1-Naphthol

1-Naphthol

SCHEMBL594288

Cl.Oc1cccc2ccccc12

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of 1-Naphthol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 known ✓ P03372 2/20 0.48
ESR2 known ✓ Q92731 2/20 0.48
EGFR known ✓ P00533 1/20 0.47
CA2 known ✓ P00918 1/20 0.47
PIK3CA known ✓ P42336 1/20 0.47
CYP1A2 P05177 2/20 0.94
PTPN22 Q9Y2R2 1/20 0.61
IDO1 P14902 1/20 0.55
HSD17B10 Q99714 4/20 0.52
TDP1 Q9NUW8 3/20 0.52
TSHR P16473 2/20 0.52
MAPT P10636 2/20 0.52
HPGD P15428 2/20 0.52
ALOX15 P16050 2/20 0.52
RECQL P46063 2/20 0.52
APP P05067 1/20 0.52
THRB P10828 1/20 0.52
CASP1 P29466 1/20 0.52
SNCA P37840 1/20 0.52
NQO2 P16083 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
1-Naphthol SCHEMBL30657150 1.00 CYP1A2 (0.94) CYP1A2PTPN22IDO1HSD17B10TDP1
1-Naphthol SCHEMBL27269259 0.97 CYP1A2 (0.90) CYP1A2PTPN22IDO1HSD17B10TDP1
1-Naphthol SCHEMBL6896129 0.97 CYP1A2 (0.90) CYP1A2PTPN22IDO1HSD17B10TDP1
1-Naphthol SCHEMBL10486461 0.97 CYP1A2 (1.00) CYP1A2PTPN22IDO1HSD17B10TDP1
1-Naphthol SCHEMBL3416 0.97 CYP1A2 (1.00) CYP1A2PTPN22IDO1HSD17B10TDP1
1-Naphthol SCHEMBL273260 0.97 CYP1A2 (1.00) CYP1A2PTPN22IDO1HSD17B10TDP1
1-Naphthol SCHEMBL29767730 0.97 CYP1A2 (1.00) CYP1A2PTPN22IDO1HSD17B10TDP1
1-Naphthol SCHEMBL8904232 0.94 CYP1A2 (0.94) CYP1A2PTPN22IDO1HSD17B10TDP1
1-Naphthol SCHEMBL3924043 0.94 CYP1A2 (0.94) CYP1A2PTPN22IDO1HSD17B10TDP1
1-Naphthol SCHEMBL21490911 0.94 CYP1A2 (0.94) CYP1A2PTPN22IDO1HSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114235990-A Tuberculosis serum marker screening method and application 宁夏医科大学 2022-03-25 CN claimed
CN-112209838-A Preparation method of butenaphthol hydrochloride 鲁南制药集团股份有限公司 2021-01-12 CN claimed
CN-118045162-A Application of decorin combined with NK cells in treatment of solid tumors 北京景达生物科技有限公司 2024-05-17 CN disclosed
CN-114269756-B 4-Oxo-3, 4-dihydropyrido [3,4-D ] pyrimidine compounds that inhibit EIF4E 效应疗法股份有限公司 2024-05-14 CN disclosed
CN-117357503-B Use of p-hydroxyphenylacetamide in the treatment of psychotic disorders 中国人民解放军军事科学院军事医学研究院 2024-03-08 CN disclosed
CN-117545748-A Benzimidazolyl GLP-1GPCR receptor agonists, pharmaceutical compositions comprising the same, and methods of use thereof 卡莫特医疗有限公司 2024-02-09 CN disclosed
CN-117357503-A Use of p-hydroxyphenylacetamide in the treatment of psychotic disorders 中国人民解放军军事科学院军事医学研究院 2024-01-09 CN disclosed
CN-117043154-A GPCR receptor agonists, pharmaceutical compositions comprising same, and methods of use thereof 卡莫特医疗有限公司 2023-11-10 CN disclosed
CN-114235990-A Tuberculosis serum marker screening method and application 宁夏医科大学 2022-03-25 CN disclosed
CN-111183134-A Heterocyclic compound and organic light-emitting device comprising the same LT素材株式会社 2020-05-19 CN disclosed
US-8704348-B2 Polyol photosensitizers, carrier gas UV laser ablation sensitizers, and other additives and methods for making and using same NDSU RESEARCH FOUNDATION (US) 2014-04-22 US disclosed
US-8114567-B2 Polyol photosensitizers, carrier gas UV laser ablation sensitizers, and other additives and methods for making and using same NDSU RESEARCH FOUNDATION (US) 2012-02-14 US disclosed
US-20090184417-A1 POLYOL PHOTOSENSITIZERS, CARRIER GAS UV LASER ABLATION SENSITIZERS, AND OTHER ADDITIVES AND METHODS FOR MAKING AND USING SAME NDSU RESEARCH FOUNDATION 2009-07-23 US disclosed
WO-2007124073-A2 POLYOL PHOTOSENSITIZERS, CARRIER GAS UV LASER ABLATION SENSITIZERS, AND OTHER ADDITIVES AND METHODS FOR MAKING AND USING SAME NDSU RESEARCH FOUNDATION (US) 2007-11-01 WO disclosed
CN-1747944-A Blue light-emitting compound, method for producing same, and light-emitting element using same HIROSE ENGINEERING CO LTD (JP) 2006-03-15 CN disclosed
WO-2000056691-A1 SYNTHESIS OF VAPOL LIGANDS ARCH DEVELOPMENT CORPORATION (US) 2000-09-28 WO disclosed
EP-0476016-A1 THERAPEUTICALLY USEFUL 2-AMINOTETRALIN DERIVATIVES PHARMACIA & UPJOHN COMPANY (US) 1992-03-25 EP disclosed
WO-1990015047-A1 THERAPEUTICALLY USEFUL 2-AMINOTETRALIN DERIVATIVES THE UPJOHN COMPANY (US) 1990-12-13 WO disclosed
CN-88102538-A New dicyclic compound, its preparation method and the pharmaceutical composition that contains this compounds 1988-12-07 CN disclosed
EP-0205180-A1 Process for preparing virtually spherical catalyst particles and a process for polymerizing alkenes-1 and for copolymerizing alkenes-1 with each other and/or with ethylene while applying such spherical catalyst particles STAMICARBON B.V. (NL) 1986-12-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090184417-A1 POLYOL PHOTOSENSITIZERS, CARRIER GAS UV LASER ABLATION SENSITIZERS, AND OTHER ADDITIVES AND METHODS FOR MAKING AND USING SAME OTC, ODC1, OXGR1 ESR1 1614/4885ESR2 2349/4885EGFR 1514/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.