Phosphocholine

Phosphocholine

SCHEMBL2456733

C=C(C)C(=O)[O-].C[N+](C)(C)CCOP(=O)(O)O.Cl

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Phosphocholine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 known ✓ P08912 5/20 0.40
CHRM1 known ✓ P11229 5/20 0.40
CHRM3 known ✓ P20309 5/20 0.40
CHRM2 known ✓ P08172 4/20 0.40
CHRM4 known ✓ P08173 4/20 0.40
CHRNA7 known ✓ P36544 3/20 0.40
HTR1A known ✓ P08908 2/20 0.40
CHRNB4 known ✓ P30926 1/20 0.40
CHRNA3 known ✓ P32297 1/20 0.40
GAA known ✓ P10253 1/20 0.39
ADRA1A known ✓ P35348 2/20 0.38
ESR1 known ✓ P03372 1/20 0.38
AGTR1 known ✓ P30556 1/20 0.38
KCNH2 known ✓ Q12809 1/20 0.38
ADRA2A known ✓ P08913 1/20 0.36
ADRA1D known ✓ P25100 1/20 0.35
HTR1D known ✓ P28221 1/20 0.35
HTR2C known ✓ P28335 1/20 0.35
ADRA1B known ✓ P35368 1/20 0.35
DRD3 known ✓ P35462 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phosphocholine SCHEMBL27766488 0.98 CHRM5 (0.41) CHRM5CHRM1CHRM3CHRM2CHRM4
Phosphocholine SCHEMBL28014826 0.88 SMN1; SMN2 (0.52) CHRM5CHRM1CHRM3CHRM2CHRM4
Phosphocholine SCHEMBL1802772 0.86 CHRM5 (0.42) CHRM5CHRM1CHRM3CHRM2CHRM4
Phosphocholine SCHEMBL8773456 0.86 SMN1; SMN2 (0.42) CHRM5CHRM1CHRM3CHRM2CHRM4
Phosphocholine SCHEMBL19386099 0.85 CHRM5 (0.44) CHRM5CHRM1CHRM3CHRM2CHRM4
Phosphocholine SCHEMBL1085846 0.84 CHRM5 (0.47) CHRM5CHRM1CHRM3CHRM2CHRM4
Phosphocholine SCHEMBL27757850 0.84 LPAR3 (0.45) CHRM5CHRM1CHRM3CHRM2CHRM4
Phosphocholine SCHEMBL18148995 0.83 SMN1; SMN2 (0.39) CHRM5CHRM1CHRM3CHRM2CHRM4
Methacrylic Acid SCHEMBL28639506 0.83 SMN1; SMN2 (0.42) CHRM5CHRM1CHRM3CHRM2CHRM4
Phosphocholine SCHEMBL23466865 0.82 LPAR3 (0.43) CHRM5CHRM1CHRM3CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 175 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260072020-A1 PRINTABLE MOLECULE-SELECTIVE CORE-SHELL NANOPARTICLES FOR WEARABLE AND IMPLANTABLE SENSING CALIFORNIA INST OF TECHN (US) 2026-03-12 US claimed
US-20250188521-A1 NUCLEIC ACID DELIVERY SCAFFOLDS Singular Genomics Systems, Inc. 2025-06-12 US claimed
CN-119529204-A Triblock expansion viscosity-increasing carbon dioxide channeling profile control agent and preparation method thereof 中国石油大学(华东) 2025-02-28 CN claimed
US-12220550-B2 Transdermal delivery device, methods of using and making the same BUDDHIST TZU CHI MEDICAL FOUNDATION (TW) 2025-02-11 US claimed
US-20240167087-A1 MULTI-DIMENSIONAL POLYMER SCAFFOLDS FOR NUCLEIC ACID ANALYSES FIRST-CITIZENS BANK & TRUST COMPANY 2024-05-23 US claimed
US-20240167089-A1 NANOARRAYS AND METHODS OF USE THEREOF FIRST-CITIZENS BANK & TRUST COMPANY 2024-05-23 US claimed
EP-4371653-A1 FABRICATION OF FILTRATION MEMBRANES Trustees of Tufts College (US) 2024-05-22 EP claimed
CN-114957721-B Zwitterionic hydrogel and preparation method and application thereof 四川大学 2024-04-26 CN claimed
CN-117757127-A Preparation method of polyethylene material with biocompatibility and application of polyethylene material in medical field 华东理工大学 2024-03-26 CN claimed
US-11884977-B2 Nanoarrays and methods of use thereof Singular Genomics Systems, Inc. (US) 2024-01-30 US claimed
US-20180001278-A1 ZWITTERIONIC COPOLYMERS FOR FOULING RESISTANT FILTRATION MEMBRANES TRUSTEES OF TUFTS COLLEGE 2018-01-04 US claimed
US-9750852-B2 Modification of bioabsorbable stent to reduce thrombogenecity ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2017-09-05 US claimed
US-20160375143-A1 MIKTO-ARM BRANCHED POLYMERS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2016-12-29 US claimed
US-20160303523-A1 ZWITTERION-CONTAINING MEMBRANES TUFTS UNIVERSITY (US) 2016-10-20 US claimed
US-20160296676-A1 MODIFICATION OF BIOABSORBABLE STENT TO REDUCE THROMBOGENECITY ABBOTT CARDIOVASCULAR SYSTEMS INC (US) 2016-10-13 US claimed
EP-3074440-A1 MIKTO-ARM BRANCHED POLYMERS Commonwealth Scientific & Industrial Research Organisation ( C.S.I.R.O. ) (AU) 2016-10-05 EP claimed
WO-2016109621-A1 ZWITTERIONIC COPOLYMERS FOR FOULING RESISTANT FILTRATION MEMBRANES TUFTS UNIVERSITY (US) 2016-07-07 WO claimed
WO-2015077831-A1 MIKTO-ARM BRANCHED POLYMERS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2015-06-04 WO claimed
WO-2014190398-A1 INHIBITION OF AMYLOID FIBRIL FORMATION THE UNIVERSITY OF MELBOURNE (AU) 2014-12-04 WO claimed
US-20120290075-A1 MODIFICATION OF BIOABSORBABLE STENT TO REDUCE THROMBOGENECITY ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2012-11-15 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160375143-A1 MIKTO-ARM BRANCHED POLYMERS MACO1, PCNA, IPO7 CHRM5 4089/4885CHRM1 3738/4885CHRM3 3148/4885
US-20260072020-A1 PRINTABLE MOLECULE-SELECTIVE CORE-SHELL NANOPARTICLES FOR WEARABLE AND IMPLANTABLE SENSING MIF, HMOX2, HMOX1 CHRM5 2389/4885CHRM1 2135/4885CHRM3 1963/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.