SCHEMBL14744248

SCHEMBL14744248

Cc1cc(N)cc(F)c1Br

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
TSHR P16473 3/20 0.38
CYP3A4 P08684 2/20 0.35
MAPK1 P28482 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
KDM1A O60341 4/20 0.33
KDM1B Q8NB78 2/20 0.33
CYP1A2 P05177 1/20 0.33
ALOX15 P16050 1/20 0.33
CASP7 P55210 1/20 0.33
HIF1A Q16665 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PDE10A Q9Y233 1/20 0.33
CASP1 P29466 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL238421 0.82 KDM1A (0.44) ALDH1A1TSHRCYP3A4MAPK1GAA
SCHEMBL525424 0.82 ALDH1A1 (0.47) ALDH1A1TSHRCYP3A4MAPK1GAA
SCHEMBL30695922 0.75 ALDH1A1 (0.41) ALDH1A1TSHRCYP3A4MAPK1MAPT
SCHEMBL5306395 0.75 ALDH1A1 (0.41) ALDH1A1TSHRCYP3A4MAPK1MAPT
SCHEMBL29664557 0.75 NQO2 (0.32) KDM1AKDM1B
SCHEMBL29863733 0.75 RAPGEF4 (0.40) MAPK1KDM1AKDM1B
SCHEMBL13550059 0.75 NQO2 (0.32) KDM1AKDM1B
SCHEMBL1043169 0.75 RAPGEF4 (0.40) MAPK1KDM1AKDM1B
SCHEMBL20843494 0.75 ALDH1A1 (0.43) ALDH1A1TSHRCYP3A4MAPK1GAA
SCHEMBL15573628 0.75 ALDH1A1 (0.41) ALDH1A1TSHRCYP3A4MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 133 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260085067-A1 CYCLIC SULFONAMIDE RIBONUCLEOTIDE REDUCTASE (RNR) INHIBITORS AND USES THEREOF BOUNDLESS BIO INC (US) 2026-03-26 US disclosed
EP-4482579-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH LPA RECEPTOR ACTIVITY LHOTSE BIO INC (US) 2026-02-18 EP disclosed
US-12534453-B2 Inhibitors of glycogen synthase 1 (GYS1) and methods of use thereof MAZE THERAPEUTICS, INC. (US) 2026-01-27 US disclosed
US-12516059-B2 Pyrazolopyridine compounds and uses thereof INCYTE CORPORATION (US) 2026-01-06 US disclosed
US-20250388565-A1 ESTROGEN RECEPTOR ALPHA DEGRADERS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. 2025-12-25 US disclosed
US-12428375-B2 Compounds and compositions for treating conditions associated with LPA receptor activity LHOTSE BIO, INC. (US) 2025-09-30 US disclosed
US-12391663-B2 Isoindolinone compounds MONTE ROSA THERAPEUTICS AG (CH) 2025-08-19 US disclosed
US-12384778-B2 Pyrazolopyridine compounds and uses thereof INCYTE CORPORATION (US) 2025-08-12 US disclosed
EP-4587437-A1 CYCLIC SULFONAMIDE RIBONUCLEOTIDE REDUCTASE (RNR) INHIBITORS AND USES THEREOF Boundless Bio, Inc. (US) 2025-07-23 EP disclosed
EP-4543871-A1 ESTROGEN RECEPTOR ALPHA DEGRADERS AND USE THEREOF Relay Therapeutics, Inc. (US) 2025-04-30 EP disclosed
EP-3107900-B1 5-BENZYLISOQUINOLEINE DERIVATIVES FOR THE TREATMENT OF CARDIOVASCULAR DISEASES SERVIER LAB (FR) 2017-11-15 EP disclosed
US-9809553-B2 Isoquinoline compounds, a process for their preparation, and pharmaceutical compositions containing them LES LABORATOIRES SERVIER (FR) 2017-11-07 US disclosed
US-20170137385-A1 ISOQUINOLINE COMPOUNDS, A PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2017-05-18 US disclosed
EP-2870143-B1 TRIAZOLE COMPOUNDS AS ANTIVIRALS HOFFMANN LA ROCHE (CH) 2017-05-17 EP disclosed
EP-3107900-A1 DERIVATIVES OF 5-BENZYLISOQUINOLINE FOR THE TREATMENT OF CARDIOVASCULAR DISEASES Les Laboratoires Servier (FR) 2016-12-28 EP disclosed
US-9487488-B2 Sulfonamide compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2016-11-08 US disclosed
US-20150307454-A1 Sulfonamide Compound KALLYOPE, INC. 2015-10-29 US disclosed
WO-2015124877-A1 DERIVATIVES OF 5-BENZYLISOQUINOLINE FOR THE TREATMENT OF CARDIOVASCULAR DISEASES LES LABORATOIRES SERVIER (FR) 2015-08-27 WO disclosed
EP-2896613-A1 SULFONAMIDE COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2015-07-22 EP disclosed
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12384778-B2 Pyrazolopyridine compounds and uses thereof PDXK, PCK1, PGK1 ALDH1A1 2205/4885TSHR 4733/4885CYP3A4 1456/4885
US-12391663-B2 Isoindolinone compounds CYP4F2, AOC2, AOC3 ALDH1A1 1142/4885TSHR 1114/4885CYP3A4 684/4885
US-20250388565-A1 ESTROGEN RECEPTOR ALPHA DEGRADERS AND METHODS OF USE THEREOF ESRRA, ESRRB, ESR2 ALDH1A1 1679/4885TSHR 68/4885CYP3A4 672/4885
US-20260085067-A1 CYCLIC SULFONAMIDE RIBONUCLEOTIDE REDUCTASE (RNR) INHIBITORS AND USES THEREOF RRM1, RRM2B, RRM2 ALDH1A1 998/4885TSHR 76/4885CYP3A4 1636/4885
US-12534453-B2 Inhibitors of glycogen synthase 1 (GYS1) and methods of use thereof GYS1, GYS2, GBA1 ALDH1A1 2276/4885TSHR 3968/4885CYP3A4 3399/4885
US-20170137385-A1 ISOQUINOLINE COMPOUNDS, A PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM MYLK, MYLK2, MYLK3 ALDH1A1 3415/4885TSHR 4698/4885CYP3A4 1738/4885
US-20150307454-A1 Sulfonamide Compound TRPM8, TRPM5, TRPM7 ALDH1A1 2634/4885TSHR 799/4885CYP3A4 1795/4885
US-12428375-B2 Compounds and compositions for treating conditions associated with LPA receptor activity LPAR2, LPAR1, LPAR6 ALDH1A1 1863/4885TSHR 1333/4885CYP3A4 4716/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.