Hydrochloric Acid

Hydrochloric Acid

SCHEMBL874057

Cl.Cl.Nc1ccc(-c2ccc(N)c(N)c2)cc1N

nearest known ligand 0.93

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Hydrochloric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 known ✓ Q12809 2/20 0.58
CYP19A1 known ✓ P11511 2/20 0.50
GAA known ✓ P10253 2/20 0.42
HSP90AA1 known ✓ P07900 1/20 0.42
ESR2 known ✓ Q92731 1/20 0.41
TDP1 Q9NUW8 6/20 0.93
KMT2A Q03164 5/20 0.93
MEN1 O00255 4/20 0.93
CYP3A4 P08684 8/20 0.57
ALDH1A1 P00352 7/20 0.57
TSHR P16473 4/20 0.57
MAPK1 P28482 2/20 0.57
ALOX15 P16050 6/20 0.52
HSD17B10 Q99714 5/20 0.52
CYP17A1 P05093 2/20 0.50
CYP11B1 P15538 2/20 0.50
CYP11B2 P19099 2/20 0.50
SMN1; SMN2 Q16637 3/20 0.48
TP53 P04637 1/20 0.48
THRB P10828 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL504482 1.00 TDP1 (0.93) TDP1KMT2AMEN1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL2565398 1.00 TDP1 (0.93) TDP1KMT2AMEN1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL29378721 1.00 TDP1 (0.93) TDP1KMT2AMEN1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL29497777 1.00 TDP1 (0.93) TDP1KMT2AMEN1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL94882 1.00 TDP1 (0.93) TDP1KMT2AMEN1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL30078382 0.97 TDP1 (0.88) TDP1KMT2AMEN1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL28836366 0.97 TDP1 (0.88) TDP1KMT2AMEN1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL1646515 0.97 TDP1 (0.88) TDP1KMT2AMEN1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL9355084 0.97 TDP1 (0.88) TDP1KMT2AMEN1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL866164 0.97 TDP1 (0.88) TDP1KMT2AMEN1KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220354902-A1 METHODS OF GENERATING, REPAIRING AND/OR MAINTAINING CONNECTIVE TISSUE IN VIVO MESOBLAST, INC. (US) 2022-11-10 US disclosed
EP-3424514-B1 TNAP+ MESENCHYMAL PRECURSOR CELLS FOR USE IN TREATING CONNECTIVE TISSUE DISEASES MESOBLAST INC (US) 2022-05-11 EP disclosed
US-10609922-B2 Protection of progenitor cells and regulation of their differentiation PROTEOBIOACTIVES PTY LTD (AU) 2020-04-07 US disclosed
US-20200101118-A1 METHODS OF GENERATING, REPAIRING AND/OR MAINTAINING CONNECTIVE TISSUE IN VIVO MESOBLAST, INC. (US) 2020-04-02 US disclosed
US-10322166-B2 Composition and method for the treatment or prevention of spinal disorders KUNOVUS PTY LTD (AU) 2019-06-18 US disclosed
EP-3424514-A1 METHOD FOR GENERATING, REPAIRING AND/OR MAINTAINING CONNECTIVE TISSUE IN VIVO Mesoblast, Inc. (US) 2019-01-09 EP disclosed
EP-2185165-B1 STRO-1bright CELLS FOR USE IN TREATING CONNECTIVE TISSUE DISEASES MESOBLAST INC (US) 2018-10-03 EP disclosed
US-20180206480-A1 PROTECTION OF PROGENITOR CELLS AND REGULATION OF THEIR DIFFERENTIATION PROTEOBIOACTIVES PTY LTD (AU) 2018-07-26 US disclosed
US-9888679-B2 Protection of progenitor cells and regulation of their differentiation PROTEOBIOACTIVES PTY LTD (AU) 2018-02-13 US disclosed
EP-2229436-B1 PROTECTION OF PROGENITOR CELLS AND REGULATION OF THEIR DIFFERENTIATION PROTEOBIOACTIVES PTY LTD (AU) 2017-08-30 EP disclosed
EP-0960117-B1 FIBROBLAST GROWTH FACTOR HOMOLOGOUS FACTORS (FHFs) AND METHODS OF USE UNIV JOHNS HOPKINS MED (US) 2007-04-18 EP disclosed
EP-1763362-A1 USE OF MORPHOGENIC PROTEINS FOR TREATING CARTILAGE DEFECTS STRYKER CORPORATION (US) 2007-03-21 EP disclosed
US-20060194726-A1 Methods of treating cartilage defects STRYKER CORPORATION 2006-08-31 US disclosed
WO-2005115438-A1 USE OF MORPHOGENIC PROTEINS FOR TREATING CARTILAGE DEFECTS STRYKER CORPORATION (US) 2005-12-08 WO disclosed
US-20040102379-A1 Fibroblast growth factor homologous factors (FHFs) and methods of use THE JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE 2004-05-27 US disclosed
US-6635744-B1 Substantially pure fibroblast growth factor homologous factor-4 polypeptide having specified amino acid sequence; diagnosis and treatment of neurodegenerative and neoplastic disorders THE JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE 2003-10-21 US disclosed
EP-0960117-A4 FIBROBLAST GROWTH FACTOR HOMOLOGOUS FACTORS (FHFs) AND METHODS OF USE UNIV JOHNS HOPKINS MED (US) 2000-06-14 EP disclosed
US-6020189-A Fibroblast growth factor homologous factors (FHFs) and methods of use THE JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 2000-02-01 US disclosed
EP-0960117-A1 FIBROBLAST GROWTH FACTOR HOMOLOGOUS FACTORS (FHFs) AND METHODS OF USE THE JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 1999-12-01 EP disclosed
WO-1998008864-A1 FIBROBLAST GROWTH FACTOR HOMOLOGOUS FACTORS (FHFs) AND METHODS OF USE THE JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 1998-03-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10609922-B2 Protection of progenitor cells and regulation of their differentiation CD44, MCL1, NES KCNH2 4383/4885CYP19A1 4732/4885GAA 1551/4885
US-20180206480-A1 PROTECTION OF PROGENITOR CELLS AND REGULATION OF THEIR DIFFERENTIATION CD44, MCL1, NES KCNH2 4383/4885CYP19A1 4732/4885GAA 1551/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.