Imidazole Acetic Acid

Imidazole Acetic Acid

SCHEMBL45374

Cl.O=C(O)Cc1c[nH]cn1

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Imidazole Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 known ✓ P31644 4/20 0.38
GABRB2 known ✓ P47870 4/20 0.38
GABRA1 known ✓ P14867 3/20 0.38
GABRA4 known ✓ P48169 3/20 0.38
GABRP known ✓ O00591 2/20 0.32
GABRD known ✓ O14764 2/20 0.32
GABRB1 known ✓ P18505 2/20 0.32
GABRG2 known ✓ P18507 2/20 0.32
GABRB3 known ✓ P28472 2/20 0.32
GABRA3 known ✓ P34903 2/20 0.32
GABRA2 known ✓ P47869 2/20 0.32
GABRE known ✓ P78334 2/20 0.32
GABRA6 known ✓ Q16445 2/20 0.32
GABRG1 known ✓ Q8N1C3 2/20 0.32
GABRG3 known ✓ Q99928 2/20 0.32
GABRQ known ✓ Q9UN88 2/20 0.32
CA2 known ✓ P00918 1/20 0.30
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Imidazole Acetic Acid SCHEMBL28497348 1.00 ALDH1A1 (0.41) ALDH1A1KDM4EMAPTPMP22GABRR1
Imidazole Acetic Acid SCHEMBL637983 0.98
Imidazole Acetic Acid SCHEMBL27340954 0.98
Imidazole Acetic Acid SCHEMBL9099789 0.98 GABRR1 (0.41) ALDH1A1KDM4EMAPTPMP22GABRR1
Imidazole Acetic Acid SCHEMBL27315430 0.96 GABRR1 (0.40) ALDH1A1KDM4EMAPTPMP22GABRR1
Imidazole Acetic Acid SCHEMBL2787422 0.96 GABRR1 (0.40) ALDH1A1KDM4EMAPTPMP22GABRR1
Imidazole Acetic Acid SCHEMBL14742176 0.82 GABRR1 (0.32) ALDH1A1KDM4EMAPTGABRR1HSD17B10
Hydrochloric Acid SCHEMBL424014 0.82 HTT (0.33) CA2
SCHEMBL2029405 0.82 KDM4E (0.35) ALDH1A1KDM4EMAPTGABRR1HSD17B10
Hydrochloric Acid SCHEMBL2693228 0.82 HTT (0.33) CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 396 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12409150-B2 pH-sensitive carbon nanoparticles, preparation method therefor, and drug delivery using same PCE TECH CO., LTD. (KR) 2025-09-09 US claimed
EP-4430102-B1 POLYOXAZOLINE BASED THERMAL LATENT CURING AGENTS FOR THERMOSET RESINS UNIV SABANCI (TR) 2025-06-25 EP claimed
WO-2025049588-A1 NOVEL TREATMENTS FOR OPTIC NEUROPATHIES AND GLAUCOMA THE TRUSTEES OF INDIANA UNIVERSITY (US) 2025-03-06 WO claimed
EP-4444058-A1 PEROVSKITE SOLAR CELL AND PHOTOVOLTAIC MODULE Contemporary Amperex Technology (Hong Kong) Limited (HK) 2024-10-09 EP claimed
US-20240324253-A1 PEROVSKITE SOLAR CELL AND PHOTOVOLTAIC MODULE CONTEMPORARY AMPEREX TECHNOLOGY (HONG KONG) LIMITED (CN) 2024-09-26 US claimed
EP-4430102-A1 POLYOXAZOLINE BASED THERMAL LATENT CURING AGENTS FOR THERMOSET RESINS Sabanci Üniversitesi (TR) 2024-09-18 EP claimed
EP-4271159-A1 PEROVSKITE SOLAR CELL, AND PHOTOVOLTAIC ASSEMBLY Contemporary Amperex Technology Co., Limited (CN) 2023-11-01 EP claimed
CN-116965169-A Perovskite solar cell, photovoltaic module 宁德时代新能源科技股份有限公司 2023-10-27 CN claimed
WO-2023103650-A1 PEROVSKITE SOLAR CELL AND PHOTOVOLTAIC MODULE 宁德时代新能源科技股份有限公司 2023-06-15 WO claimed
CN-116261336-A Perovskite solar cell and photovoltaic module 宁德时代新能源科技股份有限公司 2023-06-13 CN claimed
US-20110206617-A1 MODIFIED POLYSACCHARIDES FOR DRUG AND CONTRAST AGENT DELIVERY WILLIAM MARSH RICE UNIVERSITY 2011-08-25 US claimed
EP-0743574-B1 Migration imaging members XEROX CORP (US) 2000-12-27 EP claimed
EP-0743573-B1 Method for obtaining image contrast migration imaging members XEROX CORP (US) 2000-09-06 EP claimed
EP-0615856-B1 Recording sheets containing tetrazolium, indolinium, imidazole and imidazolinium compounds XEROX CORP (US) 1997-05-14 EP claimed
EP-0743574-A2 Migration imaging members XEROX CORPORATION (US) 1996-11-20 EP claimed
EP-0743573-A2 Method for obtaining image contrast migration imaging members XEROX CORPORATION (US) 1996-11-20 EP claimed
US-5563014-A SOFTENABLE LAYER CONTAINIG PHOTOSENSITIVE MARKING MATERIAL; TRANSPARENTIZING AGENT XEROX CORPORATION (US) 1996-10-08 US claimed
US-5514505-A SELECTIVE TRANSPARENTIZATION OF PHOTOSENSITIVE MIGRATION MARKING PARTICLES EMBEDDED NEAR THE SURFACE OF A SOFTENABLE LAYER SUPPORTED BY AN ELECTROCONDUCTIVE SUBSTRATE XEROX CORPORATION (US) 1996-05-07 US claimed
US-5457486-A Thermal printing XEROX CORPORATION (US) 1995-10-10 US claimed
EP-0615856-A1 Recording sheets containing tetrazolium, indolinium, imidazole and imidazolinium compounds XEROX CORPORATION (US) 1994-09-21 EP claimed