Predicted protein targets (top 14)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | FDPS | P14324 | 1/20 | 0.91 |
| ▸ | BLM | P54132 | 1/20 | 0.91 |
| ▸ | TDP1 | Q9NUW8 | 1/20 | 0.91 |
| ▸ | CA4 | P22748 | 1/20 | 0.37 |
| ▸ | CA2 | P00918 | 1/20 | 0.36 |
| ▸ | INPPL1 | O15357 | 2/20 | 0.35 |
| ▸ | INPP5A | Q14642 | 2/20 | 0.35 |
| ▸ | SMPD1 | P17405 | 1/20 | 0.35 |
| ▸ | INPP5B | P32019 | 1/20 | 0.35 |
| ▸ | BTN3A1 | O00481 | 2/20 | 0.35 |
| ▸ | ITPR3 | Q14573 | 3/20 | 0.33 |
| ▸ | SLC34A1 | Q06495 | 1/20 | 0.33 |
| ▸ | ITPR2 | Q14571 | 1/20 | 0.33 |
| ▸ | ITPR1 | Q14643 | 1/20 | 0.33 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| Pyrophosphoric Acid SCHEMBL27784233 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 | |
| Pyrophosphoric Acid SCHEMBL621307 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 | |
| Pyrophosphoric Acid SCHEMBL28370379 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 | |
| Pyrophosphoric Acid SCHEMBL2460231 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 | |
| Pyrophosphoric Acid SCHEMBL5550825 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 | |
| Pyrophosphoric Acid SCHEMBL18670528 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 | |
| Pyrophosphoric Acid SCHEMBL4418859 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 | |
| Pyrophosphoric Acid SCHEMBL440052 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 | |
| Pyrophosphoric Acid SCHEMBL21433694 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 | |
| Pyrophosphoric Acid SCHEMBL7650519 | 1.00 | FDPS (0.91) | FDPSBLMTDP1CA4CA2 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 246 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-20210198152-A1 | CERAMIC PARTICLE AND METHOD FOR PRODUCING THE SAME | METAL INDUSTRIES RESEARCH & DEVELOPMENT CENTRE (TW) | 2021-07-01 | — | — | US | claimed |
| EP-2684849-B1 | Method and device for treating drinking water | BWT AG (AT) | 2019-10-30 | — | — | EP | claimed |
| EP-2269663-B1 | BONE GRAFT AND BIOCOMPOSITE | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2018-03-07 | — | — | EP | claimed |
| US-20170368182-A1 | Pharmaceutical Semi-Solid Gels with Entrapped Calcium Phosphate Nanoparticles | BELMONT UNIVERSITY | 2017-12-28 | — | — | US | claimed |
| EP-3229783-A1 | PHARMACEUTICAL SEMI-SOLID GELS WITH ENTRAPPED CALCIUM PHOSPHATE NANOPARTICLES | Belmont University (US) | 2017-10-18 | — | — | EP | claimed |
| US-20170175260-A1 | CERAMIC/POLYMER COMPOSITE MATERIAL AND METHOD FOR FABRICATING THE SAME | INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (TW) | 2017-06-22 | — | — | US | claimed |
| WO-2016094571-A1 | PHARMACEUTICAL SEMI-SOLID GELS WITH ENTRAPPED CALCIUM PHOSPHATE NANOPARTICLES | BELMONT UNIVERSITY (US) | 2016-06-16 | — | — | WO | claimed |
| EP-2448609-B1 | BONE GRAFT AND BIOCOMPOSITE FOR PROSTHETIC DENTISTRY | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2014-10-08 | — | — | EP | claimed |
| US-8834935-B2 | Bone graft and biocomposite for prosthetic dentistry | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2014-09-16 | — | — | US | claimed |
| WO-2014099852-A1 | IMPROVED STRUCTURING USING AN EXTERNAL STRUCTURANT AND A COSMOTROPE | THE PROCTER & GAMBLE COMPANY (US) | 2014-06-26 | — | — | WO | claimed |
| US-20140179591-A1 | STRUCTURING USING AN EXTERNAL STRUCTURANT AND A COSMOTROPE | THE PROCTER & GAMBLE COMPANY (US) | 2014-06-26 | — | — | US | claimed |
| EP-2746377-A1 | Improved structuring using an external structurant and a cosmotrope | The Procter & Gamble Company (US) | 2014-06-25 | — | — | EP | claimed |
| EP-2448609-A2 | BONE GRAFT AND BIOCOMPOSITE FOR PROSTHETIC DENTISTRY | Armbruster Biotechnology GmbH (DE) | 2012-05-09 | — | — | EP | claimed |
| US-20120107407-A1 | BONE GRAFT AND BIOCOMPOSITE FOR PROSTHETIC DENTISTRY | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2012-05-03 | — | — | US | claimed |
| WO-2011000970-A2 | BONE GRAFT AND BIOCOMPOSITE FOR PROSTHETIC DENTISTRY | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2011-01-06 | — | — | WO | claimed |
| EP-2269663-A2 | Bone graft and biocomposite for prosthetic dentistry | Armbruster Biotechnology GmbH (DE) | 2011-01-05 | — | — | EP | claimed |
| US-6689467-B1 | Composition comprising an inorganic coating and a core comprising at least a polyhydroxyl compound | RHODIA CHIMIE (FR) | 2004-02-10 | — | — | US | claimed |
| US-5783635-A | ARTIFICIAL MARBLE, PARTICLES OF CROSSLINKED DIVINYLBENZENE-STYRENE RESIN, GLASS OR ALUMINUM HYDROXIDE POWDER FILLER, BATHROOM AND KITCHEN FIXTURES AND COUNTERS | TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) | 1998-07-21 | — | — | US | claimed |
| EP-0806454-A2 | An unsaturated polyester resin composition | Takeda Chemical Industries, Ltd. (JP) | 1997-11-12 | — | — | EP | claimed |
| JP-63238022-A | — | — | None | — | — | JP | disclosed |
| JP-1101976-A | — | — | None | — | — | JP | disclosed |
| JP-1101977-A | — | — | None | — | — | JP | disclosed |
| JP-61247610-A | — | — | None | — | — | JP | disclosed |
| US-12636299-B2 | Terpenoid derivatives, pharmaceutical preparations containing these derivatives and their use in neuroprotection | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2026-05-26 | — | — | US | disclosed |
| US-12376612-B2 | Edible concentrate comprising microfibrillated cellulose | CONOPCO INC. (US) | 2025-08-05 | — | — | US | disclosed |
| US-12319694-B2 | Heterocyclic nitrogen-containing purine derivatives, pharmaceutical preparations containing these derivatives and their use in neuroprotection | UNIVERZITA PALACKEHO (CZ) | 2025-06-03 | — | — | US | disclosed |
| EP-3946271-B1 | METHOD OF PRODUCTION OF A COMPOSITE OF YEAST-DERIVED BETA GLUCAN PARTICLE WITH INCORPORATED POORLY-WATER-SOLUBLE LOW-MOLECULAR-WEIGHT COMPOUND, PHARMACEUTICAL PREPARATION AND USE THEREOF | VS CHEMICKO TECHNOLOGICKA V PRAZE (CZ) | 2024-12-25 | — | — | EP | disclosed |
| EP-3924353-B1 | HETEROCYCLIC NITROGEN-CONTAINING PURINE DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN NEUROPROTECTION | UNIV PALACKEHO (CZ) | 2024-04-24 | — | — | EP | disclosed |
| WO-2024080123-A1 | COMPOSITION | 住友化学株式会社 | 2024-04-18 | — | — | WO | disclosed |
| WO-2024063737-A1 | PRODUCTION AND USE OF BACTERIAL CELLULOSE IN PURE FORM OR BY IMPREGNATION OF VARIOUS AGENTS AND PRODUCED IN SPHERICAL FORM FOR BONE REGENERATION, ALONE AND IN COMBINATION WITH VARIOUS GRAFT MATERIALS | ATATÜRK ÜNİVERSİTESİ REKTÖRLÜĞÜ BİLİMSEL ARAŞTIRMA PROJELERİ ( BAP ) KOORDİNASYON BİRİMİ (TR) | 2024-03-28 | — | — | WO | disclosed |
| US-20230414645-A1 | TERPENOID DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN NEUROPROTECTION | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2023-12-28 | — | — | US | disclosed |
| US-20230365616-A1 | CHOLESTANE DERIVATIVES, PREPARATIONS CONTAINING THESE DERIVATIVES AND USE THEREOF | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2023-11-16 | — | — | US | disclosed |
| CN-116891957-A | Covering agent for smelting carbonless heating copper-iron alloy and preparation method thereof | 江西省科学院应用物理研究所 | 2023-10-17 | — | — | CN | disclosed |
| EP-4255916-A2 | TERPENOID DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN NEUROPROTECTION | Univerzita Palackého v Olomouci (CZ) | 2023-10-11 | — | — | EP | disclosed |
| EP-4232457-A1 | CHOLESTANE DERIVATIVES, PREPARATIONS CONTAINING THESE DERIVATIVES AND USE THEREOF | Univerzita Palackého v Olomouci (CZ) | 2023-08-30 | — | — | EP | disclosed |
| EP-4107145-B1 | PYRAZOLE-INDOLE CONJUGATES FOR PHOTODYNAMIC TREATMENT OF CANCER AND BACTERIAL INFECTIONS | UNIV PALACKEHO (CZ) | 2023-08-02 | — | — | EP | disclosed |
| WO-2023131362-A1 | PHENYLPROPANOID DERIVATIVES | USTAV EXPERIMENTALNI BOTANIKY AV ČR, V. V. I. (CZ) | 2023-07-13 | — | — | WO | disclosed |
| US-11643413-B2 | 9-(2-oxacycloalkyl)-9H-purine-2,6-diamine derivatives and their use for the treatment of skin disorders | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2023-05-09 | — | — | US | disclosed |
| EP-4107145-A1 | PYRAZOLE-INDOLE CONJUGATES FOR PHOTODYNAMIC TREATMENT OF CANCER AND BACTERIAL INFECTIONS | Univerzita Palackého v Olomouci (CZ) | 2022-12-28 | — | — | EP | disclosed |
| CN-110234237-B | Edible concentrate comprising microfibrillated cellulose | 联合利华知识产权控股有限公司 | 2022-11-08 | — | — | CN | disclosed |
| EP-4069370-A1 | PHENOLIC DIHYDROBENZOFURANE DERIVATIVES, MEDICAL AND COSMETIC PREPARATIONS CONTAINING THESE DERIVATIVES, AND USE THEREOF | Univerzita Palackého v Olomouci (CZ) | 2022-10-12 | — | — | EP | disclosed |
| US-20220192985-A1 | METHOD OF PRODUCTION OF A COMPOSITE OF YEAST-DERIVED BETA GLUCAN PARTICLE WITH INCORPORATED POORLY-WATER-SOLUBLE LOW-MOLECULAR-WEIGHT COMPOUND, PHARMACEUTICAL PREPARATION AND USE THEREOF | VYSOKA SKOLA CHEMICKO-TECHNOLOGICKA V PRAZE (CZ) | 2022-06-23 | — | — | US | disclosed |
| EP-3615535-B1 | 9-(2-OXACYCLOALKYL)-9H-PURINE-2,6-DIAMINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF SKIN DISORDERS | UNIV PALACKEHO (CZ) | 2022-06-15 | — | — | EP | disclosed |
| WO-2022117133-A2 | TERPENOID DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN NEUROPROTECTION | Univerzita Palackého v Olomouci (CZ) | 2022-06-09 | — | — | WO | disclosed |
| WO-2022083809-A1 | CHOLESTANE DERIVATIVES, PREPARATIONS CONTAINING THESE DERIVATIVES AND USE THEREOF | Univerzita Palackého v Olomouci (CZ) | 2022-04-28 | — | — | WO | disclosed |
| US-20220127269-A1 | HETEROCYCLIC NITROGEN-CONTAINING PURINE DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN NEUROPROTECTION | UNIVERZITA PALACKEHO (CZ) | 2022-04-28 | — | — | US | disclosed |
| US-11253556-B2 | Lactobacillus fermentum GKF3, composition comprising the strain and method for improving psychataxia using the same | GRAPE KING BIO LTD (TW) | 2022-02-22 | — | — | US | disclosed |
| EP-3946271-A1 | METHOD OF PRODUCTION OF A COMPOSITE OF YEAST-DERIVED BETA GLUCAN PARTICLE WITH INCORPORATED POORLY-WATER-SOLUBLE LOW-MOLECULAR-WEIGHT COMPOUND, PHARMACEUTICAL PREPARATION AND USE THEREOF | Vysoká skola chemicko-technologická v Praze (CZ) | 2022-02-09 | — | — | EP | disclosed |
| EP-3924353-A1 | HETEROCYCLIC NITROGEN-CONTAINING PURINE DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN NEUROPROTECTION | Univerzita Palackého (CZ) | 2021-12-22 | — | — | EP | disclosed |
| EP-3601287-B1 | 2,6-DISUBSTITUTED-9-CYCLOPENTYL-9H-PURINES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | UNIV PALACKEHO (CZ) | 2021-12-15 | — | — | EP | disclosed |
| US-11186583-B2 | 5-alkylthio-7-[(4-arylbenzyl)amino]-1(2)H-pyrazolo[4,3-d]pyrimidines for treatment of lymphoma | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2021-11-30 | — | — | US | disclosed |
| EP-3749670-B1 | 5-ALKYLTHIO-7-[(4-ARYLBENZYL)AMINO]-1(2)H-PYRAZOLO[4,3-D]PYRIMIDINES FOR TREATMENT OF LYMPHOMA | UNIV PALACKEHO (CZ) | 2021-10-06 | — | — | EP | disclosed |
| US-11058733-B2 | Active substances of Bifidobacterium lactis GKK2, composition comprising the same and method of promoting longevity using the same | GRAPE KING BIO LTD (TW) | 2021-07-13 | — | — | US | disclosed |
| US-20210198152-A1 | CERAMIC PARTICLE AND METHOD FOR PRODUCING THE SAME | METAL INDUSTRIES RESEARCH & DEVELOPMENT CENTRE (TW) | 2021-07-01 | — | — | US | disclosed |
| WO-2021110185-A1 | PHENOLIC DIHYDROBENZOFURANE DERIVATIVES, MEDICAL AND COSMETIC PREPARATIONS CONTAINING THESE DERIVATIVES, AND USE THEREOF | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2021-06-10 | — | — | WO | disclosed |
| US-11028087-B2 | 2,6-disubstituted-9-cyclopentyl-9H-purines, use thereof as medicaments, and pharmaceutical compositions | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2021-06-08 | — | — | US | disclosed |
| EP-3749670-A1 | 5-ALKYLTHIO-7-[(4-ARYLBENZYL)AMINO]-1(2)H-PYRAZOLO[4,3-D]PYRIMIDINES FOR TREATMENT OF LYMPHOMA | Univerzita Palackeho v Olomouci (CZ) | 2020-12-16 | — | — | EP | disclosed |
| US-20200361943-A1 | 5-ALKYLTHIO-7-[(4-ARYLBENZYL)AMINO]-1(2)H-PYRAZOLO[4,3-D]PYRIMIDINES FOR TREATMENT OF LYMPHOMA | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2020-11-19 | — | — | US | disclosed |
| WO-2020200337-A1 | METHOD OF PRODUCTION OF A COMPOSITE OF YEAST-DERIVED BETA GLUCAN PARTICLE WITH INCORPORATED POORLY-WATER-SOLUBLE LOW-MOLECULAR-WEIGHT COMPOUND, PHARMACEUTICAL PREPARATION AND USE THEREOF | VYSOKA SKOLA CHEMICKO-TECHNOLOGICKA V PRAZE (CZ) | 2020-10-08 | — | — | WO | disclosed |
| WO-2020164648-A1 | HETEROCYCLIC NITROGEN-CONTAINING PURINE DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN NEUROPROTECTION | UNIVERZITA PALACKEHO (CZ) | 2020-08-20 | — | — | WO | disclosed |
| US-20200155623-A1 | Lactobacillus Fermentum GKF3, Composition Comprising the Strain and Method for Improving Psychataxia Using the Same | GRAPE KING BIO LTD (TW) | 2020-05-21 | — | — | US | disclosed |
| US-20200157105-A1 | 9-(2-OXACYCLOALKYL)-9H-PURINE-2,6-DIAMINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF SKIN DISORDERS | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2020-05-21 | — | — | US | disclosed |
| EP-3579706-B1 | EDIBLE CONCENTRATE COMPRISING MICROFIBRILLATED CELLULOSE | UNILEVER NV (NL) | 2020-05-13 | — | — | EP | disclosed |
| EP-3325480-B1 | 5-SUBSTITUTED-7-[4-(SUBSTITUTED) BENZYL]AMINO-3-ISOPROPYLPYRAZOLO (4,3-D) PYRIMIDINES AS MEDICAMENTS | USTAV EXPERIMENTALNI BOTANIKY AV CR V V I (CZ) | 2020-04-22 | — | — | EP | disclosed |
| US-20200087306-A1 | 2,6-DISUBSTITUTED-9-CYCLOPENTYL-9H-PURINES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2020-03-19 | — | — | US | disclosed |
| EP-3615535-A1 | 9-(2-OXACYCLOALKYL)-9H-PURINE-2,6-DIAMINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF SKIN DISORDERS | Univerzita Palackého v Olomouci (CZ) | 2020-03-04 | — | — | EP | disclosed |
| US-20200054692-A1 | ACTIVE SUBSTANCES OF BIFIDOBACTERIUM LACTIS GKK2, COMPOSITION COMPRISING THE SAME AND METHOD OF PROMOTING LONGEVITY USING THE SAME | GRAPE KING BIO LTD (TW) | 2020-02-20 | — | — | US | disclosed |
| EP-3601287-A1 | 2,6-DISUBSTITUTED-9-CYCLOPENTYL-9H-PURINES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | Univerzita Palackého v Olomouci (CZ) | 2020-02-05 | — | — | EP | disclosed |
| WO-2019149295-A1 | 5-ALKYLTHIO-7-[(4-ARYLBENZYL)AMINO]-1(2)H-PYRAZOLO[4,3-D]PYRIMIDINES FOR TREATMENT OF LYMPHOMA | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2019-08-08 | — | — | WO | disclosed |
| EP-3294741-B1 | 5-SUBSTITUTED 7-[4-(2-PYRIDYL)PHENYLMETHYLAMINO]-3-ISO PROPYLPYRAZOLO[4,3-D]PYRIMIDINE DERIVATIVES, USE THEREOF AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS | USTAV EXPERIMENTALNI BOTANIKY AV CR V V I (CZ) | 2019-05-01 | — | — | EP | disclosed |
| EP-3233861-B1 | 6,8-DISUBSTITUTED-9-(HETEROCYCLYL) PURINES, COMPOSITIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN COSMETIC AND MEDICINAL APPLICATIONS | USTAV EXPERIMENTALNI BOTANIKY AV CR V V I (CZ) | 2019-04-10 | — | — | EP | disclosed |
| WO-2018196893-A1 | 9-(2-OXACYCLOALKYL)-9H-PURINE-2,6-DIAMINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF SKIN DISORDERS | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2018-11-01 | — | — | WO | disclosed |
| US-10093675-B2 | 6,8-disubstituted-9-(heterocyclyl)purines, compositions containing these derivatives and their use in cosmetic and medicinal applications | USTAV EXPERIMENTALNI BOTANIKY AV CR, V.V.I. (CZ) | 2018-10-09 | — | — | US | disclosed |
| WO-2018171819-A1 | 2,6-DISUBSTITUTED-9-CYCLOPENTYL-9H-PURINES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2018-09-27 | — | — | WO | disclosed |
| WO-2018145886-A1 | EDIBLE CONCENTRATE COMPRISING MICROFIBRILLATED CELLULOSE | UNILEVER N.V. (NL) | 2018-08-16 | — | — | WO | disclosed |
| EP-3031854-B1 | SOFT THERMOPLASTIC RESIN COMPOSITION | KANEKA CORP (JP) | 2018-06-06 | — | — | EP | disclosed |
| EP-3325480-A1 | 5-SUBSTITUTED-7-[4-(SUBSTITUTED)BENZYL]AMINO-3-ISOPROPYLPYRAZOLO(4,3-D)PYRIMIDINES AS MEDICAMENTS | Ustav Experimentalni Botaniky Av CR, V.V.I. (CZ) | 2018-05-30 | — | — | EP | disclosed |
| EP-3031855-B1 | SOFT THERMOPLASTIC RESIN COMPOSITION | KANEKA CORP (JP) | 2018-05-23 | — | — | EP | disclosed |
| US-9957273-B2 | 5-substituted 7- [4-(2-pyridyl)phenylmethylamino] -3-isopropylpyrazolo4,3-D]pyrimidine derivatives, use thereof as medicaments, and pharmaceutical compositions | USTAV EXPERIMENTALNI BOTANIKY AV CR, V.V.I. (CZ) | 2018-05-01 | — | — | US | disclosed |
| EP-3294741-A1 | 5-SUBSTITUTED 7-[4-(2-PYRIDYL)PHENYLMETHYLAMINO]-3-ISOPROPYLPYRAZOLO4,3-D]PYRIMIDINE DERIVATIVES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | Ustav Experimentalni Botaniky Av CR, V.V.I. (CZ) | 2018-03-21 | — | — | EP | disclosed |
| US-20180072736-A1 | 5-SUBSTITUTED 7-[4-(2-PYRIDYL)PHENYLMETHYLAMINO]-3-ISOPROPYLPYRAZOLO4,3-D]PYRIMIDINE DERIVATIVES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | USTAV EXPERIMENTALNI BOTANIKY AV CR, V.V.I. (CZ) | 2018-03-15 | — | — | US | disclosed |
| EP-2269663-B1 | BONE GRAFT AND BIOCOMPOSITE | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2018-03-07 | — | — | EP | disclosed |
| US-20170368182-A1 | Pharmaceutical Semi-Solid Gels with Entrapped Calcium Phosphate Nanoparticles | BELMONT UNIVERSITY | 2017-12-28 | — | — | US | disclosed |
| US-20170362236-A1 | 6,8-DISUBSTITUTED-9-(HETEROCYCLYL)PURINES, COMPOSITIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN COSMETIC AND MEDICINAL APPLICATIONS | USTAV EXPERIMENTALNI BOTANIKY AV CR, V.V.I. (CZ) | 2017-12-21 | — | — | US | disclosed |
| EP-3233861-A1 | 6,8-DISUBSTITUTED-9-(HETEROCYCLYL)PURINES, COMPOSITIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN COSMETIC AND MEDICINAL APPLICATIONS | Ustav Experimentalni Botaniky Av CR, V.V.I. (CZ) | 2017-10-25 | — | — | EP | disclosed |
| EP-1575973-B1 | SUBSTITUTION DERIVATIVES OF N SP 6 SP -BENZYLADENOSINE, METHODS OF THEIR PREPARATION, THEIR USE FOR PREPARATION OF DRUGS, COSMETIC PREPARATIONS AND GROWTH REGULATORS, PHARMACEUTICAL PREPARATIONS, COSMETIC PREPARATIONS AND GROWTH REGULATORS CONTAINING THESE COMPOUNDS | USTAV EXPERIMENTALNI BOTANIKY AV CR V V I (CZ) | 2017-08-23 | — | — | EP | disclosed |
| US-20170175260-A1 | CERAMIC/POLYMER COMPOSITE MATERIAL AND METHOD FOR FABRICATING THE SAME | INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (TW) | 2017-06-22 | — | — | US | disclosed |
| EP-2953951-B1 | N2-SUBSTITUTED-N6-(6-ARYL-PYRIDINE-3-YLMETHYL)-9-CYCLOPENTYL-9H-PURINE-2,6-DIAMINE DERIVATIVES AS TUMOR SUPPRESSOR P53 ACTIVATORS FOR INHIBITING ANGIOGENESIS AND FOR TREATING CANCER | UNIV PALACKEHO (CZ) | 2017-05-03 | — | — | EP | disclosed |
| EP-2438068-B1 | SUBSTITUTED 6-(2-HYDROXYBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THESE DERIVATIVES | Univerzita Palackého v Olomouci (CZ) | 2017-03-01 | — | — | EP | disclosed |
| US-9574082-B2 | Soft thermoplastic resin composition | KANEKA CORPORATION (JP) | 2017-02-21 | — | — | US | disclosed |
| US-9562155-B2 | Soft thermoplastic resin composition | KANEKA CORPORATION (JP) | 2017-02-07 | — | — | US | disclosed |
| WO-2017012599-A1 | 5-SUBSTITUTED-7-[4-(SUBSTITUTED)BENZYL]AMINO-3-ISOPROPYLPYRAZOLO(4,3-D)PYRIMIDINES AS MEDICAMENTS | USTAV EXPERIMENTALNI BOTANIKY AV CR, V.V.I. (CZ) | 2017-01-26 | — | — | WO | disclosed |
| WO-2016180380-A1 | 5-SUBSTITUTED 7-[4-(2-PYRIDYL)PHENYLMETHYLAMINO]-3-ISOPROPYLPYRAZOLO4,3-D]PYRIMIDINE DERIVATIVES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | USTAV EXPERIMENTALNI BOTANIKY AV CR, V.V.I. (CZ) | 2016-11-17 | — | — | WO | disclosed |
| EP-2755977-B1 | 6,8-DISUBSTITUTED PURINE COMPOSITIONS AND THEIR PHARMACEUTICAL AND COSMETIC USE | Univerzita Palackého v Olomouci (CZ) | 2016-11-02 | — | — | EP | disclosed |
| US-20160177087-A1 | SOFT THERMOPLASTIC RESIN COMPOSITION | KANEKA CORPORATION (JP) | 2016-06-23 | — | — | US | disclosed |
| WO-2016095880-A1 | 6,8-DISUBSTITUTED-9-(HETEROCYCLYL)PURINES, COMPOSITIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN COSMETIC AND MEDICINAL APPLICATIONS | USTAV EXPERIMENTALNI BOTANIKY AV CR, V.V.I. (CZ) | 2016-06-23 | — | — | WO | disclosed |
| EP-3031854-A1 | SOFT THERMOPLASTIC RESIN COMPOSITION | Kaneka Corporation (JP) | 2016-06-15 | — | — | EP | disclosed |
| EP-3031855-A1 | SOFT THERMOPLASTIC RESIN COMPOSITION | Kaneka Corporation (JP) | 2016-06-15 | — | — | EP | disclosed |
| US-20160160020-A1 | SOFT THERMOPLASTIC RESIN COMPOSITION | KANEKA CORPORATION (JP) | 2016-06-09 | — | — | US | disclosed |
| US-9334465-B2 | Structuring using an external structurant and a cosmotrope | THE PROCTER & GAMBLE COMPANY (US) | 2016-05-10 | — | — | US | disclosed |
| US-20150368248-A1 | 2-SUBSTITUTED-6-BIARYLMETHYLAMINO-9-CYCLOPENTYL-9H-PURINE DERIVATIVES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | BIOPATTERNS S.R.O. (CZ) | 2015-12-24 | — | — | US | disclosed |
| EP-2953951-A2 | 2-SUBSTITUTED-6-BIARYLMETHYLAMINO-9-CYCLOPENTYL-9H-PURINE DERIVATIVES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | Univerzita palackeho V Olomouci (CZ) | 2015-12-16 | — | — | EP | disclosed |
| US-9174990-B2 | 2-amino-9-[(2-hydroxymethyl) cyclopropylidenemethyl] purines as antiviral agents | WAYNE STATE UNIVERSITY (US) | 2015-11-03 | — | — | US | disclosed |
| US-9073961-B2 | Substitution derivatives of N6 -benzyladenosine-5′-monophosphate, methods of preparation thereof, use thereof as medicaments, and therapeutic preparations containing these compounds | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2015-07-07 | — | — | US | disclosed |
| US-9023857-B2 | Substituted 6-(2-aminobenzylamino)purine derivatives, their use as medicaments and preparations containing these compounds | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2015-05-05 | — | — | US | disclosed |
| EP-2448609-B1 | BONE GRAFT AND BIOCOMPOSITE FOR PROSTHETIC DENTISTRY | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2014-10-08 | — | — | EP | disclosed |
| EP-2391626-B1 | SUBSTITUTED 6-(2-AMINOBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND PREPARATIONS CONTAINING THESE COMPOUNDS | Univerzita Palackého v Olomouci (CZ) | 2014-10-01 | — | — | EP | disclosed |
| EP-2563801-B1 | SUBSTITUTION DERIVATIVES OF N6-BENZYLADENOSINE-5´-MONOPHOSPHATE, METHODS OF PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, AND THERAPEUTIC PREPARATION CONTAINING THESE COMPOUNDS | Univerzita Palackého v Olomouci (CZ) | 2014-09-24 | — | — | EP | disclosed |
| US-8834935-B2 | Bone graft and biocomposite for prosthetic dentistry | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2014-09-16 | — | — | US | disclosed |
| EP-2393826-B1 | NOVEL SAPONIN COMPOUNDS, METHODS OF PREPARATION THEREOF, USE THEREOF AND PHARMACEUTICAL COMPOSITIONS | UNIV W BIALYMSTOKU (PL) | 2014-08-27 | — | — | EP | disclosed |
| WO-2014121764-A2 | 2-SUBSTITUTED-6-BIARYLMETHYLAMINO-9-CYCLOPENTYL-9H-PURINE DERIVATIVES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2014-08-14 | — | — | WO | disclosed |
| EP-2430036-B1 | SUBSTITUTED 6-(BENZYLAMINO) PURINE RIBOSIDE DERIVATIVES, USE THEREOF AND COMPOSITIONS CONTAINING THESE DERIVATIVES | Univerzita Palackého v Olomouci (CZ) | 2014-07-30 | — | — | EP | disclosed |
| EP-2755977-A1 | 6, 8- DISUBSTITUTED PURINE COMPOSITIONS AND THEIR PHARMACEUTICAL AND COSMETIC USE | Univerzita Palackého v Olomouci (CZ) | 2014-07-23 | — | — | EP | disclosed |
| WO-2014099852-A1 | IMPROVED STRUCTURING USING AN EXTERNAL STRUCTURANT AND A COSMOTROPE | THE PROCTER & GAMBLE COMPANY (US) | 2014-06-26 | — | — | WO | disclosed |
| US-20140179591-A1 | STRUCTURING USING AN EXTERNAL STRUCTURANT AND A COSMOTROPE | THE PROCTER & GAMBLE COMPANY (US) | 2014-06-26 | — | — | US | disclosed |
| EP-2746377-A1 | Improved structuring using an external structurant and a cosmotrope | The Procter & Gamble Company (US) | 2014-06-25 | — | — | EP | disclosed |
| US-20140066394-A1 | Substituted 6-(Benzylamino) Purine Riboside Derivatives, Use Thereof and Compositions Containing These Derivatives | BIOPATTERNS, S.R.O (CZ) | 2014-03-06 | — | — | US | disclosed |
| EP-1419157-B1 | 6-(4-hydroxybenzylamino)purine and its use in cosmetics | USTAV EX BOTAN AKADEMIE VED CESKE REPUBLIKY (CZ) | 2013-11-27 | — | — | EP | disclosed |
| US-8552161-B2 | Saponin compounds, methods of preparation thereof, use thereof and pharmaceutical compositions | UNIWERSYTET W BIALYMSTOKU (PL) | 2013-10-08 | — | — | US | disclosed |
| US-8552013-B2 | Heterocyclic compounds based on N6-substituted adenine, methods of their preparation, their use for preparation of drugs, cosmetic preparations and growth regulators, pharmaceutical preparations, cosmetic preparations and growth regulators containing these compounds | USTAV EXPERIMENTALNI BOTANIKY AKADEMIE VED CESKE REPUBLIKY (CZ) | 2013-10-08 | — | — | US | disclosed |
| US-8492391-B2 | Substituted 6-(2-hydroxybenzylamino)purine derivatives, their use as medicaments and compositions containing these derivatives | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2013-07-23 | — | — | US | disclosed |
| US-20130072506-A1 | 6,8-DISUBSTITUTED PURINE COMPOSITIONS | ZAHAJSKA LENKA (CZ) | 2013-03-21 | — | — | US | disclosed |
| WO-2013037333-A1 | 6, 8- DISUBSTITUTED PURINE COMPOSITIONS AND THEIR PHARMACEUTICAL AND COSMETIC USE | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2013-03-21 | — | — | WO | disclosed |
| EP-2563801-A2 | SUBSTITUTION DERIVATIVES OF N6-BENZYLADENOSINE-5´-MONOPHOSPHATE, METHODS OF PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, AND THERAPEUTIC PREPARATION CONTAINING THESE COMPOUNDS | Univerzita Palackého v Olomouci (CZ) | 2013-03-06 | — | — | EP | disclosed |
| US-20130040908-A1 | SUBSTITUTION DERIVATIVES OF N6-BENZYLADENOSINE-5' -MONOPHOSPHATE, METHODS OF PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, AND THERAPEUTIC PREPARATIONS CONTAINING THESE COMPOUNDS | BIOAPEX, S.R.O. (CZ) | 2013-02-14 | — | — | US | disclosed |
| US-8232275-B2 | 2,2-bis-(hydroxymethyl)cyclopropylidenemethyl-purines and -pyrimidines as antiviral agents | WAYNE STATE UNIVERSITY (US) | 2012-07-31 | — | — | US | disclosed |
| EP-2448609-A2 | BONE GRAFT AND BIOCOMPOSITE FOR PROSTHETIC DENTISTRY | Armbruster Biotechnology GmbH (DE) | 2012-05-09 | — | — | EP | disclosed |
| US-20120107407-A1 | BONE GRAFT AND BIOCOMPOSITE FOR PROSTHETIC DENTISTRY | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2012-05-03 | — | — | US | disclosed |
| EP-2438068-A1 | SUBSTITUTED 6-(2-HYDROXYBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THESE DERIVATIVES | Univerzita Palackého v Olomouci (CZ) | 2012-04-11 | — | — | EP | disclosed |
| US-20120071433-A1 | Substituted 6-(Benzylamino) Purine Riboside Derivatives, Use Thereof and Compositions Containing These Derivatives | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2012-03-22 | — | — | US | disclosed |
| US-20120070512-A1 | Substituted 6-(2-hydroxybenzylamino)purine Derivatives, Their Use as Medicaments and Compositions Containing These Derivatives | BIOPATTERNS, S.R.O (CZ) | 2012-03-22 | — | — | US | disclosed |
| EP-2430036-A1 | SUBSTITUTED 6-(BENZYLAMINO) PURINE RIBOSIDE DERIVATIVES, USE THEREOF AND COMPOSITIONS CONTAINING THESE DERIVATIVES | Univerzita Palackého v Olomouci (CZ) | 2012-03-21 | — | — | EP | disclosed |
| US-8119614-B2 | Substitution derivatives of N6-benzyladenosine, methods of their preparation, their use for preparation of drugs, cosmetic preparations and growth regulators, pharmaceutical preparations, cosmetic preparations and growth regulators containing these compounds | USTAV EXPERIMENTALNI BOTANIKY AKADEMIE VED CESKE REPUBLIKY (CZ) | 2012-02-21 | — | — | US | disclosed |
| WO-2011134444-A9 | SUBSTITUTION DERIVATIVES OF N6-BENZYLADENOSINE-5´-MONOPHOSPHATE, METHODS OF PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, AND THERAPEUTIC PREPARATION CONTAINING THESE COMPOUNDS | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2012-02-16 | — | — | WO | disclosed |
| US-20110311652-A1 | Novel Saponin Compounds, Methods of Preparation Thereof, Use Thereof and Pharmaceutical Compositions | UNIWERSYTET W BIALYMSTOKU (PL) | 2011-12-22 | — | — | US | disclosed |
| EP-2393826-A2 | NOVEL SAPONIN COMPOUNDS, METHODS OF PREPARATION THEREOF, USE THEREOF AND PHARMACEUTICAL COMPOSITIONS | Uniwersytet w Bialymstoku (PL) | 2011-12-14 | — | — | EP | disclosed |
| EP-2391626-A2 | SUBSTITUTED 6-(2-AMINOBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND PREPARATIONS CONTAINING THESE COMPOUNDS | Univerzita Palackého v Olomouci (CZ) | 2011-12-07 | — | — | EP | disclosed |
| US-20110287111-A1 | SUBSTITUTED 6-(2-AMINOBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND PREPARATIONS CONTAINING THESE COMPOUNDS | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2011-11-24 | — | — | US | disclosed |
| US-20110275652-A1 | 2,2-BIS-(HYDROXYMETHYL)CYCLOPROPYLIDENEMETHYL-PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | WAYNE STATE UNIVERSITY | 2011-11-10 | — | — | US | disclosed |
| WO-2011134444-A2 | SUBSTITUTION DERIVATIVES OF N6-BENZYLADENOSINE-5´-MONOPHOSPHATE, METHODS OF PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, AND THERAPEUTIC PREPARATION CONTAINING THESE COMPOUNDS | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2011-11-03 | — | — | WO | disclosed |
| EP-1490368-B1 | 2,2-BIS(HYDROXYMETHYL)CYCLOPROPYLIDENEMETHYL - PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | UNIV WAYNE STATE (US) | 2011-08-03 | — | — | EP | disclosed |
| WO-2011000970-A2 | BONE GRAFT AND BIOCOMPOSITE FOR PROSTHETIC DENTISTRY | ARMBRUSTER BIOTECHNOLOGY GMBH (DE) | 2011-01-06 | — | — | WO | disclosed |
| EP-2269663-A2 | Bone graft and biocomposite for prosthetic dentistry | Armbruster Biotechnology GmbH (DE) | 2011-01-05 | — | — | EP | disclosed |
| WO-2010139288-A1 | 5,7-DISUBSTITUTED 3-ISOPROPYLPYRAZOLO[4,3-D]PYRIMIDINES FOR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS | C3 BIO GMBH (DE) | 2010-12-09 | — | — | WO | disclosed |
| WO-2010139289-A1 | SUBSTITUTED 6-(2-HYDROXYBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THESE DERIVATIVES | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2010-12-09 | — | — | WO | disclosed |
| WO-2010130233-A1 | SUBSTITUTED 6-(BENZYLAMINO) PURINE RIBOSIDE DERIVATIVES, USE THEREOF AND COMPOSITIONS CONTAINING THESE DERIVATIVES | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2010-11-18 | — | — | WO | disclosed |
| US-7816350-B2 | Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors | INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) | 2010-10-19 | — | — | US | disclosed |
| EP-2235036-A1 | SACCHARIDE LUPANE DERIVATIVES, THEIR USE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE DERIVATIVES | Universita Palackeho v Olomouci (CZ) | 2010-10-06 | — | — | EP | disclosed |
| US-20100249259-A1 | HARD FOAM | JAPAN ADVANCED INSTITUTE OF SCIENCE AND TECHNOLOGY (JP) | 2010-09-30 | — | — | US | disclosed |
| EP-2222690-A2 | NATURAL BRASSINOSTEROIDS FOR USE FOR TREATING HYPERPROLIFERATION, TREATING PROLIFERATIVE DISEASES AND REDUCING ADVERSE EFFECTS OF STEROID DYSFUNCTION IN MAMMALS, PHARMACEUTICAL COMPOSITION AND ITS USE | Ustav Organicke Chemie A Biochemie Akademie Ved Ceske Republiky (CZ) | 2010-09-01 | — | — | EP | disclosed |
| EP-1348707-B1 | Pyrazolo[4,3-d]pyrimidines, processes for their preparation and methods for therapy | USTAV EX BOTAN AV CR V V I I O (CZ) | 2010-08-25 | — | — | EP | disclosed |
| US-20100204460-A1 | NATURAL BRASSINOSTEROIDS FOR USE FOR TREATING HYPERPROLIFERATION, TREATING PROLIFERATIVE DISEASES AND REDUCING ADVERSE EFFECTS OF STEROID DYSFUNCTION IN MAMMALS, PHARMACEUTICAL COMPOSITION AND ITS USE | USTAV ORGANICKE CHEMIE A BIOCHEMIE AKADEMIE VED EESKE REPUBLIKY, V.V.I. (CZ) | 2010-08-12 | — | — | US | disclosed |
| WO-2010088866-A2 | NOVEL SAPONIN COMPOUNDS, METHODS OF PREPARATION THEREOF, USE THEREOF AND PHARMACEUTICAL COMPOSITIONS | UNIWERSYTET W BIALYMSTOKU (PL) | 2010-08-12 | — | — | WO | disclosed |
| WO-2010085924-A2 | SUBSTITUTED 6-(2-AMINOBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND PREPARATIONS CONTAINING THESE COMPOUNDS | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2010-08-05 | — | — | WO | disclosed |
| US-7745450-B2 | Pyrazolo[4,3-d]pyrimidines, processes for their preparation and methods for therapy | INSTITUTE OF EXPERIMENTAL BOTANY (CZ) | 2010-06-29 | — | — | US | disclosed |
| US-20090312392-A1 | Amino ceramide-like compounds and therapeutic methods of use | NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR | 2009-12-17 | — | — | US | disclosed |
| EP-1358172-B1 | AMINO CERAMIDE-LIKE COMPOUNDS AND THERAPEUTIC METHODS OF USE | UNIV MICHIGAN (US) | 2009-11-18 | — | — | EP | disclosed |
| EP-1490015-B1 | NOVEL 2-AMINO-9-((2-HYDROXYMETHYL) CYCLOPROPYLIDENEMETHYL) PURINES AS ANTIVIRAL AGENTS | UNIV WAYNE STATE (US) | 2009-09-23 | — | — | EP | disclosed |
| WO-2009094958-A1 | SACCHARIDE LUPANE DERIVATIVES, THEIR USE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE DERIVATIVES | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2009-08-06 | — | — | WO | disclosed |
| US-20090118308-A1 | 2,2-Bis-(hydroxymethyl)cyclopropylidenemethyl-Purines and -Pyrimidines As Antiviral Agents | WAYNE STATE UNIVERSITY (US) | 2009-05-07 | — | — | US | disclosed |
| WO-2009024103-A2 | NATURAL BRASSINOSTEROIDS FOR USE FOR TREATING HYPERPROLIFERATION, TREATING PROLIFERATIVE DISEASES AND REDUCING ADVERSE EFFECTS OF STEROID DYSFUNCTION IN MAMMALS, PHARMACEUTICAL COMPOSITION AND ITS USE | USTAV ORGANICKE CHEMIE A BIOCHEMIE AKADEMIE VED CESKE REPUBLIKY, V.V.I. (CZ) | 2009-02-26 | — | — | WO | disclosed |
| US-7393855-B2 | 2,2-bis-(hydroxymethyl)cyclopropylidenemethyl-purines and pyrimidines as antiviral agents | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2008-07-01 | — | — | US | disclosed |
| US-20080146533-A1 | Amino ceramide-like compounds and therapeutic methods of use | NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR | 2008-06-19 | — | — | US | disclosed |
| US-7335681-B2 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2008-02-26 | — | — | US | disclosed |
| US-20080014227-A1 | HETEROCYCLIC COMPOUNDS BASED ON N6-SUBSTITUTED ADENINE, METHODS OF THEIR PREPARATION, THEIR USE FOR PREPARATION OF DRUGS, COSMETIC PREPARATIONS AND GROWTH REGULATORS, PHARMACEUTICAL PREPARATIONS, COSMETIC PREPARATIONS AND GROWTH REGULATORS CONTAINING THESE COMPOUNDS | USTAV EXPERIMENTALNI BOTANIKY AKADEMIE VED CESKE REPUBLIKY (CZ) | 2008-01-17 | — | — | US | disclosed |
| US-7279482-B2 | Heterocyclic compound based on N6-substituted adenine, methods, of their preparation, their use for preparation of drugs, cosmetic preparations and growth regulators, pharmaceutical preparations, cosmetic preparations and growth regulators containing these compounds | Ústav experimentálni botaniky Akademie ved Ceské republiky (CZ) | 2007-10-09 | — | — | US | disclosed |
| US-20070225302-A1 | 2-Amino-9-[(2-hydroxymethyl) cyclopropylidenemethyl] purines as antiviral agents | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2007-09-27 | — | — | US | disclosed |
| WO-2007095666-A1 | AN IMPROVED GOLF TEE AND METHOD OF MANUFACTURE | SAFE-TEES DOWN UNDER PTY LTD (AU) | 2007-08-30 | — | — | WO | disclosed |
| US-7253185-B2 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2007-08-07 | — | — | US | disclosed |
| US-20070072916-A1 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2007-03-29 | — | — | US | disclosed |
| US-7183268-B2 | 2-amino-9-[(2-hydroxymethyl) cyclopropylidenemethyl] purine antiviral agents | WAYNE STATE UNIVERSITY (US) | 2007-02-27 | — | — | US | disclosed |
| US-7148251-B2 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2006-12-12 | — | — | US | disclosed |
| US-20060217560-A1 | Amino ceramide-like compounds and therapeutic methods of use | NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR | 2006-09-28 | — | — | US | disclosed |
| US-20060166925-A1 | Substitution derivatives of n6-benzyladenosine, methods of their preparation, their use for preparation of drugs, cosmetic preparations and growth regulators, pharmaceutical preparations, cosmetic preparations and growth regulators containing these compounds | USTAV EXPERIMENTALNI BOTANIKY AKADEMIE VED CESKE REPUBLIKY (CZ) | 2006-07-27 | — | — | US | disclosed |
| EP-1490368-A4 | 2,2-BIS(HYDROXYMETHYL)CYCLOPROPYLIDENEMETHYL - PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | UNIV WAYNE STATE (US) | 2006-07-19 | — | — | EP | disclosed |
| US-20060122203-A1 | 2-Hydroxymethylcyclopropylidenemethylpurines and - pyrimidines as antiviral agents | NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR | 2006-06-08 | — | — | US | disclosed |
| EP-1244668-B1 | PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND USE THEREOF | UNIVERSITAIRE INSTELLING ANTWE (BE) | 2006-04-05 | — | — | EP | disclosed |
| US-20060035909-A1 | 2,6,9-trisubstituted 8-azapurines such as 2-(4-aminocyclohexylamino)-6-benzylamino-9-isopropyl-8-azapurine, used as cyclin-dependent kinase inhibitors, in the treatment of skin disorders, viral infections, cancer, arthritis, lupus, diabetes, multiple sclerosis, restenosis, polycystic kidney disease, gout | UNIVERZITA PALACKEHO V OLOMOUCI (CZ) | 2006-02-16 | — | — | US | disclosed |
| EP-1490015-A4 | NOVEL 2-AMINO-9-((2-HYDROXYMETHYL) CYCLOPROPYLIDENEMETHYL) PURINES AS ANTIVIRAL AGENTS | UNIV WAYNE STATE (US) | 2005-12-28 | — | — | EP | disclosed |
| US-20050267094-A1 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN | 2005-12-01 | — | — | US | disclosed |
| US-20050239862-A1 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2005-10-27 | — | — | US | disclosed |
| US-6958345-B2 | 2-hydroxymethylcyclopropylidene methylpurines and -pyrimidines as antiviral agents | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2005-10-25 | — | — | US | disclosed |
| EP-1575973-A2 | SUBSTITUTION DERIVATIVES OF N SP 6 SP -BENZYLADENOSINE, METHODS OF THEIR PREPARATION, THEIR USE FOR PREPARATION OF DRUGS, COSMETIC PREPARATIONS AND GROWTH REGULATORS, PHARMACEUTICAL PREPARATIONS, COSMETIC PREPARATIONS AND GROWTH REGULATORS CONTAINING THESE COMPOUNDS | Ustav Experimentalni Botaniky Akademie ved Ceské Republiky (CZ) | 2005-09-21 | — | — | EP | disclosed |
| US-6916802-B2 | Amino ceramide-like compounds and therapeutic methods of use | GENZYME CORPORATION (US) | 2005-07-12 | — | — | US | disclosed |
| EP-1539760-A2 | AZAPURINE DERIVATIVES | INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) | 2005-06-15 | — | — | EP | disclosed |
| US-20050124582-A1 | 2-amino-9-[(2-hydroxymethyl) cyclopropylidenemethyl] purine antiviral agents | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2005-06-09 | — | — | US | disclosed |
| US-20050113393-A1 | 2,2-bis-(hydroxymethyl)cyclopropylidenemethyl-purines and pyrmindines as antiviral agents | WAYNE STATE UNIVERSITY (US) | 2005-05-26 | — | — | US | disclosed |
| US-6890949-B1 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2005-05-10 | — | — | US | disclosed |
| US-20050080097-A1 | Pyrazolo[4,3-D]pyrimidines, processes for their preparation and methods for therapy | USTAV EXPERIMENTALNI BOTANIKY AV CR (INSTITUTE OF EXPERIMENTAL BOTANY ACADEMY OF | 2005-04-14 | — | — | US | disclosed |
| US-20050049235-A1 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2005-03-03 | — | — | US | disclosed |
| US-20050043328-A1 | Heterocyclic compound based on n6-substituted adenine, methods, of their preparation, their use for preparation of drugs, cosmetic preparations and growth regulators, pharmaceutical preparations, cosmetic preparations and growth regulators containing these compounds | USTAV EPERIMENTALNI BOTANIKY AKADEMI VED CESKE REPUBILIKY (CZ) | 2005-02-24 | — | — | US | disclosed |
| US-20050009842-A1 | 2-hydroxymethylcyclopropylidene methylpurines and -pyrimidines as antiviral agents | NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR | 2005-01-13 | — | — | US | disclosed |
| EP-1490368-A2 | 2,2-BIS(HYDROXYMETHYL)CYCLOPROPYLIDENEMETHYL - PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | Wayne State University (US) | 2004-12-29 | — | — | EP | disclosed |
| EP-1490015-A2 | NOVEL 2-AMINO-9-((2-HYDROXYMETHYL) CYCLOPROPYLIDENEMETHYL) PURINES AS ANTIVIRAL AGENTS | Wayne State University (US) | 2004-12-29 | — | — | EP | disclosed |
| US-20040260099-A1 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN | 2004-12-23 | — | — | US | disclosed |
| EP-1165560-B1 | 2-HYDROXY METHYLCYCLOPRO PYLIDENEMETHYL PURINES AS ANTIVIRAL AGENTS | UNIV MICHIGAN (US) | 2004-11-17 | — | — | EP | disclosed |
| US-6790841-B2 | FOR THERAPY OF MAMMAL INFECTED WITH VIRUS | WAYNE STATE UNIVERSITY | 2004-09-14 | — | — | US | disclosed |
| WO-2004058791-A2 | SUBSTITUTION DERIVATIVES OF N6-BENZYLADENOSINE, METHODS OF THEIR PREPARATION, THEIR USE FOR PREPARATION OF DRUGS, COSMETIC PREPARATIONS AND GROWTH REGULATORS, PHARMACEUTICAL PREPARATIONS, COSMETIC PREPARATIONS AND GROWTH REGULATORS CONTAINING THESE COMPOUNDS | USTAV EXPERIMENTALNI BOTANIKY AKADEMIE VED CESKE REPUBLIKY (CZ) | 2004-07-15 | — | — | WO | disclosed |
| EP-1419157-A2 | HETEROCYCLIC COMPOUND BASED ON N sp 6 /sp −SUBSTITUTED ADENINE, METHODS OF THEIR PREPARATION, THEIR USE FOR PREPARATION OF DRUGS, COSMETIC PREPARATIONS AND GROWTH REGULATORS, PHARMACEUTICAL PREPARATIONS, COSMETIC PREPARATIONS AND GROWTH REGULATORS CONTAINING THESE | Ustav Experimentalni Botaniky Akademie ved Ceské Republiky (CZ) | 2004-05-19 | — | — | EP | disclosed |
| WO-2004018473-A2 | AZAPURINE DERIVATIVES | INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) | 2004-03-04 | — | — | WO | disclosed |
| EP-1384719-A1 | Inhibitors of the glucosyl ceramide synthase enzyme useful for the treatment of cancers, sphingolipidosis and microbial infections | The Regents of The University of Michigan (US) | 2004-01-28 | — | — | EP | disclosed |
| WO-2004006867-A2 | 2-AMINO-9-[(2-HYDROXYMETHYL) CYCLOPROPYLIDENEMETHYL] PURINE ANTIVIRAL AGENTS | WAYNE STATE UNIVERSITY (US) | 2004-01-22 | — | — | WO | disclosed |
| WO-2003104440-A2 | 2,2-BIS(HYDROXYMETHYL)CYCLOPROPYLIDENEMETHYL - PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | WAYNE STATE UNIVERSITY (US) | 2003-12-18 | — | — | WO | disclosed |
| EP-1358172-A2 | AMINO CERAMIDE-LIKE COMPOUNDS AND THERAPEUTIC METHODS OF USE | The Regents of The University of Michigan (US) | 2003-11-05 | — | — | EP | disclosed |
| WO-2003082872-A1 | NOVEL PYRAZOLO[4,3-D]PYRIMIDINES, PROCESSES FOR THEIR PREPARATION AND METHODS FOR THERAPY | USTAV EXPERIMENTALNI BOTANIKY AV CR (INSTITUTE OF EXPERIMENTAL BOTANY ACADEMY OF SCIENCES OF THE CZECH REPUBLIC) (CZ) | 2003-10-09 | — | — | WO | disclosed |
| US-20030187261-A1 | Purine derivatives, process for their preparation and use thereof | USTAV EXPERIMANTALNI BOTANIKY AKADEMIE VED CESKE REPUBLIKY (CZ) | 2003-10-02 | — | — | US | disclosed |
| EP-1348707-A1 | Pyrazolo[4,3-d]pyrimidines, processes for their preparation and methods for therapy | Ustav Experimentalni Botaniky AV CR (Institute of Experimental Botany Academy of Sciences of the Czech Republic) (CZ) | 2003-10-01 | — | — | EP | disclosed |
| US-6569889-B2 | Anticarcinogenic agents | THE REGENTS OF THE UNIVERSITY OF MICHIGAN | 2003-05-27 | — | — | US | disclosed |
| WO-2003040144-A2 | HETEROCYCLIC COMPOUND BASED ON N6-SUBSTITUTED ADENINE, METHODS OF THEIR PREPARATION, THEIR USE FOR PREPARATION OF DRUGS, COSMETIC PREPARATIONS AND GROWTH REGULATORS, PHARMACEUTICAL PREPARATIONS, COSMETIC PREPARATIONS AND GROWTH REGULATORS CONTAINING THESE COMPOUNDS | USTAV EXPERIMENTALNI BOTANIKY AKADEMIE VED CESKE REPUBLIKY (CZ) | 2003-05-15 | — | — | WO | disclosed |
| US-20030073680-A1 | Amino ceramide-like compounds and therapeutic methods of use | THE REGENTS OF THE UNIVERSITY OF MICHIGAN | 2003-04-17 | — | — | US | disclosed |
| WO-2002062777-A9 | AMINO CERAMIDE-LIKE COMPOUNDS AND THERAPEUTIC METHODS OF USE | UNIV MICHIGAN (US) | 2003-01-09 | — | — | WO | disclosed |
| US-20020198240-A1 | Amino ceramide - like compounds and therapeutic methods of use | REGENTS OF THE UNIVERSITY OF MICHIGAN, THE | 2002-12-26 | — | — | US | disclosed |
| US-20020193353-A1 | 2-hydroxymethylcyclopropylidenemethylpurines and -pyrimidines as antiviral agents | WAYNE STATE UNIVERSITY | 2002-12-19 | — | — | US | disclosed |
| US-20020156107-A1 | Amino ceramide - like compounds and therapeutic methods of use | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2002-10-24 | — | — | US | disclosed |
| EP-1244668-A1 | PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND USE THEREOF | UNIVERSITAIRE INSTELLING ANTWERPEN (BE) | 2002-10-02 | — | — | EP | disclosed |
| WO-2002062777-A2 | AMINO CERAMIDE-LIKE COMPOUNDS AND THERAPEUTIC METHODS OF USE | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2002-08-15 | — | — | WO | disclosed |
| WO-2000053603-A9 | 2-HYDROXY METHYLCYCLOPRO PYLIDENEMETHYL PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | UNIV MICHIGAN (US) | 2002-05-10 | — | — | WO | disclosed |
| EP-1165560-A4 | 2-HYDROXY METHYLCYCLOPRO PYLIDENEMETHYL PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | UNIV MICHIGAN (US) | 2002-04-17 | — | — | EP | disclosed |
| EP-1196406-A1 | AMINO CERAMIDE-LIKE COMPOUNDS AND THERAPEUTIC METHODS OF USE | The Regents of the University of Michigan (US) | 2002-04-17 | — | — | EP | disclosed |
| US-6352991-B1 | VIRICIDES FOR TREATMENT OF AIDS | WAYNE STATE UNIVERSITY | 2002-03-05 | — | — | US | disclosed |
| EP-1165560-A1 | 2-HYDROXY METHYLCYCLOPRO PYLIDENEMETHYL PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2002-01-02 | — | — | EP | disclosed |
| US-20010041735-A1 | Amino ceramide - like compounds and therapeutic methods of use | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2001-11-15 | — | — | US | disclosed |
| WO-2001049688-A1 | PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND USE THEREOF | UNIVERSITAIRE INSTELLING ANTWERPEN (BE) | 2001-07-12 | — | — | WO | disclosed |
| US-6255336-B1 | REDUCING CONCENTRATION OF GLYCOSPHINGOLIPIDS; SYNTHASE INHIBITORS | THE REGENTS OF THE UNIVERSITY OF MICHIGAN | 2001-07-03 | — | — | US | disclosed |
| JP-2001072502-A | SLIMICIDE | NIPPON SODA CO LTD | 2001-03-21 | — | — | JP | disclosed |
| WO-2001004108-A1 | AMINO CERAMIDE-LIKE COMPOUNDS AND THERAPEUTIC METHODS OF USE | REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2001-01-18 | — | — | WO | disclosed |
| US-6127439-A | MONOMERS ARE PARTIALLY POLYMERIZED AND THEN SUSPENDED IN WATER SO THAT THE RESULTING BEADS CONTAIN FROM 3 TO 40 WEIGHT % WATER WHICH ACTS AS SOLE OR A PREDOMINANT BLOWING AGENT | NOVA CHEMICALS (INTERNATIONAL) S.A. (CH) | 2000-10-03 | — | — | US | disclosed |
| EP-0912630-B1 | PROCESS FOR THE PREPARATION OF POLYMER PARTICLES | SHELL INT RESEARCH (NL) | 2000-09-20 | — | — | EP | disclosed |
| WO-2000053603-A1 | 2-HYDROXY METHYLCYCLOPRO PYLIDENEMETHYL PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 2000-09-14 | — | — | WO | disclosed |
| EP-0912630-A1 | PROCESS FOR THE PREPARATION OF POLYMER PARTICLES | SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) | 1999-05-06 | — | — | EP | disclosed |
| US-5783635-A | ARTIFICIAL MARBLE, PARTICLES OF CROSSLINKED DIVINYLBENZENE-STYRENE RESIN, GLASS OR ALUMINUM HYDROXIDE POWDER FILLER, BATHROOM AND KITCHEN FIXTURES AND COUNTERS | TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) | 1998-07-21 | — | — | US | disclosed |
| WO-1998030563-A1 | 2-HYDROXYMETHYLCYCLOPROPYLI- DENEMETHYLPURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) | 1998-07-16 | — | — | WO | disclosed |
| WO-1998001501-A1 | PROCESS FOR THE PREPARATION OF POLYMER PARTICLES | SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) | 1998-01-15 | — | — | WO | disclosed |
| EP-0806454-A2 | An unsaturated polyester resin composition | Takeda Chemical Industries, Ltd. (JP) | 1997-11-12 | — | — | EP | disclosed |
| US-5429762-A | Cooling agent | JAPAN PIONICS CO., LTD. (JP) | 1995-07-04 | — | — | US | disclosed |
| EP-0608789-A1 | Cooling agent | JAPAN PIONICS CO., LTD. (JP) | 1994-08-03 | — | — | EP | disclosed |
| EP-0474639-A1 | GENERAL PURPOSE FERTILISER | McKenzie, David Lawrence (GB) | 1992-03-18 | — | — | EP | disclosed |
| WO-1990011265-A2 | GENERAL PURPOSE FERTILISER | MCKENZIE DAVID LAWRENCE (GB) | 1990-10-04 | — | — | WO | disclosed |
| JP-H01101976-A | BONE CEMENT COMPONENT | SUMITOMO CEMENT CO LTD | 1989-04-19 | — | — | JP | disclosed |
| JP-H01101977-A | MANUFACTURE OF APATITE COVER | SUMITOMO CEMENT CO LTD | 1989-04-19 | — | — | JP | disclosed |
| JP-S63238022-A | ISOLATION OF HBE ANTIGEN | KURARAY CO LTD | 1988-10-04 | — | — | JP | disclosed |
| EP-0169926-B1 | POLYESTER COMPOSITION | TEIJIN LIMITED (JP) | 1988-05-18 | — | — | EP | disclosed |
| JP-S61247610-A | PREPARATION OF TRICALCIUM DIPHOSPHATE | KANTO KAGAKU KK | 1986-11-04 | — | — | JP | disclosed |
| EP-0169926-A1 | Polyester composition | TEIJIN LIMITED (JP) | 1986-02-05 | — | — | EP | disclosed |
| US-4563207-A | MANURE, POTASSIUM COMPOUND, PHOSPHATE AND CALCIUM CARBONATE | MCKENZIE DAVID L | 1986-01-07 | — | — | US | disclosed |
| US-4513114-A | CONTAINING DISPERSOID PARTICLES OR AGGLOMERATES | TEIJIN LIMITED (JP) | 1985-04-23 | — | — | US | disclosed |
| US-4513114-A | CONTAINING DISPERSOID PARTICLES OR AGGLOMERATES | TEIJIN LIMITED (JP) | 1985-04-23 | — | — | US | disclosed |
Patent text — is the patent's own abstract consistent with the prediction?
For each of this compound's patents that has machine-readable text (49 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.
| Patent | Title | Text reads most about | Predicted target · text-rank |
|---|---|---|---|
| US-20110287111-A1 | SUBSTITUTED 6-(2-AMINOBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND PREPARATIONS CONTAINING THESE COMPOUNDS | CDK6, CCNI, CDK2 | FDPS 866/4885BLM 1536/4885TDP1 273/4885 |
| US-20140066394-A1 | Substituted 6-(Benzylamino) Purine Riboside Derivatives, Use Thereof and Compositions Containing These Derivatives | PNP, NUDT1, TYMP | FDPS 1369/4885BLM 561/4885TDP1 329/4885 |
| US-20180072736-A1 | 5-SUBSTITUTED 7-[4-(2-PYRIDYL)PHENYLMETHYLAMINO]-3-ISOPROPYLPYRAZOLO4,3-D]PYRIMIDINE DERIVATIVES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | CDK5, CDK2, CDK4 | FDPS 2091/4885BLM 3742/4885TDP1 1976/4885 |
| US-20040260099-A1 | Amino ceramide-like compounds and therapeutic methods of use | UGCG, CERS2, CERT1 | FDPS 357/4885BLM 4857/4885TDP1 2029/4885 |
| US-20110275652-A1 | 2,2-BIS-(HYDROXYMETHYL)CYCLOPROPYLIDENEMETHYL-PURINES AND -PYRIMIDINES AS ANTIVIRAL AGENTS | TPMT, HPRT1, MTAP | FDPS 585/4885BLM 1871/4885TDP1 286/4885 |
| US-20080014227-A1 | HETEROCYCLIC COMPOUNDS BASED ON N6-SUBSTITUTED ADENINE, METHODS OF THEIR PREPARATION, THEIR USE FOR PREPARATION OF DRUGS, COSMETIC PREPARATIONS AND GROWTH REGULATORS, PHARMACEUTICAL PREPARATIONS, COSMETIC PREPARATIONS AND GROWTH REGULATORS CONTAINING THESE COMPOUNDS | TYMP, CCNB1, CCNA2 | FDPS 346/4885BLM 1594/4885TDP1 967/4885 |
| US-12636299-B2 | Terpenoid derivatives, pharmaceutical preparations containing these derivatives and their use in neuroprotection | GALC, HK1, SNCA | FDPS 3194/4885BLM 4827/4885TDP1 1367/4885 |
| US-20100204460-A1 | NATURAL BRASSINOSTEROIDS FOR USE FOR TREATING HYPERPROLIFERATION, TREATING PROLIFERATIVE DISEASES AND REDUCING ADVERSE EFFECTS OF STEROID DYSFUNCTION IN MAMMALS, PHARMACEUTICAL COMPOSITION AND ITS USE | BRDT, NR5A1, BRSK2 | FDPS 1796/4885BLM 3752/4885TDP1 3392/4885 |
| US-20060166925-A1 | Substitution derivatives of n6-benzyladenosine, methods of their preparation, their use for preparation of drugs, cosmetic preparations and growth regulators, pharmaceutical preparations, cosmetic preparations and growth regulators containing these compounds | ADAR, ADORA2A, AMPD2 | FDPS 1069/4885BLM 1256/4885TDP1 1147/4885 |
| US-20050080097-A1 | Pyrazolo[4,3-D]pyrimidines, processes for their preparation and methods for therapy | CBR3, DHFR, AKR1C3 | FDPS 812/4885BLM 400/4885TDP1 2367/4885 |
| US-20090312392-A1 | Amino ceramide-like compounds and therapeutic methods of use | UGCG, CERS2, SGMS1 | FDPS 523/4885BLM 4798/4885TDP1 2433/4885 |
| US-20020198240-A1 | Amino ceramide - like compounds and therapeutic methods of use | UGCG, CERS2, CERT1 | FDPS 357/4885BLM 4857/4885TDP1 2029/4885 |
| US-20050239862-A1 | Amino ceramide-like compounds and therapeutic methods of use | UGCG, CERS2, CERT1 | FDPS 438/4885BLM 4856/4885TDP1 2567/4885 |
| US-20060122203-A1 | 2-Hydroxymethylcyclopropylidenemethylpurines and - pyrimidines as antiviral agents | HPRT1, TPMT, NUDT1 | FDPS 1644/4885BLM 1690/4885TDP1 377/4885 |
| US-20050043328-A1 | Heterocyclic compound based on n6-substituted adenine, methods, of their preparation, their use for preparation of drugs, cosmetic preparations and growth regulators, pharmaceutical preparations, cosmetic preparations and growth regulators containing these compounds | ATIC, UMPS, CCNB1 | FDPS 304/4885BLM 1551/4885TDP1 1656/4885 |
| US-20050009842-A1 | 2-hydroxymethylcyclopropylidene methylpurines and -pyrimidines as antiviral agents | TPMT, HPRT1, MTAP | FDPS 1541/4885BLM 1693/4885TDP1 366/4885 |
| US-20200087306-A1 | 2,6-DISUBSTITUTED-9-CYCLOPENTYL-9H-PURINES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | FLT3, CDK9, CDK6 | FDPS 826/4885BLM 1656/4885TDP1 802/4885 |
| US-20120071433-A1 | Substituted 6-(Benzylamino) Purine Riboside Derivatives, Use Thereof and Compositions Containing These Derivatives | CD38, NUDT1, PNP | FDPS 1123/4885BLM 861/4885TDP1 367/4885 |
| US-20220127269-A1 | HETEROCYCLIC NITROGEN-CONTAINING PURINE DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN NEUROPROTECTION | NME4, NLN, PNP | FDPS 1168/4885BLM 1942/4885TDP1 63/4885 |
| US-20010041735-A1 | Amino ceramide - like compounds and therapeutic methods of use | UGCG, CERS2, CERT1 | FDPS 458/4885BLM 4837/4885TDP1 2739/4885 |
| US-20150368248-A1 | 2-SUBSTITUTED-6-BIARYLMETHYLAMINO-9-CYCLOPENTYL-9H-PURINE DERIVATIVES, USE THEREOF AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS | ENTPD5, PNP, HCCS | FDPS 421/4885BLM 920/4885TDP1 2150/4885 |
| US-20170362236-A1 | 6,8-DISUBSTITUTED-9-(HETEROCYCLYL)PURINES, COMPOSITIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN COSMETIC AND MEDICINAL APPLICATIONS | PNP, UNG, NUDT1 | FDPS 514/4885BLM 680/4885TDP1 47/4885 |
| US-20200361943-A1 | 5-ALKYLTHIO-7-[(4-ARYLBENZYL)AMINO]-1(2)H-PYRAZOLO[4,3-D]PYRIMIDINES FOR TREATMENT OF LYMPHOMA | TK1, DCK, CCNK | FDPS 2001/4885BLM 2796/4885TDP1 324/4885 |
| US-20200157105-A1 | 9-(2-OXACYCLOALKYL)-9H-PURINE-2,6-DIAMINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF SKIN DISORDERS | ADORA2A, UNG, P2RY6 | FDPS 1612/4885BLM 1739/4885TDP1 31/4885 |
| US-20120070512-A1 | Substituted 6-(2-hydroxybenzylamino)purine Derivatives, Their Use as Medicaments and Compositions Containing These Derivatives | CDK6, CCNI, CDK2 | FDPS 1027/4885BLM 1075/4885TDP1 484/4885 |
| US-20130040908-A1 | SUBSTITUTION DERIVATIVES OF N6-BENZYLADENOSINE-5' -MONOPHOSPHATE, METHODS OF PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, AND THERAPEUTIC PREPARATIONS CONTAINING THESE COMPOUNDS | MTAP, RNMT, NUDT1 | FDPS 723/4885BLM 311/4885TDP1 767/4885 |
| US-10093675-B2 | 6,8-disubstituted-9-(heterocyclyl)purines, compositions containing these derivatives and their use in cosmetic and medicinal applications | PNP, UNG, NUDT1 | FDPS 514/4885BLM 680/4885TDP1 47/4885 |
| US-20050267094-A1 | Amino ceramide-like compounds and therapeutic methods of use | UGCG, CERS2, SGMS1 | FDPS 523/4885BLM 4798/4885TDP1 2433/4885 |
| US-20050113393-A1 | 2,2-bis-(hydroxymethyl)cyclopropylidenemethyl-purines and pyrmindines as antiviral agents | TPMT, HPRT1, MTAP | FDPS 793/4885BLM 1759/4885TDP1 280/4885 |
| US-20080146533-A1 | Amino ceramide-like compounds and therapeutic methods of use | UGCG, CERS2, SGMS1 | FDPS 523/4885BLM 4798/4885TDP1 2433/4885 |
| US-20230414645-A1 | TERPENOID DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES AND THEIR USE IN NEUROPROTECTION | HTT, SNCA, BDNF | FDPS 562/4885BLM 4405/4885TDP1 458/4885 |
| US-11643413-B2 | 9-(2-oxacycloalkyl)-9H-purine-2,6-diamine derivatives and their use for the treatment of skin disorders | ADORA2A, UNG, P2RY6 | FDPS 1612/4885BLM 1739/4885TDP1 31/4885 |
| US-20230365616-A1 | CHOLESTANE DERIVATIVES, PREPARATIONS CONTAINING THESE DERIVATIVES AND USE THEREOF | BAD, CYP27A1, NPC1L1 | FDPS 1098/4885BLM 2220/4885TDP1 1031/4885 |
| US-20030187261-A1 | Purine derivatives, process for their preparation and use thereof | DCK, DTYMK, CCNK | FDPS 499/4885BLM 2208/4885TDP1 1089/4885 |
| US-20070225302-A1 | 2-Amino-9-[(2-hydroxymethyl) cyclopropylidenemethyl] purines as antiviral agents | HAVCR2, ORC3, HPRT1 | FDPS 2146/4885BLM 2783/4885TDP1 1514/4885 |
| US-20110311652-A1 | Novel Saponin Compounds, Methods of Preparation Thereof, Use Thereof and Pharmaceutical Compositions | CYP4A11, CYP11B1, CYP11B2 | FDPS 402/4885BLM 2281/4885TDP1 4478/4885 |
| US-20030073680-A1 | Amino ceramide-like compounds and therapeutic methods of use | UGCG, CERS2, SGMS1 | FDPS 523/4885BLM 4798/4885TDP1 2433/4885 |
| US-11028087-B2 | 2,6-disubstituted-9-cyclopentyl-9H-purines, use thereof as medicaments, and pharmaceutical compositions | FLT3, CDK9, CDK6 | FDPS 826/4885BLM 1656/4885TDP1 802/4885 |
| US-20090118308-A1 | 2,2-Bis-(hydroxymethyl)cyclopropylidenemethyl-Purines and -Pyrimidines As Antiviral Agents | TPMT, HPRT1, MTAP | FDPS 585/4885BLM 1871/4885TDP1 286/4885 |
| US-20070072916-A1 | Amino ceramide-like compounds and therapeutic methods of use | UGCG, CERS2, CERT1 | FDPS 357/4885BLM 4857/4885TDP1 2029/4885 |
| US-20050049235-A1 | Amino ceramide-like compounds and therapeutic methods of use | UGCG, CERS2, SGMS1 | FDPS 523/4885BLM 4798/4885TDP1 2433/4885 |
| US-20020193353-A1 | 2-hydroxymethylcyclopropylidenemethylpurines and -pyrimidines as antiviral agents | TPMT, HPRT1, MTAP | FDPS 1922/4885BLM 1729/4885TDP1 266/4885 |
| US-11186583-B2 | 5-alkylthio-7-[(4-arylbenzyl)amino]-1(2)H-pyrazolo[4,3-d]pyrimidines for treatment of lymphoma | TK1, DCK, CCNK | FDPS 2001/4885BLM 2796/4885TDP1 324/4885 |
| US-20130072506-A1 | 6,8-DISUBSTITUTED PURINE COMPOSITIONS | UNG, PNP, UMPS | FDPS 613/4885BLM 532/4885TDP1 45/4885 |
| US-20060035909-A1 | 2,6,9-trisubstituted 8-azapurines such as 2-(4-aminocyclohexylamino)-6-benzylamino-9-isopropyl-8-azapurine, used as cyclin-dependent kinase inhibitors, in the treatment of skin disorders, viral infections, cancer, arthritis, lupus, diabetes, multiple sclerosis, restenosis, polycystic kidney disease, gout | CDK8, CDK6, CDK1 | FDPS 2309/4885BLM 4722/4885TDP1 1166/4885 |
| US-20050124582-A1 | 2-amino-9-[(2-hydroxymethyl) cyclopropylidenemethyl] purine antiviral agents | HAVCR2, ORC3, NSUN2 | FDPS 2365/4885BLM 2818/4885TDP1 1454/4885 |
| US-12319694-B2 | Heterocyclic nitrogen-containing purine derivatives, pharmaceutical preparations containing these derivatives and their use in neuroprotection | NME4, NLN, PNP | FDPS 1168/4885BLM 1942/4885TDP1 63/4885 |
| US-20060217560-A1 | Amino ceramide-like compounds and therapeutic methods of use | UGCG, CERS2, CERT1 | FDPS 357/4885BLM 4857/4885TDP1 2029/4885 |
| US-20020156107-A1 | Amino ceramide - like compounds and therapeutic methods of use | UGCG, CERS2, CERT1 | FDPS 357/4885BLM 4857/4885TDP1 2029/4885 |
“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.