Morpholine

Morpholine

SCHEMBL337059

C1COCCN1.Cl

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Morpholine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morpholine SCHEMBL17336349 1.00
Morpholine SCHEMBL29440831 1.00 MEN1 (0.85)
Morpholine SCHEMBL4620513 1.00
Morpholine SCHEMBL10782491 1.00 MEN1 (0.85)
Morpholine SCHEMBL25338784 0.96
Morpholine SCHEMBL2164566 0.96
Morpholine SCHEMBL15789175 0.96
Morpholine SCHEMBL31312337 0.96
Hydrochloric Acid SCHEMBL8586805 0.96 KDM4E (0.92)
Morpholine SCHEMBL27466765 0.96

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1539 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122057566-A Ionic liquid catalyst for preparing methacrolein and preparation method thereof 中国科学院过程工程研究所 2026-05-19 CN claimed
CN-120022522-A Drug-loaded microneedle, drug-loaded microneedle patch and electrically-controlled drug release microneedle system 成都邦迈医创科技有限公司 2025-05-23 CN claimed
CN-119978822-A Antistatic silicone rubber composition and preparation method thereof 杭州之江有机硅化工有限公司 2025-05-13 CN claimed
CN-118684636-B Synthesis process of 4-morpholine-1-phenylmercapto-2-butanone 上海优合贝德医药科技有限公司 2025-03-11 CN claimed
CN-118684636-A Synthesis process of 4-morpholine-1-phenylmercapto-2-butanone 上海优合贝德医药科技有限公司 2024-09-24 CN claimed
WO-2024105225-A1 SYNERGISTIC COMBINATIONS OF A SIGMA RECEPTOR 1 (S1R) ANTAGONIST AND A SOLUBLE EPOXIDE HYDROLASE INHIBITOR (SEHI) AND THEIR USE IN THE TREATMENT OF PAIN UNIVERSITAT DE BARCELONA (ES) 2024-05-23 WO claimed
CN-118028412-A Extraction processing technology of rice protein 安徽稼仙金佳粮集团股份有限公司 2024-05-14 CN claimed
CN-117986139-A Synthesis method of 1- (biphenyl-4-yl) -2-methyl-2-aminopropane-1-ketone 深圳有为技术控股集团有限公司 2024-05-07 CN claimed
EP-4315482-A1 HALOGEN COMPLEXING AGENTS BOUND TO THE CATHODE SURFACE IN A STATIC ZINC HALIDE BATTERY EOS Energy Technology Holdings, LLC (US) 2024-02-07 EP claimed
CN-108350005-B Chiral agent for preparing homogeneous oligomer 卫材R&D管理有限公司 2024-02-06 CN claimed
EP-0843592-A1 DEHALOGENATION OF HALOGENATED HYDROCARBONS IN AQUEOUS COMPOSITIONS MONSANTO COMPANY (US) 1998-05-27 EP claimed
CN-1171398-A Process for preparing morpholine hydrochloride as precursor of monoxydine hydrochloride LU XINGHAI (CN) 1998-01-28 CN claimed
WO-1997004868-A1 DEHALOGENATION OF HALOGENATED HYDROCARBONS IN AQUEOUS COMPOSITIONS MONSANTO COMPANY (US) 1997-02-13 WO claimed
US-4915169-A Method for controlling the pH of steam fluids using heterocyclic, multifunctional, nitrogen-containing compounds CHEVRON RESEARCH COMPANY (US) 1990-04-10 US claimed
US-4845219-A ANTITUMOR, ANTOCOAGULANT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-07-04 US claimed
EP-0255366-A2 Nitrogen- and sulfur-containing lipid compound, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-02-03 EP claimed
EP-0209274-A2 Furanone derivatives ELI LILLY AND COMPANY (US) 1987-01-21 EP claimed
CN-86104450-A The preparation method of furanone derivatives 1986-12-31 CN claimed
US-4287284-A AND A DEVELOPER OF BUTYL METHACRYLATE-STYRENE RESIN OR BUTADIENE-STYRENE RESIN WITH CARBON BLACK, AND A CARRIER OF POLYVINYLIDENE FLUORIDE COATED STEEL XEROX CORPORATION (US) 1981-09-01 US claimed
US-4097479-A FROM ORGANIC NITRILE AND AZIDE ANION, AMINE SOLVENT MILES LABORATORIES, INC. (US) 1978-06-27 US claimed