Cystamine

Cystamine

SCHEMBL320311

Cl.Cl.NCCSSCCN

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Cystamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 1.00
TDP1 Q9NUW8 4/20 1.00
EHMT2 Q96KQ7 1/20 1.00
TSHR P16473 2/20 0.91
THPO P40225 1/20 0.91
CYP1A2 P05177 1/20 0.35
NOS1 P29475 1/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 2/20 0.33
ALDH1A1 P00352 2/20 0.33
BLM P54132 1/20 0.33
CYP3A4 P08684 1/20 0.33
APEX1 P27695 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TRPA1 O75762 1/20 0.33
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cystamine SCHEMBL196510 1.00
Cystamine SCHEMBL28842776 1.00 MAPT (1.00) MAPTTDP1EHMT2TSHRTHPO
Cystamine SCHEMBL28235943 1.00 MAPT (1.00) MAPTTDP1EHMT2TSHRTHPO
Cystamine SCHEMBL345893 1.00 MAPT (1.00) MAPTTDP1EHMT2TSHRTHPO
Cystamine SCHEMBL28418529 0.96 MAPT (0.92) MAPTTDP1EHMT2TSHRTHPO
Cystamine SCHEMBL7903150 0.96 MAPT (0.92) MAPTTDP1EHMT2TSHRTHPO
Cystamine SCHEMBL28409923 0.96 MAPT (0.92) MAPTTDP1EHMT2TSHRTHPO
Cystamine SCHEMBL43866 0.95
Cystamine SCHEMBL3648870 0.95 TSHR (1.00) MAPTTDP1EHMT2TSHRTHPO
Cystamine SCHEMBL11040994 0.95

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3226 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026105108-A2 AN ERGOTHIONEINE-CURCUMIN SYNERGISTIC ANTI-INFLAMMATORY AND ANTI-AGING COMPLEX COMPOSITION AND A PREPARATION METHOD THEREOF ZIRAOUI ANAS (EG) 2026-05-21 WO claimed
US-20260139097-A1 SELF-HEALING MULTI-COMPONENT POLYIMIDE COMPOSITION AND FILM, AND METHOD FOR MANUFACTURING THE SAME KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2026-05-21 US claimed
CN-122060219-A Degradable environment-friendly flame retardant and preparation method thereof 江西砥石矿纤技术有限公司 2026-05-19 CN claimed
CN-122056827-A Nanometer ophthalmic gel preparation for treating corneal epithelial injury 福州大学附属省立医院 2026-05-19 CN claimed
CN-122013511-A First bath dipping liquid for two-bath dipping method of fiber framework material 浙江海利得科技有限公司 2026-05-12 CN claimed
CN-122005429-A Medicine-carrying microneedle patch for inhibiting keloid hyperplasia and preparation method thereof 中国人民解放军总医院海南医院 2026-05-12 CN claimed
EP-4678163-A2 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING NAIL AND SKIN TINEA Chang, Byeung Mo (KR) 2026-01-14 EP claimed
CN-118388745-B Polyurethane elastomer material and preparation method thereof 菁彩新材料(安徽)有限公司 2025-06-24 CN claimed
CN-120114530-A Glutaraldehyde gel and preparation method thereof 沈阳望力生物科技有限公司 2025-06-10 CN claimed
CN-117428874-B High-antibacterial mildew-proof composite board for furniture and manufacturing process thereof 上海拉迷家具有限公司 2025-06-03 CN claimed
WO-2001084976-A2 SELF-NEUTRALIZING PERMANENT WAVE COMPOSITION AND METHOD THEREFOR SHISEIDO CO., LTD. (JP) 2001-11-15 WO claimed
US-6132955-A Method for derivitizing electrodes and assay methods using such derivitized electrodes IGEN INTERNATIONAL, INC. (US) 2000-10-17 US claimed
US-6008328-A PURIFYING PROTEIN BY CATION EXCHANGE RESIN THEN PASSING THROUGH AN MOLECULAR WEIGHT EXCLUSION MATRIX, RECOVERING THE PURIFIED PROTEIN AMGEN INC. (US) 1999-12-28 US claimed
CN-1034077-C Process for preparing pyrido [2, 3-f ] [1, 4] thiazepines ORTHO PHARMA CORP (US) 1997-02-19 CN claimed
WO-1996036870-A1 METHOD FOR DERIVITIZING ELECTRODES AND ASSAY METHODS USING SUCH DERIVITIZED ELECTRODES IGEN, INC. (US) 1996-11-21 WO claimed
EP-0462696-B1 Novel pyrido [2,3-f][1,4] thiazepines and pyrido [3,2-b][1,5] benzothiazepines ORTHO PHARMA CORP (US) 1995-08-09 EP claimed
EP-0502131-A1 PRODUCTION OF MULTIMERIC GLYCOPROTEINS THROUGH CHEMICAL COUPLING BIOGEN, INC. (US) 1992-09-09 EP claimed
WO-1992005188-A1 PRODUCTION OF MULTIMERIC GLYCOPROTEINS THROUGH CHEMICAL COUPLING BIOGEN, INC. (US) 1992-04-02 WO claimed
EP-0462696-A1 Novel pyrido [2,3-f][1,4] thiazepines and pyrido [3,2-b][1,5] benzothiazepines ORTHO PHARMACEUTICAL CORPORATION (US) 1991-12-27 EP claimed
CN-1056880-A Novel pyrido [2, 3-f ] [1, 4] thiazepines and pyrido [3, 2-b ] [1, 5] benzothiazepines ORTHO PHARMA CORP (US) 1991-12-11 CN claimed