Pyromellitic Acid

Pyromellitic Acid

SCHEMBL11316481

Cl.Cl.O=C(O)c1cc(C(=O)O)c(C(=O)O)cc1C(=O)O

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Pyromellitic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 known ✓ P00918 4/20 0.43
PTGS2 known ✓ P35354 2/20 0.43
SLC6A2 known ✓ P23975 1/20 0.41
SLC6A4 known ✓ P31645 1/20 0.41
DRD3 known ✓ P35462 1/20 0.41
KDR known ✓ P35968 1/20 0.40
ALDH1A1 P00352 6/20 0.50
ALOX15 P16050 2/20 0.50
CYP1A2 P05177 1/20 0.50
KMT2A Q03164 4/20 0.46
TDP1 Q9NUW8 4/20 0.46
MEN1 O00255 3/20 0.46
POLB P06746 2/20 0.46
THRB P10828 2/20 0.46
RECQL P46063 2/20 0.46
USP2 O75604 1/20 0.46
MAPT P10636 1/20 0.46
PKM P14618 1/20 0.46
APEX1 P27695 1/20 0.46
BLM P54132 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyromellitic Acid SCHEMBL338944 1.00 ALDH1A1 (0.50) ALDH1A1ALOX15CYP1A2KMT2ATDP1
Pyromellitic Acid SCHEMBL895352 1.00 ALDH1A1 (0.50) ALDH1A1ALOX15CYP1A2KMT2ATDP1
Pyromellitic Acid SCHEMBL338946 1.00 ALDH1A1 (0.50) ALDH1A1ALOX15CYP1A2KMT2ATDP1
Pyromellitic Acid SCHEMBL11316473 1.00 ALDH1A1 (0.50) ALDH1A1ALOX15CYP1A2KMT2ATDP1
Pyromellitic Acid SCHEMBL22127 0.96 ALDH1A1 (0.53) ALDH1A1ALOX15CYP1A2KMT2ATDP1
Pyromellitic Acid SCHEMBL22443 0.96 ALDH1A1 (0.53) ALDH1A1ALOX15CYP1A2KMT2ATDP1
Pyromellitic Acid SCHEMBL692530 0.92 ALDH1A1 (0.50) ALDH1A1ALOX15CYP1A2KMT2ATDP1
Pyromellitic Acid SCHEMBL9485109 0.92 ALDH1A1 (0.50) ALDH1A1ALOX15CYP1A2KMT2ATDP1
Pyromellitic Acid SCHEMBL22982083 0.92 ALDH1A1 (0.50) ALDH1A1ALOX15CYP1A2KMT2ATDP1
Pyromellitic Acid SCHEMBL21328420 0.92 ALDH1A1 (0.50) ALDH1A1ALOX15CYP1A2KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112973473-A Reverse osmosis composite membrane resisting biological pollution and preparation method thereof 天津工业大学 2021-06-18 CN claimed
CN-111187413-A Sulfonated polyethyleneimine, nanofiltration membrane and preparation method thereof 东华大学 2020-05-22 CN claimed
US-20230318146-A1 NONAQUEOUS ELECTROLYTE SECONDARY BATTERY SEPARATOR SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2023-10-05 US disclosed
CN-112973473-A Reverse osmosis composite membrane resisting biological pollution and preparation method thereof 天津工业大学 2021-06-18 CN disclosed
US-20150361257-A1 METHOD FOR PRODUCING SUBSTRATE HAVING PATTERN AND RESIN COMPOSITION FOR HYDROFLUORIC ACID ETCHING NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2015-12-17 US disclosed
US-4243743-A CARBOXYL-CONTAINING POLYAMIDE, UNSATURATED AMINE OR QUATERNARY AMMONIUM SALT TORAY INDUSTRIES, INC. (JP) 1981-01-06 US disclosed