SCHEMBL9967799

SCHEMBL9967799

CN(C)C(=O)Nc1ccc(S(=O)(=O)NC(=O)c2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 1/20 0.62
MEN1 O00255 4/20 0.58
KMT2A Q03164 4/20 0.58
LMNA P02545 3/20 0.58
L3MBTL1 Q9Y468 2/20 0.58
FLT1 P17948 2/20 0.58
FLT4 P35916 2/20 0.58
KDR P35968 2/20 0.58
CA12 O43570 2/20 0.56
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
CA9 Q16790 2/20 0.56
HTT P42858 2/20 0.54
MAPT P10636 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
PRMT1 Q99873 1/20 0.54
HPGD P15428 1/20 0.51
BCL2L1 Q07817 1/20 0.51
MCL1 Q07820 1/20 0.51
MMP2 P08253 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26342886 0.89 MEN1 (0.56) BDKRB1MEN1KMT2ALMNAL3MBTL1
SCHEMBL21086881 0.89 MEN1 (0.56) BDKRB1MEN1KMT2ALMNAL3MBTL1
SCHEMBL21844845 0.86 MEN1 (0.58) MEN1KMT2ALMNAL3MBTL1FLT1
SCHEMBL9467928 0.86 GPR17 (0.52) BDKRB1LMNAFLT1FLT4KDR
SCHEMBL9967797 0.84 CA1 (0.64) BDKRB1MEN1KMT2ALMNAL3MBTL1
SCHEMBL15624637 0.83 FLT1 (0.64) BDKRB1LMNAFLT1FLT4KDR
SCHEMBL6295620 0.82 MEN1 (0.65) MEN1KMT2ALMNAL3MBTL1FLT1
SCHEMBL28113465 0.82 BDKRB1 (0.63) BDKRB1MEN1KMT2ALMNAL3MBTL1
SCHEMBL9467720 0.82 CA12 (0.51) BDKRB1MEN1KMT2ALMNAFLT1
SCHEMBL9971694 0.81 FLT1 (0.63) MEN1KMT2ALMNAL3MBTL1FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 141 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240239755-A1 SUBSTITUTED PYRIDAZINONES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-07-18 US disclosed
US-20240025862-A1 SUBSTITUTED N-PHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-01-25 US disclosed
US-11834434-B2 Substituted 2-heteroaryloxypyridines and salts thereof and their use as herbicidal agents BAYER AKTIENGESELLSCHAFT (DE) 2023-12-05 US disclosed
US-20230303549-A1 SUBSTITUTED HETEROARYLOXYPYRIDINES, THE SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2023-09-28 US disclosed
US-20230180757-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-06-15 US disclosed
US-20230180758-A1 SUBSTITUTED PYRROLINE-2-ONES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-06-15 US disclosed
US-20230167088-A1 1-PYRAZINYLPYRAZOLYL-3-OXYALKYL ACIDS AND THEIR DERIVATIVES, AND THEIR USE FOR CONTROL OF UNDESIRED PLANT GROWTH BAYER AKTIENGESELLSCHAFT (DE) 2023-06-01 US disclosed
US-20230159472-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-05-25 US disclosed
US-20230150953-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-05-18 US disclosed
US-20230151025-A1 SUBSTITUTED THIAZOLOPYRIDINES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AG (DE) 2023-05-18 US disclosed
US-20100255995-A1 HERBICIDE/AZOLE COMBINATION BAYER CROPSCIENCE AG (DE) 2010-10-07 US disclosed
US-20100248965-A1 HERBICIDAL COMBINATION BAYER CROPSCIENCE AG 2010-09-30 US disclosed
US-20100240536-A1 PYRIMIDIN-4-YLPROPANEDINITRILE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2010-09-23 US disclosed
US-20100167935-A1 Pyrimidine derivatives and their use for controlling undesired plant growth BAYER CROPSCIENCE AG (DE) 2010-07-01 US disclosed
US-20100167934-A1 PYRIMIDINE DERIVATIVES AND THEIR USE FOR CONTROLLING UNDESIRED PLANT GROWTH BAYER CROPSCIENCE AG (DE) 2010-07-01 US disclosed
US-20100137139-A1 HERBICIDE/SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 US disclosed
US-20100137136-A1 HERBICIDE/SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 US disclosed
US-20100137138-A1 HERBICIDE/SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 US disclosed
US-20100137137-A1 HERBICIDE/SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 US disclosed
US-20100062939-A1 Herbicide/Safener Combination Comprising Dimethoxytriazinyl-Substituted Difluoromethanesulfonylanilides BAYER CROPSCIENCE AG (DE) 2010-03-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (20 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137138-A1 HERBICIDE/SAFENER COMBINATION DDT, GSTO1, GAP43 BDKRB1 4814/4885MEN1 4051/4885KMT2A 2182/4885
US-20230150953-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES DDT, ZDHHC2, DDAH1 BDKRB1 3028/4885MEN1 3475/4885KMT2A 730/4885
US-20100137136-A1 HERBICIDE/SAFENER COMBINATION DDT, GAP43, CYP2W1 BDKRB1 4826/4885MEN1 3652/4885KMT2A 1948/4885
US-20100255995-A1 HERBICIDE/AZOLE COMBINATION HTT, SOD1, ABAT BDKRB1 4702/4885MEN1 4024/4885KMT2A 1412/4885
US-20100167935-A1 Pyrimidine derivatives and their use for controlling undesired plant growth TYMS, TYMP, UMPS BDKRB1 4177/4885MEN1 4628/4885KMT2A 2327/4885
US-20230167088-A1 1-PYRAZINYLPYRAZOLYL-3-OXYALKYL ACIDS AND THEIR DERIVATIVES, AND THEIR USE FOR CONTROL OF UNDESIRED PLANT GROWTH AGPS, CBR3, HPD BDKRB1 3791/4885MEN1 4795/4885KMT2A 3622/4885
US-20230180757-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES AND THEIR USE AS HERBICIDES DDT, DAO, IDH2 BDKRB1 3566/4885MEN1 3762/4885KMT2A 495/4885
US-20240239755-A1 SUBSTITUTED PYRIDAZINONES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES PNPO, WEE1, PDXK BDKRB1 4285/4885MEN1 4547/4885KMT2A 2299/4885
US-20100137137-A1 HERBICIDE/SAFENER COMBINATION DDT, CYP2W1, GAP43 BDKRB1 4768/4885MEN1 3489/4885KMT2A 1867/4885
US-20100137139-A1 HERBICIDE/SAFENER COMBINATION CYP2W1, DDT, CBR3 BDKRB1 2197/4885MEN1 2602/4885KMT2A 1782/4885
US-20230303549-A1 SUBSTITUTED HETEROARYLOXYPYRIDINES, THE SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS DDT, AGPS, GMDS BDKRB1 3449/4885MEN1 4575/4885KMT2A 2025/4885
US-11834434-B2 Substituted 2-heteroaryloxypyridines and salts thereof and their use as herbicidal agents DDT, AGPS, GMDS BDKRB1 3939/4885MEN1 4581/4885KMT2A 1300/4885
US-20230180758-A1 SUBSTITUTED PYRROLINE-2-ONES AND THEIR USE AS HERBICIDES DDT, HPD, ALDH18A1 BDKRB1 4784/4885MEN1 4567/4885KMT2A 1688/4885
US-20100248965-A1 HERBICIDAL COMBINATION DDT, AADAC, AS3MT BDKRB1 4093/4885MEN1 4086/4885KMT2A 131/4885
US-20230151025-A1 SUBSTITUTED THIAZOLOPYRIDINES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES TST, DDT, GMDS BDKRB1 4160/4885MEN1 4379/4885KMT2A 2454/4885
US-20240025862-A1 SUBSTITUTED N-PHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES PFAS, DDT, NOTUM BDKRB1 4718/4885MEN1 4557/4885KMT2A 1736/4885
US-20230159472-A1 SUBSTITUTED ISOPHTHALIC ACID DIAMIDES DDT, IDH2, DAO BDKRB1 4241/4885MEN1 3793/4885KMT2A 696/4885
US-20100062939-A1 Herbicide/Safener Combination Comprising Dimethoxytriazinyl-Substituted Difluoromethanesulfonylanilides DDT, CYP2W1, AS3MT BDKRB1 3742/4885MEN1 1695/4885KMT2A 107/4885
US-20100240536-A1 PYRIMIDIN-4-YLPROPANEDINITRILE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS DDT, PLPBP, HPD BDKRB1 4013/4885MEN1 3857/4885KMT2A 2759/4885
US-20100167934-A1 PYRIMIDINE DERIVATIVES AND THEIR USE FOR CONTROLLING UNDESIRED PLANT GROWTH TYMS, TYMP, UMPS BDKRB1 4327/4885MEN1 4352/4885KMT2A 2672/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.