Toluene

Toluene

SCHEMBL6928034

Cc1ccccc1.Cl.N

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Toluene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Toluene SCHEMBL8015120 1.00 ACHE (0.85)
Toluene SCHEMBL11113893 1.00 ACHE (0.85)
Toluene SCHEMBL11742959 1.00 ACHE (0.85)
Toluene SCHEMBL27781947 0.96 ACHE (0.79)
Toluene SCHEMBL11741374 0.96 ACHE (0.79)
Toluene SCHEMBL180839 0.96
Toluene SCHEMBL628172 0.96
Toluene SCHEMBL15009 0.96
Toluene SCHEMBL522792 0.96 ACHE (0.92)
Toluene SCHEMBL7591772 0.96 ACHE (0.92)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118320794-B Adsorbing material for dioxin in flue gas and preparation method thereof 杭州回水科技股份有限公司 2024-08-23 CN claimed
CN-118320794-A Adsorbing material for dioxin in flue gas and preparation method thereof 杭州回水科技股份有限公司 2024-07-12 CN claimed
CN-1293705-A Heat transpiration preparation and method of the heat transpiration EARTH CHEMICAL CO (JP) 2001-05-02 CN claimed
CN-114127121-B Methods and compositions for promoting and enhancing T cell mediated immune responses through ADCC targeting of CD39 expressing cells 北京恩瑞尼生物科技股份有限公司 2025-04-11 CN disclosed
CN-119604610-A Vectors and methods for in vivo antibody production 瑞泽恩制药公司 2025-03-11 CN disclosed
CN-119409834-A Methods and compositions for promoting and enhancing T cell mediated immune responses through ADCC targeting of CD39 expressing cells 北京恩瑞尼生物科技股份有限公司 2025-02-11 CN disclosed
CN-118320794-B Adsorbing material for dioxin in flue gas and preparation method thereof 杭州回水科技股份有限公司 2024-08-23 CN disclosed
CN-118401547-A Interleukin-12 self-replicating RNA and methods 嘉晨西海(杭州)生物技术有限公司 2024-07-26 CN disclosed
CN-118382433-A RNA formulations and lipids 嘉晨西海(杭州)生物技术有限公司 2024-07-23 CN disclosed
CN-118320794-A Adsorbing material for dioxin in flue gas and preparation method thereof 杭州回水科技股份有限公司 2024-07-12 CN disclosed
CN-111032619-B Adamantylmethylamine derivatives and their use as medicaments 国立大学法人东北大学 2023-07-18 CN disclosed
CN-1068588-C 1H-indole-3-acetamide splA2 inhibitors LILLY CO ELI (US) 2001-07-18 CN disclosed
CN-1293705-A Heat transpiration preparation and method of the heat transpiration EARTH CHEMICAL CO (JP) 2001-05-02 CN disclosed
CN-1284135-A Rapid method for assessment of inhibition and kill of anaerobic bacteria by toxic compounds NALCO CHEMICAL CO (US) 2001-02-14 CN disclosed
EP-1051510-A1 A RAPID METHOD FOR THE ASSESSMENT OF THE INHIBITION AND KILL OF ANAEROBIC BACTERIA BY TOXIC COMPOUNDS NALCO CHEMICAL COMPANY (US) 2000-11-15 EP disclosed
WO-1999034013-A1 A RAPID METHOD FOR THE ASSESSMENT OF THE INHIBITION AND KILL OF ANAEROBIC BACTERIA BY TOXIC COMPOUNDS NALCO CHEMICAL COMPANY (US) 1999-07-08 WO disclosed
US-4780252-A FORMING SALT WITH SINGLE ISOMERS OF OPTICAL ACTIVE AMINE IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-10-25 US disclosed
US-4683089-A SEPARATION OF OPTICAL ISOMERS, INSECTICIDES IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1987-07-28 US disclosed
EP-0010874-B1 PROCESS FOR SEPARATING OPTICAL ISOMERS OF SUBSTITUTED CYCLOPROPANE CARBOXYLIC ACIDS; AMINE SALTS OF SUBSTITUTED CYCLOPROPANE CARBOXYLIC ACIDS; A SUBSTITUTED CYCLOPROPANE CARBOXYLIC ACID IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-06-22 EP disclosed
EP-0010874-A1 Process for separating optical isomers of substituted cyclopropane carboxylic acids; amine salts of substituted cyclopropane carboxylic acids; a substituted cyclopropane carboxylic acid IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1980-05-14 EP disclosed