SCHEMBL2540289

SCHEMBL2540289

NS(=O)(=O)c1nn2cc(-c3ccccc3)nc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 1.00
KMT2A Q03164 2/20 1.00
CA12 O43570 10/20 0.67
CA1 P00915 10/20 0.67
CA2 P00918 10/20 0.67
CA9 Q16790 10/20 0.67
TP53 P04637 6/20 0.60
SMN1; SMN2 Q16637 5/20 0.58
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
ALOX15 P16050 2/20 0.58
NFKB1 P19838 1/20 0.58
NFKB2 Q00653 1/20 0.58
RELA Q04206 1/20 0.58
KDM4E B2RXH2 1/20 0.56
HSD17B10 Q99714 1/20 0.56
F2RL3 Q96RI0 2/20 0.55
PKM P14618 1/20 0.55
RECQL P46063 1/20 0.55
MAPT P10636 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2981652 0.99 MEN1 (0.97) MEN1KMT2ACA12CA1CA2
SCHEMBL13204703 0.97 MEN1 (0.95) MEN1KMT2ACA12CA1CA2
SCHEMBL13204667 0.90 MEN1 (0.81) MEN1KMT2ACA12CA1CA2
SCHEMBL2969028 0.89 MEN1 (0.81) MEN1KMT2ACA12CA1CA2
SCHEMBL2978970 0.89 MEN1 (0.81) MEN1KMT2ACA12CA1CA2
SCHEMBL2977101 0.89 MEN1 (0.79) MEN1KMT2ACA12CA1CA2
SCHEMBL2970463 0.87 MEN1 (0.78) MEN1KMT2ACA12CA1CA2
SCHEMBL2979747 0.87 MEN1 (0.78) MEN1KMT2ACA12CA1CA2
SCHEMBL2979379 0.87 MEN1 (0.76) MEN1KMT2ACA12CA1CA2
SCHEMBL2985683 0.87 MEN1 (0.76) MEN1KMT2ACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 292 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12383558-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2025-08-12 US claimed
EP-4556010-A2 JAK INHIBITORS FOR USE IN THE PREVENTION OR TREATMENT OF A VIRAL DISEASE CAUSED BY A CORONAVIRIDAE Emory University (US) 2025-05-21 EP claimed
US-20240415838-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION UNIV EMORY (US) 2024-12-19 US claimed
WO-2024144816-A1 TREATMENT OF IMMUNOLOGICALLY COLD SOLID TUMORS CANTEX PHARMACEUTICALS, INC. (US) 2024-07-04 WO claimed
US-20240173322-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS UNIV EMORY (US) 2024-05-30 US claimed
US-11969427-B2 Use of TREM-1 inhibitors for treatment, elimination and eradication of HIV-1 infection EMORY UNIVERSITY (US) 2024-04-30 US claimed
EP-3194572-B1 MEDIA FOR CULTURING PLURIPOTENT STEM CELLS YEDA RES & DEV (IL) 2023-10-25 EP claimed
US-11744831-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2023-09-05 US claimed
US-20220313696-A9 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION UNIV EMORY (US) 2022-10-06 US claimed
US-20220307034-A1 INHIBITING APE2 EXPRESSION IN A SUBJECT TREATED WITH A DRUG AGENT THAT CAUSES INCREASED APE2 EXPRESSION THE CLEVELAND CLINIC FOUNDATION 2022-09-29 US claimed
US-20220211706-A1 Methods and Compositions for Treating Cancer UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2022-07-07 US claimed
US-20220110939-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS UNIV EMORY (US) 2022-04-14 US claimed
US-11285154-B2 Methods and compositions for treating cancer UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS (US) 2022-03-29 US claimed
US-20220040185-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION UNIV EMORY (US) 2022-02-10 US claimed
US-20170097334-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2017-04-06 US claimed
US-20160115518-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-04-28 US claimed
US-20110263554-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR WARF - WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2011-10-27 US claimed
WO-2010053573-A2 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR KAWAOKA YOSHIHIRO (US) 2010-05-14 WO claimed
US-20050069492-A1 Imidazo [2,1-b]-1,3,4-thiadiazole suflonamides PHARMASCIENCE INC. (CA) 2005-03-31 US claimed
WO-2026098574-A1 DRUG FOR BRONCHOPULMONARY DYSPLASIA AND USE METHOD THEREFOR 中国福利会国际和平妇幼保健院 2026-05-15 WO disclosed
EP-4735462-A1 COMPOUNDS AND USES THEREFOR GLYCOSYNNOVATIONS PTY LTD (AU) 2026-05-06 EP disclosed
EP-4735463-A1 COMPOUNDS AND USES THEREFOR GLYCOSYNNOVATIONS PTY LTD (AU) 2026-05-06 EP disclosed
US-20260097028-A1 Methods of Treating Myeloproliferative Neoplasms KARTOS THERAPEUTICS INC (US) 2026-04-09 US disclosed
US-12570957-B2 Isolated naive pluripotent stem cells and methods of generating same YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2026-03-10 US disclosed
US-20260028583-A1 ISOLATED NAIVE PLURIPOTENT STEM CELLS AND METHODS OF GENERATING SAME YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2026-01-29 US disclosed
US-20250387383-A1 METHODS OF TREATING MYELOPROLIFERATIVE NEOPLASMS KARTOS THERAPEUTICS, INC. (US) 2025-12-25 US disclosed
EP-4667054-A2 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY Novartis AG (CH) 2025-12-24 EP disclosed
US-12460207-B2 Inhibiting APE2 expression in a subject treated with a drug agent that causes increased APE2 expression THE CLEVELAND CLINIC FOUNDATION (US) 2025-11-04 US disclosed
EP-4629993-A1 METHODS OF TREATING MYELOPROLIFERATIVE NEOPLASMS Kartos Therapeutics (US) 2025-10-15 EP disclosed
US-12427149-B2 Methods and compositions for the prevention and treatment of hearing loss Ting Theropeutics, Inc. (US) 2025-09-30 US disclosed
US-12414981-B2 JNK inhibitors for use in treating and preventing neurodegenerative disorders NORTHWESTERN UNIVERSITY (US) 2025-09-16 US disclosed
US-20250270310-A1 TREATMENT OF KIDNEY INJURY NATIONAL UNIVERSITY OF SINGAPORE (SG) 2025-08-28 US disclosed
US-12390479-B2 Nitric oxide-releasing antibacterial compounds, formulations, and methods pertaining thereto KNOW BIO, LLC (US) 2025-08-19 US disclosed
US-12383558-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2025-08-12 US disclosed
EP-3980400-B1 PEPTIDOMIMETICS FOR THE TREATMENT OF CORONAVIRUS AND PICORNAVIRUS INFECTIONS UNIV EMORY (US) 2025-08-06 EP disclosed
US-20250237642-A1 PREDICTIVE MODEL FOR VARIANTS ASSOCIATED WITH DRUG RESISTANCE AND THERANOSTIC APPLICATIONS THEREOF UNIV EMORY (US) 2025-07-24 US disclosed
EP-3880660-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2025-07-02 EP disclosed
EP-4565577-A1 INHIBITORS AND USES THEREFOR Macquarie University (AU) 2025-06-11 EP disclosed
EP-4556010-A2 JAK INHIBITORS FOR USE IN THE PREVENTION OR TREATMENT OF A VIRAL DISEASE CAUSED BY A CORONAVIRIDAE Emory University (US) 2025-05-21 EP disclosed
US-20250145945-A1 CULTURE MEDIA FOR CULTURING PLURIPOTENT STEM CELLS IN SUSPENSION ACCELLTA LTD. (IL) 2025-05-08 US disclosed
CN-113677706-B Treatment of liver toxicity 新加坡保健服务私人有限公司 2025-05-02 CN disclosed
US-20250127786-A1 Compositions and Methods for the Prevention and Treatment of Hearing Loss TING THERAPEUTICS, INC. (US) 2025-04-24 US disclosed
CN-113166065-B Compounds and compositions for treating disorders associated with NLRP activity 诺华股份有限公司 2025-04-15 CN disclosed
US-20250114389-A1 NUCLEOSIDES AND NUCLEOTIDES ANALOGS AS ANTIVIRAL AGENTS UNIV EMORY (US) 2025-04-10 US disclosed
US-12268681-B2 Methods of treating myeloproliferative neoplasms KARTOS THERAPEUTICS, INC. (US) 2025-04-08 US disclosed
US-12268723-B2 Peptidomimetics for the treatment of coronavirus and picorna virus infections EMORY UNIVERSITY (US) 2025-04-08 US disclosed
US-20250099454-A1 COMBINATION OF 8-CHLORO-N-(4-(TRIFLUOROMETHOXY)PHENYL)QUINOLIN-2-AMINE AND ITS DERIVATIVES WITH A JAK INHIBITOR ABIVAX (FR) 2025-03-27 US disclosed
US-20250092126-A1 TREATMENT AND PREVENTION OF ALCOHOLIC LIVER DISEASE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2025-03-20 US disclosed
US-12252709-B2 Culture media for culturing pluripotent stem cells in suspension ACCELLTA LTD. (IL) 2025-03-18 US disclosed
US-20250082608-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE SINGAPORE HEALTH SERVICES PTE LTD. (SG) 2025-03-13 US disclosed
US-12234284-B2 Treatment of kidney injury NATIONAL UNIVERSITY OF SINGAPORE (SG) 2025-02-25 US disclosed
WO-2025028555-A1 CASK DISORDER TREATING AGENT AND TREATMENT METHOD 国立大学法人信州大学 2025-02-06 WO disclosed
WO-2025000059-A1 COMPOUNDS AND USES THEREFOR Glycosynnovations Pty Ltd (AU) 2025-01-02 WO disclosed
WO-2025000061-A1 COMPOUNDS AND USES THEREFOR Glycosynnovations Pty Ltd (AU) 2025-01-02 WO disclosed
US-20250000364-A1 GASTROINTESTINAL TRACT DETECTION METHODS, DEVICES AND SYSTEMS GLAS USA LLC 2025-01-02 US disclosed
US-20240415838-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION UNIV EMORY (US) 2024-12-19 US disclosed
US-20240408145-A1 Gene Therapy OSPEDALE SAN RAFFAELE SRL (IT) 2024-12-12 US disclosed
EP-3914698-B1 CULTURE MEDIA FOR PLURIPOTENT STEM CELLS YEDA RES & DEV (IL) 2024-12-11 EP disclosed
US-20240400983-A1 CELL AGGREGATE INCLUDING PITUITARY HORMONE-PRODUCING CELLS AND METHOD FOR PRODUCING SAME Sumitomo Pharma Co., Ltd. (JP) 2024-12-05 US disclosed
EP-4469049-A1 COMBINATION OF 8-CHLORO-N-(4-(TRIFLUOROMETHOXY)PHENYL)QUINOLIN-2-AMINE AND ITS DERIVATIVES WITH A JAK INHIBITOR ABIVAX (FR) 2024-12-04 EP disclosed
US-12157768-B2 Anti-LILRB2 antibodies and methods of use thereof ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2024-12-03 US disclosed
US-20240391884-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2024-11-28 US disclosed
US-20240392241-A1 METHOD FOR PRODUCING CELL MASS INCLUDING PITUITARY TISSUE AND CELL MASS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2024-11-28 US disclosed
CN-118873822-A Treatment of gastrointestinal disorders with TNF inhibitors 比奥拉治疗股份有限公司 2024-11-01 CN disclosed
EP-4448096-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE Singapore Health Services Pte. Ltd. (SG) 2024-10-23 EP disclosed
CN-118767143-A Compositions and methods for preventing and treating hearing loss 听治疗有限责任公司 2024-10-15 CN disclosed
CN-118785907-A Combination of 8-chloro-N- (4- (trifluoromethoxy) phenyl) quinolin-2-amine and its derivatives with a JAK inhibitor ABIVAX公司 2024-10-15 CN disclosed
US-20240318144-A1 MEDIA FOR CULTURING NAIVE HUMAN PLURIPOTENT STEM CELLS YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2024-09-26 US disclosed
US-12089916-B2 Gastrointestinal tract detection methods, devices and systems BIORA THERAPEUTICS, INC. (US) 2024-09-17 US disclosed
US-12084424-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2024-09-10 US disclosed
EP-4419543-A1 GENE THERAPY Ospedale San Raffaele S.r.l. (IT) 2024-08-28 EP disclosed
WO-2024171957-A1 TRANSPLANTATION OF PITUITARY HORMONE-PRODUCING CELLS 国立大学法人東海国立大学機構 2024-08-22 WO disclosed
EP-3221446-B1 IN VITRO PRODUCTION OF EXPANDED POTENTIAL STEM CELLS GENOME RES LTD (GB) 2024-08-21 EP disclosed
CN-114981298-B Compositions and methods for preventing and treating hearing loss 听治疗有限责任公司 2024-08-20 CN disclosed
US-20240262857-A1 NOVEL UNIVERSAL ANTI-RNA VIRUS AGENTS EMORY UNIVERSITY 2024-08-08 US disclosed
US-20240261243-A1 NITRIC OXIDE DONORS, COMPOSITIONS, AND METHODS OF USE KNOW BIO, LLC (US) 2024-08-08 US disclosed
EP-4410962-A1 CELL AGGREGATE INCLUDING PITUITARY HORMONE-PRODUCING CELLS AND METHOD FOR PRODUCING SAME Sumitomo Pharma Co., Ltd. (JP) 2024-08-07 EP disclosed
EP-4410832-A2 TREATMENT OF A DISEASE OF THE GASTROINTESTINAL TRACT WITH A TNF INHIBITOR Biora Therapeutics, Inc. (US) 2024-08-07 EP disclosed
EP-4410963-A1 METHOD FOR PRODUCING CELL MASS INCLUDING PITUITARY TISSUE AND CELL MASS Sumitomo Chemical Company, Limited (JP) 2024-08-07 EP disclosed
EP-3554342-B1 TREATMENT OF A DISEASE OF THE GASTROINTESTINAL TRACT WITH A TNF INHIBITOR BIORA THERAPEUTICS INC (US) 2024-07-24 EP disclosed
US-20240238323-A1 MODIFIED NUCLEOSIDES AND NUCLEOTIDES ANALOGS AS ANTIVIRAL AGENTS FOR CORONA AND OTHER VIRUSES EMORY UNIVERSITY 2024-07-18 US disclosed
CN-118318033-A Cell aggregate comprising pituitary hormone-producing cells and method for producing the same 住友制药株式会社 2024-07-09 CN disclosed
WO-2024144816-A1 TREATMENT OF IMMUNOLOGICALLY COLD SOLID TUMORS CANTEX PHARMACEUTICALS, INC. (US) 2024-07-04 WO disclosed
US-20240216413-A1 THIONUCLEOSIDES AS ANTIVIRAL AGENTS EMORY UNIVERSITY (US) 2024-07-04 US disclosed
CN-107898790-B Antiviral JAK inhibitors for the treatment or prevention of retroviral and other viral infections 埃默里大学 2024-06-21 CN disclosed
WO-2024124240-A1 METHODS OF TREATING MYELOPROLIFERATIVE NEOPLASMS KARTOS THERAPEUTICS (US) 2024-06-13 WO disclosed
EP-4376948-A1 TREATMENT AND PREVENTION OF ALCOHOLIC LIVER DISEASE Boehringer Ingelheim International GmbH (DE) 2024-06-05 EP disclosed
US-20240173322-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS UNIV EMORY (US) 2024-05-30 US disclosed
US-20240156913-A1 TREATMENT AND PREVENTION OF METABOLIC DISEASES SINGAPORE HEALTH SERVICES PTE LTD. (SG) 2024-05-16 US disclosed
CN-118043447-A Method for preparing cell population containing pituitary tissue and cell population 住友化学株式会社 2024-05-14 CN disclosed
US-20240139315-A1 COMPOSITIONS AND METHODS FOR PREVENTION AND TREATMENT OF HEARING LOSS ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. 2024-05-02 US disclosed
US-11969427-B2 Use of TREM-1 inhibitors for treatment, elimination and eradication of HIV-1 infection EMORY UNIVERSITY (US) 2024-04-30 US disclosed
CN-110430801-B Treatment of gastrointestinal disorders with TNF inhibitors 比奥拉治疗股份有限公司 2024-04-30 CN disclosed
CN-117881403-A Thionucleosides as antiviral agents 爱莫里大学 2024-04-12 CN disclosed
EP-4349820-A2 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY Novartis AG (CH) 2024-04-10 EP disclosed
CN-117858711-A Nucleoside and nucleotide analogs as antiviral agents 爱莫里大学 2024-04-09 CN disclosed
CN-117769427-A Modified nucleosides and nucleotide analogues as antiviral agents for coronaviruses and other viruses 埃默里大学 2024-03-26 CN disclosed
US-11920164-B2 Media for culturing naive human pluripotent stem cells YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2024-03-05 US disclosed
US-11913018-B2 In vitro production of expanded potential stem cells GENOME RESEARCH LIMITED (GB) 2024-02-27 US disclosed
EP-3658539-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2024-02-21 EP disclosed
EP-4319764-A2 THIONUCLEOSIDES AS ANTIVIRAL AGENTS Emory University (US) 2024-02-14 EP disclosed
EP-4319762-A2 NUCLEOSIDES AND NUCLEOTIDES ANALOGS AS ANTIVIRAL AGENTS Emory University (US) 2024-02-14 EP disclosed
EP-4319763-A2 MODIFIED NUCLEOSIDES AND NUCLEOTIDES ANALOGS AS ANTIVIRAL AGENTS FOR CORONA AND OTHER VIRUSES Emory University (US) 2024-02-14 EP disclosed
CN-111655228-B Compositions and methods for preventing and treating hearing loss 听治疗有限责任公司 2024-02-09 CN disclosed
CN-111094242-B Compounds and compositions for treating disorders associated with NLRP activity 诺华股份有限公司 2024-02-09 CN disclosed
WO-2024026540-A1 INHIBITORS AND USES THEREFOR MACQUARIE UNIVERSITY (AU) 2024-02-08 WO disclosed
EP-3870261-B1 INGESTIBLE DEVICE FOR DELIVERY OF THERAPEUTIC AGENT TO THE GASTROINTESTINAL TRACT BIORA THERAPEUTICS INC (US) 2024-01-31 EP disclosed
US-11883491-B2 Compositions and methods for prevention and treatment of hearing loss ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2024-01-30 US disclosed
EP-4309722-A2 INGESTIBLE DEVICE FOR DELIVERY OF THERAPEUTIC AGENT TO THE GASTROINTESTINAL TRACT Biora Therapeutics, Inc. (US) 2024-01-24 EP disclosed
EP-3880673-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2024-01-03 EP disclosed
EP-3880659-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2024-01-03 EP disclosed
US-20230416211-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-12-28 US disclosed
US-20230399393-A1 METHODS TO EXTEND HEALTH-SPAN AND TREAT AGE-RELATED DISEASES NATIONAL UNIVERSITY OF SINGAPORE (SG) 2023-12-14 US disclosed
CN-117209447-A Compounds and compositions for treating disorders associated with NLRP activity 诺华股份有限公司 2023-12-12 CN disclosed
CN-117143042-A Compounds and compositions for treating disorders associated with NLRP activity 诺华股份有限公司 2023-12-01 CN disclosed
US-11813270-B2 Nitric oxide-releasing antibacterial compounds, formulations, and methods pertaining thereto KNOW BIO, LLC (US) 2023-11-14 US disclosed
US-11813311-B2 Treatment and prevention of metabolic diseases SINGAPORE HEALTH SERVICES PTE LTD. (SG) 2023-11-14 US disclosed
EP-3194572-B1 MEDIA FOR CULTURING PLURIPOTENT STEM CELLS YEDA RES & DEV (IL) 2023-10-25 EP disclosed
US-11787858-B2 Anti-LILRB3 antibodies and methods of use thereof ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-10-17 US disclosed
US-20230312700-A1 TREATMENT OF A DISEASE OF THE GASTROINTESTINAL TRACT WITH A TNF INHIBITOR GLAS USA LLC 2023-10-05 US disclosed
EP-4252629-A2 GASTROINTESTINAL TRACT DETECTION METHODS, DEVICES AND SYSTEMS Biora Therapeutics, Inc. (US) 2023-10-04 EP disclosed
CN-116829583-A Methods for extending the health period and treating age-related disorders 新加坡国立大学 2023-09-29 CN disclosed
WO-2023172635-A1 PREDICTIVE MODEL FOR VARIANTS ASSOCIATED WITH DRUG RESISTANCE AND THERANOSTIC APPLICATIONS THEREOF EMORY UNIVERSITY (US) 2023-09-14 WO disclosed
CN-116726362-A Methods and devices for treating diseases with biologic therapeutic agents 比奥拉治疗股份有限公司 2023-09-12 CN disclosed
CN-116726361-A Methods and devices for treating diseases with biologic therapeutic agents 比奥拉治疗股份有限公司 2023-09-12 CN disclosed
EP-4237448-A1 METHODS TO EXTEND HEALTH-SPAN AND TREAT AGE-RELATED DISEASES National University of Singapore (SG) 2023-09-06 EP disclosed
CN-111094243-B Compounds and compositions for treating disorders associated with NLRP activity 诺华股份有限公司 2023-09-05 CN disclosed
US-11744831-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2023-09-05 US disclosed
US-11744831-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2023-09-05 US disclosed
EP-4232146-A1 METHODS OF TREATING AND PREDICTING NON-RESPONSE TO ANTI-TNF TREATMENT IN SUBJECTS WITH GASTROINTESTINAL TRACT DISEASES Biora Therapeutics, Inc. (US) 2023-08-30 EP disclosed
US-11724992-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-08-15 US disclosed
US-11718631-B2 Sulphonamides and compositions thereof for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-08-08 US disclosed
WO-2023139233-A1 COMBINATION OF 8-CHLORO-N-(4-(TRIFLUOROMETHOXY)PHENYL)QUINOLIN-2-AMINE AND ITS DERIVATIVES WITH A JAK INHIBITOR ABIVAX (FR) 2023-07-27 WO disclosed
EP-4215196-A1 COMBINATION OF 8-CHLORO-N-(4-(TRIFLUOROMETHOXY)PHENYL)QUINOLIN-2-AMINE AND ITS DERIVATIVES WITH A JAK INHIBITOR ABIVAX (FR) 2023-07-26 EP disclosed
US-11707610-B2 Ingestible device for delivery of therapeutic agent to the gastrointestinal tract BIORA THERAPEUTICS, INC. (US) 2023-07-25 US disclosed
EP-4208029-A1 NITRIC OXIDE DONORS, COMPOSITIONS, AND METHODS OF USE KNOW Bio, LLC (US) 2023-07-12 EP disclosed
US-20230212279-A1 TREATMENT AND PREVENTION OF DISEASE CAUSED BY TYPE IV COLLAGEN DYSFUNCTION SINGAPORE HEALTH SERVICES PTE, LTD. (SG) 2023-07-06 US disclosed
WO-2023111196-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE SINGAPORE HEALTH SERVICES PTE. LTD. (SG) 2023-06-22 WO disclosed
US-20230149315-A1 INGESTIBLE DEVICE FOR DELIVERY OF THERAPEUTIC AGENT TO THE GASTROINTESTINAL TRACT GLAS USA LLC 2023-05-18 US disclosed
WO-2023066735-A1 GENE THERAPY OSPEDALE SAN RAFFAELE S.R.L. (IT) 2023-04-27 WO disclosed
CN-113348011-B Method and apparatus for treating disease with biotherapeutic agents 比奥拉治疗股份有限公司 2023-04-18 CN disclosed
WO-2023054395-A1 CELL AGGREGATE INCLUDING PITUITARY HORMONE-PRODUCING CELLS AND METHOD FOR PRODUCING SAME 住友ファーマ株式会社 2023-04-06 WO disclosed
WO-2023054396-A1 METHOD FOR PRODUCING CELL MASS INCLUDING PITUITARY TISSUE AND CELL MASS 住友化学株式会社 2023-04-06 WO disclosed
US-20230079631-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-03-16 US disclosed
US-20230062815-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-03-02 US disclosed
US-20230063462-A1 SULFONIMIDAMIDE COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-03-02 US disclosed
US-20230059136-A1 THE COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-02-23 US disclosed
US-20230051589-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-02-16 US disclosed
US-20230031406-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-02-02 US disclosed
WO-2023006765-A1 TREATMENT AND PREVENTION OF ALCOHOLIC LIVER DISEASE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-02-02 WO disclosed
CN-115666704-A Ingestible device for delivery of therapeutic agents to the gastrointestinal tract 比奥拉治疗股份有限公司 2023-01-31 CN disclosed
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US-20230011652-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-01-12 US disclosed
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WO-2023277135-A1 METHOD FOR PRODUCING CELLS CONSTITUTING NASAL EPITHELIUM, AND CELL POPULATION INCLUDING CELLS CONSTITUTING NASAL EPITHELIUM OR PROGENITOR CELLS THEREOF 住友化学株式会社 2023-01-05 WO disclosed
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US-20220387397-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-12-08 US disclosed
WO-2022251663-A2 NOVEL UNIVERSAL ANTI-RNA VIRUS AGENTS EMORY UNIVERSITY (US) 2022-12-01 WO disclosed
EP-4093205-A1 NITRIC OXIDE-RELEASING ANTIBACTERIAL COMPOUNDS, FORMULATIONS, AND METHODS PERTAINING THERETO KNOW Bio, LLC (US) 2022-11-30 EP disclosed
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US-20220340591-A1 SULPHONAMIDES AND COMPOSITIONS THEREOF FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-10-27 US disclosed
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WO-2022217155-A2 THIONUCLEOSIDES AS ANTIVIRAL AGENTS EMORY UNIVERSITY (US) 2022-10-13 WO disclosed
WO-2022217153-A2 NUCLEOSIDES AND NUCLEOTIDES ANALOGS AS ANTIVIRAL AGENTS EMORY UNIVERSITY (US) 2022-10-13 WO disclosed
WO-2022217154-A2 MODIFIED NUCLEOSIDES AND NUCLEOTIDES ANALOGS AS ANTIVIRAL AGENTS FOR CORONA AND OTHER VIRUSES EMORY UNIVERSITY (US) 2022-10-13 WO disclosed
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US-20220307034-A1 INHIBITING APE2 EXPRESSION IN A SUBJECT TREATED WITH A DRUG AGENT THAT CAUSES INCREASED APE2 EXPRESSION THE CLEVELAND CLINIC FOUNDATION 2022-09-29 US disclosed
US-11439802-B2 Ingestible device for delivery of therapeutic agent to the gastrointestinal tract BIORA THERAPEUTICS, INC. (US) 2022-09-13 US disclosed
US-11433073-B2 Compositions and methods for the prevention and treatment of hearing loss TING THERAPEUTICS LLC (US) 2022-09-06 US disclosed
US-20220273753-A1 PEPTIDOMIMETICS FOR THE TREATMENT OF CORONAVIRUS AND PICORNAVIRUS INFECTIONS EMORY UNIVERSITY 2022-09-01 US disclosed
US-20220273196-A1 INGESTIBLE DEVICE AND ASSOCIATED METHODS GLAS USA LLC 2022-09-01 US disclosed
CN-114981298-A Compositions and methods for preventing and treating hearing loss 听治疗有限责任公司 2022-08-30 CN disclosed
US-20220267276-A1 NLRP MODULATORS NOVARTIS INFLAMMASOME RESEARCH, INC. 2022-08-25 US disclosed
US-20220265660-A1 METHODS AND COMPOSITIONS FOR THE PREVENTION AND TREATMENT OF HEARING LOSS TING THERAPEUTICS LLC (US) 2022-08-25 US disclosed
WO-2022170396-A1 AGENTS AND METHODS FOR THERAPY AND PROPHYLAXIS ViraLok Therapeutics Pty Ltd (AU) 2022-08-18 WO disclosed
US-20220249814-A1 METHODS AND DEVICES FOR TREATING A DISEASE WITH BIOTHERAPEUTICS GLAS USA LLC 2022-08-11 US disclosed
US-20220244263-A1 METHODS FOR TREATING SMALL CELL NEUROENDOCRINE AND RELATED CANCERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-08-04 US disclosed
US-20220227707-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-07-21 US disclosed
US-20220211706-A1 Methods and Compositions for Treating Cancer UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2022-07-07 US disclosed
EP-3697758-B1 SULPHONAMIDES AND COMPOSITIONS THEREOF FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-07-06 EP disclosed
US-11377636-B2 Endogenous retrovirus transcription as a marker for primate naive pluripotent stem cells MAX-DELBRÜCK-CENTRUM FÜR MOLEKULARE MEDIZIN IN DER HELMHOLTZ-GEMEINSCHAFT (DE) 2022-07-05 US disclosed
US-11370763-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2022-06-28 US disclosed
US-20220160736-A1 NITRIC OXIDE-RELEASING ANTIBACTERIAL COMPOUNDS, FORMULATIONS, AND METHODS PERTAINING THERETO KNOW BIO LLC (US) 2022-05-26 US disclosed
US-11339216-B2 Treatment of kidney injury NATIONAL UNIVERSITY OF SINGAPORE (SG) 2022-05-24 US disclosed
US-20220152063-A1 NITRIC OXIDE-RELEASING ANTIBACTERIAL COMPOUNDS, FORMULATIONS, AND METHODS PERTAINING THERETO KNOW BIO LLC (US) 2022-05-19 US disclosed
US-20220145264-A1 CULTURE MEDIUM FOR MAMMALIAN EXPANDED POTENTIAL STEM CELLS, COMPOSITION, AND METHODS THEREOF THE UNIVERSITY OF HONG KONG (CN) 2022-05-12 US disclosed
US-20220133730-A1 Compositions and Methods for the Prevention and Treatment of Hearing Loss TING THERAPEUTICS LLC (US) 2022-05-05 US disclosed
WO-2022090509-A1 METHODS TO EXTEND HEALTH-SPAN AND TREAT AGE-RELATED DISEASES NATIONAL UNIVERSITY OF SINGAPORE (SG) 2022-05-05 WO disclosed
US-11319368-B2 Treatment of hepatotoxicity with IL-11 antibody SINGAPORE HEALTH SERVICES PTE LTD. (SG) 2022-05-03 US disclosed
WO-2022087313-A1 METHODS OF TREATING AND PREDICTING NON-RESPONSE TO ANTI-TNF TREATMENT IN SUBJECTS WITH GASTROINTESTINAL TRACT DISEASES PROGENITY, INC. (US) 2022-04-28 WO disclosed
CN-114364693-A Treatment and prevention of metabolic disorders 新加坡保健服务私人有限公司 2022-04-15 CN disclosed
US-20220110939-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS UNIV EMORY (US) 2022-04-14 US disclosed
EP-3980400-A1 PEPTIDOMIMETICS FOR THE TREATMENT OF CORONAVIRUS AND PICORNAVIRUS INFECTIONS Emory University (US) 2022-04-13 EP disclosed
US-11285154-B2 Methods and compositions for treating cancer UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS (US) 2022-03-29 US disclosed
WO-2022051606-A1 NITRIC OXIDE DONORS, COMPOSITIONS, AND METHODS OF USE KNOW BIO, LLC (US) 2022-03-10 WO disclosed
EP-3962936-A1 TREATMENT AND PREVENTION OF METABOLIC DISEASES Singapore Health Services Pte. Ltd. (SG) 2022-03-09 EP disclosed
US-20220056128-A1 ANTI-LILRB2 ANTIBODIES AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-02-24 US disclosed
US-20220054472-A1 Methods of Treating Myeloproliferative Neoplasms KARTOS THERAPEUTICS INC. 2022-02-24 US disclosed
US-20220040185-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION UNIV EMORY (US) 2022-02-10 US disclosed
EP-3947642-A1 CULTURE MEDIUM FOR MAMMALIAN EXPANDED POTENTIAL STEM CELLS, COMPOSITION, AND METHODS THEREOF The University of Hong Kong (CN) 2022-02-09 EP disclosed
CN-113966393-A Culture medium, composition and method for expanding latent energy stem cells of mammals 香港大学 2022-01-21 CN disclosed
US-11065254-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS (US) 2021-07-20 US disclosed
US-11052090-B2 Use of TREM-1 inhibitors for treatment, elimination and eradication of HIV-1 infection EMORY UNIVERSITY (US) 2021-07-06 US disclosed
US-11045474-B2 Antiviral JAK inhibitors useful in treating or preventing coronaviridae infections EMORY UNIVERSITY (US) 2021-06-29 US disclosed
CN-112804994-A Method for treating myeloproliferative tumors 卡托斯医疗公司 2021-05-14 CN disclosed
EP-3801476-A2 METHODS OF TREATING MYELOPROLIFERATIVE NEOPLASMS Kartos Therapeutics, Inc. (US) 2021-04-14 EP disclosed
EP-3750544-A2 JAK INHIBITORS FOR USE IN THE PREVENTION OR TREATMENT OF VIRAL INFECTION Emory University (US) 2020-12-16 EP disclosed
US-20200352948-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS UNIV EMORY (US) 2020-11-12 US disclosed
US-10821111-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2020-11-03 US disclosed
US-20200316073-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION UNIV EMORY (US) 2020-10-08 US disclosed
CN-111655228-A Compositions and methods for preventing and treating hearing loss J·左 2020-09-11 CN disclosed
US-10765679-B2 Use of TREM-1 inhibitors for treatment, elimination and eradication of HIV-1 infection EMORY UNIVERSITY (US) 2020-09-08 US disclosed
US-20200206229-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS UNIV EMORY (US) 2020-07-02 US disclosed
EP-2785184-B1 COMPOSITIONS COMPRISING JAK INHIBITORS AND HAART DRUGS FOR USE IN THE PREVENTION OR TREATMENT OF HIV UNIV EMORY (US) 2020-06-10 EP disclosed
US-20200093923-A1 COMPOSITIONS AND METHODS FOR PREVENTION AND TREATMENT OF HEARING LOSS ST. JUDE CHILDREN'S RESEARCH HOSPITALEINDHOVEN (US) 2020-03-26 US disclosed
EP-3618807-A1 COMPOSITIONS AND METHODS FOR PREVENTION AND TREATMENT OF HEARING LOSS Zuo, Jian (US) 2020-03-11 EP disclosed
US-20190134039-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2019-05-09 US disclosed
WO-2018204226-A1 COMPOSITIONS AND METHODS FOR PREVENTION AND TREATMENT OF HEARING LOSS ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2018-11-08 WO disclosed
US-10022378-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2018-07-17 US disclosed
US-10022378-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2018-07-17 US disclosed
US-20180185372-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION UNIV EMORY (US) 2018-07-05 US disclosed
US-20180185372-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION UNIV EMORY (US) 2018-07-05 US disclosed
US-20170312283-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2017-11-02 US disclosed
US-20170312283-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2017-11-02 US disclosed
US-20170191038-A1 TGFß SIGNALING INDEPENDENT NAÏVE INDUCED PLURIPOTENT STEM CELLS, METHODS OF MAKING AND USE HONG GUAN LTD (CN) 2017-07-06 US disclosed
US-9662332-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2017-05-30 US disclosed
US-9662332-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2017-05-30 US disclosed
US-20170097334-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2017-04-06 US disclosed
US-20170097334-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2017-04-06 US disclosed
WO-2017007712-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION EMORY UNIVERSITY (US) 2017-01-12 WO disclosed
US-20160115518-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-04-28 US disclosed
US-20160115518-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-04-28 US disclosed
US-9222118-B2 Screen for inhibitors of filovirus and uses therefor WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2015-12-29 US disclosed
US-9222118-B2 Screen for inhibitors of filovirus and uses therefor WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2015-12-29 US disclosed
US-9089574-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2015-07-28 US disclosed
US-9089574-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections EMORY UNIVERSITY (US) 2015-07-28 US disclosed
US-20140328793-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS EMORY UNIVERSITY (US) 2014-11-06 US disclosed
US-20140328793-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS EMORY UNIVERSITY (US) 2014-11-06 US disclosed
WO-2013082476-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS EMORY UNIVERSITY (US) 2013-06-06 WO disclosed
US-20110263554-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR WARF - WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2011-10-27 US disclosed
US-7772260-B2 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-08-10 US disclosed
US-7772260-B2 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-08-10 US disclosed
US-7772260-B2 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-08-10 US disclosed
US-7741349-B2 Imidazo[2, 1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-06-22 US disclosed
US-7741349-B2 Imidazo[2, 1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-06-22 US disclosed
US-7741349-B2 Imidazo[2, 1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-06-22 US disclosed
WO-2010053573-A2 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR KAWAOKA YOSHIHIRO (US) 2010-05-14 WO disclosed
WO-2010053573-A2 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR KAWAOKA YOSHIHIRO (US) 2010-05-14 WO disclosed
US-7714003-B2 Imidazo[2,1-b ]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-05-11 US disclosed
US-7714003-B2 Imidazo[2,1-b ]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-05-11 US disclosed
US-7714003-B2 Imidazo[2,1-b ]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-05-11 US disclosed
US-7700635-B2 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-04-20 US disclosed
US-7700635-B2 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-04-20 US disclosed
US-7700635-B2 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS INC. (CA) 2010-04-20 US disclosed
EP-1463735-B1 IMIDAZO¬2,1-B -1,3,4-THIADIAZOLE SULFONAMIDES AEGERA THERAPEUTICS INC (CA) 2009-08-12 EP disclosed
EP-1463735-B1 IMIDAZO¬2,1-B -1,3,4-THIADIAZOLE SULFONAMIDES AEGERA THERAPEUTICS INC (CA) 2009-08-12 EP disclosed
US-20090179638-A1 ASSAY FOR IDENTIFYING INHIBITORS OF NEURONAL APOPTOTIC PATHWAYS AEGERA THERAPEUTICS INC. (CA) 2009-07-16 US disclosed
US-20090179638-A1 ASSAY FOR IDENTIFYING INHIBITORS OF NEURONAL APOPTOTIC PATHWAYS AEGERA THERAPEUTICS INC. (CA) 2009-07-16 US disclosed
US-20090170845-A1 USE OF IMIDAZO[2,1-b]-1,3,4-THIADIAZOLE-2-SULFONAMIDE COMPOUNDS TO TREAT NEUROPATHIC PAIN AEGERA THERAPEUTICS INC. (CA) 2009-07-02 US disclosed
US-20090170845-A1 USE OF IMIDAZO[2,1-b]-1,3,4-THIADIAZOLE-2-SULFONAMIDE COMPOUNDS TO TREAT NEUROPATHIC PAIN AEGERA THERAPEUTICS INC. (CA) 2009-07-02 US disclosed
US-20090170845-A1 USE OF IMIDAZO[2,1-b]-1,3,4-THIADIAZOLE-2-SULFONAMIDE COMPOUNDS TO TREAT NEUROPATHIC PAIN AEGERA THERAPEUTICS INC. (CA) 2009-07-02 US disclosed
US-20090042953-A1 IMIDAZO [2,1,-b]-1,3,4-THIADIAZOLE SULFONAMIDES AEGERA THERAPEUTICS, INC. (CA) 2009-02-12 US disclosed
US-20090042953-A1 IMIDAZO [2,1,-b]-1,3,4-THIADIAZOLE SULFONAMIDES AEGERA THERAPEUTICS, INC. (CA) 2009-02-12 US disclosed
US-20090042953-A1 IMIDAZO [2,1,-b]-1,3,4-THIADIAZOLE SULFONAMIDES AEGERA THERAPEUTICS, INC. (CA) 2009-02-12 US disclosed
EP-2012782-A1 USE OF IMIDAZO[2,1-b)]-1,3,4-THIADIAZOLE-2-SULFONAMIDE COMPOUNDS TO TREAT NEUROPATHIC PAIN Aegera Therapeutics Inc. (CA) 2009-01-14 EP disclosed
US-20070265319-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-11-15 US disclosed
US-20070265319-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-11-15 US disclosed
US-20070265319-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-11-15 US disclosed
WO-2007118318-A1 USE OF IMIDAZO[2,1-b)]-1,3,4-THIADIAZOLE-2-SULFONAMIDE COMPOUNDS TO TREAT NEUROPATHIC PAIN AEGERA THERAPEUTICS INC. (CA) 2007-10-25 WO disclosed
US-20070238768-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-10-11 US disclosed
US-20070238766-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-10-11 US disclosed
US-20070238766-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-10-11 US disclosed
US-20070238768-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-10-11 US disclosed
US-20070238766-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-10-11 US disclosed
US-20070238768-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-10-11 US disclosed
WO-2007087716-A1 ASSAY FOR IDENTIFYING INHIBITORS OF NEURONAL APOPTOTIC PATHWAYS AEGERA THERAPEUTICS INC. (CA) 2007-08-09 WO disclosed
US-7230019-B2 Imidazo [2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-06-12 US disclosed
US-7230019-B2 Imidazo [2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-06-12 US disclosed
US-7230019-B2 Imidazo [2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-06-12 US disclosed
US-20070088059-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides PHARMASCIENCE INC. (CA) 2007-04-19 US disclosed
US-20070088059-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides PHARMASCIENCE INC. (CA) 2007-04-19 US disclosed
US-20070088059-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides PHARMASCIENCE INC. (CA) 2007-04-19 US disclosed
US-20070021416-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-01-25 US disclosed
US-20070021416-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-01-25 US disclosed
US-20070021416-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides AEGERA THERAPEUTICS, INC. (CA) 2007-01-25 US disclosed
US-20070021476-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides PHARMASCIENCE INC. (CA) 2007-01-25 US disclosed
US-20070021476-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides PHARMASCIENCE INC. (CA) 2007-01-25 US disclosed
US-20070021476-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides PHARMASCIENCE INC. (CA) 2007-01-25 US disclosed
US-20050069492-A1 Imidazo [2,1-b]-1,3,4-thiadiazole suflonamides PHARMASCIENCE INC. (CA) 2005-03-31 US disclosed
EP-1463735-A1 IMIDAZO[2,1-B]-1,3,4-THIADIAZOLE SULFONAMIDES Aegera Therapeutics Inc. (CA) 2004-10-06 EP disclosed
WO-2003051890-A1 IMIDAZO [2,1-B]-1,3,4-THIADIAZOLE SUFLONAMIDES AEGERA THERAPEUTICS INC. (CA) 2003-06-26 WO disclosed
WO-2003051890-A1 IMIDAZO [2,1-B]-1,3,4-THIADIAZOLE SUFLONAMIDES AEGERA THERAPEUTICS INC. (CA) 2003-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230062815-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 MEN1 3390/4885KMT2A 4441/4885CA12 2839/4885
US-20240216413-A1 THIONUCLEOSIDES AS ANTIVIRAL AGENTS MTAP, NSUN3, METTL3 MEN1 3603/4885KMT2A 1555/4885CA12 3066/4885
US-20250387383-A1 METHODS OF TREATING MYELOPROLIFERATIVE NEOPLASMS JAK2, JAK1, MPL MEN1 1150/4885KMT2A 723/4885CA12 4748/4885
US-20260028583-A1 ISOLATED NAIVE PLURIPOTENT STEM CELLS AND METHODS OF GENERATING SAME PRKD3, GSK3B, GSK3A MEN1 3714/4885KMT2A 955/4885CA12 4532/4885
US-10821111-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections JAK1, JAK3, PNP MEN1 4875/4885KMT2A 253/4885CA12 4773/4885
US-20140328793-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS JAK1, JAK3, PNP MEN1 4875/4885KMT2A 253/4885CA12 4773/4885
US-11707610-B2 Ingestible device for delivery of therapeutic agent to the gastrointestinal tract MUC1, SLC10A2, FABP2 MEN1 1260/4885KMT2A 4184/4885CA12 488/4885
US-20220054472-A1 Methods of Treating Myeloproliferative Neoplasms JAK2, JAK1, PDPK1 MEN1 1475/4885KMT2A 445/4885CA12 4734/4885
US-12089916-B2 Gastrointestinal tract detection methods, devices and systems FABP2, SI, MLNR MEN1 3932/4885KMT2A 4575/4885CA12 188/4885
US-12390479-B2 Nitric oxide-releasing antibacterial compounds, formulations, and methods pertaining thereto NOS1, NOS2, NOS3 MEN1 3202/4885KMT2A 3019/4885CA12 4564/4885
US-12570957-B2 Isolated naive pluripotent stem cells and methods of generating same GSK3B, EZH2, GSK3A MEN1 3667/4885KMT2A 313/4885CA12 4433/4885
US-20160115518-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR ZC3HAV1, WASF2, ZC3HAV1L MEN1 2749/4885KMT2A 3879/4885CA12 4598/4885
US-20230031406-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 MEN1 3390/4885KMT2A 4441/4885CA12 2839/4885
US-20230079631-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 MEN1 3390/4885KMT2A 4441/4885CA12 2839/4885
US-20090170845-A1 USE OF IMIDAZO[2,1-b]-1,3,4-THIADIAZOLE-2-SULFONAMIDE COMPOUNDS TO TREAT NEUROPATHIC PAIN SCN1B, SCN3A, SCN1A MEN1 3389/4885KMT2A 2979/4885CA12 4706/4885
US-20200352948-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS JAK1, JAK3, PNP MEN1 4793/4885KMT2A 130/4885CA12 4832/4885
US-20230051589-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 MEN1 3277/4885KMT2A 4465/4885CA12 2844/4885
US-20230023414-A1 METHODS AND DEVICES FOR TREATING A DISEASE WITH BIOTHERAPEUTICS HAVCR2, CD47, FCGR3B MEN1 903/4885KMT2A 3139/4885CA12 275/4885
US-11744831-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections JAK1, JAK3, PNP MEN1 4796/4885KMT2A 168/4885CA12 4674/4885
US-12268681-B2 Methods of treating myeloproliferative neoplasms JAK2, JAK1, PDPK1 MEN1 1475/4885KMT2A 445/4885CA12 4734/4885
US-20200206229-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS JAK1, JAK3, PNP MEN1 4875/4885KMT2A 253/4885CA12 4773/4885
US-20220110939-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS JAK1, JAK3, PNP MEN1 4796/4885KMT2A 168/4885CA12 4674/4885
US-20220387397-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 MEN1 3294/4885KMT2A 4417/4885CA12 3146/4885
US-20220339169-A1 METHODS OF TREATING OR SELECTING A TREATMENT FOR A SUBJECT RESISTANT TO TNF INHIBITOR USING A NLRP3 ANTAGONIST NLRP3, NLRP1, TNF MEN1 4298/4885KMT2A 4750/4885CA12 3752/4885
US-20220340591-A1 SULPHONAMIDES AND COMPOSITIONS THEREOF FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 MEN1 3988/4885KMT2A 2903/4885CA12 2416/4885
US-20070021476-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides SMN1; SMN2, PMP22, BDNF MEN1 3572/4885KMT2A 3862/4885CA12 3878/4885
US-20260097028-A1 Methods of Treating Myeloproliferative Neoplasms JAK2, TP53, CDKN1A MEN1 1822/4885KMT2A 1324/4885CA12 4586/4885
US-20220160736-A1 NITRIC OXIDE-RELEASING ANTIBACTERIAL COMPOUNDS, FORMULATIONS, AND METHODS PERTAINING THERETO NOS1, NOS2, NOS3 MEN1 3202/4885KMT2A 3019/4885CA12 4564/4885
US-20090042953-A1 IMIDAZO [2,1,-b]-1,3,4-THIADIAZOLE SULFONAMIDES PMP22, SMN1; SMN2, BDNF MEN1 3442/4885KMT2A 3774/4885CA12 3873/4885
US-20230011652-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 MEN1 3418/4885KMT2A 4433/4885CA12 2983/4885
US-20220152063-A1 NITRIC OXIDE-RELEASING ANTIBACTERIAL COMPOUNDS, FORMULATIONS, AND METHODS PERTAINING THERETO NOS1, NOS2, NOS3 MEN1 3202/4885KMT2A 3019/4885CA12 4564/4885
US-11718631-B2 Sulphonamides and compositions thereof for treating conditions associated with NLRP activity NLRP1, NLRP3, NOD1 MEN1 3988/4885KMT2A 2903/4885CA12 2416/4885
US-20190134039-A1 ANTIVIRAL JAK INHIBITORS USEFUL IN TREATING OR PREVENTING RETROVIRAL AND OTHER VIRAL INFECTIONS JAK1, JAK3, PNP MEN1 4875/4885KMT2A 253/4885CA12 4773/4885
US-20070265319-A1 Imidazo[2,1-b]-1,3,4-thiadiazole sulfonamides SMN1; SMN2, PMP22, BDNF MEN1 3572/4885KMT2A 3862/4885CA12 3878/4885
US-20230063462-A1 SULFONIMIDAMIDE COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 MEN1 2868/4885KMT2A 2653/4885CA12 1332/4885
US-20240408145-A1 Gene Therapy MCL1, DNASE1L3, CDKN1A MEN1 3359/4885KMT2A 764/4885CA12 4688/4885
US-20220273753-A1 PEPTIDOMIMETICS FOR THE TREATMENT OF CORONAVIRUS AND PICORNAVIRUS INFECTIONS ACE2, SARS1, VIP MEN1 1932/4885KMT2A 2906/4885CA12 1344/4885
US-20240415838-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION MERTK, PNP, HAVCR2 MEN1 3046/4885KMT2A 300/4885CA12 4746/4885
US-20240261243-A1 NITRIC OXIDE DONORS, COMPOSITIONS, AND METHODS OF USE NOS2, NOS1, NOS3 MEN1 1564/4885KMT2A 4126/4885CA12 3092/4885
US-20110263554-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR ZC3HAV1, WASF2, ZC3HAV1L MEN1 2619/4885KMT2A 3882/4885CA12 4645/4885
US-12084424-B2 Compounds and compositions for treating conditions associated with NLRP activity NLRP1, NLRP3, NOD1 MEN1 3390/4885KMT2A 4441/4885CA12 2839/4885
US-11724992-B2 Compounds and compositions for treating conditions associated with NLRP activity NLRP1, NLRP3, NOD1 MEN1 3390/4885KMT2A 4441/4885CA12 2839/4885
US-11547301-B2 Methods for collecting and testing bacteria containing samples from within the gastrointestinal tract SI, VIP, MLN MEN1 2076/4885KMT2A 4477/4885CA12 2674/4885
US-10022378-B2 Antiviral JAK inhibitors useful in treating or preventing retroviral and other viral infections JAK1, JAK3, PNP MEN1 4875/4885KMT2A 253/4885CA12 4773/4885
US-12268723-B2 Peptidomimetics for the treatment of coronavirus and picorna virus infections ACE2, SARS1, HAVCR2 MEN1 2273/4885KMT2A 2785/4885CA12 1470/4885
US-20170097334-A1 SCREEN FOR INHIBITORS OF FILOVIRUS AND USES THEREFOR ZC3HAV1, WASF2, ZC3HAV1L MEN1 2749/4885KMT2A 3879/4885CA12 4598/4885
US-20250114389-A1 NUCLEOSIDES AND NUCLEOTIDES ANALOGS AS ANTIVIRAL AGENTS PNP, MTAP, NOP2 MEN1 3159/4885KMT2A 2061/4885CA12 4128/4885
US-20250099454-A1 COMBINATION OF 8-CHLORO-N-(4-(TRIFLUOROMETHOXY)PHENYL)QUINOLIN-2-AMINE AND ITS DERIVATIVES WITH A JAK INHIBITOR JAK2, JAK1, JAK3 MEN1 1600/4885KMT2A 99/4885CA12 3782/4885
US-20200316073-A1 USE OF TREM-1 INHIBITORS FOR TREATMENT, ELIMINATION AND ERADICATION OF HIV-1 INFECTION MERTK, PNP, HAVCR2 MEN1 3046/4885KMT2A 300/4885CA12 4746/4885
US-11969427-B2 Use of TREM-1 inhibitors for treatment, elimination and eradication of HIV-1 infection MERTK, PNP, HAVCR2 MEN1 3046/4885KMT2A 300/4885CA12 4746/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.