Hydrochloric Acid

Hydrochloric Acid

SCHEMBL1064436

CC1CNCCN1S(=O)(=O)c1cccc2cnccc12.Cl.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Hydrochloric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCD known ✓ Q05655 7/20 1.00
PRKD3 known ✓ O94806 6/20 1.00
PRKCZ known ✓ Q05513 6/20 1.00
PRKCG known ✓ P05129 5/20 1.00
PRKCB known ✓ P05771 5/20 1.00
PRKCA known ✓ P17252 5/20 1.00
PRKCH known ✓ P24723 5/20 1.00
PRKCI known ✓ P41743 5/20 1.00
PRKCE known ✓ Q02156 5/20 1.00
PRKCQ known ✓ Q04759 5/20 1.00
PRKD1 known ✓ Q15139 5/20 1.00
ROCK2 known ✓ O75116 12/20 0.61
ROCK1 known ✓ Q13464 11/20 0.61
LCK known ✓ P06239 1/20 0.60
FGFR1 known ✓ P11362 1/20 0.60
FLT4 known ✓ P35916 1/20 0.60
KDR known ✓ P35968 1/20 0.60
HTR1A known ✓ P08908 1/20 0.59
ADRA2A known ✓ P08913 1/20 0.59
ADRA2B known ✓ P18089 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15093619 1.00 PRKCD (1.00) PRKCDPRKD3PRKCZPRKACAPRKCG
Hydrochloric Acid SCHEMBL29968524 1.00 PRKCD (1.00) PRKCDPRKD3PRKCZPRKACAPRKCG
Hydrochloric Acid SCHEMBL6414754 1.00 PRKCD (1.00) PRKCDPRKD3PRKCZPRKACAPRKCG
Hydrochloric Acid SCHEMBL29353191 1.00 PRKCD (1.00) PRKCDPRKD3PRKCZPRKACAPRKCG
SCHEMBL29968723 0.99 PRKCD (1.00) PRKCDPRKD3PRKCZPRKACAPRKCG
SCHEMBL190590 0.99 PRKCD (1.00) PRKCDPRKD3PRKCZPRKACAPRKCG
SCHEMBL13186235 0.99 PRKCD (1.00) PRKCDPRKD3PRKCZPRKACAPRKCG
Calcium SCHEMBL29883592 0.98 PRKCD (0.98) PRKCDPRKD3PRKCZPRKACAPRKCG
Hydrochloric Acid SCHEMBL23795291 0.94 PRKCD (0.88) PRKCDPRKD3PRKCZPRKACAPRKCG
Hydrochloric Acid SCHEMBL23795350 0.94 PRKCD (0.88) PRKCDPRKD3PRKCZPRKACAPRKCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 155 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4304717-A1 USE OF NADOLOL TO TREAT CHRONIC OBSTRUCTIVE PULMONARY DISEASE BY BLOCKAGE OF THE ARRESTIN-2 PATHWAY Chronic Airway Therapeutics Limited (AU) 2024-01-17 EP claimed
US-20230285556-A1 METHODS AND COMPOSITIONS FOR TREATING CANCER OMEROS CORPORATION 2023-09-14 US claimed
WO-2023039578-A1 METHODS AND COMPOSITIONS FOR TREATING CANCER OMEROS CORPORATION (US) 2023-03-16 WO claimed
US-20200046693-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ZELLWEGER SPECTRUM DISORDER NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2020-02-13 US claimed
US-20190331665-A1 COMPOSITIONS AND METHODS FOR IMPROVING SENSITIVITY IN CELL BASED ASSAYS BIOMADISON, INC. 2019-10-31 US claimed
US-10317394-B2 Sensitized cultured cells for botulinum toxin characterization BIOMADISON, INC. (US) 2019-06-11 US claimed
EP-2800973-B1 METHODS AND COMPOUNDS FOR INCREASING SENSITIVITY OF BOTULINUM ASSAYS BIOMADISON INC (US) 2018-05-16 EP claimed
US-20160223524-A1 SENSITIZED CULTURED CELLS FOR BOTULINUM TOXIN CHARACTERIZATION BIOMADISON, INC. 2016-08-04 US claimed
US-9303285-B2 Methods and compounds for increasing sensitivity of botulinum assays BIOMADISON, INC. (US) 2016-04-05 US claimed
US-20140024063-A1 METHODS AND COMPOUNDS FOR INCREASING SENSITIVITY OF BOTULINUM ASSAYS BIOSENTINEL, INC. 2014-01-23 US claimed
US-20030013703-A1 Upregulation of type III endothelial cell nitric oxide synthase by agents that disrupt actin cytoskeletal organization LIAO JAMES K (US) 2003-01-16 US claimed
US-20020082281-A1 UPREGULATION OF TYPE III ENDOTHELIAL CELL NITRIC OXIDE SYNTHASE BY AGENTS THAT DISRUPT ACTIN CYTOSKELETAL ORGANIZATION NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2002-06-27 US claimed
EP-0705433-A4 COMPOSITIONS AND METHODS FOR ANTI-ADDICTIVE NARCOTIC ANALGESIS ACIVITY SCREENING AND TREATMENTS UNIV CALIFORNIA (US) 2001-09-26 EP claimed
EP-0846265-A4 METHODS FOR G PROTEIN COUPLED RECEPTOR ACTIVITY SCREENING UNIV CALIFORNIA (US) 2001-06-27 EP claimed
WO-2000003746-A2 UPREGULATION OF TYPE III ENDOTHELIAL CELL NITRIC OXIDE SYNTHASE BY AGENTS THAT DISRUPT ACTIN CYTOSKELETAL ORGANIZATION THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2000-01-27 WO claimed
EP-0846265-A1 METHODS FOR G PROTEIN COUPLED RECEPTOR ACTIVITY SCREENING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-06-10 EP claimed
WO-1996037775-A1 METHODS FOR G PROTEIN COUPLED RECEPTOR ACTIVITY SCREENING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1996-11-28 WO claimed
EP-0705433-A1 COMPOSITIONS AND METHODS FOR ANTI-ADDICTIVE NARCOTIC ANALGESIS ACIVITY SCREENING AND TREATMENTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1996-04-10 EP claimed
US-5385915-A Using an enzyme inhibitor THE ROCKEFELLER UNIVERSITY (US) 1995-01-31 US claimed
WO-1995000848-A1 COMPOSITIONS AND METHODS FOR ANTI-ADDICTIVE NARCOTIC ANALGESIS ACIVITY SCREENING AND TREATMENTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-01-05 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230285556-A1 METHODS AND COMPOSITIONS FOR TREATING CANCER TP53, CD4, MCL1 PRKCD 2328/4885PRKD3 2542/4885PRKCZ 1911/4885
US-20200046693-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ZELLWEGER SPECTRUM DISORDER HSD17B4, CYP27A1, OAT PRKCD 808/4885PRKD3 1170/4885PRKCZ 560/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.