SCHEMBL10140227

SCHEMBL10140227

CNC(=O)c1cc(Cl)cc(Cl)c1NC(=O)c1cc(Cl)nn1-c1ncccc1C

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.36
KMT2A Q03164 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PPARG P37231 1/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
NTRK1 P04629 5/20 0.35
P2RX7 Q99572 1/20 0.34
EPHX2 P34913 2/20 0.34
MALT1 Q9UDY8 2/20 0.34
DHODH Q02127 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10140188 0.93 RAB9A (0.38) TRPV1KMT2AL3MBTL1PPARGRAB9A
SCHEMBL782242 0.92 MALT1 (0.38) TRPV1KMT2ANTRK1EPHX2MALT1
SCHEMBL10140197 0.91 DHODH (0.41) TRPV1KMT2AL3MBTL1PPARGRAB9A
SCHEMBL10140225 0.90 CNR1 (0.37) TRPV1KMT2AL3MBTL1RAB9ANPC1
SCHEMBL782485 0.89 MALT1 (0.39) TRPV1KMT2ARAB9ANPC1NTRK1
SCHEMBL10140216 0.88 PDE4B (0.37) KMT2AMALT1
SCHEMBL13442911 0.88 PKM (0.35) TRPV1KMT2APPARGMALT1DHODH
SCHEMBL10140154 0.86 SORT1 (0.39) TRPV1KMT2AL3MBTL1RAB9ANPC1
SCHEMBL12528237 0.85 NTRK1 (0.39) KMT2ARAB9ANPC1NTRK1MALT1
SCHEMBL10140180 0.84 DHODH (0.40) TRPV1KMT2AL3MBTL1PPARGRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9949482-B2 Fungicidal compositions SYNGENTA CROP PROTECTION, LLC (US) 2018-04-24 US disclosed
US-20170071205-A1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION, LLC (US) 2017-03-16 US disclosed
US-20160302414-A1 INSECTICIDAL COMPOUNDS SYNGENTA CROP PROTECTION LLC (US) 2016-10-20 US disclosed
US-9282743-B2 Chemical compounds SYNGENTA PARTICIPATIONS AG (CH) 2016-03-15 US disclosed
US-9096525-B2 Iminipyridine derivatives and their uses as microbiocides SYNGENTA CROP PROTECTION, LLC (US) 2015-08-04 US disclosed
US-20140148339-A1 CHEMICAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2014-05-29 US disclosed
US-8536089-B2 For controlling phytopathogenic diseases; synergistic SYNGENTA CROP PROTECTION LLC (US) 2013-09-17 US disclosed
US-20130210625-A1 SPIROHETEROCYCLIC PYRROLIDINE DERIVATIVES BASED PESTICIDES SYNGENTA CROP PROTECTION LLC (US) 2013-08-15 US disclosed
US-20120309812-A1 INSECTICIDAL COMPOUNDS SYNGENTA CROP PROTECTION LLC (US) 2012-12-06 US disclosed
US-8124566-B2 Synergistic fungicidal compositions SYNGENTA CROP PROTECTION, INC. (US) 2012-02-28 US disclosed
US-8124567-B2 Fungicidal compositions SYNGENTA CROP PROTECTION, INC. (US) 2012-02-28 US disclosed
US-20080076664-A1 Fungicidal Compositions SYNGENTA CROP PROTECTION, INC. 2008-03-27 US disclosed
US-20080070785-A1 For controlling phytopathogenic diseases; synergistic SYNGENTA CROP PROTECTION, INC. (US) 2008-03-20 US disclosed
US-20070265267-A1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION, INC. (US) 2007-11-15 US disclosed
US-20070244121-A1 Synergistic Fungicidal Compositions SYNGENTA CROP PROTECTION, INC. (US) 2007-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120309812-A1 INSECTICIDAL COMPOUNDS ACHE, AADAC, NISCH TRPV1 432/4885KMT2A 1531/4885L3MBTL1 772/4885
US-20130210625-A1 SPIROHETEROCYCLIC PYRROLIDINE DERIVATIVES BASED PESTICIDES DDT, PYCR1, PKD2 TRPV1 295/4885KMT2A 3529/4885L3MBTL1 2524/4885
US-20160302414-A1 INSECTICIDAL COMPOUNDS ACHE, AADAC, CASP3 TRPV1 1248/4885KMT2A 3045/4885L3MBTL1 1177/4885
US-20070265267-A1 FUNGICIDAL COMPOSITIONS CRY1, ERG28, DDT TRPV1 1660/4885KMT2A 1397/4885L3MBTL1 247/4885
US-20070244121-A1 Synergistic Fungicidal Compositions DDT, CRY1, HCN1 TRPV1 1081/4885KMT2A 2009/4885L3MBTL1 375/4885
US-20080070785-A1 For controlling phytopathogenic diseases; synergistic BROX, EPM2A, MANBA TRPV1 3772/4885KMT2A 3493/4885L3MBTL1 1584/4885
US-20140148339-A1 CHEMICAL COMPOUNDS DDT, CYP1B1, CYP1A1 TRPV1 347/4885KMT2A 1487/4885L3MBTL1 2310/4885
US-20170071205-A1 FUNGICIDAL COMPOSITIONS PIK3C3, CYP51A1, CYP1B1 TRPV1 2857/4885KMT2A 2404/4885L3MBTL1 2580/4885
US-20080076664-A1 Fungicidal Compositions AKR7A2, CYP51A1, TUBA3C TRPV1 2728/4885KMT2A 3265/4885L3MBTL1 173/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.