Bunitrolol

Bunitrolol

SCHEMBL6061096

CC(C)(C)NCC(O)COc1ccccc1C#N.Cl

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Bunitrolol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A known ✓ P08908 2/20 0.97
ADRA2A known ✓ P08913 2/20 0.97
ADRA2B known ✓ P18089 1/20 0.97
MAOA known ✓ P21397 1/20 0.97
HTR2B known ✓ P41595 1/20 0.97
ADRB2 known ✓ P07550 5/20 0.65
CASR known ✓ P41180 4/20 0.65
SLC6A2 known ✓ P23975 3/20 0.65
SLC6A4 known ✓ P31645 3/20 0.65
KCNH2 known ✓ Q12809 3/20 0.65
SLC6A3 known ✓ Q01959 2/20 0.65
ADRB3 known ✓ P13945 1/20 0.65
ADRB1 known ✓ P08588 1/20 0.61
CHRM1 known ✓ P11229 1/20 0.56
DRD1 known ✓ P21728 1/20 0.56
PTGS1 known ✓ P23219 1/20 0.56
ADRA1A known ✓ P35348 1/20 0.56
OPRM1 known ✓ P35372 1/20 0.56
DRD3 known ✓ P35462 1/20 0.56
MAPT P10636 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bunitrolol SCHEMBL142695 1.00 HTR1A (0.97) HTR1AADRA2AADRA2BMAOAHTR2B
Bunitrolol SCHEMBL142696 1.00 HTR1A (0.97) HTR1AADRA2AADRA2BMAOAHTR2B
Bunitrolol SCHEMBL6506350 0.99 HTR1A (1.00) HTR1AADRA2AADRA2BMAOAHTR2B
Bunitrolol SCHEMBL34721 0.99 HTR1A (1.00) HTR1AADRA2AADRA2BMAOAHTR2B
Bunitrolol SCHEMBL29354749 0.99 HTR1A (1.00) HTR1AADRA2AADRA2BMAOAHTR2B
Bunitrolol SCHEMBL34720 0.99 HTR1A (1.00) HTR1AADRA2AADRA2BMAOAHTR2B
SCHEMBL10650914 0.88 HTR1A (0.81) HTR1AADRA2AADRA2BMAOAHTR2B
Penirolol SCHEMBL1254596 0.87 HTR1A (0.79) HTR1AADRA2AADRA2BMAOAHTR2B
SCHEMBL11747215 0.87 HTR1A (0.79) HTR1AADRA2AADRA2BMAOAHTR2B
SCHEMBL10592687 0.87 HTR1A (0.78) HTR1AADRA2AADRA2BMAOAHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1322 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122040175-A Advanced pressure relief method for parallel drilling of roadway 济宁市煤矿安全生产监测监控中心 2026-05-15 CN claimed
CN-122046824-A Method and system for representing aircraft panel assembly stress distribution balance sub-region 北京科技大学 2026-05-15 CN claimed
CN-122048856-A Damaged tray detection and identification method, system and device 深圳粤十冷链机器人有限公司 2026-05-15 CN claimed
CN-121723117-B Pipeline displacement stress prediction method, device, storage medium and equipment 大唐东北电力试验研究院有限公司 2026-05-12 CN claimed
CN-122014722-A Multi-source sensing oil cylinder clamping stress non-uniformity prevention control method 深圳市博硕科技股份有限公司 2026-05-12 CN claimed
CN-121580589-A Shear-resistant-slip constitutive calculation method for split bolts in double-steel-plate shear wall 天津大学 2026-02-27 CN claimed
US-12387956-B2 Systems and methods for controlling non-uniformity APPLIED MATERIALS, INC. (US) 2025-08-12 US claimed
CN-120163324-A Efficient and accurate construction system for curve inclined bridge based on intelligent perception and cooperative control 盐城市交通投资建设控股集团有限公司 2025-06-17 CN claimed
CN-120028486-A Method for evaluating drought resistance and drought resistance gene effect of transgenic corn field 新疆维吾尔自治区农业科学院 2025-05-23 CN claimed
CN-120007253-A Explosion pre-pressure relief and anti-impact method for island working face of mine with high gas rock burst 安徽理工大学 2025-05-16 CN claimed
CN-114459648-A Multi-mode Lamb wave data fusion-based baseline-free stress online monitoring system and monitoring method 哈尔滨工业大学 2022-05-10 CN claimed
CN-114320293-A Coal pillar type rock burst control method based on electric pulse 辽宁工程技术大学 2022-04-12 CN claimed
CN-114216583-A SH guided wave-based temperature stress online monitoring system and monitoring method thereof 北京大学 2022-03-22 CN claimed
CN-114215183-A Construction method for realizing space special-shaped structure pouring by using UHPC material 中交第三航务工程局有限公司 2022-03-22 CN claimed
CN-114092293-A Mine rock and soil industry emergency linkage monitoring system and method based on precise positioning 山东泽明能源科技有限公司 2022-02-25 CN claimed
CN-114008335-A Washer fastening structure 株式会社松尾工业所 2022-02-01 CN claimed
CN-215678149-U Glass internal stress on-line measuring device 江苏华东耀皮玻璃有限公司 2022-01-28 CN claimed
CN-113967106-A Orbital defect prosthesis and processing technology thereof 苏州诺普再生医学有限公司 2022-01-25 CN claimed
CN-113962837-A Mine geotechnical engineering monitoring and evaluation emergency feedback system and method 山东泽明能源科技有限公司 2022-01-21 CN claimed
CN-110683424-B Uneven stress eliminating device for textile tows 神马实业股份有限公司 2022-01-21 CN claimed