SCHEMBL342534

SCHEMBL342534

CNC(=O)[C@@H](N)C(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.50
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
PTGS1 P23219 1/20 0.37
CIT O14578 1/20 0.34
MMP1 P03956 10/20 0.33
MMP3 P08254 9/20 0.33
MMP2 P08253 8/20 0.33
MMP9 P14780 7/20 0.33
MMP8 P22894 4/20 0.33
MMP13 P45452 3/20 0.33
ADAM17 P78536 3/20 0.32
MMP7 P09237 2/20 0.32
MMP14 P50281 2/20 0.32
TNF P01375 2/20 0.32
MMP20 O60882 1/20 0.32
ADAMTS4 O75173 1/20 0.32
MMP10 P09238 1/20 0.32
MMP12 P39900 1/20 0.32
MMP15 P51511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1174655 1.00 DPP4 (0.50) DPP4ALDH1A1MAPTPTGS1CIT
SCHEMBL343358 1.00 DPP4 (0.50) DPP4ALDH1A1MAPTPTGS1CIT
Hydrochloric Acid SCHEMBL2005453 0.97 DPP4 (0.48) DPP4ALDH1A1MAPTPTGS1CIT
Hydrochloric Acid SCHEMBL20721188 0.97 DPP4 (0.48) DPP4ALDH1A1MAPTPTGS1CIT
Hydrochloric Acid SCHEMBL2005458 0.97 DPP4 (0.48) DPP4ALDH1A1MAPTPTGS1CIT
Trifluoroacetic Acid SCHEMBL7399856 0.87 DPP4 (0.42) DPP4ALDH1A1MAPTPTGS1CIT
SCHEMBL3416457 0.82 SPHK1 (0.41) DPP4ALDH1A1MAPTPTGS1
SCHEMBL12867478 0.80 MAPT (0.34) DPP4ALDH1A1MAPTPTGS1FAP
SCHEMBL14261061 0.80 DPP4 (0.47) DPP4ALDH1A1MAPTPTGS1CIT
SCHEMBL8202933 0.80 MAPT (0.34) DPP4ALDH1A1MAPTPTGS1FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 282 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250214928-A1 Process for the preparation of marimastat, marimastat prepared by this process, a pharmaceutical composition comprising the same, and uses thereof PIKRALIDA SPOLKA Z OGRANICZONA ODPOWIEDZIALNOSCIA (PL) 2025-07-03 US claimed
US-20230364272-A1 THERANOSTIC COMPOUNDS UNIVERSITY OF CAPE TOWN (ZA) 2023-11-16 US claimed
US-20230033510-A1 Compounds and Methods for Treatment of Visceral Pain ARENA PHARMACEUTICALS, INC. 2023-02-02 US claimed
US-20210060040-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. 2021-03-04 US claimed
US-10632134-B2 Cannabinoid receptor modulators ARENA PHARMACEUTICALS, INC. (US) 2020-04-28 US claimed
US-20200078358-A1 Compounds and Methods for Treatment of Visceral Pain ARENA PHARMACEUTICALS, INC. 2020-03-12 US claimed
CN-110709085-A Compounds and methods for treating visceral pain 艾尼纳制药公司 2020-01-17 CN claimed
CN-109970708-A Cannibinoid receptor modulators 艾尼纳制药公司 2019-07-05 CN claimed
CN-103492369-B Cannabinoid receptor modulators 艾尼纳制药公司 2019-03-29 CN claimed
US-20180354907-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. 2018-12-13 US claimed
US-20120316147-A1 NOVEL PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2012-12-13 US claimed
WO-2012168350-A1 PYRIDIN- 2 -AMIDES USEFUL AS CB2 AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2012-12-13 WO claimed
US-20120214766-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. 2012-08-23 US claimed
US-20090220514-A1 ADAM10 and its Uses Related to Infection VANDERBILT UNIVERSITY 2009-09-03 US claimed
EP-1224211-B1 PROCESS FOR THE PREPARATION OF A DIPEPTIDE AND INTERMEDIATE PRODUCT IN SUCH A PROCESS DSM NV (NL) 2003-04-16 EP claimed
US-6486193-B2 ANTIARTHRITIC AGENTS; ANTIINFLAMMATORY AGENTS AVENTIS PHARMACEUTICALS INC. 2002-11-26 US claimed
EP-1224211-A1 PROCESS FOR THE PREPARATION OF A DIPEPTIDE AND INTERMEDIATE PRODUCT IN SUCH A PROCESS DSM N.V. (NL) 2002-07-24 EP claimed
US-20020037859-A1 3-substituted pyrrolidines useful as inhibitors of matrix metalloproteinases AVENTISUB INC. 2002-03-28 US claimed
EP-0818443-B1 Mercaptoketones and mercaptoalcohols, a process for their preparation and their use as inhibitors of matrix metalloproteinases AMERICAN CYANAMID CO (US) 2001-12-05 EP claimed
WO-2001030807-A1 PROCESS FOR THE PREPARATION OF A DIPEPTIDE AND INTERMEDIATE PRODUCT IN SUCH A PROCESS DSM N.V. (NL) 2001-05-03 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120214766-A1 CANNABINOID RECEPTOR MODULATORS CNR1, CNR2, TRPV1 DPP4 4074/4885ALDH1A1 3623/4885MAPT 627/4885
US-20200078358-A1 Compounds and Methods for Treatment of Visceral Pain VIP, FABP2, FABP6 DPP4 1022/4885ALDH1A1 603/4885MAPT 3544/4885
US-20180354907-A1 CANNABINOID RECEPTOR MODULATORS CNR1, CNR2, TRPV1 DPP4 4074/4885ALDH1A1 3623/4885MAPT 627/4885
US-10632134-B2 Cannabinoid receptor modulators CNR1, CNR2, GPR18 DPP4 4760/4885ALDH1A1 2571/4885MAPT 3883/4885
US-20230364272-A1 THERANOSTIC COMPOUNDS MMP12, TIMP3, CTSZ DPP4 344/4885ALDH1A1 1414/4885MAPT 689/4885
US-20210060040-A1 CANNABINOID RECEPTOR MODULATORS CNR1, CNR2, GPR18 DPP4 4760/4885ALDH1A1 2571/4885MAPT 3883/4885
US-20120316147-A1 NOVEL PYRIDINE DERIVATIVES NDUFS6, NDUFS4, NDUFV1 DPP4 2226/4885ALDH1A1 269/4885MAPT 1821/4885
US-20090220514-A1 ADAM10 and its Uses Related to Infection ADAM10, ADAM12, ADAM17 DPP4 232/4885ALDH1A1 4310/4885MAPT 3451/4885
US-20250214928-A1 Process for the preparation of marimastat, marimastat prepared by this process, a pharmaceutical composition comprising the same, and uses thereof MMP7, MMP9, MMP3 DPP4 463/4885ALDH1A1 1330/4885MAPT 407/4885
US-20230033510-A1 Compounds and Methods for Treatment of Visceral Pain VIP, FABP2, FABP6 DPP4 1022/4885ALDH1A1 603/4885MAPT 3544/4885
US-20020037859-A1 3-substituted pyrrolidines useful as inhibitors of matrix metalloproteinases MMP3, MMP1, MMP9 DPP4 329/4885ALDH1A1 281/4885MAPT 3351/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.