SCHEMBL6417124

SCHEMBL6417124

CC(C)(C)NC(=O)c1ccc(F)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
HTT P42858 1/20 0.50
PTPN1 P18031 1/20 0.48
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
ATM Q13315 1/20 0.47
MITF O75030 1/20 0.47
MAOB P27338 1/20 0.47
AOC3 Q16853 1/20 0.47
CYP2D6 P10635 1/20 0.46
SNCA P37840 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19625786 1.00 LMNA (0.50) LMNAMEN1KMT2AHTTPTPN1
SCHEMBL17865779 0.89 LMNA (0.58) LMNAHTTMAOBAOC3
SCHEMBL24554348 0.84 MEN1 (0.47) MEN1KMT2AHTTPTPN1CES2
SCHEMBL1233194 0.84 MEN1 (0.47) MEN1KMT2AHTTPTPN1CES2
SCHEMBL2522600 0.83 LMNA (0.53) LMNAKMT2AHTTMAOBAOC3
SCHEMBL1742088 0.82 EGLN1 (0.50) MEN1KMT2APTPN1CES2CES1
SCHEMBL14009645 0.82 MAOB (0.65) LMNAMEN1KMT2AHTTMAOB
SCHEMBL7753604 0.82 TRPV1 (0.59) LMNAHTTPTPN1CES2CES1
SCHEMBL3757683 0.81 NPC1 (0.52) MEN1KMT2APTPN1NPC1RAB9A
SCHEMBL12206267 0.81 KCNN4 (0.48) MEN1KMT2APTPN1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1034783-B1 AMIDE DERIVATIVES FOR THE TREATMENT OF RETINAL NEURODEGENERATIVE DISORDERS SUMITOMO PHARMA (JP) 2004-12-15 EP claimed
US-20020147204-A1 Amide derivative SUMITOMO PHARMACEUTICALS COMPANY, LIMITED 2002-10-10 US claimed
EP-1034783-A1 AMIDE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-09-13 EP claimed
CN-119192012-A Reductive amidation method of aryl fluorosulfonate and isocyanate 南京工业大学 2024-12-27 CN disclosed
US-20230041761-A1 SMALL MOLECULE MODULATORS OF SIGMA-1 AND SIGMA-2 RECEPTORS AND USES THEREOF NORTHWESTERN UNIVERSITY 2023-02-09 US disclosed
US-20220194930-A1 Matrix Metalloproteinase Inhibitors and Imaging Agents, And Methods Using Same UNIV YALE (US) 2022-06-23 US disclosed
CN-113620761-B Preparation method for synthesizing aryl aldehyde compound by reducing aryl secondary amide or aryl secondary amide derivative with phenylsilane 西北工业大学 2022-06-17 CN disclosed
CN-113620761-A Preparation method for synthesizing aryl aldehyde compound by reducing aryl secondary amide or aryl secondary amide derivative with phenylsilane 西北工业大学 2021-11-09 CN disclosed
US-11034648-B2 Cystobactamide derivatives HELMHOLTZ-ZENTRUM FÜR (DE) 2021-06-15 US disclosed
US-10968199-B2 Cycloalkyl-containing apoptosis signal-regulating kinase 1 inhibitors and methods of use thereof ENANTA PHARMACEUTICALS, INC. (US) 2021-04-06 US disclosed
US-20200283428-A1 Matrix Metalloproteinase Inhibitors and Imaging Agents, And Methods Using Same YALE UNIVERSITY 2020-09-10 US disclosed
US-20070293530-A1 SULFAMIDE AND SULFAMATE DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS METHYLGENE INC. (CA) 2007-12-20 US disclosed
US-20070149556-A1 Hydroxypyrimidinone derivatives having inhibitory activity against hiv integrase SHIONOGI & CO., LTD. (JP) 2007-06-28 US disclosed
US-6936736-B2 Amide derivative SUMITOMO MANUFACTURING COMPANY LIMITED (JP) 2005-08-30 US disclosed
EP-1034783-B1 AMIDE DERIVATIVES FOR THE TREATMENT OF RETINAL NEURODEGENERATIVE DISORDERS SUMITOMO PHARMA (JP) 2004-12-15 EP disclosed
US-20020147204-A1 Amide derivative SUMITOMO PHARMACEUTICALS COMPANY, LIMITED 2002-10-10 US disclosed
US-6384033-B1 DRUGS FOR VISION DEFECTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2002-05-07 US disclosed
EP-1184367-A1 AMIDE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2002-03-06 EP disclosed
EP-1034783-A1 AMIDE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-09-13 EP disclosed
US-5563144-A SERATONIN ANTAGONISTS FOR TREATMENT OF DISORDERS OF CENTRAL NERVOUS, CARDIOVASCULAR AND GASTROINTESTINAL SYSTEMS RHONE-POULENC RORER S.A. (FR) 1996-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11034648-B2 Cystobactamide derivatives CTH, CBS, SLC7A11 LMNA 4771/4885MEN1 2023/4885KMT2A 2115/4885
US-20070149556-A1 Hydroxypyrimidinone derivatives having inhibitory activity against hiv integrase HAT1, SULT1A1, CDK20 LMNA 3192/4885MEN1 4651/4885KMT2A 1167/4885
US-20200283428-A1 Matrix Metalloproteinase Inhibitors and Imaging Agents, And Methods Using Same MMP1, MMP3, TIMP3 LMNA 796/4885MEN1 322/4885KMT2A 3234/4885
US-10968199-B2 Cycloalkyl-containing apoptosis signal-regulating kinase 1 inhibitors and methods of use thereof BAD, BCL2, AIFM1 LMNA 2011/4885MEN1 4743/4885KMT2A 3618/4885
US-20220194930-A1 Matrix Metalloproteinase Inhibitors and Imaging Agents, And Methods Using Same MMP3, MMP1, MMP10 LMNA 927/4885MEN1 450/4885KMT2A 2836/4885
US-20070293530-A1 SULFAMIDE AND SULFAMATE DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS HDAC1, HDAC11, HAT1 LMNA 2203/4885MEN1 3832/4885KMT2A 37/4885
US-20020147204-A1 Amide derivative ALDH1A2, NR1H2, HDAC3 LMNA 2807/4885MEN1 3899/4885KMT2A 1003/4885
US-20230041761-A1 SMALL MOLECULE MODULATORS OF SIGMA-1 AND SIGMA-2 RECEPTORS AND USES THEREOF SIGMAR1, TMEM97, OPRM1 LMNA 4760/4885MEN1 4146/4885KMT2A 3188/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.