Hydrochloric Acid

Hydrochloric Acid

SCHEMBL11447743

COc1ccc(C(O)CNC(C)CCc2ccc3c(c2)OCO3)cc1C(N)=O.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Hydrochloric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 known ✓ P08588 17/20 1.00
ADRB2 known ✓ P07550 16/20 1.00
ADRB3 known ✓ P13945 15/20 1.00
ADRA1D known ✓ P25100 13/20 0.85
ADRA1A known ✓ P35348 13/20 0.85
ADRA1B known ✓ P35368 13/20 0.85
ADRA2A known ✓ P08913 2/20 0.54
GAA known ✓ P10253 1/20 0.54
ADRA2B known ✓ P18089 1/20 0.54
ADRA2C known ✓ P18825 1/20 0.54
HTR1A known ✓ P08908 1/20 0.52
SLC6A2 known ✓ P23975 1/20 0.52
SLC6A4 known ✓ P31645 1/20 0.52
OPRM1 known ✓ P35372 1/20 0.52
DRD3 known ✓ P35462 1/20 0.52
HTR2B known ✓ P41595 1/20 0.52
SLC6A3 known ✓ Q01959 1/20 0.52
SIGMAR1 known ✓ Q99720 1/20 0.52
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11467502 0.99 ADRB1 (0.98) ADRB1ADRB2ADRB3ADRA1DADRA1A
Medroxalol SCHEMBL588175 0.88 ADRB2 (1.00) ADRB1ADRB2ADRB3ADRA1DADRA1A
Medroxalol SCHEMBL31058839 0.87 ADRB2 (0.98) ADRB1ADRB2ADRB3ADRA1DADRA1A
Medroxalol SCHEMBL30371313 0.87 ADRB2 (0.98) ADRB1ADRB2ADRB3ADRA1DADRA1A
Medroxalol SCHEMBL120537 0.87 ADRB2 (0.98) ADRB1ADRB2ADRB3ADRA1DADRA1A
SCHEMBL11594732 0.82 ADRB1 (0.76) ADRB1ADRB2ADRB3ADRA1DADRA1A
SCHEMBL11457096 0.81 ADRB1 (0.69) ADRB1ADRB2ADRB3ADRA1DADRA1A
SCHEMBL11881655 0.79 ADRB2 (0.98) ADRB1ADRB2ADRB3ADRA1DADRA1A
SCHEMBL11172675 0.75 ADRB2 (0.63) ADRB1ADRB2ADRB3ADRA1DADRA1A
Hydrochloric Acid SCHEMBL11447739 0.75 ADRB2 (0.71) ADRB1ADRB2ADRB3ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4221808-A Novel antihypertensive agent RICHARDSON-MERRELL INC. (US) 1980-09-09 US claimed
US-4221808-A Novel antihypertensive agent RICHARDSON-MERRELL INC. (US) 1980-09-09 US disclosed