SCHEMBL9967797

SCHEMBL9967797

CC(=O)Nc1ccc(S(=O)(=O)NC(=O)c2ccccc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.64
CA2 P00918 1/20 0.64
MMP1 P03956 1/20 0.64
MMP2 P08253 1/20 0.64
MMP9 P14780 1/20 0.64
MMP8 P22894 1/20 0.64
MMP13 P45452 1/20 0.64
CACNA1B Q00975 1/20 0.64
APBA1 Q02410 1/20 0.64
MEN1 O00255 4/20 0.63
KMT2A Q03164 4/20 0.63
L3MBTL1 Q9Y468 3/20 0.63
LMNA P02545 2/20 0.63
FLT1 P17948 1/20 0.63
FLT4 P35916 1/20 0.63
KDR P35968 1/20 0.63
IDO1 P14902 1/20 0.62
GAA P10253 2/20 0.61
GFER P55789 1/20 0.61
BDKRB1 P46663 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfabenzamide SCHEMBL28198214 0.89 MEN1 (0.69) CA1CA2MMP1MMP2MMP9
SCHEMBL27450474 0.88 HSD17B10 (0.71) CA1CA2MMP2MMP9CACNA1B
SCHEMBL6295620 0.86 MEN1 (0.65) CA1CA2MEN1KMT2AL3MBTL1
SCHEMBL23196556 0.86 KMT2A (0.57) CA1CA2MMP2MMP9MEN1
SCHEMBL28113465 0.85 BDKRB1 (0.63) CA1CA2MMP2MMP9MEN1
SCHEMBL19749350 0.85 MEN1 (0.68) CA1CA2MMP2MMP9MEN1
SCHEMBL19629897 0.85 MEN1 (0.63) CA1CA2MMP2MMP9MEN1
SCHEMBL14585676 0.84 FLT1 (0.67) CA1CA2MEN1KMT2AL3MBTL1
SCHEMBL7774524 0.84 LMNA (0.72) CA1CA2MEN1KMT2AL3MBTL1
SCHEMBL12354484 0.84 MMP2 (0.61) CA1CA2MMP2MMP9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 120 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240239755-A1 SUBSTITUTED PYRIDAZINONES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-07-18 US disclosed
US-20230180758-A1 SUBSTITUTED PYRROLINE-2-ONES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-06-15 US disclosed
US-20230180757-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-06-15 US disclosed
US-20230167088-A1 1-PYRAZINYLPYRAZOLYL-3-OXYALKYL ACIDS AND THEIR DERIVATIVES, AND THEIR USE FOR CONTROL OF UNDESIRED PLANT GROWTH BAYER AKTIENGESELLSCHAFT (DE) 2023-06-01 US disclosed
US-20230159472-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-05-25 US disclosed
US-20230150953-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-05-18 US disclosed
US-20230151025-A1 SUBSTITUTED THIAZOLOPYRIDINES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AG (DE) 2023-05-18 US disclosed
US-20210137117-A1 HERBICIDAL MIXTURES FMC CORPORATION 2021-05-13 US disclosed
US-20190053484-A1 SOLVENT-FREE FORMULATIONS OF LOW-MELTING ACTIVE INGREDIENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-02-21 US disclosed
US-9963431-B2 Use of quinoline derivatives for improving plant yield BAYER CROPSCIENCE AG (DE) 2018-05-08 US disclosed
US-20100255995-A1 HERBICIDE/AZOLE COMBINATION BAYER CROPSCIENCE AG (DE) 2010-10-07 US disclosed
US-20100248965-A1 HERBICIDAL COMBINATION BAYER CROPSCIENCE AG 2010-09-30 US disclosed
US-20100240536-A1 PYRIMIDIN-4-YLPROPANEDINITRILE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2010-09-23 US disclosed
US-20100167935-A1 Pyrimidine derivatives and their use for controlling undesired plant growth BAYER CROPSCIENCE AG (DE) 2010-07-01 US disclosed
US-20100167934-A1 PYRIMIDINE DERIVATIVES AND THEIR USE FOR CONTROLLING UNDESIRED PLANT GROWTH BAYER CROPSCIENCE AG (DE) 2010-07-01 US disclosed
US-20100137139-A1 HERBICIDE/SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 US disclosed
US-20100137136-A1 HERBICIDE/SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 US disclosed
US-20100137138-A1 HERBICIDE/SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 US disclosed
US-20100137137-A1 HERBICIDE/SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 US disclosed
US-20100062939-A1 Herbicide/Safener Combination Comprising Dimethoxytriazinyl-Substituted Difluoromethanesulfonylanilides BAYER CROPSCIENCE AG (DE) 2010-03-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (19 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137138-A1 HERBICIDE/SAFENER COMBINATION DDT, GSTO1, GAP43 CA1 592/4885CA2 384/4885MMP1 722/4885
US-20230150953-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES DDT, ZDHHC2, DDAH1 CA1 535/4885CA2 348/4885MMP1 597/4885
US-20100137136-A1 HERBICIDE/SAFENER COMBINATION DDT, GAP43, CYP2W1 CA1 631/4885CA2 413/4885MMP1 1078/4885
US-20100255995-A1 HERBICIDE/AZOLE COMBINATION HTT, SOD1, ABAT CA1 401/4885CA2 342/4885MMP1 885/4885
US-20190053484-A1 SOLVENT-FREE FORMULATIONS OF LOW-MELTING ACTIVE INGREDIENTS CYP51A1, ABCG2, FASTKD5 CA1 2156/4885CA2 2918/4885MMP1 1362/4885
US-20100167935-A1 Pyrimidine derivatives and their use for controlling undesired plant growth TYMS, TYMP, UMPS CA1 4853/4885CA2 4425/4885MMP1 4319/4885
US-20230167088-A1 1-PYRAZINYLPYRAZOLYL-3-OXYALKYL ACIDS AND THEIR DERIVATIVES, AND THEIR USE FOR CONTROL OF UNDESIRED PLANT GROWTH AGPS, CBR3, HPD CA1 1679/4885CA2 332/4885MMP1 420/4885
US-20210137117-A1 HERBICIDAL MIXTURES DDT, MTX2, ATL3 CA1 773/4885CA2 75/4885MMP1 2099/4885
US-20230180757-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES AND THEIR USE AS HERBICIDES DDT, DAO, IDH2 CA1 580/4885CA2 249/4885MMP1 809/4885
US-20240239755-A1 SUBSTITUTED PYRIDAZINONES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES PNPO, WEE1, PDXK CA1 4238/4885CA2 1687/4885MMP1 788/4885
US-20100137137-A1 HERBICIDE/SAFENER COMBINATION DDT, CYP2W1, GAP43 CA1 346/4885CA2 339/4885MMP1 1184/4885
US-20100137139-A1 HERBICIDE/SAFENER COMBINATION CYP2W1, DDT, CBR3 CA1 948/4885CA2 502/4885MMP1 1662/4885
US-20230180758-A1 SUBSTITUTED PYRROLINE-2-ONES AND THEIR USE AS HERBICIDES DDT, HPD, ALDH18A1 CA1 2594/4885CA2 845/4885MMP1 2293/4885
US-20100248965-A1 HERBICIDAL COMBINATION DDT, AADAC, AS3MT CA1 366/4885CA2 42/4885MMP1 1139/4885
US-20230151025-A1 SUBSTITUTED THIAZOLOPYRIDINES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES TST, DDT, GMDS CA1 2280/4885CA2 284/4885MMP1 949/4885
US-20230159472-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES DDT, IDH2, DAO CA1 509/4885CA2 428/4885MMP1 1265/4885
US-20100062939-A1 Herbicide/Safener Combination Comprising Dimethoxytriazinyl-Substituted Difluoromethanesulfonylanilides DDT, CYP2W1, AS3MT CA1 384/4885CA2 198/4885MMP1 2352/4885
US-20100240536-A1 PYRIMIDIN-4-YLPROPANEDINITRILE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS DDT, PLPBP, HPD CA1 4677/4885CA2 2716/4885MMP1 4220/4885
US-20100167934-A1 PYRIMIDINE DERIVATIVES AND THEIR USE FOR CONTROLLING UNDESIRED PLANT GROWTH TYMS, TYMP, UMPS CA1 4585/4885CA2 3718/4885MMP1 4223/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.