Dipyridyl

Dipyridyl

SCHEMBL501755

Cl.Cl.c1ccc(-c2ccccn2)nc1.c1ccc(-c2ccccn2)nc1.c1ccc(-c2ccccn2)nc1

nearest known ligand 0.93

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Dipyridyl. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 known ✓ P51681 3/20 0.93
HSP90AA1 known ✓ P07900 1/20 0.74
GLA known ✓ P06280 1/20 0.62
CYP19A1 known ✓ P11511 1/20 0.50
KDM4E B2RXH2 9/20 0.93
LMNA P02545 3/20 0.93
CCR1 P32246 3/20 0.93
CCR8 P51685 3/20 0.93
CYP1A2 P05177 1/20 0.93
POLB P06746 1/20 0.93
METAP1 P53582 1/20 0.93
BLM P54132 1/20 0.93
HIF1A Q16665 1/20 0.93
DOHH Q9BU89 1/20 0.93
P4HTM Q9NXG6 1/20 0.93
NPC1 O15118 6/20 0.74
TP53 P04637 4/20 0.74
RAB9A P51151 4/20 0.74
ALOX15 P16050 3/20 0.74
SMN1; SMN2 Q16637 3/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dipyridyl SCHEMBL30443629 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL28365105 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL29064174 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL31480063 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL4263105 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL4220617 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL10395611 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL6795069 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL1450622 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL30008960 1.00 KDM4E (0.93) KDM4ELMNACCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118108753-A N, N-dialkyl thioformyl-containing 2-silicon-based indole or pyrrole compound and synthesis method and application thereof 杭州师范大学 2024-05-31 CN claimed
US-20220332902-A1 RADICAL CROSSLINKED ZWITTERIONIC GELS AND USES THEREOF COLORADO SCHOOL OF MINES 2022-10-20 US claimed
US-20120097832-A1 ELECTROSPUN LIGHT-EMITTING FIBERS CORNELL UNIVERSITY (US) 2012-04-26 US claimed
US-8106580-B2 Electrospun light-emitting fibers CORNELL UNIVERSITY (US) 2012-01-31 US claimed
US-20090198574-A1 FLYING FOAM APPARATUS AND METHOD OF MAKING FLYING FOAM GUERRA FRANCISCO 2009-08-06 US claimed
US-20090072728-A1 ELECTROSPUN LIGHT-EMITTING FIBERS CORNELL UNIVERSITY (US) 2009-03-19 US claimed
EP-4701674-A1 CROSSLINKABLE LIQUID COMPOSITION FOR USE IN A METHOD OF TREATING OR PREVENTING AN EYE DISORDER Universiteit Antwerpen (BE) 2026-03-04 EP disclosed
EP-4701622-A1 CROSSLINKABLE LIQUID COMPOSITION FOR USE IN A METHOD OF TREATING AN EYE DISORDER Universiteit Antwerpen (BE) 2026-03-04 EP disclosed
EP-3987287-B1 A METHOD FOR DETECTING AN ANALYTE PSYROS DIAGNOSTICS LTD (GB) 2025-05-14 EP disclosed
EP-4549943-A2 A METHOD FOR DETECTING AN ANALYTE Psyros Diagnostics Limited (GB) 2025-05-07 EP disclosed
CN-119039622-A Photoelectric dual-mode responsive photonic crystal hydrogel suitable for DLP three-dimensional molding 浙江理工大学 2024-11-29 CN disclosed
WO-2024223805-A1 CROSSLINKABLE LIQUID COMPOSITION FOR USE IN A METHOD OF TREATING OR PREVENTING AN EYE DISORDER UNIVERSITEIT ANTWERPEN (BE) 2024-10-31 WO disclosed
WO-2024223806-A1 CROSSLINKABLE LIQUID COMPOSITION FOR USE IN A METHOD OF TREATING AN EYE DISORDER UNIVERSITEIT ANTWERPEN (BE) 2024-10-31 WO disclosed
EP-3394179-A1 PHOTOSTABLE FLUORESCENT POLYMERIC TANDEM DYES INCLUDING LUMINESCENT METAL COMPLEXES Becton, Dickinson and Company (US) 2018-10-31 EP disclosed
WO-2017105928-A1 PHOTOSTABLE FLUORESCENT POLYMERIC TANDEM DYES INCLUDING LUMINESCENT METAL COMPLEXES BECTON, DICKINSON AND COMPANY (US) 2017-06-22 WO disclosed
US-8541940-B2 Electrospun light-emitting fibers CORNELL UNIVERSITY (US) 2013-09-24 US disclosed
US-20120097832-A1 ELECTROSPUN LIGHT-EMITTING FIBERS CORNELL UNIVERSITY (US) 2012-04-26 US disclosed
US-7883649-B2 apparatus for generating foam shapes that float in air having a container, a gas source, an aeration nozzle for aerating a gas from the gas source, an outlet, and a separator for separating extruded foam into individualized foam shapes GUERRA FRANCISCO 2011-02-08 US disclosed
US-20090198574-A1 FLYING FOAM APPARATUS AND METHOD OF MAKING FLYING FOAM GUERRA FRANCISCO 2009-08-06 US disclosed
US-5840443-A SECONDARY CELL COMPRISING ELECTROLYTE AND TWO ELECTRODES, AT LEAST ONE COMPRISING REDOX POLYMER MATERIAL WHICH CHANGES OXIDATION STATE TO TRANSFER CHARGE MIDWEST RESEARCH INSTITUTE (US) 1998-11-24 US disclosed