Fumaric Acid

Fumaric Acid

SCHEMBL2398321

O=C(O)C=CC(=O)O.c1ccc(CN2CCC(CCCc3ccc4c(c3)NCCCC4)CC2)cc1

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ACHE P22303 17/20 0.67
NPY2R P49146 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL23668767 1.00 ACHE (0.67) ACHENPY2R
SCHEMBL3341801 0.92 ACHE (0.68) ACHE
Zanapezil SCHEMBL1232176 0.86 ACHE (0.91) ACHE
Zanapezil SCHEMBL1232174 0.86 ACHE (0.91) ACHE
Fumaric Acid SCHEMBL9203761 0.85 ACHE (0.91) ACHE
Fumaric Acid SCHEMBL9203739 0.85 ACHE (0.91) ACHE
Fumaric Acid SCHEMBL6848789 0.85 ACHE (0.66) ACHE
Fumaric Acid SCHEMBL9200365 0.83 ACHE (0.91) ACHE
Fumaric Acid SCHEMBL9200378 0.83 ACHE (0.91) ACHE
SCHEMBL6262731 0.81 ACHE (0.68) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 95 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220160733-A1 COMPOSITIONS FOR IMPROVING CELL VIABILITY AND METHODS OF USE THEREOF Amylyx Pharmaceuticals Inc. 2022-05-26 US claimed
US-20190262268-A1 ORAL MODIFIED RELEASE FORMULATIONS RUBICON RES PRIVATE LIMITED (IN) 2019-08-29 US claimed
US-20170128379-A1 MODIFIED RELEASE PHARMACEUTICAL PREPARATIONS RUBICON RESEARCH PRIVATE LIMITED (IN) 2017-05-11 US claimed
WO-2016001937-A2 MODIFIED RELEASE PHARMACEUTICAL PREPARATIONS RUBICON RESEARCH PRIVATE LIMITED (IN) 2016-01-07 WO claimed
US-20240043395-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF TLR SIGNALING NEUROPORE THERAPIES, INC. 2024-02-08 US disclosed
US-20230391734-A1 SUBSTITUTED PHENYL SULFONYL PHENYL TRIAZOLE THIONES AND USES THEREOF NEUROPORE THERAPIES, INC. (US) 2023-12-07 US disclosed
US-20230265086-A1 TRI-SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES AS MODULATORS OF PI3-KINASE AND AUTOPHAGY PATHWAYS NEUROPORE THERAPIES, INC. (US) 2023-08-24 US disclosed
US-11708338-B2 Substituted phenyl sulfonyl phenyl triazole thiones and uses thereof NEUROPORE THERAPIES, INC. (US) 2023-07-25 US disclosed
US-11492348-B2 Tri-substituted aryl and heteroaryl derivatives as modulators of PI3-kinase and autophagy pathways NEUROPORE THERAPIES, INC. (US) 2022-11-08 US disclosed
US-11345713-B2 Compounds as modulators of TLR2 signaling NEUROPORE THERAPIES, INC. (US) 2022-05-31 US disclosed
US-20220160733-A1 COMPOSITIONS FOR IMPROVING CELL VIABILITY AND METHODS OF USE THEREOF Amylyx Pharmaceuticals Inc. 2022-05-26 US disclosed
EP-3946599-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF TLR SIGNALING Neuropore Therapies, Inc. (US) 2022-02-09 EP disclosed
US-20040258741-A1 Percutaneous absorption preparations HISAMITSU PHARMACEUTICAL CO., INC. (JP) 2004-12-23 US disclosed
EP-1484053-A2 Percutaneously applicable preparation and suppository containing an antidementia medicament Eisai Co., Ltd. (JP) 2004-12-08 EP disclosed
US-6815454-B2 DONEPEZIL HYDROCHLORIDE AND A ABSORPTION PROMOTER SELECTED FROM THE GROUP CONSISTING OF A HIGHER ALCOHOL, AN ESTER OF A HIGHER FATTY ACID AND A LOWER ALCOHOL AND AN ESTER OF A FATTY ACID HAVING 6-18 CARBON ATOMS AND PROPYLENE GLYCOL EISAI CO., LTD. (JP) 2004-11-09 US disclosed
US-6521639-B1 Donepezil hydrochloride and lactate of a higher alcohol; increased absorption EISAI CO., LTD. (JP) 2003-02-18 US disclosed
US-6372760-B1 COGNITION ACTIVATORS WITH ORGANIC ACID FOR DONEPEZIL EISAI CO., LTD. (JP) 2002-04-16 US disclosed
EP-1086706-A1 STABILIZED COMPOSITIONS CONTAINING NOOTROPIC DRUGS Eisai Co., Ltd. (JP) 2001-03-28 EP disclosed
US-6193993-B1 Suppository containing an antidementia medicament EISAI CO., LTD. (JP) 2001-02-27 US disclosed
EP-0947193-A2 Percutaneously applicable preparation and suppository containing an antidementia medicament Eisai Co., Ltd. (JP) 1999-10-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220160733-A1 COMPOSITIONS FOR IMPROVING CELL VIABILITY AND METHODS OF USE THEREOF HSPA9, CYP27A1, TUFM ACHE 3040/4885NPY2R 2907/4885
US-20040258741-A1 Percutaneous absorption preparations CUTA, CDH1, DSG1 ACHE 12/4885NPY2R 2963/4885
US-20240043395-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF TLR SIGNALING TLR3, TLR6, TLR4 ACHE 3591/4885NPY2R 4008/4885
US-11492348-B2 Tri-substituted aryl and heteroaryl derivatives as modulators of PI3-kinase and autophagy pathways ATG7, ULK1, BECN1 ACHE 4852/4885NPY2R 3125/4885
US-11345713-B2 Compounds as modulators of TLR2 signaling TLR2, TLR4, TLR3 ACHE 3887/4885NPY2R 3130/4885
US-11708338-B2 Substituted phenyl sulfonyl phenyl triazole thiones and uses thereof TPMT, ABCB1, DPP8 ACHE 3365/4885NPY2R 1585/4885
US-20230391734-A1 SUBSTITUTED PHENYL SULFONYL PHENYL TRIAZOLE THIONES AND USES THEREOF TPMT, ABCB1, DPP8 ACHE 3365/4885NPY2R 1585/4885
US-20230265086-A1 TRI-SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES AS MODULATORS OF PI3-KINASE AND AUTOPHAGY PATHWAYS ATG7, ULK1, BECN1 ACHE 4852/4885NPY2R 3125/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.