTIBODIES, OR FRAGMENTS THEREOF, FOR TREATING HEPATITIS B ARBUTUS BIOPHARMA CORPORATION (CA) 2021-09-16 US claimed
US-20200385721-A1 DELIVERING CRISPR THERAPEUTICS WITH LIPID NANOPARTICLES ARBUTUS BIOPHARMA CORPORATION (CA) 2020-12-10 US claimed
US-10626393-B2 Delivering CRISPR therapeutics with lipid nanoparticles ARBUTUS BIOPHARMA CORPORATION (CA) 2020-04-21 US claimed
US-20190336611-A1 HYBRID CARRIERS FOR NUCLEIC ACID CARGO CUREVAC AG (DE) 2019-11-07 US claimed
US-20190328664-A1 METHODS FOR AMELIORATING INFUSION REACTIONS ARBUTUS BIOPHARMA CORPORATION (CA) 2019-10-31 US claimed
US-10415037-B2 Compositions and methods for silencing hepatitis B virus gene expression ARBUTUS BIOPHARMA CORPORATION (CA) 2019-09-17 US claimed
US-20190032051-A1 NON-LIPOSOMAL SYSTEMS FOR NUCLEIC ACID DELIVERY PROTIVA BIOTHERAPEUTICS, INC. (CA) 2019-01-31 US claimed
US-20180245077-A1 COMPOSITIONS AND METHODS FOR TREATING HYPERTRIGLYCERIDEMIA PROTIVA BIOTHERAPEUTICS, INC. (CA) 2018-08-30 US claimed
US-20160076035-A1 COMPOSITIONS AND METHODS FOR SILENCING MARBURG VIRUS GENE EXPRESSION PROTIVA BIOTHERAPEUTICS, INC. (CA) 2016-03-17 US claimed
US-20160032320-A1 NON-LIPOSOMAL SYSTEMS FOR NUCLEIC ACID DELIVERY ARBUTUS BIOPHARMA CORPORATION (CA) 2016-02-04 US claimed
US-20140248338-A1 COMPOSITIONS AND METHODS FOR SILENCING ALDEHYDE DEHYDROGENASE PROTIVA BIOTHERAPEUTICS, INC. (CA) 2014-09-04 US claimed
US-8716464-B2 Compositions and methods for silencing Ebola virus gene expression PROTIVA BIOTHERAPEUTICS, INC. (CA) 2014-05-06 US claimed
US-20130172405-A1 COMPOSITIONS AND METHODS FOR SILENCING SMAD4 PROTIVA BIOTHERAPEUTICS INC. (CA) 2013-07-04 US claimed
US-20130122104-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS TO SOLID TUMORS PROTIVA BIOTHERAPEUTICS, INC. (CA) 2013-05-16 US claimed
US-8283333-B2 Lipid formulations for nucleic acid delivery PROTIVA BIOTHERAPEUTICS, INC. (CA) 2012-10-09 US claimed
US-20110313017-A1 SNALP FORMULATIONS CONTAINING POLYOXAZOLINE-DIALKYLOXYPROPYL CONJUGATES PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-12-22 US claimed
US-20110076335-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS TO SOLID TUMORS PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-03-31 US claimed
WO-2011011447-A1 COMPOSITIONS AND METHODS FOR SILENCING EBOLA VIRUS GENE EXPRESSION PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-01-27 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (15 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110076335-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS TO SOLID TUMORS PNLIP, CETP, NPC1L1 ALDH1A1 2057/4885CNR1 3865/4885CNR2 4215/4885
US-20210284733-A1 ANTI-PD-1 ANTIBODIES, OR FRAGMENTS THEREOF, FOR TREATING HEPATITIS B CD274, PDCD1, HAVCR2 ALDH1A1 260/4885CNR1 3309/4885CNR2 4382/4885
US-20190032051-A1 NON-LIPOSOMAL SYSTEMS FOR NUCLEIC ACID DELIVERY SNRPE, NPC1L1, LIPA ALDH1A1 3573/4885CNR1 4202/4885CNR2 4528/4885
US-20180245077-A1 COMPOSITIONS AND METHODS FOR TREATING HYPERTRIGLYCERIDEMIA APOB, APOL1, LPL ALDH1A1 4258/4885CNR1 4611/4885CNR2 4656/4885
US-10415037-B2 Compositions and methods for silencing hepatitis B virus gene expression HAVCR2, HDGF, LDLR ALDH1A1 4150/4885CNR1 3305/4885CNR2 3843/4885
US-20140248338-A1 COMPOSITIONS AND METHODS FOR SILENCING ALDEHYDE DEHYDROGENASE ALDH2, ADH1A, ALDH3A1 ALDH1A1 6/4885CNR1 3088/4885CNR2 3455/4885
US-20160076035-A1 COMPOSITIONS AND METHODS FOR SILENCING MARBURG VIRUS GENE EXPRESSION PLIN3, PLIN1, PLIN5 ALDH1A1 3280/4885CNR1 4121/4885CNR2 4502/4885
US-20110313017-A1 SNALP FORMULATIONS CONTAINING POLYOXAZOLINE-DIALKYLOXYPROPYL CONJUGATES DAZAP1, SPOP, PNKP ALDH1A1 1532/4885CNR1 4495/4885CNR2 4648/4885
US-20190328664-A1 METHODS FOR AMELIORATING INFUSION REACTIONS IL2, CD47, IL5 ALDH1A1 1351/4885CNR1 783/4885CNR2 347/4885
US-20160032320-A1 NON-LIPOSOMAL SYSTEMS FOR NUCLEIC ACID DELIVERY SNRPE, NPC1L1, LIPA ALDH1A1 3573/4885CNR1 4202/4885CNR2 4528/4885
US-20200385721-A1 DELIVERING CRISPR THERAPEUTICS WITH LIPID NANOPARTICLES LDLR, SREBF2, NPC1 ALDH1A1 1652/4885CNR1 3258/4885CNR2 3809/4885
US-10626393-B2 Delivering CRISPR therapeutics with lipid nanoparticles LDLR, SREBF2, NPC1 ALDH1A1 1652/4885CNR1 3258/4885CNR2 3809/4885
US-20130122104-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS TO SOLID TUMORS PNLIP, CETP, NPC1L1 ALDH1A1 2057/4885CNR1 3865/4885CNR2 4215/4885
US-20130172405-A1 COMPOSITIONS AND METHODS FOR SILENCING SMAD4 LDLR, SMAD3, AGO2 ALDH1A1 4490/4885CNR1 4172/4885CNR2 4285/4885
US-20190336611-A1 HYBRID CARRIERS FOR NUCLEIC ACID CARGO PHAX, LNPEP, PITPNB ALDH1A1 4507/4885CNR1 4628/4885CNR2 4726/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.