Pramoxine

Pramoxine

SCHEMBL4435138

CCCCOc1ccc(OCCCN2CCOCC2)cc1.[Cl-].[H+]

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEBDKRB2CHRM1CHRM2CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNGGUCY1A1GUCY1A2GUCY1B1GUCY1B2NAMPTPTAFRSLC10A2SLC6A2SLC6A3TACR1dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Pramoxine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 1/20 0.94
CHRM1 known ✓ P11229 1/20 0.94
ALDH1A1 P00352 6/20 0.94
HRH3 Q9Y5N1 5/20 0.94
MAPK1 P28482 2/20 0.94
CYP1A2 P05177 1/20 0.94
HTR2A P28223 1/20 0.94
SCN1A P35498 1/20 0.94
HTR2B P41595 1/20 0.94
KCNH2 Q12809 1/20 0.94
SCN2A Q99250 1/20 0.94
SIGMAR1 Q99720 1/20 0.94
SCN3A Q9NY46 1/20 0.94
LMNA P02545 3/20 0.91
USP2 O75604 2/20 0.91
THRB P10828 2/20 0.64
MAPT P10636 1/20 0.64
KMT2A Q03164 1/20 0.64
TSHR P16473 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pramoxine SCHEMBL26020 0.97 ALDH1A1 (1.00) ALDH1A1HRH3MAPK1CYP1A2CHRM2
Pramoxine SCHEMBL180542 0.95 LMNA (1.00) ALDH1A1HRH3MAPK1CYP1A2CHRM2
SCHEMBL23804878 0.92 HRH3 (0.91) ALDH1A1HRH3MAPK1CYP1A2CHRM2
SCHEMBL29508217 0.90 ALDH1A1 (0.88) ALDH1A1HRH3MAPK1CYP1A2CHRM2
Pramoxine SCHEMBL29048599 0.88 ALDH1A1 (0.83) ALDH1A1HRH3MAPK1CYP1A2CHRM2
SCHEMBL29508145 0.88 ALDH1A1 (0.82) ALDH1A1HRH3MAPK1CYP1A2CHRM2
SCHEMBL29508184 0.87 ALDH1A1 (0.81) ALDH1A1HRH3MAPK1CYP1A2CHRM2
SCHEMBL13186317 0.86 HRH3 (0.80) ALDH1A1HRH3MAPK1CYP1A2CHRM2
SCHEMBL171264 0.86 HRH3 (0.79) ALDH1A1HRH3MAPK1CYP1A2CHRM2
SCHEMBL23804879 0.86 HRH3 (0.79) ALDH1A1HRH3MAPK1CYP1A2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1366874-A Personal nursing compound JOHNSON & JOHNSON CONSUMER (US) 2002-09-04 CN claimed
US-4877781-A TIXOCORTOL PIVALATE, EPHEDRINE SULFATE, PRAMOXINE HYDROCHLORIDE; ANTIINFLAMMATORY AGENTS FOR HEMORRHOIDS LaHaye, Peter G. (US) 1989-10-31 US claimed
US-12508218-B2 Coating compositions COTY INC. (US) 2025-12-30 US disclosed
US-20250152487-A1 FRAGRANCE COMPOSITIONS AND USES THEREOF COTY INC. 2025-05-15 US disclosed
US-20250127707-A1 FRAGRANCE FORMULATION COTY INC. 2025-04-24 US disclosed
US-20250127694-A1 FRAGRANCE COMPOSITIONS AND USES THEREOF COTY INC. 2025-04-24 US disclosed
US-20250032371-A1 ETHANOL-FREE FRAGRANCE CHASSIS COTY INC. 2025-01-30 US disclosed
US-12178896-B2 Fragrance compositions and uses thereof COTY INC. (US) 2024-12-31 US disclosed
US-20230285261-A1 FRAGRANCE COMPOSITION COMPRISING A FRAGRANCE COMPONET AND A NON-ODOROUS FRAGRANCE MODULATOR JPMORGAN CHASE BANK, N.A. 2023-09-14 US disclosed
CN-116466000-A Method for rapidly determining 176 PPCPs content in source water 福建省产品质量检验研究院(福建省缺陷产品召回技术中心) 2023-07-21 CN disclosed
EP-3141239-B1 FRAGRANCE COMPOSITIONS AND USES THEREOF PROCTER & GAMBLE (US) 2023-05-10 EP disclosed
US-20160362630-A1 Fragrance Compositions and Uses Thereof THE PROCTER & GAMBLE COMPANY 2016-12-15 US disclosed
US-20160362631-A1 Fragrance Fixatives and Compositions Comprising Thereof THE PROCTER & GAMBLE COMPANY 2016-12-15 US disclosed
EP-2846788-A1 USE OF COMPOUNDS FOR THE TREATMENT OF PAIN Akron Molecules AG (AT) 2015-03-18 EP disclosed
CN-104059029-A Preparation method of pramoxine hydrochloride STONECREEK LIFE TECHNOLOGIES INC 2014-09-24 CN disclosed
WO-2013167743-A1 USE OF COMPOUNDS FOR THE TREATMENT OF PAIN AKRON MOLECULES GMBH (AT) 2013-11-14 WO disclosed
WO-2009148684-A1 BOTANICAL COMPOSITION AND ITS USES MICRO-DOSE LIFE SCIENCES, LLC (US) 2009-12-10 WO disclosed
US-20090297643-A1 BOTANICAL COMPOSITION AND ITS USES MICRO-DOSE LIFE SCIENCES, LLC (US) 2009-12-03 US disclosed
US-4877781-A TIXOCORTOL PIVALATE, EPHEDRINE SULFATE, PRAMOXINE HYDROCHLORIDE; ANTIINFLAMMATORY AGENTS FOR HEMORRHOIDS LaHaye, Peter G. (US) 1989-10-31 US disclosed
US-4877781-A TIXOCORTOL PIVALATE, EPHEDRINE SULFATE, PRAMOXINE HYDROCHLORIDE; ANTIINFLAMMATORY AGENTS FOR HEMORRHOIDS LaHaye, Peter G. (US) 1989-10-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12178896-B2 Fragrance compositions and uses thereof FHIT, ALG3, FEM1B CHRM2 3417/4885CHRM1 3097/4885ALDH1A1 275/4885
US-20250032371-A1 ETHANOL-FREE FRAGRANCE CHASSIS OR51E2, FDFT1, ELANE CHRM2 511/4885CHRM1 483/4885ALDH1A1 694/4885
US-20250127694-A1 FRAGRANCE COMPOSITIONS AND USES THEREOF TRPA1, TRPV1, NAA40 CHRM2 3657/4885CHRM1 2639/4885ALDH1A1 1624/4885
US-20250127707-A1 FRAGRANCE FORMULATION PUF60, POLM, ADH5 CHRM2 3059/4885CHRM1 1949/4885ALDH1A1 257/4885
US-20230285261-A1 FRAGRANCE COMPOSITION COMPRISING A FRAGRANCE COMPONET AND A NON-ODOROUS FRAGRANCE MODULATOR OR51E2, TRPA1, FAM120A CHRM2 1294/4885CHRM1 1014/4885ALDH1A1 1958/4885
US-20160362630-A1 Fragrance Compositions and Uses Thereof CUTA, DPM1, PLIN5 CHRM2 4240/4885CHRM1 4108/4885ALDH1A1 1263/4885
US-12508218-B2 Coating compositions TAS2R40, TAS2R20, TAS2R10 CHRM2 1456/4885CHRM1 1665/4885ALDH1A1 3806/4885
US-20250152487-A1 FRAGRANCE COMPOSITIONS AND USES THEREOF FHIT, ALG3, FEM1B CHRM2 3417/4885CHRM1 3097/4885ALDH1A1 275/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.