SCHEMBL155157

SCHEMBL155157

COC(=O)[C@@H](N)C(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.42
CA14 Q9ULX7 2/20 0.42
APLNR P35414 1/20 0.37
DGAT1 O75907 1/20 0.35
CA2 P00918 2/20 0.35
CA1 P00915 1/20 0.35
CA7 P43166 1/20 0.35
GAA P10253 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CTSK P43235 2/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
CYP2D6 P10635 1/20 0.32
PIK3CD O00329 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3002117 1.00 CA12 (0.42) CA12CA14APLNRDGAT1CA2
SCHEMBL3008075 1.00 CA12 (0.42) CA12CA14APLNRDGAT1CA2
Hydrochloric Acid SCHEMBL3014916 0.98 CA12 (0.41) CA12CA14APLNRDGAT1CA2
Oxalic Acid SCHEMBL16148596 0.95 CA12 (0.40) CA12CA14APLNRDGAT1CA2
Oxalic Acid SCHEMBL16148595 0.95 CA12 (0.40) CA12CA14APLNRDGAT1CA2
SCHEMBL13984531 0.83 MEN1 (0.42) CA12CA14APLNRCA2CA1
SCHEMBL21612221 0.83 MEN1 (0.42) CA12CA14APLNRCA2CA1
SCHEMBL12467107 0.83 MEN1 (0.42) CA12CA14APLNRCA2CA1
SCHEMBL16855011 0.80 APLNR (0.41) CA12CA14APLNRDGAT1CA2
SCHEMBL17035397 0.79 CA12 (0.47) CA12CA14APLNRDGAT1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11827612-B2 Hydroxamic acid derivative, method for producing same and use thereof INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2023-11-28 US claimed
EP-4071134-A1 HYDROXAMIC ACID DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Institute of Medicinal Biotechnology, Chinese Academy of Medical Sciences (CN) 2022-10-12 EP claimed
US-20220033369-A1 HYDROXAMIC ACID DERIVATIVE, METHOD FOR PRODUCING SAME AND USE THEREOF INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2022-02-03 US claimed
EP-3817742-B1 HETEROCYCLIC SULFONAMIDE DERIVATIVES AND PHARMACEUTICAL USES THEREOF TEMMUNE THERAPEUTICS NV (BE) 2026-04-08 EP disclosed
EP-4658667-A1 CYCLIC PEPTIDES FOR INHIBITING TNF RECEPTOR 1 ACTIVITY Merck Sharp & Dohme LLC (US) 2025-12-10 EP disclosed
US-20250082609-A1 HETEROCYCLIC SULFONAMIDE DERIVATIVES AND PHARMACEUTICAL USES THEREOF Metrion Biosciences Limited (GB) 2025-03-13 US disclosed
WO-2025031048-A1 HYDROXAMIC ACID COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND USE THEREOF AND PREPARATION METHOD THEREFOR 中国医学科学院医药生物技术研究所 2025-02-13 WO disclosed
US-20250051269-A1 PROCESS OF THE PREPARATION OF HYDROXYLAMINE DERIVATIVES INTERVET INC. (US) 2025-02-13 US disclosed
US-12220461-B2 Polypeptide-coupled small molecule compound and antiviral application thereof GUANGZHOU MEDICAL UNIVERSITY (CN) 2025-02-11 US disclosed
US-12195466-B2 Polyproline mimetics of proline-derived module-15 FORSCHUNGSVERBUND BERLIN E.V. (DE) 2025-01-14 US disclosed
EP-4452921-A1 PROCESS OF THE PREPARATION OF HYDROXYLAMINE DERIVATIVES Intervet International B.V. (NL) 2024-10-30 EP disclosed
WO-2012154204-A1 HYDROXAMIC ACID DERIVATIVES AND THEIR USE IN THE TREATMENT OF BACTERIAL INFECTIONS ACHAOGEN, INC. (US) 2012-11-15 WO disclosed
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed
US-20100190766-A1 ANTIBACTERIAL AGENTS ACHAOGEN, INC. (US) 2010-07-29 US disclosed
US-20100190766-A1 ANTIBACTERIAL AGENTS ACHAOGEN, INC. (US) 2010-07-29 US disclosed
CN-101765585-A Antibacterial agent ACHAOGEN INC 2010-06-30 CN disclosed
US-20100120872-A1 ORGANIC COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2010-05-13 US disclosed
US-20100120872-A1 ORGANIC COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2010-05-13 US disclosed
WO-2010031750-A1 ORGANIC COMPOUNDS FOR APPLICATIONS IN BACTERIAL INFECTIONS TREATMENT NOVARTIS AG (CH) 2010-03-25 WO disclosed
WO-2008154642-A2 ANTIBACTERIAL AGENTS ACHAOGEN, INC. (US) 2008-12-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250082609-A1 HETEROCYCLIC SULFONAMIDE DERIVATIVES AND PHARMACEUTICAL USES THEREOF STS, SQOR, SULT2A1 CA12 395/4885CA14 316/4885APLNR 1886/4885
US-20100190766-A1 ANTIBACTERIAL AGENTS MRPL21, SI, ABCB11 CA12 4051/4885CA14 3029/4885APLNR 3978/4885
US-20100120872-A1 ORGANIC COMPOUNDS AND THEIR USES OAT, OTC, AOX1 CA12 886/4885CA14 778/4885APLNR 3930/4885
US-12220461-B2 Polypeptide-coupled small molecule compound and antiviral application thereof PEPD, PREP, VIP CA12 2076/4885CA14 2318/4885APLNR 314/4885
US-20220033369-A1 HYDROXAMIC ACID DERIVATIVE, METHOD FOR PRODUCING SAME AND USE THEREOF HACL2, NAAA, LCT CA12 792/4885CA14 1025/4885APLNR 2006/4885
US-12195466-B2 Polyproline mimetics of proline-derived module-15 PRAP1, ENPEP, RRP15 CA12 3983/4885CA14 3931/4885APLNR 1159/4885
US-20250051269-A1 PROCESS OF THE PREPARATION OF HYDROXYLAMINE DERIVATIVES HAAO, HNMT, ADH1A CA12 2182/4885CA14 1546/4885APLNR 3485/4885
US-11827612-B2 Hydroxamic acid derivative, method for producing same and use thereof HACL2, NAAA, LCT CA12 792/4885CA14 1025/4885APLNR 2006/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.