Hydrochloric Acid

Hydrochloric Acid

SCHEMBL5154366

CNc1ccccc1CNC1CCCCC1.Cl

nearest known ligand 0.56

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Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Hydrochloric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GLA known ✓ P06280 1/20 0.46
GAA known ✓ P10253 1/20 0.45
TACR1 known ✓ P25103 1/20 0.45
HRH3 known ✓ Q9Y5N1 1/20 0.45
KDM4E B2RXH2 3/20 0.56
PKM P14618 1/20 0.56
HTT P42858 4/20 0.49
KMT2A Q03164 4/20 0.49
LMNA P02545 2/20 0.49
PABPC1 P11940 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MEN1 O00255 2/20 0.47
ALDH1A1 P00352 2/20 0.47
NPSR1 Q6W5P4 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
ALOX15 P16050 1/20 0.45
SLC2A1 P11166 1/20 0.45
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1143633 0.98 KDM4E (0.58) KDM4EPKMHTTKMT2ALMNA
SCHEMBL16313903 0.83 TAAR1 (0.50) KDM4EPKMKMT2ALMNAL3MBTL1
SCHEMBL15025473 0.83 SLC6A2 (0.50) KDM4EPKMHTTKMT2ALMNA
SCHEMBL15025562 0.81 TACR1 (0.49) KDM4EPKMKMT2AMEN1TACR1
Hydrochloric Acid SCHEMBL11779650 0.80 KDM4E (0.52) KDM4EPKMHTTKMT2ALMNA
Hydrochloric Acid SCHEMBL11781117 0.78 HTT (0.50) KDM4EPKMHTTKMT2ALMNA
SCHEMBL9346814 0.78 KDM4E (0.53) KDM4EPKMHTTKMT2ALMNA
SCHEMBL11634666 0.77 PABPC1 (0.51) KDM4EHTTKMT2APABPC1MEN1
Hydrochloric Acid SCHEMBL11684770 0.77 HTT (0.67) KDM4EHTTKMT2ALMNAPABPC1
Hydrochloric Acid SCHEMBL11687432 0.77 HTT (0.67) KDM4EHTTKMT2ALMNAPABPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776100-B1 TREATMENT OF CANCER USING BENZOIC ACID DERIVATIVES UNIV NEW YORK (US) 2016-08-31 EP disclosed
US-9018259-B2 Treatment of cancer using benzoic acid derivatives NEW YORK UNIVERSITY (US) 2015-04-28 US disclosed
US-20120329861-A1 TREATMENT OF CANCER USING BENZOIC ACID DERIVATIVES NEW YORK UNIVERSITY (US) 2012-12-27 US disclosed
US-8198328-B2 Treatment of cancer using benzoic acid derivatives NEW YORK UNIVERSITY (US) 2012-06-12 US disclosed
EP-1776100-A4 TREATMENT OF CANCER USING BENZOIC ACID DERIVATIVES UNIV NEW YORK (US) 2007-12-26 EP disclosed
EP-1776100-A2 TREATMENT OF CANCER USING BENZOIC ACID DERIVATIVES NEW YORK UNIVERSITY (US) 2007-04-25 EP disclosed
US-20050209334-A1 method of treating cancer using benzoic acid derivatives, alone or in combination with standard treatments such as chemotherapy and radiotherapy methods of screening for benzoic derivatives based on their ability to inhibit the enzyme tyrosinase or to bind to and activate PXR/SXR xenobiotic receptors. NEW YORK UNIVERSITY (US) 2005-09-22 US disclosed
WO-2005070024-A2 TREATMENT OF CANCER USING BENZOIC ACID DERIVATIVES NEW YORK UNIVERSITY (US) 2005-08-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209334-A1 method of treating cancer using benzoic acid derivatives, alone or in combination with standard treatments such as chemotherapy and radiotherapy methods of screening for benzoic derivatives based on their ability to inhibit the enzyme tyrosinase or to bind to and activate PXR/SXR xenobiotic receptors. AHR, TYR, CYP4X1 GLA 402/4885GAA 204/4885TACR1 398/4885
US-20120329861-A1 TREATMENT OF CANCER USING BENZOIC ACID DERIVATIVES AHR, TYR, CYP4X1 GLA 438/4885GAA 167/4885TACR1 271/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.