Acridine

Acridine

SCHEMBL1798660

Cl.c1ccc2nc3ccccc3cc2c1

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA known ✓ P06280 2/20 0.94
ACHE known ✓ P22303 1/20 0.94
HTR3A known ✓ P46098 1/20 0.62
GAA known ✓ P10253 2/20 0.54
CACNA1B known ✓ Q00975 1/20 0.48
MAPT P10636 3/20 0.94
ALDH1A1 P00352 3/20 0.94
HPGD P15428 3/20 0.94
NQO2 P16083 2/20 0.60
KMT2A Q03164 3/20 0.54
KDM4E B2RXH2 2/20 0.54
NPC1 O15118 2/20 0.54
POLB P06746 2/20 0.54
RAB9A P51151 2/20 0.54
LMNA P02545 1/20 0.54
PTBP1 P26599 1/20 0.54
RCE1 Q9Y256 1/20 0.54
TDP1 Q9NUW8 1/20 0.50
STAT3 P40763 1/20 0.50
MEN1 O00255 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acridine SCHEMBL30257128 1.00 MAPT (0.94) MAPTALDH1A1HPGDGLAACHE
Acridine SCHEMBL96928 1.00 MAPT (0.94) MAPTALDH1A1HPGDGLAACHE
Acridine SCHEMBL28062881 0.97 MAPT (0.88) MAPTALDH1A1HPGDGLAACHE
Acridine SCHEMBL4972293 0.97 ALDH1A1 (1.00) MAPTALDH1A1HPGDGLAACHE
Acridine SCHEMBL3045498 0.97 ALDH1A1 (1.00) MAPTALDH1A1HPGDGLAACHE
Acridine SCHEMBL8339 0.97 ALDH1A1 (1.00) MAPTALDH1A1HPGDGLAACHE
Acridine SCHEMBL1772714 0.97 ALDH1A1 (1.00) MAPTALDH1A1HPGDGLAACHE
Acridine SCHEMBL29352289 0.97 ALDH1A1 (1.00) MAPTALDH1A1HPGDGLAACHE
Acridine SCHEMBL1551975 0.94 ALDH1A1 (0.94) MAPTALDH1A1HPGDGLAACHE
Acridine SCHEMBL2401648 0.94 ALDH1A1 (0.94) MAPTALDH1A1HPGDGLAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 98 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119104733-A Serum amyloid A detection reagent and detection method based on improved spatial proximity chemiluminescence method 无锡壹闪生物科技有限公司 2024-12-10 CN claimed
CN-114874116-A Preparation method of thiosulfonate 苏州照固新材料科技有限公司 2022-08-09 CN claimed
CN-114835674-A Preparation method of aromatic thioether 苏州照固新材料科技有限公司 2022-08-02 CN claimed
CN-113125227-A Autumn aqueous solution for preparing high-resolution chromosome for karyotype analysis and application 上海乐辰生物科技有限公司 2021-07-16 CN claimed
CN-109232589-B Fluorescent probe and preparation and application thereof 贵州大学 2021-04-06 CN claimed
CN-109232589-A Fluorescent probe and preparation and application thereof 贵州大学 2019-01-18 CN claimed
CN-105418501-B 7 pairs of anisidino- benzo [c] acridine hydrochlorides and its preparation method and application 广西中医药大学 2018-04-17 CN claimed
CN-105399671-B 7 p-totuidine base benzo [c] acridine hydrochlorides and its preparation method and application 广西中医药大学 2018-04-17 CN claimed
CN-107142300-A A kind of Listeria enriched medium and preparation method 中国疾病预防控制中心传染病预防控制所 2017-09-08 CN claimed
US-20070026130-A1 Method of developing latent fingerprints ARMOR HOLDINGS FORENSICS, INC. 2007-02-01 US claimed
EP-0058591-B1 EPIMERISATION OF TRANS CHRYSANTHEMIC ACIDS AND INTERMEDIATES OBTAINED THEREFROM ROUSSEL-UCLAF (FR) 1984-10-03 EP claimed
US-4447637-A Epimerization of trans chrysanthemates ROUSSEL UCLAF (FR) 1984-05-08 US claimed
CN-119657220-A Application of acridine yellow as catalyst in TMB oxidation color reaction 甘肃政法大学 2025-03-21 CN disclosed
CN-119569654-A 9-Aminoacridine compound with multi-electron-withdrawing substituent, and preparation method and application thereof 郑州大学 2025-03-07 CN disclosed
CN-119104733-A Serum amyloid A detection reagent and detection method based on improved spatial proximity chemiluminescence method 无锡壹闪生物科技有限公司 2024-12-10 CN disclosed
US-20240150569-A1 2K-System XETOS AG (DE) 2024-05-09 US disclosed
US-4328210-A Modified Pasteurella bacteria and vaccines prepared therefrom NORDEN LABORATORIES, INC. (US) 1982-05-04 US disclosed
EP-0036995-A1 Veterinary vaccines for pasteurellosis NORDEN LABORATORIES, INC. (US) 1981-10-07 EP disclosed
US-4293545-A IMMUNOLOGY NORDEN LABORATORIES, INC. (US) 1981-10-06 US disclosed
US-3971952-A Method of detecting abnormal behavior of mammalian cells YEDA RESEARCH & DEVELOPMENT CO. LTD. (IL) 1976-07-27 US disclosed