Carbromal

Carbromal

SCHEMBL22375

CCC(Br)(CC)C(=O)NC(N)=O.CCC(Br)(CC)C(=O)NC(N)=O.Cl.Cl

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Carbromal. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CRBN known ✓ Q96SW2 1/20 0.37
NR3C1 known ✓ P04150 1/20 0.33
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbromal SCHEMBL158922 1.00 CRBN (0.37) CRBNNR3C1LMNAMAPTRAB9A
Carbromal SCHEMBL11745356 0.98 CRBN (0.36) CRBNNR3C1
Carbromal SCHEMBL22158510 0.98 CRBN (0.36) CRBNNR3C1
Carbromal SCHEMBL9356891 0.98 CRBN (0.36) CRBNNR3C1
Carbromal SCHEMBL8986675 0.98 CRBN (0.36) CRBNNR3C1
Carbromal SCHEMBL9705588 0.98 CRBN (0.36) CRBNNR3C1
Carbromal SCHEMBL261 0.98 CRBN (0.39) CRBNNR3C1MAPTRAB9ANPSR1
Carbromal SCHEMBL4351621 0.98 CRBN (0.39) CRBNNR3C1MAPTRAB9ANPSR1
Carbromal SCHEMBL15057476 0.98 CRBN (0.39) CRBNNR3C1MAPTRAB9ANPSR1
Carbromal SCHEMBL23855707 0.96 CRBN (0.34) CRBNNR3C1MAPTRAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 922 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12038559-B2 Window cover film and flexible display panel including the same SK INNOVATION CO., LTD. (KR) 2024-07-16 US claimed
US-11970579-B2 Polyamic acid resin and polyamideimide film SK INNOVATION CO., LTD. (KR) 2024-04-30 US claimed
US-11970592-B2 Window cover film and flexible display panel including the same SK INNOVATION CO., LTD. (KR) 2024-04-30 US claimed
US-11960159-B2 Polyamideimide film and flexible display panel including the same SK INNOVATION CO., LTD. (KR) 2024-04-16 US claimed
US-11921546-B2 Polyimide film and flexible display panel including the same SK INNOVATION CO., LTD. (KR) 2024-03-05 US claimed
US-20240026155-A1 Polyamideimide Film and Optical Multilayer Structure Comprising the Same SK INNOVATION CO., LTD. (KR) 2024-01-25 US claimed
US-11845842-B2 Window cover film and flexible display panel including the same SK INNOVATION CO., LTD. (KR) 2023-12-19 US claimed
US-11840631-B2 Polyimide-based film and flexible display panel including the same SK INNOVATION CO., LTD. (KR) 2023-12-12 US claimed
US-20230367040-A1 OPTICAL MULTILAYER STRUCTURE, METHOD OF MANUFACTURING THE SAME, AND WINDOW COVER FILM INCLUDING THE SAME SK INNOVATION CO., LTD. (KR) 2023-11-16 US claimed
US-20230340202-A9 Polyamideimide Film-Forming Composition, Method of Preparing the Same, and Use Thereof SK IE TECHNOLOGY CO., LTD. (KR) 2023-10-26 US claimed
WO-1994013727-A1 AROMATIC POLYAMIDE PULP BY MEANS OF CONTINUOUS TRANSFERABLE POLYMERIZATION-ORIENTATION METHOD AND A PROCESS FOR PREPARATION THEREOF KOLON INDUSTRIES, INC. (KR) 1994-06-23 WO claimed
EP-0598753-A1 MANGANESE COMPLEXES OF NITROGEN-CONTAINING MACROCYCLIC LIGANDS EFFECTIVE AS CATALYSTS FOR DISMUTATING SUPEROXIDE MONSANTO COMPANY (US) 1994-06-01 EP claimed
WO-1993002090-A1 MANGANESE COMPLEXES OF NITROGEN-CONTAINING MACROCYCLIC LIGANDS EFFECTIVE AS CATALYSTS FOR DISMUTATING SUPEROXIDE MONSANTO COMPANY (US) 1993-02-04 WO claimed
EP-0524161-A1 Manganese complexes of nitrogen containing macrocyclic ligands effective as catalysts for dismutating superoxide MONSANTO COMPANY (US) 1993-01-20 EP claimed
US-5153300-A Aromatic polyesters with high glass transition temperature, improved solvent resistance GENERAL ELECTRIC COMPANY (US) 1992-10-06 US claimed
EP-0229714-B1 POLYMERIZATION OF AROMATIC POLYAMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-05-20 EP claimed
EP-0277376-B1 AROMATIC AMIDE GROUPS-CONTAINING DIAMINES AND POLYMERS IN WHICH THESE DIAMINES ARE INCORPORATED AKZO N.V. (NL) 1991-02-27 EP claimed
EP-0277376-A1 Aromatic amide groups-containing diamines and polymers in which these diamines are incorporated AKZO N.V. (NL) 1988-08-10 EP claimed
US-4233434-A POLYMERS AND COPOLYMERS FOR USE AS FILMS, MEMBRANES, FIBERS, AND SHAPED OBJECTS A.T. RAMOT PLASTICS LTD. (IL) 1980-11-11 US claimed
US-4169932-A METHOD OF PRODUCING POLY-P-PHENYLENETEREPHTHALAMIDE OR ITS COPOLYMERS INGERSOLL EQUIPMENT CO., INC., 1979-10-02 US claimed