Triaziquone

Triaziquone

SCHEMBL62271

O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1.O=P(O)(O)O

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Triaziquone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 1/20 0.42
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
TP53 P04637 1/20 0.40
STAT3 P40763 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
APAF1 O14727 2/20 0.35
TDP2 O95551 2/20 0.35
NSD2 O96028 2/20 0.35
HKDC1 Q2TB90 2/20 0.35
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
GALK1 P51570 1/20 0.33
BLM P54132 1/20 0.33
ATM Q13315 1/20 0.33
NOD2 Q9HC29 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL3903553 1.00 DNMT1 (0.42) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL10680234 0.98 DNMT1 (0.41) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL9678206 0.95 DNMT1 (0.39) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL8848720 0.95 DNMT1 (0.39) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL23087090 0.93 DNMT1 (0.38) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL21805756 0.93 MAPT (0.39) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL21625776 0.93 MAPT (0.41) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL20515128 0.93 DNMT1 (0.40) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL3650047 0.93 DNMT1 (0.40) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL7064057 0.93 DNMT1 (0.40) DNMT1MAPTHTTTP53STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1231 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3827814-B1 OPHTHALMIC FORMULATIONS DOMPE FARM SPA (IT) 2025-12-17 EP claimed
WO-2025222268-A1 TOPICAL COMPOSITIONS AND METHODS FOR TREATING ATROPHIC VAGINITIS JASTLABS CORPORATION (CA) 2025-10-30 WO claimed
CN-119925276-A CRAC inhibitor freeze-dried powder preparation based on tromethamine phosphate salt prodrug and preparation method thereof 天津辰欣药物研究有限公司 2025-05-06 CN claimed
EP-4507722-A1 NANOEMULSION UNIVERSAL INFLUENZA VACCINE Bluewillow Biologics, Inc. (US) 2025-02-19 EP claimed
US-20240058434-A1 NANOEMULSION UNIVERSAL INFLUENZA VACCINE BLUEWILLOW BIOLOGICS, INC. (US) 2024-02-22 US claimed
WO-2023200764-A1 NANOEMULSION UNIVERSAL INFLUENZA VACCINE BLUEWILLOW BIOLOGICS, INC. (US) 2023-10-19 WO claimed
WO-2022157373-A1 COMPOSITIONS AND KITS FOR IN VIVO IMAGING OF CARDIAC SARCOIDOSIS VRIJE UNIVERSITEIT BRUSSEL (BE) 2022-07-28 WO claimed
CN-114133635-A Oxidation and corrosion resistant plastic 江苏爱唯生物科技有限公司 2022-03-04 CN claimed
CN-106442039-B Device, solution and method for sample collection 阿博根公司 2020-08-07 CN claimed
CN-107486037-B A kind of PVDF/PDA composite membrane with super hydrophilicity 福州大学 2019-11-12 CN claimed
CN-107486037-A A kind of PVDF/PDA composite membranes with super hydrophilicity 福州大学 2017-12-19 CN claimed
US-20170087089-A1 PROCESS FOR THE PREPARATION OF UNILAMELLAR LIPOSOMAL COMPOSITION SUN PHARMA ADVANCED RESEARCH COMPANY LTD (IN) 2017-03-30 US claimed
US-8217024-B2 Conjugated estrogen compositions, applicators, kits, and methods of making and use thereof TEVA WOMEN'S HEALTH, INC. (US) 2012-07-10 US claimed
EP-1971325-A2 CONJUGATED ESTROGEN COMPOSITIONS, APPLICATORS, KITS, AND METHODS OF MAKING AND USE THEREOF Duramed Pharmaceuticals, Inc. (US) 2008-09-24 EP claimed
US-20070191321-A1 Conjugated estrogen compositions, applicators, kits, and methods of making and use thereof TEVA WOMEN'S HEALTH, INC. 2007-08-16 US claimed
WO-2007076144-A2 CONJUGATED ESTROGEN COMPOSITIONS, APPLICATORS, KITS, AND METHODS OF MAKING AND USE THEREOF DURAMED PHARMACEUTICALS, INC. (US) 2007-07-05 WO claimed
EP-0034213-B1 A STABILIZED AQUEOUS COENZYME SOLUTION FOR USE IN A CLINICAL ASSAY, A METHOD OF STABILIZING A LABILE COENZYME IN AN AQUEOUS CLINICAL ASSAY SOLUTION AND A KIT FOR USE IN SAID CLINICAL ASSAY Modrovich, Ivan Endre (US) 1984-11-07 EP claimed
US-4394449-A REGENERATION OF COENZYME FOR CLINICAL ASSAYS MEDICAL ANALYSIS SYSTEMS, INC. 1983-07-19 US claimed
EP-0034213-A1 A stabilized aqueous coenzyme solution for use in a clinical assay, a method of stabilizing a labile coenzyme in an aqueous clinical assay solution and a kit for use in said clinical assay Modrovich, Ivan Endre (US) 1981-08-26 EP claimed
JP-8049282-A None JP disclosed
EP-4730479-A2 FLAME-RETARDANT NON-AQUEOUS ELECTROLYTIC SOLUTION AND SECONDARY BATTERY USING SAME Kyoto University (JP) 2026-04-22 EP disclosed
EP-4089406-B1 ION SENSOR SYSMEX CORP (JP) 2026-02-11 EP disclosed
EP-4441079-B1 SWITCHABLE POLYPEPTIDE AND ITS USE FOR GENTLE AFFINITY PURIFICATION UNIV OXFORD INNOVATION LTD (GB) 2026-02-11 EP disclosed
US-20260007731-A1 INTRANASAL POLYSACCHARIDE CONJUGATE NANOMULSION VACCINES AND METHODS OF USING THE SAME BLUEWILLOW BIOLOGICS, INC. (US) 2026-01-08 US disclosed
US-20250381246-A1 LIQUID FORMULATIONS COMPRISING MUTANT FGF-21 PEPTIDE PEGYLATED CONJUGATES 89BIO, INC. (US) 2025-12-18 US disclosed
US-20250380724-A1 METHOD FOR PRODUCING PROCESSED PLANT PROTEIN-CONTAINING COMPOSITION AMANO ENZYME INC. (JP) 2025-12-18 US disclosed
EP-3827814-B1 OPHTHALMIC FORMULATIONS DOMPE FARM SPA (IT) 2025-12-17 EP disclosed
US-20250354996-A1 SIGNAL AMPLIFICATION AND MULTIPLEXING USING MASS TAGS FOR IA-LC-MS/ MS BASED ASSAYS GENENTECH, INC. (US) 2025-11-20 US disclosed
US-20250352677-A1 METHODS AND KITS FOR PREPARING RADIONUCLIDE COMPLEXES THERAGNOSTICS LTD (GB) 2025-11-20 US disclosed
WO-2025233688-A1 MICROPLATE-BASED ELECTROPHORESIS SYSTEM AXOR BIOSYSTEMS INC. (US) 2025-11-13 WO disclosed
WO-2025222280-A1 STABLE TOPICAL COMPOSITIONS FOR TREATING ATROPHIC VAGINITIS JASTLABS CORPORATION (CA) 2025-10-30 WO disclosed
WO-2025222268-A1 TOPICAL COMPOSITIONS AND METHODS FOR TREATING ATROPHIC VAGINITIS JASTLABS CORPORATION (CA) 2025-10-30 WO disclosed
US-20250325679-A1 COMPOSITIONS AND METHODS OF TREATMENT FOR SEVERE HYPERTRIGLYCERIDEMIA 89BIO INC. (US) 2025-10-23 US disclosed
US-12447192-B1 Stable cannabinoid-comprising nanoemulsions and methods of using the same SGN NANOPHARMA INC. (US) 2025-10-21 US disclosed
EP-4619755-A1 SIGNAL AMPLIFICATION AND MULTIPLEXING USING MASS TAGS FOR IA-LC-MS/MS BASED ASSAYS Genentech, Inc. (US) 2025-09-24 EP disclosed
US-12411103-B2 Electrode, method for manufacturing electrode, ion sensor, in-vivo component measuring device, and in-vivo component measuring method SYSMEX CORPORATION (JP) 2025-09-09 US disclosed
US-20250246685-A1 FLAME-RETARDANT NON-AQUEOUS ELECTROLYTIC SOLUTION AND SECONDARY BATTERY USING SAME KYOTO UNIVERSITY (JP) 2025-07-31 US disclosed
US-12371521-B2 Photosensitive composition, hologram recording medium using the same, hologram optical element, and method of forming hologram diffraction grating Sony Group Corporation (JP) 2025-07-29 US disclosed
US-12350314-B2 Liquid formulations comprising mutant FGF-21 peptide pegylated conjugates 89BIO, INC. (US) 2025-07-08 US disclosed
EP-4577563-A2 METHODS OF TREATMENT OF NASH USING MUTANT FGF-21 PEPTIDE CONJUGATES 89Bio, Inc. (US) 2025-07-02 EP disclosed
US-12345718-B2 Method for determining the haemoglobin content of an erythroid cell UNIVERSITÉ PARIS EST CRÉTEIL VAL DE MARNE (FR) 2025-07-01 US disclosed
CN-120202411-A Signal amplification and multiplexing for IA-LC-MS/MS based assays using mass labels 基因泰克公司 2025-06-24 CN disclosed
US-20250170249-A1 COMPOSITIONS AND METHODS OF TREATMENT FOR SEVERE HYPERTRIGLYCERIDEMIA 89BIO, INC. (US) 2025-05-29 US disclosed
US-20250161331-A1 ANTI-INFLAMMATORY DRUG-CANNABINOID-COMPRISING NANOEMULSIONS AND METHODS OF USING THE SAME SGN NANOPHARMA INC. (US) 2025-05-22 US disclosed
EP-4548771-A1 METHOD FOR PRODUCING PROCESSED PLANT PROTEIN-CONTAINING COMPOSITION Amano Enzyme Inc. (JP) 2025-05-07 EP disclosed
CN-119925276-A CRAC inhibitor freeze-dried powder preparation based on tromethamine phosphate salt prodrug and preparation method thereof 天津辰欣药物研究有限公司 2025-05-06 CN disclosed
EP-4543479-A1 COMPOSITIONS AND METHODS OF TREATMENT FOR SEVERE HYPERTRIGLYCERIDEMIA 89Bio, Inc. (US) 2025-04-30 EP disclosed
CN-119816317-A Compositions and methods for treating severe hypertriglyceridemia 89生物公司 2025-04-11 CN disclosed
US-20250108136-A1 METHODS AND KITS FOR PREPARING RADIONUCLIDE COMPLEXES THERAGNOSTICS LIMITED (GB) 2025-04-03 US disclosed
US-20250082615-A1 SOLID DISPERSION OF RIFAXIMIN LUPIN LIMITED (IN) 2025-03-13 US disclosed
WO-2025043155-A1 THERAPEUTIC REGIMENS AND METHODS OF TREATMENT OF NASH USING MUTANT FGF-21 PEPTIDE CONJUGATES 89BIO, INC. (US) 2025-02-27 WO disclosed
EP-4507722-A1 NANOEMULSION UNIVERSAL INFLUENZA VACCINE Bluewillow Biologics, Inc. (US) 2025-02-19 EP disclosed
CN-119451579-A Method for producing processed plant protein-containing composition 天野酶制品株式会社 2025-02-14 CN disclosed
CN-119367551-A Liquid formulations comprising mutant FGF-21 peptide pegylated conjugates 89生物公司 2025-01-28 CN disclosed
US-20250002528-A1 SWITCHABLE POLYPEPTIDE AND ITS USE FOR GENTLE AFFINITY PURIFICATION OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2025-01-02 US disclosed
EP-4482485-A1 ANTI-INFLAMMATORY DRUG-CANNABINOID-COMPRISING NANOEMULSIONS AND METHODS OF USING THE SAME SGN Nanopharma Inc. (US) 2025-01-01 EP disclosed
CN-112472796-B Methods of diagnosing or treating neurological disorders using P75ECD and/or P75 上海澳宗生物科技有限公司 2024-12-24 CN disclosed
US-20240415929-A1 FORMULATIONS COMPRISING A TRIS BUFFER AND A PROTEIN AMGEN INC. (US) 2024-12-19 US disclosed
EP-3535589-B1 METHOD FOR DETERMINING THE HEMOGLOBIN F CONTENT OF AN ERYTHROID CELL UNIV PARIS VAL DE MARNE (FR) 2024-12-04 EP disclosed
CN-117120070-B Liquid formulations comprising mutant FGF-21 peptide pegylated conjugates 89生物公司 2024-11-15 CN disclosed
EP-4441079-A1 SWITCHABLE POLYPEPTIDE AND ITS USE FOR GENTLE AFFINITY PURIFICATION Oxford University Innovation Limited (GB) 2024-10-09 EP disclosed
EP-4058059-B1 NANOEMULSION COMPOSITIONS FOR TREATING AEROALLERGEN ASSOCIATED ALLERGY AND INFLAMMATION UNIV MICHIGAN REGENTS (US) 2024-10-09 EP disclosed
US-12109277-B2 Methods and kits for preparing radionuclide complexes THERAGNOSTICS LIMITED (GB) 2024-10-08 US disclosed
CN-114870061-B Air spray based on virus blocking agent and application thereof 康码(上海)生物科技有限公司 2024-09-24 CN disclosed
US-12098168-B2 XylR mutant for improved xylose utilization or improved co-utilization of glucose and xylose preliminary GENOMATICA, INC. (US) 2024-09-24 US disclosed
US-20240307492-A1 LIQUID FORMULATIONS COMPRISING MUTANT FGF-21 PEPTIDE PEGYLATED CONJUGATES 89BIO, INC. (US) 2024-09-19 US disclosed
EP-4428982-A1 FLAME-RETARDANT NON-AQUEOUS ELECTROLYTIC SOLUTION AND SECONDARY BATTERY USING SAME Kyoto University (JP) 2024-09-11 EP disclosed
US-20240252620-A1 COMBINED AGONIST ADJUVANT FOR CORONAVIRUS VACCINE THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2024-08-01 US disclosed
CN-118406674-A DNA repair enzyme extraction method 杭州合碳创物科技有限公司 2024-07-30 CN disclosed
CN-118389457-A Peptide ligase and use thereof 牛津大学创新有限公司 2024-07-26 CN disclosed
US-12036293-B2 Methods and kits for preparing radionuclide complexes THERAGNOSTICS LIMITED (GB) 2024-07-16 US disclosed
US-12036284-B2 Compositions and methods of treatment for severe hypertriglyceridemia 89BIO, INC. (US) 2024-07-16 US disclosed
US-12029708-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2024-07-09 US disclosed
US-20240165277-A1 METHODS AND KITS FOR PREPARING RADIONUCLIDE COMPLEXES THERAGNOSTICS LIMITED (GB) 2024-05-23 US disclosed
WO-2024108178-A1 SIGNAL AMPLIFICATION AND MULTIPLEXING USING MASS TAGS FOR IA-LC-MS/MS BASED ASSAYS GENENTECH, INC. (US) 2024-05-23 WO disclosed
CN-110582566-B Peptide ligase and use thereof 牛津大学创新有限公司 2024-05-10 CN disclosed
WO-2024044680-A2 METHODS OF TREATMENT OF NASH USING MUTANT FGF-21 PEPTIDE CONJUGATES 89BIO, INC. (US) 2024-02-29 WO disclosed
US-20240058434-A1 NANOEMULSION UNIVERSAL INFLUENZA VACCINE BLUEWILLOW BIOLOGICS, INC. (US) 2024-02-22 US disclosed
EP-3843701-B1 BACTERIOCINS TO IMPROVE VAGINAL COLONIZATION OF HYDROGEN PEROXIDE PRODUCING LACTOBACILLUS FOR FEMALE REPRODUCTIVE HEALTH OSEL INC (US) 2024-02-21 EP disclosed
US-20240042016-A1 NANOEMULSION VACCINE COMPOSITIONS AND METHODS FOR SUPPRESSING REACTIVITY TO MULTIPLE FOOD ALLERGENS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2024-02-08 US disclosed
EP-4304625-A1 LIQUID FORMULATIONS COMPRISING MUTANT FGF-21 PEPTIDE PEGYLATED CONJUGATES 89Bio, Inc. (US) 2024-01-17 EP disclosed
WO-2024010056-A1 SECONDARY BATTERY ダイキン工業株式会社 2024-01-11 WO disclosed
WO-2024010057-A1 NEGATIVE ELECTRODE, BATTERY, AND METHOD FOR COVERING BATTERY MATERIAL ダイキン工業株式会社 2024-01-11 WO disclosed
CN-110545845-B anti-CD 33 antibody agents 纪念斯隆凯特琳癌症中心 2024-01-05 CN disclosed
WO-2024004947-A1 METHOD FOR PRODUCING PROCESSED PLANT PROTEIN-CONTAINING COMPOSITION 天野エンザイム株式会社 2024-01-04 WO disclosed
WO-2023249003-A1 SURFACE TREATMENT AGENT FOR ELECTRODE MATERIAL, POSITIVE ELECTRODE ACTIVE MATERIAL, CURRENT COLLECTOR FOIL, NEGATIVE ELECTRODE ACTIVE MATERIAL, CONDUCTIVE AID, ELECTRODE, BATTERY, METHOD FOR MANUFACTURING POSITIVE ELECTRODE ACTIVE MATERIAL, METHOD FOR MANUFACTURING CURRENT COLLECTOR FOIL, METHOD FOR MANUFACTURING NEGATIVE ELECTRODE ACTIVE MATERIAL, METHOD FOR MANUFACTURING CONDUCTIVE AID, AND METHOD FOR MANUFACTURING ELECTRODE ダイキン工業株式会社 2023-12-28 WO disclosed
US-20230414768-A1 COMPOSITIONS AND METHODS OF TREATMENT FOR SEVERE HYPERTRIGLYCERIDEMIA 89BIO, INC. (US) 2023-12-28 US disclosed
WO-2023250493-A1 COMPOSITIONS AND METHODS OF TREATMENT FOR SEVERE HYPERTRIGLYCERIDEMIA 89BIO INC. (US) 2023-12-28 WO disclosed
US-11850275-B2 Liquid formulations comprising mutant FGF-21 peptide pegylated conjugates 89BIO, INC. (US) 2023-12-26 US disclosed
WO-2023232096-A1 AIR SPRAY BASED ON VIRUS BLOCKING AGENT, AND USE THEREOF 康码(上海)生物科技有限公司 2023-12-07 WO disclosed
US-11826436-B2 Methods and kits for preparing radionuclide complexes THERAGNOSTICS LIMITED (GB) 2023-11-28 US disclosed
CN-117120070-A Liquid formulations comprising mutant FGF-21 peptide pegylated conjugates 89生物公司 2023-11-24 CN disclosed
CN-117100874-A Nanoparticle, preparation and application thereof, eye disease medicine comprising nanoparticle and preparation thereof 苏州维益生物科技有限公司 2023-11-24 CN disclosed
EP-2735562-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS INC (US) 2023-11-15 EP disclosed
EP-4271406-A1 NANOEMULSION VACCINE COMPOSITIONS AND METHODS FOR SUPPRESSING REACTIVITY TO MULTIPLE FOOD ALLERGENS The Regents of The University of Michigan (US) 2023-11-08 EP disclosed
US-20230338471-A1 LIQUID FORMULATIONS COMPRISING MUTANT FGF-21 PEPTIDE PEGYLATED CONJUGATES 89BIO, INC. (US) 2023-10-26 US disclosed
US-20230330202-A1 NANOEMULSION AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-10-19 US disclosed
WO-2023200764-A1 NANOEMULSION UNIVERSAL INFLUENZA VACCINE BLUEWILLOW BIOLOGICS, INC. (US) 2023-10-19 WO disclosed
US-20230288429-A1 REAL TIME ELECTRONIC CELL SENSING SYSTEMS AND APPLICATIONS FOR CELL-BASED ASSAYS AGILENT TECHNOLOGIES, INC. 2023-09-14 US disclosed
WO-2023133143-A1 INTRANASAL POLYSACCHARIDE CONJUGATE NANOEMULSION VACCINES AND METHODS OF USING THE SAME BLUEWILLOW BIOLOGICS, INC. (US) 2023-07-13 WO disclosed
US-20230218549-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. 2023-07-13 US disclosed
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US-20230145666-A1 REAL TIME ELECTRONIC CELL SENSING SYSTEMS AND APPLICATIONS FOR CELL-BASED ASSAYS AGILENT TECHNOLOGIES, INC. 2023-05-11 US disclosed
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US-11604197-B2 Real time electronic cell sensing systems and applications for cell-based assays AGILENT TECHNOLOGIES, INC. (US) 2023-03-14 US disclosed
US-11596669-B2 Liquid formulations comprising mutant FGF-21 peptide pegylated conjugates 89BIO, INC. (US) 2023-03-07 US disclosed
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US-20230011185-A1 LAMINATE, METHOD FOR MANUFACTURING LAMINATE, AND METHOD FOR MANUFACTURING SEMICONDUCTOR SUBSTRATE TOKYO OHKA KOGYO CO., LTD. (JP) 2023-01-12 US disclosed
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US-20220387316-A1 NANOEMULSION COMPOSITIONS FOR TREATING AEROALLERGEN ASSOCIATED ALLERGY AND INFLAMMATION NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-12-08 US disclosed
WO-2022251406-A1 COMBINED AGONIST ADJUVANT FOR CORONAVIRUS VACCINE THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2022-12-01 WO disclosed
EP-4089406-A1 ELECTRODE, ELECTRODE MANUFACTURING METHOD, ION SENSOR, IN VIVO COMPONENT MEASURING DEVICE, AND IN VIVO COMPONENT MEASURING METHOD SYSMEX CORPORATION (JP) 2022-11-16 EP disclosed
US-20220339304-A1 METHODS AND KITS FOR PREPARING RADIONUCLIDE COMPLEXES THERAGNOSTICS LIMITED (GB) 2022-10-27 US disclosed
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CN-115181616-A Nucleic acid scavenger based on virus blocking agent and application thereof 康码(上海)生物科技有限公司 2022-10-14 CN disclosed
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CN-111635752-B Gold nanorod/DNA/carbon dot nano hybrid material and preparation method and application thereof 中国科学院理化技术研究所 2022-09-23 CN disclosed
US-20220296678-A1 LIQUID FORMULATIONS COMPRISING MUTANT FGF-21 PEPTIDE PEGYLATED CONJUGATES 89BIO, INC. (US) 2022-09-22 US disclosed
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US-11446261-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2022-09-20 US disclosed
WO-2022192601-A1 LIQUID FORMULATIONS COMPRISING MUTANT FGF-21 PEPTIDE PEGYLATED CONJUGATES 89BIO, INC. (US) 2022-09-15 WO disclosed
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CN-114929271-A Nanoemulsion compositions for the treatment of aeroallergen-related allergies and inflammation 密歇根大学董事会 2022-08-19 CN disclosed
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EP-4043961-A1 2K SYSTEM Xetos AG (DE) 2022-08-17 EP disclosed
EP-4043962-A1 PHOTOPOLYMERIZABLE COMPOSITION Xetos AG (DE) 2022-08-17 EP disclosed
CN-114870061-A Air spray based on virus blocking agent and application thereof 康码(上海)生物科技有限公司 2022-08-09 CN disclosed
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WO-2022156908-A1 METHOD FOR PREPARING A LYOPHILIZED COMPOSITION VRIJE UNIVERSITEIT BRUSSEL (BE) 2022-07-28 WO disclosed
WO-2022156907-A1 METHOD AND KIT FOR LABELING A BIOMOLECULE WITH ONE OR MORE DETECTABLE LABELS, INCLUDING A RADIOLABEL VRIJE UNIVERSITEIT BRUSSEL (BE) 2022-07-28 WO disclosed
WO-2022157373-A1 COMPOSITIONS AND KITS FOR IN VIVO IMAGING OF CARDIAC SARCOIDOSIS VRIJE UNIVERSITEIT BRUSSEL (BE) 2022-07-28 WO disclosed
WO-2022153616-A1 HOLOGRAM RECORDING MEDIUM, HOLOGRAM OPTICAL ELEMENT, OPTICAL DEVICE, OPTICAL COMPONENT, AND METHOD FOR FORMING HOLOGRAM DIFFRACTION GRATING ソニーグループ株式会社 2022-07-21 WO disclosed
WO-2022145446-A1 CHLORINATED POLYOLEFIN COMPOSITION 昭和電工株式会社 2022-07-07 WO disclosed
WO-2022145447-A1 CHLORINATED-POLYOLEFIN COMPOSITION 昭和電工株式会社 2022-07-07 WO disclosed
WO-2022147173-A1 NANOEMULSION VACCINE COMPOSITIONS AND METHODS FOR SUPPRESSING REACTIVITY TO MULTIPLE FOOD ALLERGENS THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2022-07-07 WO disclosed
WO-2022138893-A1 NONAQUEOUS ELECTROLYTIC SOLUTION AND NONAQUEOUS ELECTROLYTIC SOLUTION BATTERY MUアイオニックソリューションズ株式会社 2022-06-30 WO disclosed
WO-2022124382-A1 PROVIDED ARE A NEGATIVE ELECTRODE MATERIAL IN A CONTAINER, A TRANSPORTATION METHOD FOR NEGATIVE ELECTRODE MATERIAL, A NEGATIVE ELECTRODE MATERIAL STORAGE CONTAINER, A STORAGE METHOD FOR NEGATIVE ELECTRODE MATERIAL, AND A MANUFACTURING METHOD FOR NEGATIVE ELECTRODE MATERIAL. 昭和電工マテリアルズ株式会社 2022-06-16 WO disclosed
WO-2022123701-A1 PACKED NEGATIVE ELECTRODE MATERIAL, NEGATIVE ELECTRODE MATERIAL TRANSPORTATION METHOD, NEGATIVE ELECTRODE MATERIAL STORAGE CONTAINER, AND NEGATIVE ELECTRODE MATERIAL STORAGE METHOD 昭和電工マテリアルズ株式会社 2022-06-16 WO disclosed
EP-2417249-B1 DNA-CELL CONJUGATES UNIV CALIFORNIA (US) 2022-06-08 EP disclosed
WO-2022107255-A1 LITHIUM ION SECONDARY BATTERY AND SEPARATION MEMBRANE 昭和電工マテリアルズ株式会社 2022-05-27 WO disclosed
WO-2022102623-A1 METHOD AND KIT FOR TRANSPARENTIZING BIOLOGICAL MATERIAL 住友化学株式会社 2022-05-19 WO disclosed
EP-3998289-A1 PHOTOSENSITIVE COMPOSITION AND A HOLOGRAM STORAGE MEDIUM USING SAME, HOLOGRAM OPTICAL ELEMENT, AND HOLOGRAM DIFFRACTION GRATING FORMING METHOD Sony Group Corporation (JP) 2022-05-18 EP disclosed
US-20220105172-A1 HERPES SIMPLEX VIRUS NANOEMULSION VACCINES AND METHODS OF USING THE SAME BLUEWILLOW BIOLOGICS, INC. (US) 2022-04-07 US disclosed
WO-2022054737-A1 FLUORINATED CARBOXYLIC ACID SALT COMPOUND ダイキン工業株式会社 2022-03-17 WO disclosed
WO-2022045282-A1 POLYMERIZATION CATALYST COMPOSITION, METHOD FOR PRODUCING POLYMERIZATION CATALYST COMPOSITION, AND METHOD FOR PRODUCING CONJUGATED DIENE POLYMER DIC株式会社 2022-03-03 WO disclosed
WO-2022045059-A1 RESIN COMPOSITION, CURED PRODUCT, MULTILAYER BODY, METHOD FOR PRODUCING CURED PRODUCT, AND SEMICONDUCTOR DEVICE 富士フイルム株式会社 2022-03-03 WO disclosed
EP-3354650-B1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMA (US) 2022-02-16 EP disclosed
US-11231427-B2 Method for determining the haemoglobin F content of an erythroid cell UNIVERSITE PARIS EST CRETEIL VAL DE MARNE (FR) 2022-01-25 US disclosed
US-20210353713-A1 FORMULATIONS COMPRISING A TRIS BUFFER AND A PROTEIN AMGEN INC. (US) 2021-11-18 US disclosed
US-11166924-B2 N-methyl-d-aspartate receptor allosteric modulators and methods for their use QINGDAO PRIMEDICINE PHARMACEUTICAL COMPANY, LTD. (CN) 2021-11-09 US disclosed
EP-3010501-B1 ESTROGEN RECEPTOR MODULATOR AND USES THEREOF SERAGON PHARMACEUTICALS INC (US) 2021-11-03 EP disclosed
EP-3610005-B1 PEPTIDE LIGASE AND USE THEREOF UNIV OXFORD INNOVATION LTD (GB) 2021-09-29 EP disclosed
US-11120993-B2 Diffusing agent composition and method of manufacturing semiconductor substrate TOKYO OHKA KOGYO CO., LTD. (JP) 2021-09-14 US disclosed
US-20210275628-A1 BACTERIOCINS TO IMPROVE VAGINAL COLONIZATION OF HYDROGEN PEROXIDE PRODUCING LACTOBACILLUS FOR FEMALE REPRODUCTIVE HEALTH OSEL, INC. 2021-09-09 US disclosed
US-20210275557-A1 MODIFIED AMINOGLYCOSIDE COMPOUNDS AND USES THEREOF IN DISABLING BACTERIAL RIBOSOME TECHNION RESEARCH & DEVELOPMENT FOUNDATION LIMITED (IL) 2021-09-09 US disclosed
CN-106794222-B Methods of diagnosing or treating neurological disorders using P75ECD and/or P75 苏州澳宗生物科技有限公司 2021-08-24 CN disclosed
CN-113274355-A Rifaximin solid dispersion 鲁平有限公司 2021-08-20 CN disclosed
WO-2021140933-A1 ELECTRODE, ELECTRODE MANUFACTURING METHOD, ION SENSOR, IN VIVO COMPONENT MEASURING DEVICE, AND IN VIVO COMPONENT MEASURING METHOD シスメックス株式会社 2021-07-15 WO disclosed
EP-3843701-A2 BACTERIOCINS TO IMPROVE VAGINAL COLONIZATION OF HYDROGEN PEROXIDE PRODUCING LACTOBACILLUS FOR FEMALE REPRODUCTIVE HEALTH Osel, Inc. (US) 2021-07-07 EP disclosed
US-11046746-B2 Method of treatment of cerebral amyloid angiopathy with P75ECD peptide and/or P75ECD-FC fusion protein SUZHOU AUZONE BIOLOGICAL TECHNOLOGY CO., LTD 2021-06-29 US disclosed
CN-110218778-B PCR reaction system, reagent, kit and PCR method 珠海宝锐生物科技有限公司 2021-05-28 CN disclosed
WO-2021095574-A1 ELECTRODE AND ELECTROCHEMICAL DEVICE ダイキン工業株式会社 2021-05-20 WO disclosed
US-20210138094-A1 METHODS AND KITS FOR PREPARING RADIONUCLIDE COMPLEXES THERAGNOSTICS LIMITED (GB) 2021-05-13 US disclosed
CN-112638970-A Polyurethane resin composition and method for insulating building 株式会社日本雅克 2021-04-09 CN disclosed
US-10961232-B2 Substituted pyrazines as ATR kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2021-03-30 US disclosed
CN-112472796-A Methods of diagnosing or treating neurological disorders using P75ECD and/or P75 苏州澳宗生物科技有限公司 2021-03-12 CN disclosed
WO-2021020020-A1 ADDITIVE COMPOSITION 株式会社ADEKA 2021-02-04 WO disclosed
US-10889622-B2 Peptide ligase and use thereof OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2021-01-12 US disclosed
EP-3303326-B1 HETEROCYCLIC ESTROGEN RECEPTOR MODULATORS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2020-12-16 EP disclosed
US-20200375959-A1 SOLID DISPERSION OF RIFAXIMIN LUPIN LIMITED (IN) 2020-12-03 US disclosed
US-20200373162-A1 DIFFUSING AGENT COMPOSITION AND METHOD OF MANUFACTURING SEMICONDUCTOR SUBSTRATE TOKYO OHKA KOGYO CO., LTD. (JP) 2020-11-26 US disclosed
EP-3273982-B1 METHOD OF DIAGNOSIS OR TREATMENT OF NEUROLOGICAL DISORDERS WITH P75ECD AND/OR P75 SUZHOU AUZONE BIOLOGICAL TECH CO LTD (CN) 2020-11-18 EP disclosed
WO-2020218321-A1 WATER-SOLUBLE FILM AND PACKAGING 株式会社クラレ 2020-10-29 WO disclosed
US-10809222-B2 Opioid detection based on high quality graphene transistor arrays and a synthetic mu receptor THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2020-10-20 US disclosed
WO-2020184650-A1 CURABLE COMPOSITION, CURED PRODUCT, OPTICAL MEMBER, LENS, AND METHOD FOR MANUFACTURING OPTICAL MEMBER 富士フイルム株式会社 2020-09-17 WO disclosed
CN-111635752-A Gold nanorod/DNA/carbon dot nano hybrid material and preparation method and application thereof 中国科学院理化技术研究所 2020-09-08 CN disclosed
US-10716770-B2 Nicotinic receptor non-competitive antagonists CATALYST BIOSCIENCES, INC. (US) 2020-07-21 US disclosed
EP-3653733-A1 METHODS AND COMPOSITIONS FOR DETERMINING RESISTANCE TO ANDROGEN RECEPTOR THERAPY Aragon Pharmaceuticals, Inc. (US) 2020-05-20 EP disclosed
US-20200115422-A1 PEPTIDE LIGASE AND USE THEREOF OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2020-04-16 US disclosed
EP-3268337-B1 METHODS AND KITS FOR PREPARING RADIONUCLIDE COMPLEXES THERAGNOSTICS LTD (GB) 2020-04-01 EP disclosed
WO-2020047203-A2 BACTERIOCINS TO IMPROVE VAGINAL COLONIZATION OF HYDROGEN PEROXIDE PRODUCING LACTOBACILLUS FOR FEMALE REPRODUCTIVE HEALTH OSEL, INC. (US) 2020-03-05 WO disclosed
US-20200062719-A1 Application of Imidazopyridine Derivatives in Regenerative Medicine UNIVERSITY OF HEIDELBERG (DE) 2020-02-27 US disclosed
CN-107438615-B Method and kit for preparing radionuclide complexes 施拉格诺斯迪克斯有限公司 2020-02-21 CN disclosed
EP-3611256-A1 APPLICATION OF IMIDAZOPYRIDINE DERIVATIVES IN REGENERATIVE MEDICINE Universität Heidelberg (DE) 2020-02-19 EP disclosed
EP-3610005-A1 PEPTIDE LIGASE AND USE THEREOF Oxford University Innovation Limited (GB) 2020-02-19 EP disclosed
US-10549259-B2 Carbide derived carbon for use in chemical scrubbers BAE SYSTEMS INFORMATION AND ELECTRONIC SYSTEMS INTEGRATION INC. (US) 2020-02-04 US disclosed
CN-110582566-A Peptide ligase and uses thereof 牛津大学创新有限公司 2019-12-17 CN disclosed
CN-110545845-A anti-CD 33 antibody agents MEMORIAL SLOAN KETTERING CANCER CENTER 2019-12-06 CN disclosed
EP-2734512-B1 METHODS FOR SELECTIVE OXIDATION OF ALPHA TOCOTRIENOL IN THE PRESENCE OF NON-ALPHA TOCOTRIENOLS BIOELECTRON TECH CORP (US) 2019-11-20 EP disclosed
US-10479784-B2 Substituted pyrazin-2-amines as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2019-11-19 US disclosed
CN-107486037-B A kind of PVDF/PDA composite membrane with super hydrophilicity 福州大学 2019-11-12 CN disclosed
EP-2877599-B1 METHODS AND COMPOSITIONS FOR DETERMINING RESISTANCE TO ANDROGEN RECEPTOR THERAPY ARAGON PHARMACEUTICALS INC (US) 2019-10-23 EP disclosed
WO-2019189413-A1 NONAQUEOUS ELECTROLYTE SOLUTION AND ENERGY DEVICE USING SAME 三菱ケミカル株式会社 2019-10-03 WO disclosed
WO-2019188207-A1 ELECTROLYTE SOLUTION, ELECTROCHEMICAL DEVICE, LITHIUM ION SECONDARY BATTERY, MODULE AND COMPOUND ダイキン工業株式会社 2019-10-03 WO disclosed
WO-2019189414-A1 NONAQUEOUS ELECTROLYTE SOLUTION AND ELECTRICITY STORAGE DEVICE USING SAME 三菱ケミカル株式会社 2019-10-03 WO disclosed
WO-2019181240-A1 ELECTROLYTIC SOLUTION, ELECTROCHEMICAL DEVICE, LITHIUM ION SECONDARY BATTERY, AND MODULE ダイキン工業株式会社 2019-09-26 WO disclosed
EP-3535589-A1 METHOD FOR DETERMINING THE HAEMOGLOBIN F CONTENT OF AN ERYTHROID CELL Université Paris-Est Créteil Val de Marne (FR) 2019-09-11 EP disclosed
US-20190254991-A1 Nicotinic Receptor Non-Competitive Antagonists CATALYST BIOSCIENCES INC (US) 2019-08-22 US disclosed
CN-107353304-B Phosphoric acid safe ground azoles amine trishydroxymethylaminomethane salt and its crystal form A, preparation method and application 浙江普洛得邦制药有限公司 2019-08-13 CN disclosed
WO-2019150823-A1 COMPOSITION, FILM, LAMINATE STRUCTURE, LIGHT-EMITTING DEVICE, AND DISPLAY 住友化学株式会社 2019-08-08 WO disclosed
WO-2019150896-A1 ELECTROLYTE, ELECTROCHEMICAL DEVICE, LITHIUM ION SECONDARY BATTERY, AND MODULE ダイキン工業株式会社 2019-08-08 WO disclosed
WO-2019150895-A1 ELECTROLYTE, ELECTROCHEMICAL DEVICE, LITHIUM ION SECONDARY BATTERY, AND MODULE ダイキン工業株式会社 2019-08-08 WO disclosed
EP-3515427-A2 N-METHYL-D-ASPARTATE RECEPTOR ALLOSTERIC MODULATORS AND METHODS FOR THEIR USE Qingdao Primedicine Pharmaceutical Co., Ltd (CN) 2019-07-31 EP disclosed
US-20190216753-A1 N-METHYL-D-ASPARTATE RECEPTOR ALLOSTERIC MODULATORS AND METHODS FOR THEIR USE QINGDAO PRIMEDICINE PHARMACEUTICAL COMPANY, LTD. (CN) 2019-07-18 US disclosed
CN-109996539-A N-methyl-D-aspartate receptor allosteric modulators and its application method 青岛普美圣医药科技有限公司 2019-07-09 CN disclosed
EP-2791133-B1 FLUORINATED ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS INC (US) 2019-04-17 EP disclosed
US-10258582-B2 Nicotinic receptor non-competitive antagonists CATALYST BIOSCIENCES, INC. (US) 2019-04-16 US disclosed
US-10227334-B2 Estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2019-03-12 US disclosed
CN-107414069-B Silver nanoparticle disk, preparation method and Gin Nanometer globoid and assembly using its preparation 国家纳米科学中心 2019-03-12 CN disclosed
US-20190047995-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED 2019-02-14 US disclosed
US-10202325-B2 Methods for selective oxidation of alpha tocotrienol in the presence of non-alpha tocotrienols BIOELECTRON TECHNOLOGY CORPORATION (US) 2019-02-12 US disclosed
CN-105451735-B azetidine estrogen receptor modulators and uses thereof 西拉根制药公司 2019-01-11 CN disclosed
CN-105324115-B estrogen receptor modulators and uses thereof 赛拉根医药股份有限公司 2019-01-04 CN disclosed
CN-109071482-A Carry the flavonoids type compound of O- rhamnopyranosyl residue 汉堡大学 2018-12-21 CN disclosed
CN-109072271-A The method for being used to prepare rhamnopyranosyl flavonoids 汉堡大学 2018-12-21 CN disclosed
US-10151697-B2 Two-color fluorescence localization super-resolution biological microscopy method and system SHENZHEN NANOBIOIMAGING LIMITED (CN) 2018-12-11 US disclosed
EP-3010502-B1 AZETIDINE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS INC (US) 2018-11-21 EP disclosed
EP-2493456-B1 SOLID DISPERSION OF RIFAXIMIN LUPIN LTD (IN) 2018-11-21 EP disclosed
US-20180319730-A1 METHODS FOR SELECTIVE OXIDATION OF ALPHA TOCOTRIENOL IN THE PRESENCE OF NON-ALPHA TOCOTRIENOLS BIOELECTRON TECHNOLOGY CORPORATION (US) 2018-11-08 US disclosed
WO-2018189517-A1 PEPTIDE LIGASE AND USE THEREOF OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2018-10-18 WO disclosed
EP-2828243-B1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS INC (US) 2018-10-17 EP disclosed
US-10100308-B2 Method for selectively inhibiting ACAT1 in the treatment of neurodegenerative diseases TRUSTEES OF DARTMOUTH COLLEGE (US) 2018-10-16 US disclosed
US-20180287146-A1 LITHIUM POWDER, LITHIUM ION SECONDARY BATTERY NEGATIVE ELECTRODE USING THE SAME, AND LITHIUM ION SECONDARY BATTERY USING THE LITHIUM ION SECONDARY BATTERY NEGATIVE ELECTRODE TDK CORPORATION (JP) 2018-10-04 US disclosed
US-20180271806-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS CATALYST BIOSCIENCES, INC. 2018-09-27 US disclosed
CN-105121413-B Polycyclic estrogen receptor modulators and uses thereof 赛拉根医药股份有限公司 2018-09-14 CN disclosed
US-10058534-B2 Benzothiophene derivatives and compositions thereof as selective estrogen receptor degraders NOVARTIS AG (CH) 2018-08-28 US disclosed
US-10053451-B2 Heterocyclic estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2018-08-21 US disclosed
EP-3357917-A1 ANDROGEN RECEPTOR MODULATORS AND USES THEREOF Aragon Pharmaceuticals, Inc. (US) 2018-08-08 EP disclosed
EP-3354650-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2018-08-01 EP disclosed
US-10029971-B2 Methods for selective oxidation of alpha tocotrienol in the presence of non-alpha tocotrienols BIOELECTRON TECHNOLOGY CORPORATION (US) 2018-07-24 US disclosed
US-10023556-B2 Androgen receptor modulators and uses thereof ARAGON PHARMACEUTICALS, INC. (US) 2018-07-17 US disclosed
EP-3337855-A1 FLAME-RETARDANT THERMOPLASTIC POLYURETHANE BASF SE (DE) 2018-06-27 EP disclosed
EP-3337850-A1 FLAME-RETARDANT THERMOPLASTIC POLYURETHANE BASF SE (DE) 2018-06-27 EP disclosed
US-20180170996-A1 METHOD OF DIAGNOSIS OR TREATMENT OF NEUROLOGICAL DISORDERS WITH P75ECD AND/OR P75 SHANGHAI AUZONE BIOLOGICAL TECHNOLOGY CO., LTD (CN) 2018-06-21 US disclosed
US-20180170922-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED 2018-06-21 US disclosed
US-9969970-B2 DNA-cell conjugates THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-05-15 US disclosed
CN-107907399-A A kind of preparation method for the mountant that can mark nucleus at the same time 遵义医学院 2018-04-13 CN disclosed
EP-3303326-A1 HETEROCYCLIC ESTROGEN RECEPTOR MODULATORS AND USES THEREOF H. Hoffnabb-La Roche Ag (CH) 2018-04-11 EP disclosed
US-20180092996-A1 METHODS AND KITS FOR PREPARING RADIONUCLIDE COMPLEXES THERAGNOSTICS LIMITED (GB) 2018-04-05 US disclosed
EP-2718309-B1 TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS KEYGENE NV (NL) 2018-04-04 EP disclosed
US-9932388-B2 Chromatographic process for producing high purity fibrinogen and thrombin HEMARUS THERAPEUTICS LIMITED (IN) 2018-04-03 US disclosed
EP-3124481-B1 ANDROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS INC (US) 2018-03-28 EP disclosed
CN-107735026-A The method for measuring tear component in ocular fluid samples 黛尔格诺斯蒂尔有限公司 2018-02-23 CN disclosed
EP-3273982-A1 METHOD OF DIAGNOSIS OR TREATMENT OF NEUROLOGICAL DISORDERS WITH P75ECD AND/OR P75 Fujian Tiantai Medical Technology Co. Ltd. (CN) 2018-01-31 EP disclosed
US-9873684-B2 Estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2018-01-23 US disclosed
EP-3268337-A1 METHODS AND KITS FOR PREPARING RADIONUCLIDE COMPLEXES Theragnostics Limited (GB) 2018-01-17 EP disclosed
US-9868704-B2 Estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2018-01-16 US disclosed
US-9855270-B2 Methods and compositions for modulating estrogen receptor mutants GENENTECH, INC. (US) 2018-01-02 US disclosed
CN-107531722-A Heterocyclic estrogen receptor modulators and uses thereof 豪夫迈·罗氏有限公司 2018-01-02 CN disclosed
CN-107486037-A A kind of PVDF/PDA composite membranes with super hydrophilicity 福州大学 2017-12-19 CN disclosed
CN-105008343-B Alternatively benzothiophene derivative of property ERs degradation agent and combinations thereof 诺华股份有限公司 2017-12-08 CN disclosed
EP-2376485-B1 PYRAZINE DERIVATIVES USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMA (US) 2017-12-06 EP disclosed
CN-107438615-A For preparing the method and kit of radionuclide complex compound 施拉格诺斯迪克斯有限公司 2017-12-05 CN disclosed
CN-107414069-A Silver nanoparticle disk, its preparation method and the Gin Nanometer globoid and assembly using its preparation 国家纳米科学中心 2017-12-01 CN disclosed
US-20170335293-A1 Modified Luciferases And Uses Thereof TARGETING SYSTEMS 2017-11-23 US disclosed
CN-107353304-A Phosphoric acid safe ground azoles amine trishydroxymethylaminomethane salt and its crystal formation A, preparation method and application 浙江普洛得邦制药有限公司 2017-11-17 CN disclosed
CN-104515760-B Two Colour Fluorescence positions super-resolution biology microscope method and system 深圳市纳观生物有限公司 2017-10-31 CN disclosed
US-20170297991-A1 METHODS FOR SELECTIVE OXIDATION OF ALPHA TOCOTRIENOL IN THE PRESENCE OF NON-ALPHA TOCOTRIENOLS PTC THERAPEUTICS, INC. 2017-10-19 US disclosed
US-20170292128-A1 METHOD FOR SELECTIVELY INHIBITING ACAT1 IN THE TREATMENT OF NEURODEGENERATIVE DISEASES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2017-10-12 US disclosed
US-20170284941-A1 TWO-COLOR FLUORESCENCE LOCALIZATION SUPER-RESOLUTION BIOLOGICAL MICROSCOPY METHOD AND SYSTEM NINGBO INVIEW INTELLIGENT TECHNOLOGY CO., LTD (CN) 2017-10-05 US disclosed
US-20170275273-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF GENENTECH, INC. (US) 2017-09-28 US disclosed
US-20170247713-A1 TRICHOME-SPECIFIC TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS KEYGENE N.V. (NL) 2017-08-31 US disclosed
EP-3205648-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF Seragon Pharmaceuticals, Inc. (US) 2017-08-16 EP disclosed
US-9732328-B2 Modified luciferases and uses thereof TARGETING SYSTEMS (US) 2017-08-15 US disclosed
CN-106983749-A Androgen receptor modifier and application thereof 亚拉冈制药公司 2017-07-28 CN disclosed
US-20170196840-A1 METHODS AND COMPOSITIONS FOR DETERMINING RESISTANCE TO ANDROGEN RECEPTOR THERAPY ARAGON PHARMACEUTICALS INC (US) 2017-07-13 US disclosed
US-9701674-B2 Substituted pyrazines as ATR kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-07-11 US disclosed
US-9689018-B2 Mixed cell diagnostic systems for detection of respiratory, herpes and enteric viruses DIAGNOSTIC HYBRIDS, INC. (US) 2017-06-27 US disclosed
CN-106831755-A Benzamide compound and its salt form and purposes 阿腾弩阿公司 2017-06-13 CN disclosed
US-9670264-B2 Water soluble G-protein coupled receptor THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2017-06-06 US disclosed
US-20170151204-A1 USE OF LEUKOTRIENE B4 IN COMBINATION WITH A TOLL-LIKE RECEPTOR LIGAND, A RIG-I-LIKE RECEPTOR LIGAND, OR A NOD-LIKE RECEPTOR LIGAND TO ENHANCE THE INNATE IMMUNE RESPONSE UNIVERSITé LAVAL (CA) 2017-06-01 US disclosed
CN-106794222-A Methods of diagnosing or treating neurological disorders using P75ECD and/or P75 福建天泰医药科技有限公司 2017-05-31 CN disclosed
US-9655880-B2 Azetidine estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2017-05-23 US disclosed
CN-103724322-B Androgen receptor modulators and uses thereof 亚拉冈制药公司 2017-05-03 CN disclosed
US-9617602-B2 Methods and compositions for determining resistance to androgen receptor therapy ARAGON PHARMACEUTICALS, INC. (US) 2017-04-11 US disclosed
EP-3150196-A1 PROCESS FOR THE PREPARATION OF UNILAMELLAR LIPOSOMAL COMPOSITION Sun Pharma Advanced Research Company Ltd (IN) 2017-04-05 EP disclosed
US-20170087089-A1 PROCESS FOR THE PREPARATION OF UNILAMELLAR LIPOSOMAL COMPOSITION SUN PHARMA ADVANCED RESEARCH COMPANY LTD (IN) 2017-03-30 US disclosed
CN-106518856-A Pyrazine derivatives useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2017-03-22 CN disclosed
US-9598473-B2 Trichome-specific transcription factor modulating terpene biosynthesis KEYGENE N.V. (NL) 2017-03-21 US disclosed
US-20170071878-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS CATALYST BIOSCIENCES INC (US) 2017-03-16 US disclosed
CN-103842563-B Protein exhibiting expression method 亲和生物科学公司 2017-03-15 CN disclosed
CN-106496210-A It is used as the compound of ATR kinase inhibitors 沃泰克斯药物股份有限公司 2017-03-15 CN disclosed
CN-106496209-A It is used as the compound of ATR kinase inhibitors 沃泰克斯药物股份有限公司 2017-03-15 CN disclosed
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EP-2824102-B1 Androgen receptor modulators and uses thereof ARAGON PHARMACEUTICALS INC (US) 2017-02-01 EP disclosed
EP-3116496-A1 METHODS AND COMPOSITIONS FOR MODULATING ESTROGEN RECEPTOR MUTANTS F. Hoffmann-La Roche AG (CH) 2017-01-18 EP disclosed
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CN-104114551-B Fluorinated estrogen receptor modulators and uses thereof 塞拉根制药公司 2017-01-18 CN disclosed
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US-9532974-B2 Nicotinic receptor non-competitive antagonists TARGACEPT, INC. (US) 2017-01-03 US disclosed
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US-20160367526-A1 AZETIDINE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF GENENTECH, INC. (US) 2016-12-22 US disclosed
US-20160355508-A1 POLYCYCLIC ESTROGEN RECEPTOR MODULATORS AND USES THEREOF GENENTECH, INC. (US) 2016-12-08 US disclosed
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US-20160347742-A1 HETEROCYCLIC ESTROGEN RECEPTOR MODULATORS AND USES THEREOF GENENTECH, INC. (US) 2016-12-01 US disclosed
EP-2431037-B1 (2S,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofuran-2-carboxamide, novel salt forms, and methods of use thereof ATTENUA INC (US) 2016-11-30 EP disclosed
CN-102300862-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2016-11-23 CN disclosed
US-9499538-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS, INC. (US) 2016-11-22 US disclosed
US-20160319238-A1 DNA-CELL CONJUGATES ENERGY, UNITED STATES DEPARTMENT OF 2016-11-03 US disclosed
US-9481664-B2 Androgen receptor modulators and uses thereof ARAGON PHARMACEUTICALS, INC. (US) 2016-11-01 US disclosed
US-20160311809-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2016-10-27 US disclosed
US-9475798-B2 Azetidine estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2016-10-25 US disclosed
US-20160297767-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF GENENTECH, INC. (US) 2016-10-13 US disclosed
EP-2465501-B1 Method for the preparation of (2S,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofuran-2-carboxamide ATTENUA INC (US) 2016-10-05 EP disclosed
WO-2016150403-A1 METHOD OF DIAGNOSIS OR TREATMENT OF NEUROLOGICAL DISORDERS WITH P75ECD AND/OR P75 FUJIAN TIANTAI MEDICAL TECHNOLOGY CO. LTD (CN) 2016-09-29 WO disclosed
WO-2016142702-A1 METHODS AND KITS FOR PREPARING RADIONUCLIDE COMPLEXES THERAGNOSTICS LIMITED (GB) 2016-09-15 WO disclosed
US-20160264944-A1 Modified Luciferases And Uses Thereof TARGETING SYSTEMS 2016-09-15 US disclosed
US-20160264617-A1 Integrated Approach to the Isolation and Purification of Antibodies ABBOTT LABORATORIES 2016-09-15 US disclosed
CN-102884057-B Androgen receptor modulators and uses thereof 亚拉冈制药公司 2016-09-14 CN disclosed
US-9399646-B2 Estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2016-07-26 US disclosed
US-9388414-B2 Method for selectively inhibiting ACAT1 in the treatment of neurodegenerative diseases TRUSTEES OF DARTMOUTH COLLEGE (US) 2016-07-12 US disclosed
US-9388413-B2 Method for selectively inhibiting ACAT1 in the treatment of neurodegenerative diseases TRUSTEES OF DARTMOUTH COLLEGE (US) 2016-07-12 US disclosed
EP-2809647-B1 MGLU 2/3 AGONISTS LILLY CO ELI (US) 2016-07-06 EP disclosed
US-9365557-B2 Substituted pyrazin-2-amines as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2016-06-14 US disclosed
WO-2016084097-A1 PROCESS FOR PRODUCING FIBRINOGEN AND THROMBIN HEMARUS THERAPEUTICS LTD. (IN) 2016-06-02 WO disclosed
US-9353401-B2 Multiplex assays with multiple luciferases reporters and uses thereof TARGETING SYSTEMS (US) 2016-05-31 US disclosed
EP-2721012-B1 BICYCLO(3.1.0)HEXANE-2,6-DICARBOXYLIC ACID DERIVATIVES AS MGLU2 RECEPTOR AGONIST LILLY CO ELI (US) 2016-05-25 EP disclosed
US-20160137719-A1 PROCESS FOR PRODUCING HIGH PURITY FIBRINOGEN AND THROMBIN FOR FIBRIN SEALANT ICHOR BIOLOGICS PRIVATE LIMITED (IN) 2016-05-19 US disclosed
US-20160123919-A1 OPIOID DETECTION BASED ON HIGH QUALITY GRAPHENE TRANSISTOR ARRAYS AND A SYNTHETIC MU RECEPTOR THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2016-05-05 US disclosed
US-9327036-B2 DNA-cell conjugates THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-05-03 US disclosed
US-20160102130-A1 WATER SOLUBLE G-PROTEIN COUPLED RECEPTOR THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2016-04-14 US disclosed
CN-105461736-A PHOSPHOINOSITIDE 3-KINASE INHIBITOR WITH A ZINC BINDING MOIETY CURIS INC 2016-04-06 CN disclosed
US-20160090377-A1 AZETIDINE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF GENENTECH, INC. (US) 2016-03-31 US disclosed
US-20160090378-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF GENENTECH, INC. (US) 2016-03-31 US disclosed
US-9296710-B2 Bicyclo (3.1.0) hexane-2, 6-dicarboxylic acid derivatives as mGlu2 receptor agonist ELI LILLY AND COMPANY (US) 2016-03-29 US disclosed
EP-2989440-A2 OPIOID DETECTION BASED ON HIGH QUALITY GRAPHENE TRANSISTOR ARRAYS AND A SYNTHETIC MU RECEPTOR The Trustees Of The University Of Pennsylvania (US) 2016-03-02 EP disclosed
EP-2970130-A1 POLYCYCLIC ESTROGEN RECEPTOR MODULATORS AND USES THEREOF Seragon Pharmaceuticals, Inc. (US) 2016-01-20 EP disclosed
US-20160008323-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS TARGACEPT INC (US) 2016-01-14 US disclosed
US-20160002138-A1 METHODS FOR SELECTIVE OXIDATION OF ALPHA TOCOTRIENOL IN THE PRESENCE OF NON-ALPHA TOCOTRIENOLS PTC THERAPEUTICS, INC. 2016-01-07 US disclosed
WO-2015184105-A1 METHOD FOR SELECTIVELY INHIBITING ACAT1 IN THE TREATMENT OF NEURODEGENERATIVE DISEASES TRUSTEES OF DARTMOUTH COLLEGE (US) 2015-12-03 WO disclosed
US-9193714-B2 Fluorinated estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS, INC. (US) 2015-11-24 US disclosed
US-9187460-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS, INC. (US) 2015-11-17 US disclosed
US-9162957-B2 Methods for oxidation of alpha tocotrienol in the presence of non-alpha tocotrienols EDISON PHARMACEUTICALS, INC. (US) 2015-10-20 US disclosed
US-20150258099-A1 METHODS AND COMPOSITIONS FOR MODULATING ESTROGEN RECEPTOR MUTANTS GENENTECH, INC. (US) 2015-09-17 US disclosed
WO-2015136017-A1 METHODS AND COMPOSITIONS FOR MODULATING ESTROGEN RECEPTOR MUTANTS F. HOFFMANN-LA ROCHE AG (CH) 2015-09-17 WO disclosed
US-20150252426-A1 METHODS AND COMPOSITIONS FOR DETERMINING RESISTANCE TO ANDROGEN RECEPTOR THERAPY ARAGON PHARMACEUTICALS, INC. 2015-09-10 US disclosed
US-9108944-B2 Androgen receptor modulators and uses thereof ARAGON PHARMACEUTICALS, INC. (US) 2015-08-18 US disclosed
CN-103464108-B A kind of golden palladium bimetallic satellite structure assembly and its preparation method and application STATE NANOMETER SCIENCE CENTER (CN) 2015-07-29 CN disclosed
US-9078871-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS, INC. (US) 2015-07-14 US disclosed
US-9081009-B2 Oxidized cardiolipin and uses to detect cardiolipin antibodies THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2015-07-14 US disclosed
US-20150182529-A1 ANDROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS INC (US) 2015-07-02 US disclosed
US-9051204-B2 Nontoxic polysiloxane material for producing biologically resorbable and/or bioactive articles containing polysiloxane material, its production and use BAYER INNOVATION GMBH (DE) 2015-06-09 US disclosed
EP-2877599-A1 METHODS AND COMPOSITIONS FOR DETERMINING RESISTANCE TO ANDROGEN RECEPTOR THERAPY Aragon Pharmaceuticals, Inc. (US) 2015-06-03 EP disclosed
EP-0925369-B2 UNIVERSAL TEST SYSTEMS AND METHODS OF USE THEREOF FOR IDENTIFYING MULTIPLE FAMILIES OF MICROORGANISMS SIEMENS HEALTHCARE DIAGNOSTICS (US) 2015-05-20 EP disclosed
EP-2271936-B1 IN VITRO METHOD TO DETERMINE WHETHER A DRUG CANDIDATE ACTIVE AGAINST A TARGET PROTEIN IS ACTIVE AGAINST A VARIANT OF SAID PROTEIN VALNEVA (FR) 2015-05-06 EP disclosed
CN-104533251-A Polyurethane embossment fireproof door and production process thereof ZHOU DONGPING 2015-04-22 CN disclosed
US-20150105403-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS, INC. 2015-04-16 US disclosed
CN-104515760-A Double-color fluorescence positioning super-resolution biological microscopy method and system NANOBIOIMAGING LTD 2015-04-15 CN disclosed
US-20150079161-A1 METHOD FOR SELECTIVELY INHIBITING ACAT1 IN THE TREATMENT OF NEURODEGENERATIVE DISEASES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-03-19 US disclosed
EP-2735562-B1 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS INC (US) 2015-03-11 EP disclosed
US-20150056627-A1 APTAMERS THE UNIVERSITY OF CHESTER (GB) 2015-02-26 US disclosed
US-20150051187-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED 2015-02-19 US disclosed
US-8956880-B2 Detection of micro-organisms MICAP PLC (GB) 2015-02-17 US disclosed
US-20150045386-A1 (2S,3R)-N-2-3-PYRIDINYLMETHYL-1-AZABICYCLO 2.2.2 OCT-3-YL BENZOFURAN-2-CARBOXAMIDE, NOVEL SALT FORMS, AND METHODS OF USE THEREOF ATTENUA, INC. 2015-02-12 US disclosed
US-20150038535-A1 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMA (US) 2015-02-05 US disclosed
US-20150031016-A1 Mixed Cell Diagnostic Systems For Detection Of Respiratory, Herpes and Enteric Viruses DIAGNOSTIC HYBRIDS INC. (US) 2015-01-29 US disclosed
US-20150031661-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-01-29 US disclosed
EP-2828243-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF Seragon Pharmaceuticals, Inc. (US) 2015-01-28 EP disclosed
US-8937064-B2 Pyrazolo[1,5-a]pyrimidines useful as JAK2 inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-01-20 US disclosed
EP-2824102-A1 Androgen receptor modulators and uses thereof Aragon Pharmaceuticals, Inc. (US) 2015-01-14 EP disclosed
EP-1948193-B1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMA (US) 2015-01-07 EP disclosed
US-20150005286-A1 FLUORINATED ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS, INC. 2015-01-01 US disclosed
US-20140364450-A1 AMINOPYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED 2014-12-11 US disclosed
US-20140364427-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS, INC. 2014-12-11 US disclosed
EP-2809647-A1 MGLU 2/3 AGONISTS Eli Lilly and Company (US) 2014-12-10 EP disclosed
US-8906603-B2 Modified cardiolipin and uses therefor THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES, CENTERS FOR DISEASE CONTROL AND PREVENTION (US) 2014-12-09 US disclosed
WO-2014176544-A1 WATER SOLUBLE G-PROTEIN COUPLED RECEPTOR THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2014-10-30 WO disclosed
WO-2014176524-A2 OPIOID DETECTION BASED ON HIGH QUALITY GRAPHENE TRANSISTOR ARRAYS AND A SYNTHETIC MU RECEPTOR THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2014-10-30 WO disclosed
US-20140322800-A1 OXIDIZED CARDIOLIPIN AND USES TO DETECT CARDIOLIPIN ANTIBODIES THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF 2014-10-30 US disclosed
US-20140315877-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS TARGACEPT INC (US) 2014-10-23 US disclosed
EP-2791133-A1 FLUORINATED ESTROGEN RECEPTOR MODULATORS AND USES THEREOF Seragon Pharmaceuticals, Inc. (US) 2014-10-22 EP disclosed
EP-2791132-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF Seragon Pharmaceuticals, Inc. (US) 2014-10-22 EP disclosed
US-8865751-B2 Thiazoles, imidazoles, and pyrazoles useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-21 US disclosed
US-20140308340-A1 METHOD FOR SELECTIVELY INHIBITING ACAT1 IN THE TREATMENT OF NEURODEGENERATIVE DISEASES TRUSTEES OF DARTMOUTH COLLEGE (US) 2014-10-16 US disclosed
US-20140303137-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED 2014-10-09 US disclosed
US-8853244-B2 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-07 US disclosed
US-8853382-B2 Expression of antibody or a fragment thereof in lactobacillus HERA PHARMACEUTICALS, INC. (US) 2014-10-07 US disclosed
US-8853423-B2 Indane estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS, INC. (US) 2014-10-07 US disclosed
CN-102695701-B MGLU2 agonists ELI LILLY AND CO. (US) 2014-10-01 CN disclosed
US-8846715-B2 (2S,3R)-N-(2((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofuran-2-carboxamide novel salt forms, and methods of use thereof TARGACEPT, INC. (US) 2014-09-30 US disclosed
US-20140288185-A1 NICOTINIC RECEPTOR NON-COMPETITIVE MODULATORS TARGACEPT, INC. 2014-09-25 US disclosed
US-20140288169-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS TARGACEPT, INC. (US) 2014-09-25 US disclosed
WO-2014151899-A1 POLYCYCLIC ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS, INC. (US) 2014-09-25 WO disclosed
EP-2152696-B1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMA (US) 2014-09-24 EP disclosed
US-8841308-B2 Pyrazin-2-amines useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-09-23 US disclosed
US-20140256703-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED 2014-09-11 US disclosed
EP-2773609-A2 NICOTINIC RECEPTOR NON-COMPETITIVE MODULATORS Targacept, Inc. (US) 2014-09-10 EP disclosed
EP-2773759-A1 APTAMERS DuPont Nutrition Biosciences ApS (DK) 2014-09-10 EP disclosed
US-8828673-B2 Mixed cell diagnostic systems for detection of respiratory, herpes and enteric viruses DIAGNOSTIC HYBRIDS INC (US) 2014-09-09 US disclosed
US-20140249332-A1 METHODS FOR SELECTIVE OXIDATION OF ALPHA TOCOTRIENOL IN THE PRESENCE OF NON-ALPHA TOCOTRIENOLS PTC THERAPEUTICS, INC. 2014-09-04 US disclosed
US-20140221414-A1 SOLID DISPERSION OF RIFAXIMIN LUPIN LIMITED (IN) 2014-08-07 US disclosed
EP-2758395-A1 COMPOUNDS USEFUL AS INHIBITORS OF CHOLINE KINASE Vertex Pharmaceuticals Inc. (US) 2014-07-30 EP disclosed
US-8785444-B2 Thiazoles and pyrazoles useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-07-22 US disclosed
US-8778619-B2 Oxidized cardiolipin and uses to detect cardiolipin antibodies THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2014-07-15 US disclosed
US-20140194444-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED 2014-07-10 US disclosed
EP-2751101-A1 COMPOUNDS USEFUL AS INHIBITORS OF CHOLINE KINASE Vertex Pharmaceuticals Incorporated (US) 2014-07-09 EP disclosed
US-20140187781-A1 AMINOPYRIDINES AND AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-07-03 US disclosed
EP-1831168-B1 PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY PROTEIN KINASES FOR THE TREATMENT OF INFLAMMATORY, PROLIFERATIVE AND IMMUNOLOGICALLY-MEDIATED DISEASES. VERTEX PHARMA (US) 2014-07-02 EP disclosed
US-8759389-B1 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-06-24 US disclosed
US-20140173771-A1 TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS Stichting Techno. Topinstituut Groene Genetica (Foundation Techno. top Institute Green Genetics) 2014-06-19 US disclosed
US-8741932-B2 Imidazopyridine derivatives Piramal Enterprises Limited (IN) 2014-06-03 US disclosed
EP-2734512-A1 METHODS FOR SELECTIVE OXIDATION OF ALPHA TOCOTRIENOL IN THE PRESENCE OF NON-ALPHA TOCOTRIENOLS Edison Pharmaceuticals, Inc. (US) 2014-05-28 EP disclosed
EP-2735562-A1 Estrogen receptor modulators and uses thereof Seragon Pharmaceuticals, Inc. (US) 2014-05-28 EP disclosed
US-8735593-B2 Aminopyridines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-05-27 US disclosed
US-20140141099-A1 DRUG DISCOVERY METHODS VERTEX PHARMACEUTICALS INCORPORATED 2014-05-22 US disclosed
US-20140113944-A1 BICYCLO (3.1.0) HEXANE-2, 6-DICARBOXYLIC ACID DERIVATIVES AS MGLU2 RECEPTOR AGONIST ELI LILLY AND COMPANY (US) 2014-04-24 US disclosed
US-20140113005-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-04-24 US disclosed
EP-2721012-A1 BICYCLO (3.1.0) HEXANE- 2, 6 -DICARBOXYLIC ACID DERIVATIVES AS MGLU2 RECEPTOR AGONIST Eli Lilly and Company (US) 2014-04-23 EP disclosed
US-8703810-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS, INC. (US) 2014-04-22 US disclosed
US-20140107095-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS, INC. (US) 2014-04-17 US disclosed
EP-2718309-A1 TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS Stichting Technologisch Topinstituut Groene Genetica (Foundation Technological Top Institute Green Genetics) (NL) 2014-04-16 EP disclosed
US-20140087398-A1 OXIDIZED CARDIOLIPIN AND USES TO DETECT CARDIOLIPIN ANTIBODIES Arlington Scientific, Inc. (US) 2014-03-27 US disclosed
US-8680062-B2 System for delivering therapeutic agents into living cells and cells nuclei Deliversir Ltd. (IL) 2014-03-25 US disclosed
EP-1765819-B1 AZAINDOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2014-03-12 EP disclosed
US-8664219-B2 Aminopyrimidines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-03-04 US disclosed
CN-103596933-A Bicyclo (3.1.0) hexane- 2, 6 -dicarboxylic acid derivatives as MGLU2 receptor agonist LILLY CO ELI 2014-02-19 CN disclosed
US-20140038935-A1 DIHYDRODIAZEPINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-02-06 US disclosed
US-20140037754-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-02-06 US disclosed
WO-2014018926-A1 METHODS AND COMPOSITIONS FOR DETERMINING RESISTANCE TO ANDROGEN RECEPTOR THERAPY ARAGON PHARMACEUTICALS, INC. (US) 2014-01-30 WO disclosed
US-8637511-B2 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-01-28 US disclosed
US-20140024673-A1 (2S,3R)-N-(2-((3-PYRIDINYL)METHYL)-1-AZABICYCLO[2.2.2]OCT-3-YL)BENZYOFURN-2-CARBOXAMIDE, NOVEL SALT FORMS, AND METHODS OF USE THEREOF TARGACEPT,INC. (US) 2014-01-23 US disclosed
US-20140018352-A1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-01-16 US disclosed
WO-2014004417-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS TARGACEPT, INC. (US) 2014-01-03 WO disclosed
CN-103464108-A Gold-palladium thermometal satellite structure assembly as well as preparation method and application thereof NAT CT NANOSCIENCE NCNST CHINA 2013-12-25 CN disclosed
US-20130323819-A1 EXPRESSION OF ANTIBODY OR A FRAGMENT THEREOF IN LACTOBACILLUS HERA PHARMACEUTICALS, INC. 2013-12-05 US disclosed
US-20130324725-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED 2013-12-05 US disclosed
US-8598361-B2 Process for preparing 5-fluoro-1H-pyrazolo [3,4-B] pyridin-3-amine and derivatives therof VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-12-03 US disclosed
US-20130310433-A1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED 2013-11-21 US disclosed
WO-2013171281-A1 HYDANTOIN AND THIOHYDANTOIN DERIVATIVES AS ANTIVIRAL DRUGS VIVALIS (FR) 2013-11-21 WO disclosed
US-20130310428-A1 THERMO-STABLE, ARSENIC-FREE SYNERGISTIC BIOCIDE CONCENTRATE COMPOSITION FOR POLYMER MATRICES AND PROCESS FOR PREPARING SAME ISP INVESTMENTS INC. (US) 2013-11-21 US disclosed
EP-2190849-B1 4-(9-(3,3-DIFLUOROCYCLOPENTYL)-5,7,7-TRIMETHYL-6-OXO-6,7,8,9-TETRAHYDRO-5H-PYRIMIDO[4,5-B[1,4]DIAZEPIN-2-YLAMINO)-3-METHOXYBENZAMIDE DERIVATIVES AS INHIBITORS OF THE HUMAN PROTEIN KINASES PLK1 TO PLK4 FOR THE TREATMENT OF PROLIFERATIVE DISEASES VERTEX PHARMA (US) 2013-11-20 EP disclosed
EP-2664616-A1 Hydantoin and thiohydantoin derivatives as antiviral drugs Vivalis (FR) 2013-11-20 EP disclosed
EP-2661421-A2 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS Targacept, Inc. (US) 2013-11-13 EP disclosed
US-8575214-B2 MGlu 2/3 agonists ELI LILLY AND COMPANY (US) 2013-11-05 US disclosed
US-20130281445-A1 COMPOUNDS USEFUL AS INHIBITORS OF CHOLINE KINASE VERTEX PHARMACEUTICALS INCORPORATED 2013-10-24 US disclosed
US-8557818-B2 Compounds useful as protein kinase inhibitors VERTEX PHAMACEUTICALS INCORPORATED (US) 2013-10-15 US disclosed
US-8557833-B2 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-10-15 US disclosed
US-20130267498-A1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED 2013-10-10 US disclosed
US-20130261114-A1 COMPOUNDS USEFUL AS INHIBITORS OF CHOLINE KINASE VERTEX PHARMACEUTICALS INCORPORATED 2013-10-03 US disclosed
WO-2013142266-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS, INC. (US) 2013-09-26 WO disclosed
EP-1949108-B1 MODIFIED CARDIOLIPIN AND USES THEREFOR US GOV HEALTH & HUMAN SERV (US) 2013-09-25 EP disclosed
US-8541446-B2 (2S,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofurn-2-carboxamide, novel salt forms, and methods of use thereof TARGACEPT, INC. (US) 2013-09-24 US disclosed
US-20130245273-A1 AMINOPYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-09-19 US disclosed
EP-2516406-B1 MGLU2 AGONISTS LILLY CO ELI (US) 2013-09-18 EP disclosed
US-20130236496-A1 USE OF LEUKOTRIENE B4 IN COMBINATION WITH A TOLL-LIKE RECEPTOR LIGAND, A RIG-I-LIKE RECEPTOR LIGAND, OR A NOD-LIKE RECEPTOR LIGAND TO ENHANCE THE INNATE IMMUNE RESPONSE UNIVERSITE DE LAVAL (CA) 2013-09-12 US disclosed
EP-2134707-B1 Aminopyrimidines useful as inhibitors of protein kinases VERTEX PHARMA (US) 2013-09-11 EP disclosed
US-20130231333-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2013-09-05 US disclosed
EP-1951715-B1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMA (US) 2013-09-04 EP disclosed
US-8524902-B2 [1,2,4]triazolo[4,3-f]pteridines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-09-03 US disclosed
US-8518953-B2 Aminopyrimidines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-08-27 US disclosed
WO-2013116174-A1 MGLU 2/3 AGONISTS ELI LILLY AND COMPANY (US) 2013-08-08 WO disclosed
US-20130197079-A1 MGLU 2/3 AGONISTS ELI LILY AND COMPANY (US) 2013-08-01 US disclosed
EP-2616445-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF Aragon Pharmaceuticals, Inc. (US) 2013-07-24 EP disclosed
US-20130184259-A1 PYRIDONES USEFUL AS INHIBITORS OF KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-07-18 US disclosed
CN-101420955-B Dihydrodiazepines useful as inhibitors of protein kinases VERTEX PHARMA 2013-07-17 CN disclosed
US-8481578-B2 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-07-09 US disclosed
WO-2013090836-A1 FLUORINATED ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2013-06-20 WO disclosed
WO-2013090829-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2013-06-20 WO disclosed
CN-202994798-U Diagnostic kit for diagnosis of rheumatoid arthritis SHANGHAI KEXIN BIOTECH CO LTD 2013-06-12 CN disclosed
US-8461149-B2 Compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-06-11 US disclosed
US-8455534-B2 Estrogen receptor modulators and uses thereof ARAGON PHARMACEUTICALS, INC. (US) 2013-06-04 US disclosed
US-8455507-B2 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-06-04 US disclosed
US-20130137746-A1 INDANE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2013-05-30 US disclosed
WO-2013067105-A2 NICOTINIC RECEPTOR NON-COMPETITIVE MODULATORS TARGACEPT, INC. (US) 2013-05-10 WO disclosed
WO-2013064818-A1 APTAMERS DUPONT NUTRITION BIOSCIENCES APS (DK) 2013-05-10 WO disclosed
US-20130116258-A1 ANDROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2013-05-09 US disclosed
US-20130116232-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2013-05-09 US disclosed
US-20130116228-A1 THIAZOLES AND PYRAZOLES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-05-09 US disclosed
CN-101360997-B Modified cardiolipin and uses therefor US GOVERNMENT (US) 2013-05-01 CN disclosed
US-8426425-B2 Aminopyrimidines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-04-23 US disclosed
US-20130096302-A1 PYRROLOPYRAZINES AND PYRAZOLOPYRAZINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED 2013-04-18 US disclosed
EP-2580210-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF Aragon Pharmaceuticals, Inc. (US) 2013-04-17 EP disclosed
US-20130090479-A1 THIAZOLES, IMIDAZOLES, AND PYRAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-04-11 US disclosed
EP-2576496-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS Targacept, Inc. (US) 2013-04-10 EP disclosed
US-8410112-B2 Compounds useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-04-02 US disclosed
US-8410133-B2 Aminopyridines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-04-02 US disclosed
WO-2013043961-A1 COMPOUNDS USEFUL AS INHIBITORS OF CHOLINE KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-03-28 WO disclosed
WO-2013043960-A1 COMPOUNDS USEFUL AS INHIBITORS OF CHOLINE KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-03-28 WO disclosed
US-8399478-B2 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-03-19 US disclosed
US-8399458-B2 Compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-03-19 US disclosed
US-8394952-B2 Dihydrodiazepines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-03-12 US disclosed
US-8383633-B2 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-02-26 US disclosed
US-8372835-B2 Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-02-12 US disclosed
US-8372850-B2 Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-02-12 US disclosed
WO-2013013078-A1 METHODS FOR SELECTIVE OXIDATION OF ALPHA TOCOTRIENOL IN THE PRESENCE OF NON-ALPHA TOCOTRIENOLS EDISON PHARMECEUTICALS, INC. (US) 2013-01-24 WO disclosed
EP-2545025-A1 SYNTHESIS OF ALPHA-TOCOPHEROLQUINONE DERIVATIVES, AND METHODS OF USING THE SAME Edison Pharmaceuticals, Inc. (US) 2013-01-16 EP disclosed
US-20130012561-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2013-01-10 US disclosed
EP-2182949-B1 (2S,3R)-N-(2-((3-PYRIDINYL)METHYL)-1-AZABICYCLO[2.2.2]OCT-3-YL)BENZOFURAN-2-CARBOXAMIDE, NOVEL SALT FORMS, AND METHODS OF USE THEREOF TARGACEPT INC (US) 2013-01-02 EP disclosed
EP-2536708-A2 ANDROGEN RECEPTOR MODULATORS AND USES THEREOF Aragon Pharmaceuticals, Inc. (US) 2012-12-26 EP disclosed
US-8338597-B2 Pyridones useful as inhibitors of kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-12-25 US disclosed
WO-2012173850-A1 BICYCLO (3.1.0) HEXANE- 2, 6 -DICARBOXYLIC ACID DERIVATIVES AS MGLU2 RECEPTOR AGONIST ELI LILLY AND COMPANY (US) 2012-12-20 WO disclosed
EP-2176261-B1 PROCESS FOR PREPARING 5-FLUORO-1H-PYRAZOLO [3, 4-B] PYRIDIN-3-AMINE AND DERIVATIVES THEREOF VERTEX PHARMA (US) 2012-12-19 EP disclosed
WO-2012169893-A1 TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS STICHTING TECHNOLOGISCH TOPINSTITUUT GROENE GENETICA (FOUNDATION TECHNOLOGICAL TOP INSTITUTE GREEN GENETICS) (NL) 2012-12-13 WO disclosed
US-8318184-B2 MGLU2 agonists ELI LILLY AND COMPANY (US) 2012-11-27 US disclosed
US-20120277425-A1 TETRAHYDROPTERIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-11-01 US disclosed
EP-2516406-A1 MGLU2 AGONISTS Eli Lilly and Company (US) 2012-10-31 EP disclosed
US-8299112-B2 Estrogen receptor modulators and uses thereof ARAGON PHARMACEUTICALS, INC. (US) 2012-10-30 US disclosed
US-8288400-B2 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-10-16 US disclosed
EP-2007757-B1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2012-10-03 EP disclosed
CN-102695701-A MGLU2 agonists LILLY CO ELI 2012-09-26 CN disclosed
WO-2012125735-A1 AN INTEGRATED APPROACH TO THE ISOLATION AND PURIFICATION OF ANTIBODIES ABOTT LABORATORIES (US) 2012-09-20 WO disclosed
US-20120238730-A1 INTEGRATED APPROACH TO THE ISOLATION AND PURIFICATION OF ANTIBODIES ABBOTT LABORATORIES (US) 2012-09-20 US disclosed
US-8268811-B2 Thiazoles and pyrazoles useful as kinase inhibitors VERTEX PHARMACEUTICALS INC. (US) 2012-09-18 US disclosed
US-20120232275-A1 PROCESS FOR PREPARING 5-FLUORO-1H-PYRAZOLO [3,4-B] PYRIDIN-3-AMINE AND DERIVATIVES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-09-13 US disclosed
US-20120232072-A1 IMIDAZOPYRIDINE DERIVATIVES PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-09-13 US disclosed
EP-2496577-A1 IMIDAZOPYRIDINE DERIVATIVES Piramal Life Sciences Limited (IN) 2012-09-12 EP disclosed
EP-2493456-A2 SOLID DISPERSION OF RIFAXIMIN Lupin Limited (IN) 2012-09-05 EP disclosed
EP-2019826-B1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2012-08-29 EP disclosed
US-20120214833-A1 SOLID DISPERSION OF RIFAXIMIN LUPIN LIMITED (IN) 2012-08-23 US disclosed
US-8247393-B2 Conjugated estrogen compositions, applicators, kits, and methods of making and use thereof TEVA WOMEN'S HEALTH, INC. (US) 2012-08-21 US disclosed
US-8242272-B2 Process for preparing 5-fluoro-1H-pyrazolo [3,4-B] pyridin-3-amine and derivatives thereof VERTEX PHARMACEUTICALS INC. (US) 2012-08-14 US disclosed
US-8236832-B2 Thiazoles, imidazoles, and pyrazoles useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INC. (US) 2012-08-07 US disclosed
US-20120196276-A1 Mixed Cell Diagnostic Systems For Detection Of Respiratory, Herpes and Enteric Viruses QUIDEL CORPORATION 2012-08-02 US disclosed
US-20120189579-A1 SUBSTITUTED PYRROLIDINONE AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE VIVALIS (FR) 2012-07-26 US disclosed
US-20120190699-A1 PYRIDONES USEFUL AS INHIBITORS OF KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-07-26 US disclosed
US-20120183577-A1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-07-19 US disclosed
WO-2012093174-A1 1-(6-MEMBERED AZO-HETEROCYCLIC)-2,5-DIHYDRO-1H-PYRROL-2-ONE DERIVATIVES AS ANTI-HEPATITIS C VIRUS, THE PHARMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE VIVALIS (FR) 2012-07-12 WO disclosed
WO-2012094437-A2 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS TARGACEPT, INC. (US) 2012-07-12 WO disclosed
EP-2474546-A1 Thiophene-carboxamides useful as inhibitors of protein kinases Vertex Pharmaceuticals Inc. (US) 2012-07-11 EP disclosed
US-8217024-B2 Conjugated estrogen compositions, applicators, kits, and methods of making and use thereof TEVA WOMEN'S HEALTH, INC. (US) 2012-07-10 US disclosed
US-20120165378-A1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-28 US disclosed
EP-2467364-A2 NITROGEN-CONTAINING COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF ATRIAL FIBRILLATION Otsuka Pharmaceutical Co., Ltd. (JP) 2012-06-27 EP disclosed
US-8206675-B2 Nontoxic polyethoxysiloxane material or the production of biologically resorbable and/or bioactive articles containing polyethoxysiloxane material, the production thereof, and the use thereof BAYER INNOVATION GMBH (DE) 2012-06-26 US disclosed
US-20120156705-A1 LUCIFERASES AND USES THEREOF TARGETING SYSTEMS (US) 2012-06-21 US disclosed
EP-2465501-A1 (2S,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofuran-2-carboxamide, novel salt forms, and methods of preparation Targacept Inc. (US) 2012-06-20 EP disclosed
US-20120149898-A1 DIHYDRODIAZEPINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-14 US disclosed
EP-1989205-B1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2012-06-13 EP disclosed
US-20120142660-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-07 US disclosed
US-20120142088-A1 DNA-CELL CONJUGATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-06-07 US disclosed
US-8188134-B2 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-05-29 US disclosed
US-20120129885-A1 (2S,3R)-N-(2-((3-PYRIDINYL)METHYL)-1-AZABICYCLO[2.2.2]OCT-3-YL)BENZOFURN-2-CARBOXAMIDE, NOVEL SALT FORMS, AND METHODS OF USE THEREOF TARGACEPT, INC. (US) 2012-05-24 US disclosed
US-20120128630-A1 1-(6 MEMBERS AZO-HETEROCYCLIC)-PYRROLIN-2-ONE COMPOUNDS AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARAMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE VIVALIS (FR) 2012-05-24 US disclosed
WO-2012037411-A9 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed
US-20120122879-A1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-05-17 US disclosed
EP-2451453-A1 SUBSTITUTED PYRROLIDINONE AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE Vivalis (FR) 2012-05-16 EP disclosed
EP-2451800-A1 1-(6 MEMBERS AZO-HETEROCYCLIC)-PYRROLIN-2-ONE COMPOUNDS AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE Vivalis (FR) 2012-05-16 EP disclosed
WO-2012037410-A9 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-05-10 WO disclosed
WO-2012019058-A9 EXPRESSION OF ANTIBODY OR A FRAGMENT THEREOF IN LACTOBACILLUS HERA PHARMACEUTICALS, INC. (US) 2012-04-26 WO disclosed
US-20120095014-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-04-19 US disclosed
US-8142997-B2 Mixed cell diagnostic systems for detection of respiratory, herpes and enteric viruses Diagnostic Hybrids, Inc—Quidel Corporation (US) 2012-03-27 US disclosed
US-20120071535-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 US disclosed
WO-2012037410-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 WO disclosed
WO-2012037411-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 WO disclosed
EP-2431037-A1 (2S,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofuran-2-carboxamide, novel salt forms, and methods of use thereof Targacept, Inc. (US) 2012-03-21 EP disclosed
EP-1919891-B1 3,5-DISUBSTITUTED PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY OF NON-RECEPTOR TYROSINE KINASES VERTEX PHARMA (US) 2012-03-07 EP disclosed
US-8129387-B2 Substituted 5,6-dihydroimidazo[1,5-F]pteridines useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-03-06 US disclosed
US-8129399-B2 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-03-06 US disclosed
EP-1778637-B1 FKBP-binding composition and pharmaceutical use thereof AVENTIS PHARMA INC (US) 2012-02-22 EP disclosed
US-8119659-B2 (2S,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofuran-2-carboxamide, novel salt forms, and methods of use thereof TARGACEPT, INC. (US) 2012-02-21 US disclosed
US-20120040020-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-16 US disclosed
EP-2418210-A1 Thiophene-carboxamides useful as inhibitors of protein kinases Vertex Pharmceuticals Incorporated (US) 2012-02-15 EP disclosed
EP-2417249-A1 DNA-CELL CONJUGATES The Regents of the University of California (US) 2012-02-15 EP disclosed
WO-2012019054-A2 EXPRESSION OF ANTIBODY OR A FRAGMENT THEREOF IN LACTOBACILLUS HERA PHARMACEUTICALS, INC. (US) 2012-02-09 WO disclosed
WO-2012019058-A1 EXPRESSION OF ANTIBODY OR A FRAGMENT THEREOF IN LACTOBACILLUS HERA PHARMACEUTICALS, INC. (US) 2012-02-09 WO disclosed
US-20120028965-A1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-02 US disclosed
US-8101770-B2 Pyridones useful as inhibitors of kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-01-24 US disclosed
WO-2012000082-A1 USE OF LEUKOTRIENE B4 IN COMBINATION WITH A TOLL-LIKE RECEPTOR LIGAND, A RIG-L-LIKE RECEPTOR LIGAND OR A NOD-LIKE RECEPTOR LIGAND TO ENHANCE THE INNATE IMMUNE RESPONSE UNIVERSITé LAVAL (CA) 2012-01-05 WO disclosed
US-20110315625-A1 DETECTION OF MICRO-ORGANISMS MILLIPORE CORPORATION (US) 2011-12-29 US disclosed
WO-2011159769-A2 INDANE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2011-12-22 WO disclosed
WO-2011156518-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2011-12-15 WO disclosed
WO-2011149859-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS TARGACEPT, INC. (US) 2011-12-01 WO disclosed
WO-2011149862-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS MODULATORS TARGACEPT, INC. (US) 2011-12-01 WO disclosed
CN-102264721-A Compounds useful as inhibitors of ATR kinase 2011-11-30 CN disclosed
US-8067417-B2 Imidazo[1,2-F]pteridines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-11-29 US disclosed
US-20110288095-A1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-11-24 US disclosed
EP-2007732-B1 THIAZOLES, IMIDAZOLES, AND PYRAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2011-11-23 EP disclosed
US-20110269732-A1 DRUG DISCOVERY METHODS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-11-03 US disclosed
US-20110263720-A1 SYNTHESIS OF ALPHA-TOCOPHEROLQUINONE DERIVATIVES, AND METHODS OF USING THE SAME PENWEST PHARMACEUTICALS CO. (US) 2011-10-27 US disclosed
US-20110263859-A1 (2S, 3R)-N-(2-((3-PYRIDINYL)METHYL)-1-AZABICYCLO[2.2.2]OCT-3-YL)BENZOFURAN-2-CARBOXAMIDE, NOVEL SALT FORMS, AND METHODS OF USE THEREOF TARGACEPT, INC. (US) 2011-10-27 US disclosed
US-20110263575-A1 Compounds Useful as Protein Kinase Inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2011-10-27 US disclosed
EP-2376485-A1 PYRAZINE DERIVATIVES USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2011-10-19 EP disclosed
US-8039206-B1 Detection of micro-organisms MILLIPORE CORPORATION (US) 2011-10-18 US disclosed
US-8039661-B2 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-10-18 US disclosed
US-20110251085-A1 IN VITRO METHOD TO DETERMINE WHETHER A DRUG CANDIDATE ACTIVE AGAINST A TARGET PROTEIN IS ACTIVE AGAINST A VARIANT OF SAID PROTEIN VIVALIS (FR) 2011-10-13 US disclosed
EP-2094712-B1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2011-10-12 EP disclosed
EP-1919906-B1 3, 5-DISUBSTITUTED PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY OF NON-RECEPTOR TYROSINE KINASES VERTEX PHARMA (US) 2011-10-12 EP disclosed
EP-2370424-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2011-10-05 EP disclosed
EP-2137183-B1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2011-09-28 EP disclosed
US-8022202-B2 Dihydrodiazepines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-09-20 US disclosed
WO-2011112679-A1 SYNTHESIS OF ALPHA-TOCOPHEROLQUINONE DERIVATIVES, AND METHODS OF USING THE SAME PENWEST PHARMACEUTICALS CO. (US) 2011-09-15 WO disclosed
US-20110223659-A1 Compositions And Methods For Detecting Severe Acute Respiratory Syndrome Coronavirus DIAGNOSTIC HYBRIDS, INC. 2011-09-15 US disclosed
US-20110224197-A1 PYRIMIDINES AND PYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-09-15 US disclosed
US-8017619-B2 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-09-13 US disclosed
WO-2011103202-A2 ANDROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2011-08-25 WO disclosed
US-20110190507-A1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-08-04 US disclosed
US-20110178146-A1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-07-21 US disclosed
US-7981906-B2 (2S,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl-benzofuran-2-carboxamide, novel salt forms, and methods of use thereof TARGACEPT, INC. (US) 2011-07-19 US disclosed
WO-2011084437-A1 MGLU2 AGONISTS ELI LILLY AND COMPANY (US) 2011-07-14 WO disclosed
US-20110152334-A1 MGLU2 AGONISTS ELI LILLY AND COMPANY (US) 2011-06-23 US disclosed
US-20110136143-A1 MODIFIED CARDIOLIPIN AND USES THEREFOR THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF 2011-06-09 US disclosed
EP-2325184-A1 Azaindoles useful as inhibitors of protein kinases Vertex Pharmceuticals Incorporated (US) 2011-05-25 EP disclosed
US-20110118255-A1 PYRAZOLO[1,5-a]PYRIMIDINES USEFUL AS JAK2 INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-05-19 US disclosed
WO-2011055320-A1 IMIDAZOPYRIDINE DERIVATIVES PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-05-12 WO disclosed
WO-2011051971-A2 SOLID DISPERSION OF RIFAXIMIN LUPIN LIMITED (IN) 2011-05-05 WO disclosed
EP-2316835-A1 Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases Vertex Pharmceuticals Incorporated (US) 2011-05-04 EP disclosed
EP-1951716-B1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMA (US) 2011-05-04 EP disclosed
US-20110081364-A1 PYRROLOPYRAZINES AND PYRAZOLOPYRAZINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED 2011-04-07 US disclosed
US-7915305-B2 To treat autoimmune, inflammatory, proliferative, hyperproliferative,neurodegenerative or immunologically-mediated diseases; useful for the study of kinases in biological and pathological phenomena; study of intracellular signal transduction pathways mediated by such kinases, and comparative evaluation VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-03-29 US disclosed
EP-2295413-A1 Indazole compounds useful as protein kinase inhibitors Vertex Pharmaceuticals Incorporated (US) 2011-03-16 EP disclosed
EP-2295412-A1 Indazole compounds useful as protein kinase inhibitors Vertex Pharmaceuticals Incorporated (US) 2011-03-16 EP disclosed
US-20110060013-A1 THIAZOLES AND PYRAZOLES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-03-10 US disclosed
WO-2011025980-A1 MODIFIED LUCIFERASES AND USES THEREOF TARGETING SYSTEMS (US) 2011-03-03 WO disclosed
EP-2289486-A1 Conjugated estrogen compositions, applicators, kits, and methods of making and use thereof Teva Women's Health, Inc. (US) 2011-03-02 EP disclosed
EP-2289487-A1 Conjugated estrogen compositions, applicators, kits, and methods of making and use thereof Teva Women's Health, Inc. (US) 2011-03-02 EP disclosed
WO-2011021726-A2 NITROGEN-CONTAINING COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-02-24 WO disclosed
US-20110046104-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-02-24 US disclosed
US-7888043-B2 Modified cardiolipin and uses therefor THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES, CENTERS FOR DISEASE CONTROL AND PREVENTION (US) 2011-02-15 US disclosed
EP-2102210-B1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2011-02-09 EP disclosed
US-20110020377-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-01-27 US disclosed
US-20110021559-A1 AMINOPYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-01-27 US disclosed
US-20110021519-A1 TETRAHYDROPTERIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-01-27 US disclosed
US-20110020469-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-01-27 US disclosed
US-20110020376-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-01-27 US disclosed
US-7872129-B2 Compositions useful as inhibitors of GSK-3 VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-01-18 US disclosed
US-20110009023-A1 NONTOXIC POLYSILOXANE MATERIAL FOR PRODUCING BIOLOGICALLY RESORBABLE AND/OR BIOACTIVE ARTICLES CONTAINING POLYSILOXANE MATERIAL, ITS PRODUCTION AND USE BAYER INNOVATION GMBH (DE) 2011-01-13 US disclosed
WO-2011004018-A1 SUBSTITUTED PYRROLIDINONE AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE VIVALIS (FR) 2011-01-13 WO disclosed
WO-2011004017-A1 1-(6 MEMBERS AZO-HETEROCYCLIC)-PYRROLIN-2-ONE COMPOUNDS AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE VIVALIS (FR) 2011-01-13 WO disclosed
EP-2271936-A1 IN VITRO METHOD TO DETERMINE WHETHER A DRUG CANDIDATE ACTIVE AGAINST A TARGET PROTEIN IS ACTIVE AGAINST A VARIANT OF SAID PROTEIN Vivalis (FR) 2011-01-12 EP disclosed
EP-2262498-A2 PYRIMIDINES AND PYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmceuticals Incorporated (US) 2010-12-22 EP disclosed
US-7855214-B2 Fused cyclic systems useful as inhibitors of TEC family protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-12-21 US disclosed
US-20100317641-A1 THIAZOLES AND PYRAZOLES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-12-16 US disclosed
US-7851495-B2 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-12-14 US disclosed
US-20100310675-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-12-09 US disclosed
US-7846655-B2 Compositions and methods for detecting a non plus-stranded RNA virus DIAGNOSTIC HYBRIDS, INC. (US) 2010-12-07 US disclosed
EP-2252618-A1 PYRAZOLO [1,5-a] PYRIMIDINES USEFUL AS JAK2 INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2010-11-24 EP disclosed
US-7838517-B2 Compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-11-23 US disclosed
EP-2249430-A1 COMPOSITE MATERIAL, PHOTOELECTRIC CONVERSION MATERIAL, DYE-SENSITIZED SOLAR CELL, DYE-SENSITIZED SOLAR CELL DEVICE, MANUFACTURING METHOD FOR PHOTOELECTRIC CONVERSION DEVICE, AND METHOD OF ANALYZING OXYGEN TITANIUM CRYSTAL STRUCTURE The University of Tokyo (JP) 2010-11-10 EP disclosed
US-7829590-B2 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2010-11-09 US disclosed
US-20100280026-A1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-11-04 US disclosed
US-7820685-B2 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-10-26 US disclosed
US-20100266690-A1 STABILIZER CONCENTRATE FOR MATRIX COMPOSITIONS PROCESSED AT ELEVATED TEMPERATURES TROY TECHNOLOGY II, INC. 2010-10-21 US disclosed
US-7816490-B2 Specific inhibitors of NFAT activation by calcineurin and their use in treating immune-related diseases IMMUNE DISEASE INSTITUTE, INC. (US) 2010-10-19 US disclosed
WO-2010118235-A1 DNA-CELL CONJUGATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2010-10-14 WO disclosed
EP-1812440-B1 PYRAZOLO[1,5-A]PYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2010-09-22 EP disclosed
US-7795259-B2 Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-09-14 US disclosed
US-20100222318-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-09-02 US disclosed
EP-1983987-B1 DIHYDRODIAZEPINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2010-09-01 EP disclosed
US-7786130-B2 Pyridones useful as inhibitors of kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-08-31 US disclosed
US-7786283-B2 BRI constructs and methods of using MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2010-08-31 US disclosed
US-20100215772-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-08-26 US disclosed
US-7777042-B2 N-sulfonylpipecolic acid derivative FKBP binding composition and pharmaceutical use thereof AVENTIS PHARMACEUTICALS INC. (US) 2010-08-17 US disclosed
CN-101801959-A Aminopyrimidines useful as kinase inhibitors VERTEX PHARMA 2010-08-11 CN disclosed
US-7767672-B2 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-08-03 US disclosed
US-20100190765-A1 DIHYDRODIAZEPINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-07-29 US disclosed
US-7763629-B2 Tetrahydropteridines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-07-27 US disclosed
US-20100184980-A1 Process for Preparing 5-Fluoro-1H-Pyrazolo [3,4-b] Pyridin-3-amine and Derivatives Thereof VERTEX PHARMACEUTICALS INCORPORATED 2010-07-22 US disclosed
EP-2099787-B1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2010-07-21 EP disclosed
CN-101784273-A (2S,3R) -N- (2- ((3-pyridinyl) methyl) -1-azabicyclo [2.2.2] oct-3-yl) benzofuran-2-carboxamide, novel salt forms, and methods of use thereof TARGACEPT INC 2010-07-21 CN disclosed
US-20100173280-A1 Systems for Detection and Production of Respiratory, Herpes and Enteric Viruses DIAGNOSTIC HYBRIDS, INC (US) 2010-07-08 US disclosed
US-20100174045-A1 NONTOXIC POLYETHOXYSILOXANE MATERIAL OR THE PRODUCTION OF BIOLOGICALLY RESORBABLE AND OR BIOACTIVE ARTICLES CONTAINING POLYETHOXYSILOXANE MATERIAL, THE PRODUCTION THEREOF, AND THE USE THEREOF JIANGSU SYNECOUN MEDICAL TECHNOLOGY CO., LTD. (CN) 2010-07-08 US disclosed
EP-2203054-A1 STABILIZER CONCENTRATE FOR MATRIX COMPOSITIONS PROCESSED AT ELEVATED TEMPERATURES Isp Investments Inc. (US) 2010-07-07 EP disclosed
WO-2010071837-A1 PYRAZINE DERIVATIVES USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-06-24 WO disclosed
US-20100137305-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-06-03 US disclosed
EP-2190849-A2 COMPOUNDS USEFUL AS PROTEIN KINASES INHIBITORS Vertex Pharmceuticals Incorporated (US) 2010-06-02 EP disclosed
WO-2009145814-A9 PYRIMIDINES AND PYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-05-14 WO disclosed
WO-2010054398-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-05-14 WO disclosed
EP-2182949-A1 (2S,3R)-N-(2-((3-PYRIDINYL)METHYL)-1-AZABICYCLO[2.2.2]OCT-3-YL)BENZOFURAN-2-CARBOXAMIDE, NOVEL SALT FORMS, AND METHODS OF USE THEREOF Targacept Inc. (US) 2010-05-12 EP disclosed
US-20100099686-A1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED 2010-04-22 US disclosed
EP-2176261-A1 PROCESS FOR PREPARING 5-FLUORO-1H-PYRAZOLO [3, 4-B] PYRIDIN-3-AMINE AND DERIVATIVES THEREOF Vertex Pharmaceuticals Incorporated (US) 2010-04-21 EP disclosed
US-7700609-B2 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-04-20 US disclosed
US-7691885-B2 Pyridones useful as inhibitors of kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-04-06 US disclosed
CN-101687852-A Thiazoles and pyrazoles useful as kinase inhibitors VERTEX PHARMA 2010-03-31 CN disclosed
EP-2164842-A2 THIAZOLES AND PYRAZOLES USEFUL AS KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2010-03-24 EP disclosed
CN-101679378-A Thiazoles and pyrazoles as kinase inhibitors VERTEX PHARMA 2010-03-24 CN disclosed
CN-101679387-A Aminopyrimidines useful as kinase inhibitors VERTEX PHARMA 2010-03-24 CN disclosed
CN-101679386-A Aminopyrimidines useful as kinase inhibitors VERTEX PHARMA 2010-03-24 CN disclosed
CN-101675041-A Aminopyrimidines useful as kinase inhibitors VERTEX PHARMA 2010-03-17 CN disclosed
EP-1451366-B1 MOLECULAR DETECTION SYSTEMS UTILIZING REITERATIVE OLIGONUCLEOTIDE SYNTHESIS RIBOMED BIOTECHNOLOGIES INC (US) 2010-03-10 EP disclosed
EP-2155730-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2010-02-24 EP disclosed
US-20100037713-A1 Pharmaceutical Analysis Apparatus and Method SMITHKLINE BEECHAM CORPORATION 2010-02-18 US disclosed
EP-2152696-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2010-02-17 EP disclosed
EP-2152694-A2 THIAZOLES AND PYRAZOLES USEFUL AS KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2010-02-17 EP disclosed
EP-2086965-B1 AMINOPYRIDINES AND AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2010-02-10 EP disclosed
US-7659283-B2 Pyrrolo [3,2-C] pyridines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-02-09 US disclosed
EP-2148931-A2 DRUG DISCOVERY METHODS FOR AURORA KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2010-02-03 EP disclosed
US-20100022502-A1 AMINOPYRIDINES AND AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-01-28 US disclosed
US-20100022507-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-01-28 US disclosed
EP-2146982-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2010-01-27 EP disclosed
EP-2142537-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2010-01-13 EP disclosed
EP-2137183-A2 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals Incorporated (US) 2009-12-30 EP disclosed
EP-2134707-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals, Inc. (US) 2009-12-23 EP disclosed
EP-2134709-A1 AMINOPYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals, Inc. (US) 2009-12-23 EP disclosed
EP-2131816-A1 PHARMACEUTICAL ANALYSIS APPARATUS AND METHOD Smithkline Beecham Corporation (US) 2009-12-16 EP disclosed
US-20090306155-A1 THIAZOLES, IMIDAZOLES, AND PYRAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-12-10 US disclosed
EP-1692140-B1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-12-09 EP disclosed
WO-2009145814-A2 PYRIMIDINES AND PYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-12-03 WO disclosed
US-7622463-B2 Dihydrodiazepines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-11-24 US disclosed
US-20090286840-A1 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2009-11-19 US disclosed
US-20090286222-A1 Mixed Cell Diagnostic Systems For Detection Of Respiratory, Herpes And Enteric Viruses QUIDEL CORPORATION 2009-11-19 US disclosed
US-20090281082-A1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-11-12 US disclosed
EP-2111223-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-10-28 EP disclosed
EP-2102210-A2 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS Vertex Pharmceuticals Incorporated (US) 2009-09-23 EP disclosed
US-7592169-B2 Methods and compositions for treatment and prevention of HSV-2 infections and conditions MEDIMMUNE, LLC (US) 2009-09-22 US disclosed
WO-2009112592-A1 IN VITRO METHOD TO DETERMINE WHETHER A DRUG CANDIDATE ACTIVE AGAINST A TARGET PROTEIN IS ACTIVE AGAINST A VARIANT OF SAID PROTEIN VIVALIS (FR) 2009-09-17 WO disclosed
EP-2099787-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals, Inc. (US) 2009-09-16 EP disclosed
EP-2101173-A1 In vitro method to determine whether a drug candidate active against a target protein is active against a variant of said protein Vivalis (FR) 2009-09-16 EP disclosed
US-7589214-B2 2-Cyclopentyl-4-(4-phenoxyphenyl)thiazole-5-carboxamide; amidation; oxidation; cyclization; VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-09-15 US disclosed
EP-2094712-A2 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS Vertex Pharmceuticals Incorporated (US) 2009-09-02 EP disclosed
EP-1798556-B1 Device for the early and rapid immunochromatographic detection of HIV and uses thereof JORDANIAN PHARMACEUTICAL MFG (JO) 2009-08-26 EP disclosed
EP-2086965-A1 AMINOPYRIDINES AND AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals, Inc. (US) 2009-08-12 EP disclosed
EP-1501797-B1 3-(SUBSTITUTED AMINO)-1H-INDOLE-2-CARBOXYLIC ACID ESTER AND 3-(SUBSTITUTED AMINO)-BENZO[B]THIOPHENE-2-CARBOXYLIC ACID ESTER DERIVATIVES AS INTERLEUKIN-4 GENE EXPRESSION INHIBITORS AVENTIS PHARMA INC (US) 2009-08-05 EP disclosed
US-20090186422-A1 SPECIFIC INHIBITORS OF NFAT ACTIVATION BY CALCINEURIN AND THEIR USE IN TREATING IMMUNE-RELATED DISEASES THE CBR INSTITUTE FOR BIOMEDICAL RESEARCH, INC., A MASSACHUSETTS CORPORATION 2009-07-23 US disclosed
US-20090181938-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-07-16 US disclosed
WO-2009085913-A1 PYRAZOLO [1,5-a] PYRIMIDINES USEFUL AS JAK2 INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-07-09 WO disclosed
EP-2076122-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-07-08 EP disclosed
CN-101466380-A Methods and compositions for the treatment of parkinson's disease MCLEAN HOSPITAL CORP (US) 2009-06-24 CN disclosed
US-7541165-B2 Molecular detection systems utilizing reiterative oligonucleotide synthesis RIBOMED BIOTECHNOLOGIES, INC. (US) 2009-06-02 US disclosed
US-20090118278-A1 COMPOSITIONS USEFUL AS INHIBITORS OF GSK-3 VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-05-07 US disclosed
WO-2009058216-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-05-07 WO disclosed
US-7528142-B2 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-05-05 US disclosed
US-7528138-B2 Pyrazolo[1,5-a]pyrimidines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-05-05 US disclosed
CN-101420955-A Dihydrodiazepines useful as inhibitors of protein kinases VERTEX PHARMA (US) 2009-04-29 CN disclosed
WO-2009046172-A1 STABILIZER CONCENTRATE FOR MATRIX COMPOSITIONS PROCESSED AT ELEVATED TEMPERATURES ISP INVESTMENTS INC. (US) 2009-04-09 WO disclosed
US-20090062292-A1 Tetrahydropteridines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2009-03-05 US disclosed
EP-2027116-A2 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals Incorporated (US) 2009-02-25 EP disclosed
EP-1107665-B1 METHOD OF DIAGNOSIS OF PROSTATE CANCER UROPATH PTY LTD (AU) 2009-02-25 EP disclosed
WO-2009023269-A2 4-(9-(3, 3-DIFLUOROCYCLOPENTYL) -5, 7, 7-TRIMETHYL-6-OXO-6, 7, 8, 9-TETRAHYDRO-5H-PYRIMIDO [4, 5-B[1, 4] DIAZEPIN-2-YLAMINO)-3-METHOXYBENZAMIDE DERIVATIVES AS INHIBITORS OF THE HUMAN PROTEIN KINASES PLK1 TO PLK4 FOR THE TREATMENT OF PROLIFERATIVE DISEASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-02-19 WO disclosed
US-20090048290-A1 2S,3R)-N-(2-((3-PYRIDINYL)METHYL)-1-AZABICYCLO[2.2.2]OCT-3-YL-BENZYOFURAN-2-CARBOXAMIDE, NOVEL SALT FORMS, AND METHODS OF USE THEREOF TRAMES BIO, INC. 2009-02-19 US disclosed
US-7491730-B2 Compositions useful as inhibitors of GSK-3 VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-02-17 US disclosed
WO-2009018415-A1 PROCESS FOR PREPARING 5-FLUORO-1H-PYRAZOLO [3, 4-B] PYRIDIN-3-AMINE AND DERIVATIVES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-02-05 WO disclosed
WO-2009018505-A1 (2S,3R)-N-(2-((3-PYRIDINYL)METHYL)-1-AZABICYCLO[2.2.2]OCT-3-YL)BENZOFURAN-2-CARBOXAMIDE, NOVEL SALT FORMS, AND METHODS OF USE THEREOF TARGACEPT, INC. (US) 2009-02-05 WO disclosed
EP-2019826-A1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals, Inc. (US) 2009-02-04 EP disclosed
CN-101360997-A Modified cardiolipin and uses therefor US GOV HEALTH & HUMAN SERV (US) 2009-02-04 CN disclosed
WO-2009005794-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-01-08 WO disclosed
EP-2010542-A2 4,5-DIHYDRO-[1,2,4]TRIAZOLO[4,3-F]PTERIDINES AS PROTEIN KINASE PLK1 INHIBITORS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS Vertex Pharmaceuticals Incorporated (US) 2009-01-07 EP disclosed
US-7473775-B2 Abortive promoter cassettes RIBOMED BIOTECHNOLOGIES, INC. (US) 2009-01-06 US disclosed
EP-2007757-A2 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmceuticals Incorporated (US) 2008-12-31 EP disclosed
EP-2007732-A2 THIAZOLES, IMIDAZOLES, AND PYRAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals, Inc. (US) 2008-12-31 EP disclosed
US-7470511-B2 Methods for determining nucleic acid methylation RIBOMED BIOTECHNOLOGIES, INC. (US) 2008-12-30 US disclosed
EP-2004645-A2 PYRROLO(3,2-C) PYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals, Inc. (US) 2008-12-24 EP disclosed
US-7468462-B2 Therapeutic agents for the treatment of cancer, metabolic diseases and skin disorders AUSPEX PHARMACEUTICALS (US) 2008-12-23 US disclosed
US-7468261-B2 Molecular detection systems utilizing reiterative oligonucleotide synthesis RIBOMED BIOTECHNOLOGIES, INC. (US) 2008-12-23 US disclosed
US-20080311597-A1 Modified Cardiolipin and Uses Therefor THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES CENTERS FOR DISEASE CONTROL AND PREVENTION 2008-12-18 US disclosed
WO-2008147626-A2 THIAZOLES AND PYRAZOLES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-12-04 WO disclosed
WO-2008137619-A2 THIAZOLES AND PYRAZOLES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-11-13 WO disclosed
WO-2008137621-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-11-13 WO disclosed
WO-2008137622-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-11-13 WO disclosed
EP-1989205-A2 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmceuticals Incorporated (US) 2008-11-12 EP disclosed
WO-2008131103-A2 DRUG DISCOVERY METHODS FOR AURORA KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-10-30 WO disclosed
EP-1983987-A2 DIHYDRODIAZEPINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals Incorporated (US) 2008-10-29 EP disclosed
US-7442508-B2 Mixture of biological cells, used for detection and medical diagnosis of viruses; microbiology; Detecting and differentiating viruses or intracellular parasites present in a specimen; inoculating culture with pathogen and observing for its presence DIAGNOSTIC HYBRIDS, INC. (US) 2008-10-28 US disclosed
WO-2008128009-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-10-23 WO disclosed
US-7435588-B2 Systems for detection and production of respiratory, herpes and enteric viruses DIAGNOSTIC HYBRIDS, INC. (US) 2008-10-14 US disclosed
WO-2008115973-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-09-25 WO disclosed
EP-1971325-A2 CONJUGATED ESTROGEN COMPOSITIONS, APPLICATORS, KITS, AND METHODS OF MAKING AND USE THEREOF Duramed Pharmaceuticals, Inc. (US) 2008-09-24 EP disclosed
WO-2008112642-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-09-18 WO disclosed
WO-2008112651-A2 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-09-18 WO disclosed
WO-2008112646-A1 AMINOPYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-09-18 WO disclosed
WO-2008109723-A1 PHARMACEUTICAL ANALYSIS APPARATUS AND METHOD SMITHKLINE BEECHAM CORPORATION (US) 2008-09-12 WO disclosed
EP-1954277-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS Vertex Pharmceuticals Incorporated (US) 2008-08-13 EP disclosed
EP-1951716-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS Vertex Pharmaceuticals, Inc. (US) 2008-08-06 EP disclosed
EP-1951715-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2008-08-06 EP disclosed
EP-1948193-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2008-07-30 EP disclosed
EP-1949108-A2 MODIFIED CARDIOLIPIN AND USES THEREFOR THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2008-07-30 EP disclosed
WO-2008089405-A1 COMPOSITION OF MULTIPLE HORMONES DELIVERED VAGINALLY IN A SINGLE CREAM NEUROSCI, INC. (US) 2008-07-24 WO disclosed
EP-1945811-A2 SYSTEMS FOR DETECTION AND PRODUCTION OF RESPIRATORY, HERPES AND ENTERIC VIRUSES Diagnostic Hybrids (US) 2008-07-23 EP disclosed
US-20080167289-A1 Dihydrodiazepines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2008-07-10 US disclosed
WO-2008077086-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-06-26 WO disclosed
WO-2008076392-A2 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-06-26 WO disclosed
US-20080139556-A1 FKBP BINDING COMPOSITION AND PHARMACEUTICAL USE THEREOF AVENTIS PHARMACEUTICALS INC. (US) 2008-06-12 US disclosed
US-20080132481-A1 INTERLEUKIN-4 GENE EXPRESSION INHIBITORS AVENTIS PHARMACEUTICALS INC. 2008-06-05 US disclosed
WO-2008060597-A2 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-05-22 WO disclosed
WO-2008057940-A1 AMINOPYRIDINES AND AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-05-15 WO disclosed
EP-1919906-A1 3, 5-DISUBSTITUTED PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY OF NON-RECEPTOR TYROSINE KINASES Vertex Pharmaceuticals Incorporated (US) 2008-05-14 EP disclosed
EP-1919891-A1 3,5-DISUBSTITUTED PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY OF NON-RECEPTOR TYROSINE KINASES Vertex Pharmaceuticals Incorporated (US) 2008-05-14 EP disclosed
US-20080108546-A1 Novel Human Card-Only Protein That Inhibits Pro-Il-1 Beta Maturation VLAAMS INTERUNIVERSITAIR INSTITUUT (BE) 2008-05-08 US disclosed
US-20080076115-A1 Compositions and Methods for Detecting Severe Acute Respiratory Syndrome Coronavirus DIAGNOSTIC HYBRIDGS, INC. 2008-03-27 US disclosed
US-20080070965-A1 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2008-03-20 US disclosed
US-20080070882-A1 Vaginal cream compositions, kits thereof and methods of using thereof TEVA WOMEN'S HEALTH, INC. 2008-03-20 US disclosed
EP-1660487-B1 PYRROLE COMPOSITIONS USEFUL AS INHIBITORS OF C-MET VERTEX PHARMA (US) 2008-03-19 EP disclosed
US-20080051377-A1 Conjugated estrogen compositions, applicators, kits, and methods of making and use thereof DURAMED PHARMACEUTICALS, INC. (US) 2008-02-28 US disclosed
US-20080045570-A1 To treat autoimmune, inflammatory, proliferative, hyperproliferative,neurodegenerative or immunologically-mediated diseases; useful for the study of kinases in biological and pathological phenomena; study of intracellular signal transduction pathways mediated by such kinases, and comparative evaluation VERTEX PHARMACEUTICALS INCORPORATED 2008-02-21 US disclosed
US-20080032963-A1 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-02-07 US disclosed
US-20080004234-A1 System for delivering therapeutic agents into living cells and cells nuclei SEGEV LABORATORIES LIMITED (IL) 2008-01-03 US disclosed
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed
US-20070298065-A1 2-Cyclopentyl-4-(4-phenoxyphenyl)thiazole-5-carboxamide; amidation; oxidation; cyclization; VERTEX PHARMACEUTICALS INCORPORATED 2007-12-27 US disclosed
WO-2007139816-A2 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-12-06 WO disclosed
WO-2007139795-A1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-12-06 WO disclosed
EP-1622923-A4 MOLECULAR DETECTION SYSTEMS UTILIZING REITERATIVE OLIGONUCLEOTIDE SYNTHESIS RIBOMED BIOTECHNOLOGIES INC (US) 2007-11-28 EP disclosed
US-20070259869-A1 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-11-08 US disclosed
EP-1109552-A4 NOVEL DNA-CLEAVING ANTITUMOR AGENTS RES DEV FOUNDATION (US) 2007-11-07 EP disclosed
US-20070249031-A1 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-10-25 US disclosed
WO-2007120760-A2 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-10-25 WO disclosed
WO-2007120752-A2 4, 5-DIHYDRO- [1, 2, 4] TRIAZOLO [4, 3-F] PTERIDINES AS PROTEIN KINASE PLK1 INHIBITORS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-10-25 WO disclosed
WO-2007117692-A2 THIAZOLES, IMIDAZOLES, AND PYRAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-10-18 WO disclosed
US-20070219205-A1 Thiophene-carboxamides useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2007-09-20 US disclosed
EP-1834947-A2 3-substituted amino-1H-indole-2-carboxylic acid and 3-substituted amino-benzo[B]thiophene-2carboxylic acid derivatives as interleukin-4 gene expression inhibitors Aventis Pharmaceuticals, Inc. (US) 2007-09-19 EP disclosed
CN-101037438-A Compositions useful as inhibitors of GSK-3 VERTEX PHARMA (US) 2007-09-19 CN disclosed
US-20070213327-A1 Pyrrolo [3,2-C] pyridines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2007-09-13 US disclosed
EP-1831168-A1 PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY PROTEIN KINASES FOR THE TREATMENT OF INFLAMMATORY, PROLIFERATIVE AND IMMUNOLOGICALLY-MEDIATED DISEASES. Vertex Pharmaceuticals Incorporated (US) 2007-09-12 EP disclosed
WO-2007095188-A2 DIHYDRODIAZEPINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-08-23 WO disclosed
WO-2007095223-A2 PYRROLO(3,2-C) PYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-08-23 WO disclosed
US-20070191321-A1 Conjugated estrogen compositions, applicators, kits, and methods of making and use thereof TEVA WOMEN'S HEALTH, INC. 2007-08-16 US disclosed
EP-1814882-A1 PYRROLOPYRAZINES AND PYRAZOLOPYRAZINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals Incorporated (US) 2007-08-08 EP disclosed
US-20070179125-A1 Aminopyrimidines useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2007-08-02 US disclosed
US-20070179156-A1 Pyridones useful as inhibitors of kinases VERTEX PHARMACEUTICALS INCORPORATED 2007-08-02 US disclosed
WO-2007087283-A2 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-08-02 WO disclosed
EP-1812440-A1 PYRAZOLOÝ1,5-a¨PYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals, Inc. (US) 2007-08-01 EP disclosed
US-20070155794-A1 Pyridones useful as inhibitors of kinases VERTEX PHARMACEUTICALS INCORPORATED 2007-07-05 US disclosed
WO-2007076144-A2 CONJUGATED ESTROGEN COMPOSITIONS, APPLICATORS, KITS, AND METHODS OF MAKING AND USE THEREOF DURAMED PHARMACEUTICALS, INC. (US) 2007-07-05 WO disclosed
EP-1360274-B1 DETECTION OF MICRO-ORGANISMS MILLIPORE CORP (US) 2007-07-04 EP disclosed
EP-1485376-B1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2007-06-27 EP disclosed
WO-2007068310-A1 DEVICE FOR THE EARLY AND RAPID IMMUNOCHROMATOGRAPHIC DETECTION OF HIV AND USES THEREOF THE JORDANIAN PHARMACEUTICAL MANUFACTURING CO. (JO) 2007-06-21 WO disclosed
EP-1798556-A1 Device for the early and rapid immunochromatographic detection of HIV and uses thereof The Jordanian Pharmaceutical Manufacturing Co. (JO) 2007-06-20 EP disclosed
CN-1319968-C Pyrazole compositions useful as inhibitors of GSK-3 VERTEX PHARMA (US) 2007-06-06 CN disclosed
US-7226738-B2 Molecular detection systems utilizing reiterative oligonucleotide synthesis RIBOMED BIOTECHNOLOGIES, INC. (US) 2007-06-05 US disclosed
WO-2007061793-A2 MODIFIED CARDIOLIPIN AND USES THEREFOR THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SCIENCES, CENTERS FOR DISEASE CONTROL AND PREVENTION (US) 2007-05-31 WO disclosed
WO-2007059299-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-05-24 WO disclosed
WO-2007056164-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-05-18 WO disclosed
WO-2007056221-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-05-18 WO disclosed
WO-2007056163-A2 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-05-18 WO disclosed
EP-1147188-B1 INTERNAL RIBOSOME ENTRY SITE (IRES), VECTOR CONTAINING SAME AND THE USES THEREOF VLAAMS INTERUNIV INST BIOTECH (BE) 2007-05-16 EP disclosed
EP-1784192-A2 VAGINAL CREAM COMPOSITIONS, KITS THEREOF AND METHODS OF USING THEREOF Duramed Pharmaceuticals, Inc. (US) 2007-05-16 EP disclosed
EP-1501796-B1 3-(PYRIDINYL-AMINO)-1H-INDOLE-2-CARBOXYLIC ACID DERIVATIVES AS INTERLEUKIN-4 GENE EXPRESSION INHIBITORS AVENTIS PHARMA INC (US) 2007-05-09 EP disclosed
US-20070099296-A1 Compositions and methods for determining susceptibility of hepatitis C virus to anti-viral drugs MONOGRAM BIOSCIENCES, INC. 2007-05-03 US disclosed
EP-1778637-A2 FKBP BINDING COMPOSITION AND PHARMACEUTICAL USE THEREOF Aventis Pharmaceuticals, Inc. (US) 2007-05-02 EP disclosed
US-20070078189-A1 Novel therapeutic agents for the treatment of cancer, metabolic diseases and skin disorders AUSPEX PHARMACEUTICALS (US) 2007-04-05 US disclosed
WO-2007035856-A2 SYSTEMS FOR DETECTION AND PRODUCTION OF RESPIRATORY, HERPES AND ENTERIC VIRUSES DIAGNOSTIC HYBRIDS (US) 2007-03-29 WO disclosed
EP-1765819-A1 AZAINDOLES USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals Incorporated (US) 2007-03-28 EP disclosed
US-20070065939-A1 Systems for detection and production of respiratory, herpes and enteric viruses UNIVERSITY HOSPITALS OF CLEVELAND (US) 2007-03-22 US disclosed
WO-2007027729-A1 3, 5-DISUBSTITUTED PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY OF NON-RECEPTOR TYROSINE KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-03-08 WO disclosed
WO-2007027594-A1 3,5-DISUBSTITUTED PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY OF NON-RECEPTOR TYROSINE KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-03-08 WO disclosed
US-20070048774-A1 Continuous in-vitro evolution DIATECH PTY LTD. 2007-03-01 US disclosed
US-20070042403-A1 Specific inhibitors of NFAT activation by calcineurin and their use in treating immune-related diseases CENTER FOR BLOOD RESEARCH, INC. 2007-02-22 US disclosed
EP-1751182-A1 A NOVEL HUMAN CARD-ONLY PROTEIN THAT INHIBITS PRO-IL-1 BETA; MATURATION VIB vzw (BE) 2007-02-14 EP disclosed
US-7169925-B2 Indole derivatives as interleukin-4 gene expression inhibitors AVENTIS PHARMACEUTICALS INC. (US) 2007-01-30 US disclosed
EP-1739087-A1 Pyrazole compositions useful as inhibitors of gsk-3 Vertex Pharmaceuticals Incorporated (US) 2007-01-03 EP disclosed
US-20060286667-A1 Mixture of biological cells, used for detection and medical diagnosis of viruses; microbiology; Detecting and differentiating viruses or intracellular parasites present in a specimen; inoculating culture with pathogen and observing for its presence DIAGNOSTIC HYBRIDS, INC. (US) 2006-12-21 US disclosed
US-20060258662-A1 Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2006-11-16 US disclosed
EP-1716151-A1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals Incorporated (US) 2006-11-02 EP disclosed
US-7129042-B2 detecting the presence SARS-coronavirus sgRNA in a sample; DIAGNOSTIC HYBRIDS, INC. (US) 2006-10-31 US disclosed
US-20060236435-A1 Chimeric plant promoters and plants containing the same MERISTEM THERAPEUTICS 2006-10-19 US disclosed
EP-1385840-B1 SULFONAMIDES SMITHKLINE BEECHAM CORP (US) 2006-10-04 EP disclosed
US-20060204964-A1 Molecular detection systems utilizing reiterative oligonucleotide synthesis HANNA MICHELLE M 2006-09-14 US disclosed
EP-1451366-A4 MOLECULAR DETECTION SYSTEMS UTILIZING REITERATIVE OLIGONUCLEOTIDE SYNTHESIS RIBOMED BIOTECHNOLOGIES INC (US) 2006-09-13 EP disclosed
EP-1532145-B1 PYRAZOLE COMPOSITIONS USEFUL AS INHIBITORS OF GSK-3 VERTEX PHARMA (US) 2006-09-13 EP disclosed
US-20060188942-A1 Detection of Micro-Organisms MICAP PLC (GB) 2006-08-24 US disclosed
EP-1692140-A1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals Incorporated (US) 2006-08-23 EP disclosed
US-20060183911-A1 Pyridones useful as inhibitors of kinases VERTEX PHARMACEUTICALS INCORPORATED 2006-08-17 US disclosed
US-7091204-B2 Sulfonamides SMITHKLINE BEECHAM CORPORATION (US) 2006-08-15 US disclosed
US-20060177640-A1 Laminated film and method for producing same TORAY INDUSTRIES, INC. (JP) 2006-08-10 US disclosed
US-20060173055-A1 (4-(4-(2,3-difluorophenyl)-4H-1,2,4-triazol-3-yl)-1H-pyrrol-2-yl)(2H-pyrrol-1(5H)-yl)methanone; anticarcinogenic, antiproliferative and antimetastasis agent; inhibitors of c-Met protein kinase VERTEX PHARMACEUTICALS INCORPORATED 2006-08-03 US disclosed
CN-1812973-A Indazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICAL CO LTD (US) 2006-08-02 CN disclosed
US-7084241-B2 Specific inhibitors of NFAT activation by calcineurin and their use in treating immune-related diseases THE CBR INSTITUTE FOR BIOMEDICAL RESEARCH, INC. (US) 2006-08-01 US disclosed
US-20060166936-A1 Diaminotriazole compounds useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2006-07-27 US disclosed
US-20060160763-A1 System for delivering therapeutic agents into living cells and cells nuclei SEGEV LABORATORIES LIMITED (IL) 2006-07-20 US disclosed
EP-1220935-B1 SYNTHETIC AND CHIMERIC PROMOTERS, EXPRESSION CASSETTES, PLASMIDS, VECTORS, TRANSGENIC PLANTS AND SEEDS CONTAINING THEM, AND METHOD FOR PRODUCING THEM MERISTEM THERAPEUTICS (FR) 2006-07-19 EP disclosed
WO-2006065946-A1 PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY PROTEIN KINASES FOR THE TREATMENT OF INFLAMMATORY, PROLIFERATIVE AND IMMUNOLOGICALLY-MEDIATED DISEASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-06-22 WO disclosed
US-20060135537-A1 Pyrazolo[1,5-a]pyrimidines useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2006-06-22 US disclosed
US-20060122213-A1 Azaindoles useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2006-06-08 US disclosed
WO-2006058074-A1 PYRROLOPYRAZINES AND PYRAZOLOPYRAZINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-06-01 WO disclosed
EP-1660487-A1 PYRROLE COMPOSITIONS USEFUL AS INHIBITORS OF C-MET Vertex Pharmaceuticals Incorporated (US) 2006-05-31 EP disclosed
WO-2006052913-A1 PYRAZOLO[1,5-a]PYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-05-18 WO disclosed
US-7045319-B2 Molecular detection systems utilizing reiterative oligonucleotide synthesis RIBOMED BIOTECHNOLOGIES, INC. (US) 2006-05-16 US disclosed
WO-2006050249-A1 DIAMINOTRIAZOLE COMPOUNDS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-05-11 WO disclosed
US-7041687-B2 Indazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-05-09 US disclosed
US-20060094105-A1 Mixed cell diagnostic systems for detection of respiratory, herpes and enteric viruses UNIVERSITY HOSPITALS OF CLEVELAND (US) 2006-05-04 US disclosed
US-7026349-B2 Sulfonamides SMITHKLINE BEECHAM CORPORATION (US) 2006-04-11 US disclosed
US-7019008-B2 Pyrrolidine sulfonamides SMITHKLINE BEECHAM CORPORATION (US) 2006-03-28 US disclosed
WO-2006023496-A2 VAGINAL CREAM COMPOSITIONS, KITS THEREOF AND METHODS OF USING THEREOF DURAMED PHARMACEUTICALS, INC. (US) 2006-03-02 WO disclosed
CN-1243545-C DNA-cleaving antitumor agents RES DEV FOUNDATION (US) 2006-03-01 CN disclosed
US-20060040904-A1 Vaginal cream compositions, kits thereof and methods of using thereof DURAMED PHARMACEUTICALS, INC. 2006-02-23 US disclosed
EP-1622923-A2 MOLECULAR DETECTION SYSTEMS UTILIZING REITERATIVE OLIGONUCLEOTIDE SYNTHESIS Ribomed Biotechnologies, Inc. (US) 2006-02-08 EP disclosed
WO-2006012256-A2 FKBP BINDING COMPOSITION AND PHARMACEUTICAL USE THEREOF AVENTIS PHARMACEUTICALS INC. (US) 2006-02-02 WO disclosed
WO-2006010084-A2 A SYSTEM FOR DELIVERING THERAPEUTIC AGENTS INTO LIVING CELLS AND CELL NUCLEI SEGEV LABORATORIES LIMITED (IL) 2006-01-26 WO disclosed
US-20060008895-A1 Microarray chip for detection of immunoglobulin CHENG LOONG CORPORATION (TW) 2006-01-12 US disclosed
WO-2006004984-A1 AZAINDOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-12 WO disclosed
EP-1351688-A4 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2006-01-04 EP disclosed
EP-1385495-A4 SULFONAMIDES SMITHKLINE BEECHAM CORP (US) 2005-12-21 EP disclosed
EP-1165815-B1 CHIMERIC EXPRESSION PROMOTERS ORIGINATING FROM COMMELINA YELLOW MOTTLE VIRUS AND CASSAVA VEIN MOSAIC VIRUS MERISTEM THERAPEUTICS (FR) 2005-12-21 EP disclosed
WO-2005118632-A1 A NOVEL HUMAN CARD-ONLY PROTEIN THAT INHIBITS PRO-IL-1β MATURATION VIB VZW (BE) 2005-12-15 WO disclosed
EP-1399137-A4 SULFONAMIDES SMITHKLINE BEECHAM CORP (US) 2005-12-14 EP disclosed
EP-1385840-A4 SULFONAMIDES SMITHKLINE BEECHAM CORP (US) 2005-11-23 EP disclosed
EP-1385507-A4 SULFONAMIDES SMITHKLINE BEECHAM CORP (US) 2005-11-23 EP disclosed
US-6963021-B2 Chimeric expression promoters originating from commelina yellow mottle virus and cassava vein mosaic virus MERISTEM THERAPEUTICS (FR) 2005-11-08 US disclosed
WO-2005094324-A2 MIXED CELL DIAGNOSTIC SYSTEMS DIAGNOSTIC HYBRIDS, INC. (US) 2005-10-13 WO disclosed
WO-2005095406-A1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-10-13 WO disclosed
CN-1681815-A Pyrazole compositions useful as inhibitors of GSK-3 VERTEX PHARMA (US) 2005-10-12 CN disclosed
EP-1582340-A1 LAMINATED FILM AND METHOD FOR PRODUCING SAME TORAY INDUSTRIES, INC. (JP) 2005-10-05 EP disclosed
US-20050209255-A1 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2005-09-22 US disclosed
EP-0804565-B1 TETRACYCLINE-REGULATED TRANSCRIPTIONAL MODULATORS TET SYSTEMS HOLDING GMBH & CO (DE) 2005-09-21 EP disclosed
EP-1575365-A1 ACTIVE INSECTICIDE MATERIAL, PREPARATION METHOD AND USES THEREOF UNIVERSITE JOSEPH FOURIER (GRENOBLE 1) (FR) 2005-09-21 EP disclosed
US-6946291-B2 Mixed cell diagnostic systems UNIVERSITY HOSPITALS OF CLEVELAND (US) 2005-09-20 US disclosed
US-20050197345-A1 urotensin II receptor antagonists; cardiovascular disorders; vasodilating agents; Benzo[b]thiophene-2-carboxylic acid [(S)-1-(2-{4-[3-chloro-4-(piperidin-4-yloxy)-benzenesulfonyl]-piperazin-1-yl}-ethylcarbamoyl)-3-methyl-butyl]- SMITHKLINE BEECHAM CORPORATION 2005-09-08 US disclosed
EP-1385830-A4 SULFONAMIDES SMITHKLINE BEECHAM CORP (US) 2005-08-17 EP disclosed
US-6919470-B2 Aryl and heteroaryl sulfonates BAYER AKTIENGESELLSCHAFT (DE) 2005-07-19 US disclosed
US-20050148603-A1 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2005-07-07 US disclosed
US-6914124-B2 Tetracycline-regulated transcriptional activator fusion proteins TET SYSTEMS HOLDING GMBH & CO. KG (DE) 2005-07-05 US disclosed
US-6908948-B1 DNA-cleaving antitumor agents RESEARCH DEVELOPMENT FOUNDATION (US) 2005-06-21 US disclosed
US-20050112142-A1 Methods and compositions for treatment and prevention of HSV-2 infections and conditions MEDIMMUNE, LLC 2005-05-26 US disclosed
EP-1532145-A1 PYRAZOLE COMPOSITIONS USEFUL AS INHIBITORS OF GSK-3 Vertex Pharmaceuticals Incorporated (US) 2005-05-25 EP disclosed
WO-2005042767-A2 COMPOSITIONS AND METHODS FOR DETECTING SEVERE ACUTE RESPIRATORY SYNDROME CORONAVIRUS DIAGNOSTIC HYBRIDS, INC. (US) 2005-05-12 WO disclosed
US-20050101650-A1 Pyrrole compositions useful as inhibitors of c-Met VERTEX PHARMACEUTICALS INCORPORATED 2005-05-12 US disclosed
US-20050095582-A1 Compositions and methods for detecting severe acute respiratory syndrome coronavirus DIAGNOSTIC HYBRIDS, INC. (US) 2005-05-05 US disclosed
WO-2005037843-A1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-04-28 WO disclosed
US-20050064414-A1 Molecular detection systems utilizing reiterative oligonucleotide synthesis RIBOMED BIOTECHNOLOGIES, INC. 2005-03-24 US disclosed
EP-1381365-A4 PYRROLIDINE SULFONAMIDES SMITHKLINE BEECHAM CORP (US) 2005-03-23 EP disclosed
EP-0722492-B1 STABILISATION OF PROTEINS IN SOLUTION UNIV LEEDS INNOVATIONS LTD (GB) 2005-03-09 EP disclosed
EP-1385841-A4 SULFONAMIDES SMITHKLINE BEECHAM CORP (US) 2005-03-02 EP disclosed
US-20050043536-A1 antagonists of urotensin II; for example, 2,6-Dichloro-N-[3-(dimethylamino-ethoxy)4-trifluoromethyl-phenyl]-4trifluoromethyl-benzenesulfonamide SMITHKLINE BEECHAM CORPORATION 2005-02-24 US disclosed
WO-2005016920-A1 PYRROLE COMPOSITIONS USEFUL AS INHIBITORS OF C-MET VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-02-24 WO disclosed
US-20050026150-A1 Molecular detection systems utilizing reiterative oligonucleotide synthesis RIBOMED BIOTECHNOLOGIES, INC. 2005-02-03 US disclosed
EP-1501797-A1 3-SUBSTITUTED AMINO-1H-INDOLE-2-CARBOXYLIC ACID AND 3-SUBSTITUTED AMINO-BENZO[B]THIOPHENE-2-CARBOXYLIC ACID DERIVATIVES AS INTERLEUKIN-4 GENE EXPRESSION INHIBITORS Aventis Pharmaceuticals, Inc. (US) 2005-02-02 EP disclosed
EP-1501796-A1 3-SUBSTITUTED AMINO-1H-INDOLE-2-CARBOXYLIC ACID AND 3-SUBSTITUTED AMINO-BENZO[B]THIOPHENE-2-CARBOXYLIC ACID DERIVATIVES AS INTERLEUKIN-4 GENE EXPRESSION INHIBITORS Aventis Pharmaceuticals Inc. (US) 2005-02-02 EP disclosed
US-6849635-B2 Sulfonamides SMITHKLINE BEECHAM CORPORATION (US) 2005-02-01 US disclosed
US-6846928-B2 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-01-25 US disclosed
EP-1485376-A1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals Incorporated (US) 2004-12-15 EP disclosed
US-20040234996-A1 Molecular detection systems utilizing reiterative oligonucleotide synthesis RIBOMED BIOTECHNOLOGIES, INC. 2004-11-25 US disclosed
US-6818655-B2 2-AMINOQUINOLINES; CARDIOVASCULAR, GASTROINTESTINAL, PYSCHOLOGICAL, RESPIRATORY AND NERVOUS SYSTEM DISORDERS SMITHKLINE BEECHAM CORPORATION 2004-11-16 US disclosed
WO-2004096997-A2 MOLECULAR DETECTION SYSTEMS UTILIZING REITERATIVE OLIGONUCLEOTIDE SYNTHESIS RIBOMED BIOTECHNOLOGIES, INC. (US) 2004-11-11 WO disclosed
US-20040214886-A1 Phenoxyphenyl alkanesulphonates BAYER AKTIENGESELLSCHAFT (DE) 2004-10-28 US disclosed
EP-1467972-A1 INDAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2004-10-20 EP disclosed
EP-1246619-B1 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-10-20 EP disclosed
US-20040198979-A1 Sulfonamides SMITHKLINE BEECHAM CORPORATION 2004-10-07 US disclosed
EP-1248607-A4 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-10-06 EP disclosed
US-20040175724-A1 Molecular detection systems utilizing reiterative oligonucleotide synthesis DESIGNER GENES, INC. 2004-09-09 US disclosed
US-20040170965-A1 Mixed cell diagnostic systems QUIDEL CORPORATION 2004-09-02 US disclosed
EP-1451366-A2 MOLECULAR DETECTION SYSTEMS UTILIZING REITERATIVE OLIGONUCLEOTIDE SYNTHESIS Ribomed Biotechnologies, Inc. (US) 2004-09-01 EP disclosed
US-6783756-B2 INTRODUCING INTO THE CELL A NUCLEIC ACID MOLECULE ENCODING A TETRACYCLINE-CONTROLLABLE TRANSACTIVATOR (TTA) COMPRISING TET REPRESSOR OPERABLY LINKED TO A POLYPEPTIDE WHICH OR ACTIVATES TRANSCRIPTION IN EUCARYOTIC CELL; MODULATING ABBOTT GMBH & CO., KG (DE) 2004-08-31 US disclosed
WO-2004069200-A2 SPECIFIC INHIBITORS OF NFAT ACTIVATION BY CALCINEURIN AND THEIR USE IN TREATING IMMUNE-RELATED DISEASES THE CBR INSTITUTE FOR BIOMEDICAL RESEARCH, INC. (US) 2004-08-19 WO disclosed
US-20040157257-A1 Abortive promoter cassettes RIBOMED BIOTECHNOLOGIES, INC. (US) 2004-08-12 US disclosed
EP-0642666-B2 HEPATITIS C ASSAY ABBOTT LAB (US) 2004-08-11 EP disclosed
EP-1387679-A4 SULFONAMIDES SMITHKLINE BEECHAM CORP (US) 2004-08-11 EP disclosed
US-20040152893-A1 Sulfonamides SMITHKLINE BEECHAM CORPORATION 2004-08-05 US disclosed
US-20040152895-A1 Sulfonamides SMITHKLINE BEECHAM CORPORATION 2004-08-05 US disclosed
WO-2004064525-A1 ACTIVE INSECTICIDE MATERIAL, PREPARATION METHOD AND USES THEREOF UNIVERSITE JOSEPH FOURIER (GRENOBLE 1) (FR) 2004-08-05 WO disclosed
US-20040152906-A1 Sulfonamides SHELL OIL COMPANY 2004-08-05 US disclosed
US-20040152692-A1 Urotensin antagonist; therapy for congestive heart failure; antiischemic agents; cardiovascular disorders; strokes; hypotensive agents; respiratory system disorders; restenosis; antiinflammatory agents; psychological disorders SMITHKLINE BEECHAM CORPORATION 2004-08-05 US disclosed
US-20040152891-A1 Sulfonamides SMITHKLINE BEECHAM CORPORATION 2004-08-05 US disclosed
US-20040142948-A1 Sulfonamides DHANAK DASHYANT (US) 2004-07-22 US disclosed
US-20040142923-A1 Pyrrolidine sulfonamides SMITHKLINE BEECHAM CORPORATION 2004-07-22 US disclosed
EP-1359915-A4 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM (US) 2004-07-21 EP disclosed
US-6764852-B2 NUCLEOTIDE SEQUENCE ENABLING A CELL CYCLE DEPENDENT INITIATION OF TRANSLATION OF MRNA. VLAAMS INTERUNIVERSITAIR INSTITUUT VOOR BIOTECHNOLOGIE VZW (BE) 2004-07-20 US disclosed
US-20040137461-A1 Molecular detection systems utilizing reiterative oligonucleotide synthesis DESIGNER GENES, INC. 2004-07-15 US disclosed
US-20040138224-A1 Pyrrolidine sulfonamides SMITHKLINE BEECHAM CORPORATION 2004-07-15 US disclosed
US-20040131701-A1 Method to treat infectious diseases and/or to enhance antimicrobial efficacy of drugs VIROCELL INC. 2004-07-08 US disclosed
US-6756409-B2 FOR THERAPY AND PROPHYLAXIS OF PAIN AND/OR NEURODEGENERATIVE DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 2004-06-29 US disclosed
EP-1233774-A4 UROTENSIN-II ANALOGS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
WO-2004043368-A2 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2004-05-27 WO disclosed
WO-2004043948-A1 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2004-05-27 WO disclosed
WO-2004043366-A2 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2004-05-27 WO disclosed
WO-2004043917-A1 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2004-05-27 WO disclosed
WO-2004043463-A2 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2004-05-27 WO disclosed
WO-2004043369-A2 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2004-05-27 WO disclosed
US-20040096821-A1 Detection of micro-organisms EMD MILLIPORE CORPORATION 2004-05-20 US disclosed
US-20040082566-A1 Pyrrolidine sulfonamides SMITHKLINE BEECHAM CORPORATION 2004-04-29 US disclosed
US-20040063757-A1 Urotensin-ll receptor antagonists SMITHKLINEE BEECHAM CORPORATION 2004-04-01 US disclosed
EP-1399137-A1 SULFONAMIDES SmithKline Beecham Corporation (US) 2004-03-24 EP disclosed
US-20040054162-A1 Molecular detection systems utilizing reiterative oligonucleotide synthesis RIBOMED BIOTECHNOLOGIES, INC. 2004-03-18 US disclosed
US-20040053963-A1 Urotensin-II receptor antagonists SMITHKLINE BEECHAM CORPORATION 2004-03-18 US disclosed
EP-1198554-B1 DETECTION OF MICRO-ORGANISMS MICAP PLC (GB) 2004-03-10 EP disclosed
US-6703211-B1 CELLULAR DETECTION EVEN IN A LARGE BACKGROUND OF ADENOSINE TRIPHOSPHATE (ATP) IN THE SAMPLE, USES ENDOGENOUS ENZYMES TO CONVERT ADENOSINE MONOPHOSPHATE (AMP) TO ATP AND DCTP; FOOD AND WATER SAFETY PROMEGA CORPORATION 2004-03-09 US disclosed
US-20040039017-A1 Urotensin-II receptor antagonists SMITHKLINE BEECHAM CORPORATION 2004-02-26 US disclosed
US-20040039007-A1 Compositions useful as inhibitors of GSK-3 VERTEX PHARMACEUTICALS INCORPORATED 2004-02-26 US disclosed
WO-2004013140-A1 PYRAZOLE COMPOSITIONS USEFUL AS INHIBITORS OF GSK-3 VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-02-12 WO disclosed
EP-1387679-A1 SULFONAMIDES SmithKline Beecham Corporation (US) 2004-02-11 EP disclosed
EP-1385840-A1 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2004-02-04 EP disclosed
EP-1385841-A1 SULFONAMIDES SmithKline Beecham Corporation (US) 2004-02-04 EP disclosed
EP-1385507-A1 SULFONAMIDES SmithKline Beecham Corporation (US) 2004-02-04 EP disclosed
EP-1385830-A1 SULFONAMIDES SmithKline Beecham Corporation (US) 2004-02-04 EP disclosed
EP-1385495-A2 SULFONAMIDES SmithKline Beecham Corporation (US) 2004-02-04 EP disclosed
US-6686345-B2 INCLUDES AN AZA-ENEDIYNE, AZA-ENYNE ALLENE, OR AN AZA-DIALLENE; ARE PREFERABLY NON-HYDROLYZABLE, CATIONIC COMPOUNDS THAT BIND TO NUCLEIC ACIDS. RESEARCH DEVELOPMENT FOUNDATION 2004-02-03 US disclosed
US-20040018606-A1 Control of protein systemic delivery by hypoxia using a tet-HIF1-alpha chimeric transactivator BOHL DELPHINE (FR) 2004-01-29 US disclosed
EP-1381365-A1 PYRROLIDINE SULFONAMIDES SmithKline Beecham Corporation (US) 2004-01-21 EP disclosed
EP-1351687-A4 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-01-21 EP disclosed
US-20040010029-A1 Indole derivatives as interleukin -4 gene expression inhibitors AVENTIS PHARMACEUTICALS INC. 2004-01-15 US disclosed
US-20040009968-A1 Indazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2004-01-15 US disclosed
EP-1379237-A2 PYRROLIDINE SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2004-01-14 EP disclosed
EP-1379519-A1 PYRROLIDINE SULFONAMIDES SmithKline Beecham Corporation (US) 2004-01-14 EP disclosed
EP-1379503-A1 PYRROLIDINE SULFONAMIDES SmithKline Beecham Corporation (US) 2004-01-14 EP disclosed
US-6677157-B1 SIGNIFICANT REDUCTION OR ABSENCE OF PROSTATE SECRETORY GRANULES, EOSINOPHILIC BODIES, DECAPITATED CYTOPLASMIC BODIES AND/OR CORPORA AMYLACEA INDICATIVE OF ADENOCARCINOMA UROPATH PTY LTD., A.C.N. (AU) 2004-01-13 US disclosed
US-20040006123-A1 Interleukin-4 gene expression inhibitors AVENTIS PHARMACEUTICALS INC. 2004-01-08 US disclosed
US-20040002117-A1 Specific inhibitors of NFAT activation by calcineurin and their use in treating immune-related diseases CBR INSTITUTE OF BIOMEDICAL RESEARCH, INC., THE 2004-01-01 US disclosed
US-20040003417-A1 ANIMALS TRANSGENIC FOR A TETRACYCLINE-REGULATED TRANSCRIPTIONAL INHIBITOR TET SYSTEMS HOLDING GMBH & CO. KG (DE) 2004-01-01 US disclosed
US-20030232802-A1 Aryl and heteroaryl sulfonates HEIL MARKUS (DE) 2003-12-18 US disclosed
US-20030225073-A1 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2003-12-04 US disclosed
US-20030221204-A1 BRI constructs and methods of using MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH 2003-11-27 US disclosed
WO-2003093492-A2 COMPOSITIONS AND METHODS FOR DETERMINING SUSCEPTIBILITY OF HEPATITIS C VIRUS TO ANTI-VIRAL DRUGS VIROLOGIC, INC. (US) 2003-11-13 WO disclosed
EP-1360274-A1 DETECTION OF MICRO-ORGANISMS Fluid Technologies Plc (GB) 2003-11-12 EP disclosed
EP-1359915-A1 UROTENSIN-II RECEPTOR ANTAGONISTS Smithkline Beecham (US) 2003-11-12 EP disclosed
WO-2003091215-A1 3-SUBSTITUTED AMINO-1H-INDOLE-2-CARBOXYLIC ACID AND 3-SUBSTITUTED AMINO-BENZO’ B! THIOPHENE-2-CARBOXYLIC ACID DERIVATIVES AS INTERIEUKIN-4 GENE EXPRESSION INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2003-11-06 WO disclosed
WO-2003091214-A1 3-SUBSTITUTED AMINO-1H-INDOLE-2-CARBOXYLIC ACID AND 3-SUBSTITUTED AMINO-BENZO AVENTIS PHARMACEUTICALS INC. (US) 2003-11-06 WO disclosed
US-20030203356-A1 RNase L activator-antisense complexes THE CLEVELAND CLINIC FOUNDATION (US) 2003-10-30 US disclosed
EP-1351688-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2003-10-15 EP disclosed
EP-1351687-A2 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2003-10-15 EP disclosed
US-6627735-B2 Nucleotide sequences coding polypeptide for use in the treatment and diagnosis of diabetes ZYMOGENETICS, INC. 2003-09-30 US disclosed
WO-2003078423-A1 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS, INC. (US) 2003-09-25 WO disclosed
EP-1343507-A2 METHOD TO TREAT INFECTIOUS DISEASES AND/OR TO ENHANCE ANTIMICROBIAL EFFICACY OF DRUGS Virocell Inc. (CA) 2003-09-17 EP disclosed
EP-1244452-B1 CARBOXAMIDE DERIVATES OF PYRROLIDINE AND PIPERIDINE AS UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2003-09-17 EP disclosed
US-20030170820-A1 Continuous in- vitro evolution DIATECH PTY LTD. (AU) 2003-09-11 US disclosed
US-20030166067-A1 Comprises nucleotide sequences coding pancreatic polypeptide comprising tyrosine phosphatase activity for use in diagnosing, preventing and treating diabetes and autoimmune disorders; immunoassay; drug screening ZYMOGENETICS, INC. 2003-09-04 US disclosed
US-6605639-B1 Treating and/or preventing diseases alleviated by retinoid X receptor ligand dependent transcriptional regulation using ascochlorin or derivatives NUCLEAR RECEPTOR RESEARCH, LTD. (JP) 2003-08-12 US disclosed
WO-2003064397-A1 INDAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2003-08-07 WO disclosed
WO-2003062258-A1 RNASE L ACTIVATOR-ANTISENSE COMPLEXES THE CLEVELAND CLINIC FOUNDATION (US) 2003-07-31 WO disclosed
US-20030138774-A1 Methods and apparatus for separating and detecting nucleic acid EXACT SCIENCES CORPORATION 2003-07-24 US disclosed
US-6596476-B1 Kit for use in detection of viral diseases ABBOTT LABORATORIES 2003-07-22 US disclosed
US-6593083-B1 For the detection of antibodies in body fluids; contacting the sample with polypeptide or fusion protein; detecting the antibody-polypeptide complex DEVARE SUSHIL G (US) 2003-07-15 US disclosed
US-20030100580-A1 Urotensin-II receptor antagonists SMITHKLINE BEECHAM CORPORATION 2003-05-29 US disclosed
US-20030099950-A1 Molecular detection systems utilizing reiterative oligonucleotide synthesis RIBOMED BIOTECHNOLOGIES, INC. 2003-05-29 US disclosed
EP-0925369-B1 UNIVERSAL TEST SYSTEMS AND METHODS OF USE THEREOF FOR IDENTIFYING MULTIPLE FAMILIES OF MICROORGANISMS DADE MICROSAN INC (US) 2003-05-28 EP disclosed
WO-2003038042-A2 MOLECULAR DETECTION SYSTEMS UTILIZING REITERATIVE OLIGONUCLEOTIDE SYNTHESIS RIBOMED BIOTECHNOLOGIES, INC. (US) 2003-05-08 WO disclosed
EP-1233776-A4 UROTENSIN-II CYCLIC ANALOGS SMITHKLINE BEECHAM CORP (US) 2003-05-07 EP disclosed
EP-1246619-A4 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2003-05-02 EP disclosed
US-6548609-B2 Epoxidation of vegetable oils using organic acid with oxygenated water or peracetic acid to obtain epoxydized oils and/or mixtures of esters of epoxydized unsaturated acids; reacting with alcohol or amine or alcoholamine RESINAS Y MATERIALES S.A. DE C.V. (MX) 2003-04-15 US disclosed
US-6544992-B1 Carbonylamino pyrrolidine and piperidine derivatives SMITHKLINE BEECHAM CORPORATION 2003-04-08 US disclosed
EP-1107665-A4 METHOD OF DIAGNOSIS OF PROSTATE CANCER UROPATH PTY LTD (AU) 2003-04-02 EP disclosed
EP-1293575-A2 Universal test system and methods of use thereof for indentifying multiple families of microorganisms Dade Microsan Inc. (US) 2003-03-19 EP disclosed
EP-1285965-A1 Bifactorial endosperm box, trans-activating factor that binds thereto, and method of regulation of promoter activity MERISTEM THERAPEUTICS (FR) 2003-02-26 EP disclosed
WO-2003014349-A1 BIFACTORIAL ENDOSPERM BOX, TRANS-ACTIVATING FACTOR THAT BINDS THERETO, AND METHOD OF REGULATION OF PROMOTER ACTIVITY MERISTEM THERAPEUTICS SA (FR) 2003-02-20 WO disclosed
US-20030028011-A1 Compositions and methods for determining susceptibility of hepatitis C virus to anti-viral drugs VIROLOGIC, INC. 2003-02-06 US disclosed
US-20030028922-A1 Chimeric expression promoters originating from commelina yellow mottle virus and cassava vein mosaic virus MERISTEM THERAPEUTICS (FR) 2003-02-06 US disclosed
US-6514970-B1 Pyrrolidines such as benzo(b)thiophene-2-carboxylic acid ((S)-1-((S)-1-(4-(1-benzyl-piperidin-4-yloxy)-3-chloro-benzyl)-pyrrolidin-3 -ylcarbamoyl)-3- methyl-butyl)-amide SMITHKLINE BEECHAM CORPORATION 2003-02-04 US disclosed
US-20030022315-A1 Tetracycline-inducible transcriptional inhibitor fusion proteins BASF AKTIENGESELLSCHAFT AND KNOLL AKTIENGESELLSCHAFT 2003-01-30 US disclosed
US-20030022934-A1 Phenoxyphenyl alkanesulphonates BAYER AKTIENGESELLSCHAFT (DE) 2003-01-30 US disclosed
US-6511812-B1 Adding denatured and/or purified bacterial enzyme; recombinant antigens expressed as fusion proteins with a bacterial enzyme which is CKS ABBOTT LABORATORIES 2003-01-28 US disclosed
EP-1244452-A4 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2003-01-15 EP disclosed
WO-2001053817-A9 METHODS OF AND APPARATUS FOR SEPARATING AND DETECTING NUCLEIC ACID MOSAIC TECHNOLOGIES (US) 2003-01-09 WO disclosed
WO-2003002754-A2 BRI CONSTRUCTS AND METHODS OF USING MAYO FOUNDATION FOR MEDICAL EDUCATION & RESEARCH (US) 2003-01-09 WO disclosed
EP-1105428-A4 NOVEL CLEAVED FRAGMENTS OF FIBRINOGEN NEW YORK BLOOD CT INC (US) 2003-01-02 EP disclosed
WO-2002089785-A1 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-11-14 WO disclosed
US-20020168722-A1 Novel cleaved fragments of fibrinogen NATIONAL INSTITUTES OF HEALTH-DEITR 2002-11-14 US disclosed
WO-2002090337-A1 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-11-14 WO disclosed
WO-2002089792-A1 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-11-14 WO disclosed
WO-2002090348-A1 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-11-14 WO disclosed
WO-2002090353-A1 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-11-14 WO disclosed
WO-2002089740-A2 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-11-14 WO disclosed
WO-2002089793-A1 SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-11-14 WO disclosed
EP-1255983-A2 METHODS OF AND APPARATUS FOR SEPARATING AND DETECTING NUCLEIC ACID Mosaic Technologies (US) 2002-11-13 EP disclosed
US-20020155443-A1 Metal binding DNA interactive compounds BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2002-10-24 US disclosed
US-20020152487-A1 Transgenic organisms having tetracycline-regulated transcriptional regulatory systems BASF AKTIENGESELLSCHAFT 2002-10-17 US disclosed
US-20020152489-A1 Transgenic organisms having tetracycline-regulated transcriptional regulatory systems BASF AKTIENGESELLSCHAFT 2002-10-17 US disclosed
EP-1248607-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-10-16 EP disclosed
WO-2002078641-A2 PYRROLIDINE SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-10-10 WO disclosed
WO-2002079155-A1 PYRROLIDINE SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-10-10 WO disclosed
WO-2002078707-A1 PYRROLIDINE SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-10-10 WO disclosed
WO-2002079188-A1 PYRROLIDINE SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-10-10 WO disclosed
EP-1246619-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2002-10-09 EP disclosed
EP-1244452-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-10-02 EP disclosed
US-20020132797-A1 DNA-cleaving antitumor agents NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2002-09-19 US disclosed
US-20020132300-A1 Specific inhibitors of NFAT activation by calcineurin and their use in treating immune-related diseases CENTER FOR BLOOD RESEARCH 2002-09-19 US disclosed
EP-1233776-A1 UROTENSIN-II CYCLIC ANALOGS SMITHKLINE BEECHAM CORPORATION (US) 2002-08-28 EP disclosed
EP-1233774-A1 UROTENSIN-II ANALOGS SmithKline Beecham Corporation (US) 2002-08-28 EP disclosed
WO-2002062941-A1 DETECTION OF MICRO-ORGANISMS MICAP PLC (GB) 2002-08-15 WO disclosed
US-20020102616-A1 Islet cell antigen 1851 ZYMOGENETICS, INC. 2002-08-01 US disclosed
WO-2002058702-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (GB) 2002-08-01 WO disclosed
EP-1220935-A1 SYNTHETIC AND CHIMERIC PROMOTERS, EXPRESSION CASSETTES, PLASMIDS, VECTORS, TRANSGENIC PLANTS AND SEEDS CONTAINING THEM, AND METHOD FOR PRODUCING THEM MERISTEM THERAPEUTICS (FR) 2002-07-10 EP disclosed
US-6416963-B1 CONTACTING FIBRINOGEN DIGEST COMPRISING ALPHAE CX FIBRINOGEN PRODUCED BY PROTEOLYTIC ENZYME DIGESTION WITH AT LEAST ONE ANTIBODY THAT SPECIFICALLY BINDS TO ALPHAE C DOMAIN OF FIBRINOGEN, SELECTIVELY REMOVING ALPHAE CX FIBRINOGEN NEW YORK BLOOD CENTER 2002-07-09 US disclosed
US-20020086426-A1 Tetracycline-regulated transcriptional activator fusion proteins BASF AKTIENGESELLSCHAFT (DE) 2002-07-04 US disclosed
US-20020083486-A1 Chimeric plant promoters and plants containing the same MERISTEM THERAPEUTICS (FR) 2002-06-27 US disclosed
US-20020077307-A1 METHODS FOR REGULATING GENE EXPRESSION TET SYSTEMS HOLDING GMBH & CO. KG (DE) 2002-06-20 US disclosed
WO-2002047456-A2 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2002-06-20 WO disclosed
WO-2002047687-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2002-06-20 WO disclosed
CN-1348436-A Novel ligands of nuclear receptors PPAR's NUCLEAR RECEPTOR RES LTD (JP) 2002-05-08 CN disclosed
US-20020049181-A1 Novel internal ribosome entry site, vector containing same and uses thereof VLAAMS INTERUNIVERSITAIR INSTITUUT VOOR (BE) 2002-04-25 US disclosed
EP-1198554-A2 DETECTION OF MICRO-ORGANISMS FSM Technologies Limited (GB) 2002-04-24 EP disclosed
WO-2002009677-A2 METHOD TO TREAT INFECTIOUS DISEASES AND/OR TO ENHANCE ANTIMICROBIAL EFFICACY OF DRUGS VIROCELL INC. (CA) 2002-02-07 WO disclosed
EP-1176134-A1 LIGANDS OF NUCLEAR RECEPTORS PPAR'S Nuclear Receptor Research Limited (JP) 2002-01-30 EP disclosed
EP-0666910-B1 METHOD OF CLEAVING SPECIFIC STRANDS OF RNA US GOV HEALTH & HUMAN SERV (US) 2002-01-30 EP disclosed
EP-1165815-A1 CHIMERIC EXPRESSION PROMOTERS ORIGINATING FROM COMMELINA YELLOW MOTTLE VIRUS AND CASSAVA VEIN MOSAIC VIRUS MERISTEM THERAPEUTICS (FR) 2002-01-02 EP disclosed
EP-1163351-A1 CHIMERIC PROMOTERS BASED ON THE PLASTOCYANIN PETE PROMOTER FROM PEA MERISTEM THERAPEUTICS (FR) 2001-12-19 EP disclosed
EP-1153138-A1 DETECTION OF CELLS USING THE LUCIFERASE/LUCIFERIN REACTION PROMEGA CORPORATION (US) 2001-11-14 EP disclosed
EP-0688360-B1 BONE STIMULATING FACTOR OSTEOPHARM INC (CA) 2001-11-14 EP disclosed
EP-1147188-A1 INTERNAL RIBOSOME ENTRY SITE (IRES), VECTOR CONTAINING SAME AND THE USES THEREOF Vlaams Interuniversitair Instituut voor Biotechnologie vzw. (BE) 2001-10-24 EP disclosed
EP-1142870-A1 NOVEL LIGANDS OF NUCLEAR RECEPTOR Nuclear Receptor Research Limited (JP) 2001-10-10 EP disclosed
US-6300093-B1 AN ISOLATED POLYNUCLEOTIDE ENCODING A MACAQUE ISLET CELL ANTIGEN POLYPEPTIDE THAT FORMS AN IMMUNE COMPLEX WITH AN AUTOANTIBODY FROM PATIENTS AT RISK FOR INSULIN-DEPENDENT DIABETES MELLITUS; THRAPY AND DIAGNOSIS ZYMOGENETICS, INC. 2001-10-09 US disclosed
US-6297284-B1 AZA-ENEDIYNE, AZA-ENYNE ALLENE, OR AN AZA-DIALLENE CATIONIC COMPOUNDS THAT BIND TO NUCLEIC ACIDS. RESEARCH DEVELOPMENT FOUNDATION 2001-10-02 US disclosed
WO-2001070217-A1 DNA-CLEAVING ANTITUMOR AGENTS RESEARCH DEVELOPMENT FOUNDATION (US) 2001-09-27 WO disclosed
CN-1313766-A Novel DNA-cleaving antitumor agents RES EDVELOPMENT FOUNDATION (US) 2001-09-19 CN disclosed
US-6271369-B1 OLIGONUCLEOTIDES WHICH TARGET MIRCOORGANISM TRANSCRIPTS; FOR THE TREATMENT OF VIRAL DISEASE AND CANCER THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2001-08-07 US disclosed
US-6271348-B1 FUSION PROTEIN WHICH INHIBITS TRANSCRIPTION IN EUKARYOTIC CELLS; FOR USE AS A TOOL IN GENE REGULATION BASF AKTIENGESELLSCHAFT (DE) 2001-08-07 US disclosed
EP-1120466-A2 Use of negative regulation elements for nerve-specific expression of transgenes Aventis Pharma S.A. (FR) 2001-08-01 EP disclosed
WO-2001053817-A2 METHODS OF AND APPARATUS FOR SEPARATING AND DETECTING NUCLEIC ACID MOSAIC TECHNOLOGIES (US) 2001-07-26 WO disclosed
US-20010008026-A1 SYSTEM FOR TISSUE-RESTRICTED GENE RECOMBINATION BAYLOR COLLEGE OF MEDICINE 2001-07-12 US disclosed
WO-2001045700-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-06-28 WO disclosed
WO-2001045694-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-06-28 WO disclosed
WO-2001045711-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-06-28 WO disclosed
EP-1109552-A1 NOVEL DNA-CLEAVING ANTITUMOR AGENTS RESEARCH DEVELOPMENT FOUNDATION (US) 2001-06-27 EP disclosed
US-6252136-B1 GENETICALLY ENGINEERED PLANT; FOR THE CONTROL OF GENE EXPRESSION IN CELLS; FOR TREATMENT OF ARTHRITIS AND INFLAMMATION; WOUND HEALING; FOR TREATMENT OF CANCER; GENE THERAPY BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed
EP-1107665-A1 METHOD OF DIAGNOSIS OF PROSTATE CANCER Uropath PTY. Ltd. (AU) 2001-06-20 EP disclosed
EP-1105428-A1 NOVEL CLEAVED FRAGMENTS OF FIBRINOGEN THE NEW YORK BLOOD CENTER, INC. (US) 2001-06-13 EP disclosed
US-6242667-B1 PLANT HAVING TRANSCRIPTIONAL REGULATORY SEQUENCE LINKED TO POLYNUCLEOTIDE ENCODING A FUSION PROTEIN OF A MUTATED TET REPRESSOR AND A TRANSCRIPTION ACTIVATOR; FUSION PROTEIN ACTIVATES TRANSCRIPTION OF A TET OPERATOR LINKED GENE BASF AKTIENGESELLSCHAFT (DE) 2001-06-05 US disclosed
WO-2001037780-A2 UROTENSIN-II ANALOGS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-31 WO disclosed
WO-2001037856-A1 UROTENSIN-II CYCLIC ANALOGS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-31 WO disclosed
EP-1092771-A2 Tetracycline-regulated transcriptional modulators BASF AKTIENGESELLSCHAFT (DE) 2001-04-18 EP disclosed
US-6214805-B1 GENES, GENE SIGNALS, GENOMES RNA STRANDS AND RESPIRATORY SYNCYTIAL VIRUS WITH PROMOTERS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2001-04-10 US disclosed
WO-2001023593-A1 SYNTHETIC AND CHIMERIC PROMOTERS, EXPRESSION CASSETTES, PLASMIDS, VECTORS, TRANSGENIC PLANTS AND SEEDS CONTAINING THEM, AND METHOD FOR PRODUCING THEM MERISTEM THERAPEUTICS (FR) 2001-04-05 WO disclosed
WO-2001011006-A2 DETECTION OF MICRO-ORGANISMS FLUID TECHNOLOGIES PLC (GB) 2001-02-15 WO disclosed
US-6172189-B1 POLYPEPTIDE FOR THE DETECTION OF ANTIBODIES ASSOCIATED WITH PREFERENTIAL VIRAL DISEASES AND INFECTION ABBOTT LABORATORIES 2001-01-09 US disclosed
EP-1053341-A1 USE OF NEGATIVE REGULATION ELEMENTS FOR NERVE-SPECIFIC EXPRESSION OF TRANSGENES Aventis Pharma S.A. (FR) 2000-11-22 EP disclosed
US-6136954-A POLYPEPTIDE WHICH ACTIVATES TRANSCRIPTION IN EUCARYOTIC CELLS IN THE PRESENCE OF ANTIBIOTIC; FOR ANALYSIS OF CELLULAR PROTEINS BASF AKTIENGESELLSCHAFT (US) 2000-10-24 US disclosed
US-6133229-A STABILIZING AQUEOUS ENZYME WITH AQUEOUS SOLUTION COMPRISING TRIS/HYDROXYMETHYL/METHYL COMPOUND, CATIONIC POLYELECTROLYTE, POLYOL, SALT OF CALCIUM, MAGNESIUM AND/OR COBALT THE UNIVERSITY OF LEEDS INNOVATIONS, LTD. (GB) 2000-10-17 US disclosed
WO-2000058485-A1 CHIMERIC EXPRESSION PROMOTERS ORIGINATING FROM COMMELINA YELLOW MOTTLE VIRUS AND CASSAVA VEIN MOSAIC VIRUS MERISTEM THERAPEUTICS (FR) 2000-10-05 WO disclosed
WO-2000056906-A1 CHIMERIC PROMOTERS BASED ON THE PLASTOCYANIN PETE PROMOTER FROM PEA MERISTEM THERAPEUTICS (FR) 2000-09-28 WO disclosed
EP-1033992-A1 RNASE L ACTIVATORS AND ANTISENSE OLIGONUCLEOTIDES EFFECTIVE TO TREAT RSV INFECTIONS THE CLEVELAND CLINIC FOUNDATION (US) 2000-09-13 EP disclosed
WO-2000049171-A1 DETECTION OF CELLS USING THE LUCIFERASE/LUCIFERIN REACTION PROMEGA CORPORATION (US) 2000-08-24 WO disclosed
WO-2000044896-A1 INTERNAL RIBOSOME ENTRY SITE (IRES), VECTOR CONTAINING SAME AND USES THEREOF VLAAMS INTERUNIVERSITAIR INSTITUUT VOOR BIOTECHNOLOGIE VZW (BE) 2000-08-03 WO disclosed
US-6096740-A BLOCK N-METHYL-ASPARTATE RAMOT UNIVERSITY AUTHORITY FOR APPLIED RESEARCH AND INDUSTRIAL DEVELOPMENT LTD. (IL) 2000-08-01 US disclosed
WO-2000003709-A9 NOVEL DNA-CLEAVING ANTITUMOR AGENTS UNIV TEXAS (US) 2000-07-20 WO disclosed
EP-1007655-A1 RNASE L ACTIVATORS AND ANTISENSE OLIGONUCLEOTIDES EFFECTIVE TO TREAT RSV INFECTIONS NATIONAL INSTITUTES OF HEALTH (US) 2000-06-14 EP disclosed
EP-0642666-B1 HEPATITIS C ASSAY ABBOTT LAB (US) 2000-04-12 EP disclosed
WO-2000011947-A1 METHOD OF DIAGNOSIS OF PROSTATE CANCER UROPATH PTY. LTD. (AU) 2000-03-09 WO disclosed
WO-2000009562-A1 NOVEL CLEAVED FRAGMENTS OF FIBRINOGEN THE NEW YORK BLOOD CENTER, INC. (US) 2000-02-24 WO disclosed
WO-2000003709-A1 NOVEL DNA-CLEAVING ANTITUMOR AGENTS RESEARCH DEVELOPMENT FOUNDATION (US) 2000-01-27 WO disclosed
US-6004941-A INTRODUCING NUCLEIC ACID ENCODING FUSION PROTEIN WHICH ACTIVATES TRANSCRIPTION AND COMPRISES A POLYPEPTIDE THAT BINDS TO TETRACYCLINE OPERATOR BASF AKTIENGESELLSCHAFT (DE) 1999-12-21 US disclosed
US-5998602-A RNase L activators and antisense oligonucleotides effective to treat RSV infections THE CLEVELAND CLINIC FOUINDATION AND GOVERNMENT (US) 1999-12-07 US disclosed
US-5977345-A PRELOADING BIOPOLYMER BEADS WITH ORGANIC SOLVENT, ADDING BIFUNCTIONAL REAGENT DISSOLVED IN ORGANIC SOLVENT MIXTURE, REACTING ONE FUNCTIONALITY OF REAGENT WITH THE POLYMER; FOR IONIC BINDING SITES PRIMARILY WITHIN INTERIOR VIRGINIA TECH INTELLECTUAL PROPERTIES, INC (US) 1999-11-02 US disclosed
EP-0472207-B1 Hepatitis C assay utilizing recombinant antigens ABBOTT LAB (US) 1999-10-13 EP disclosed
US-5945581-A GENETIC ENGINEERING CORNELL RESEARCH FOUNDATION, INC. (US) 1999-08-31 US disclosed
WO-1999041396-A1 USE OF NEGATIVE REGULATION ELEMENTS FOR NERVE-SPECIFIC EXPRESSION OF TRANSGENES AVENTIS PHARMA S.A. (FR) 1999-08-19 WO disclosed
WO-1999040930-A1 SPECIFIC INHIBITORS OF NFAT ACTIVATION BY CALCINEURIN AND THEIR USE IN TREATING IMMUNE-RELATED DISEASES CENTER FOR BLOOD RESEARCH, INC. (US) 1999-08-19 WO disclosed
EP-0929683-A1 DIABETES MELLITUS 37 kD AUTOANTIGEN PROTEIN-TYROSINE PHOSPHATASE ZymoGenetics, Inc. (US) 1999-07-21 EP disclosed
US-5922328-A HERPES SIMPLEX AVIRON (US) 1999-07-13 US disclosed
US-5922927-A Methods for producing tetracycline-regulated transgenic mice BASF AKTIENGESELLSCHAFT (DE) 1999-07-13 US disclosed
EP-0925369-A1 UNIVERSAL TEST SYSTEMS AND METHODS OF USE THEREOF FOR IDENTIFYING MULTIPLE FAMILIES OF MICROORGANISMS Dade Microsan Inc. (US) 1999-06-30 EP disclosed
US-5912411-A Mice transgenic for a tetracycline-inducible transcriptional activator UNIVERSITY OF HEIDELBERG (DE) 1999-06-15 US disclosed
WO-1999022742-A1 RNASE L ACTIVATORS AND ANTISENSE OLIGONUCLEOTIDES EFFECTIVE TO TREAT RSV INFECTIONS THE CLEVELAND CLINIC FOUNDATION (US) 1999-05-14 WO disclosed
US-5888760-A COMBINATION OF NON-REDUNDANT TESTS IN REACTION CHAMBERS CONTAINING SUBSTRATES FOR ENZYMATIC CLASSIFICATION BY DETECTION OF FLUORESCENT OR COLORIMETRIC PRODUCTS FORMED DADE MICROSCAN INC. (US) 1999-03-30 US disclosed
US-5888981-A INTRODUCING INTO CELL A NUCLEIC ACID MOLECULE ENCODING A TETRACYCLINE-CONTROLLABLE TRANSACTIVATOR COMPRISING A TET REPRESSOR OPERABLY LINKED TO A POLYPEPTIDE WHICH ACTIVATES TRANSCRIPTION IN EUCARYOTIC CELLS, MODULATING CONCENTRATION BASF AKTIENGESELLSCHAFT (DE) 1999-03-30 US disclosed
US-5866755-A Animals transgenic for a tetracycline-regulated transcriptional inhibitor BASF AKTIENGELLSCHAFT (DE) 1999-02-02 US disclosed
US-5859310-A Mice transgenic for a tetracycline-controlled transcriptional activator BASF AKTIENGESELLSCHAFT (DE) 1999-01-12 US disclosed
US-5854010-A Bioassay for detecting 2,3,7,8-tetrachlorodibenzo-para-dioxin and TCDD-like compounds and novel recombinant cell line useful therefor XENOBIOTIC DETECTION SYSTEMS INTERNATIONAL, INC. 1998-12-29 US disclosed
US-5850025-A Protection of plants against plant pathogens SIBIA NEUROSCIENCES, INC. (US) 1998-12-15 US disclosed
EP-0760099-A4 METHOD AND REAGENTS USEFUL FOR IMPROVING IMMUNOASSAY SPECIFICITY ABBOTT LAB (US) 1998-12-09 EP disclosed
WO-1998045469-A1 UNIVERSAL TEST SYSTEMS AND METHODS OF USE THEREOF FOR IDENTIFYING MULTIPLE FAMILIES OF MICROORGANISMS DADE MICROSCAN INC. (US) 1998-10-15 WO disclosed
US-5814618-A TETRACYCLINE-RESPONSIVE FUSION PROTEINS BASF AKTIENGESELLSCHAFT (DE) 1998-09-29 US disclosed
EP-0649905-B1 Methods of detection of mutagens using luminescence gene TOYODA CHUO KENKYUSHO KK (JP) 1998-09-23 EP disclosed
US-5789156-A NUCLEIC ACIDS ENCODING FUSION PROTEINS WHICH INHIBITSTRANSCRIPTION OF EUKARYOTIC CELLS BASF AG (DE) 1998-08-04 US disclosed
WO-1997009999-A9 METHODS AND COMPOSITIONS FOR TREATMENT OF HSV-2 INFECTIONS AND CONDITIONS 1997-11-06 WO disclosed
EP-0804565-A1 TETRACYCLINE-REGULATED TRANSCRIPTIONAL MODULATORS Bujard, Hermann (DE) 1997-11-05 EP disclosed
US-5677289-A ANTIBODY OLIGONUCLEOTIDE THE CLEVELAND CLINIC FOUNDATION (US) 1997-10-14 US disclosed
WO-1997032984-A1 DIABETES MELLITUS 37 kD AUTOANTIGEN PROTEIN-TYROSINE PHOSPHATASE ZYMOGENETICS, INC. (US) 1997-09-12 WO disclosed
US-5665579-A TRANSGENIC TOMATO PLANTS GENETICALLY ENGINEERED THE SALK INSTITUTE BIOTECHNOLOGY/INDUSTRIAL ASSOCIATES, INC. (US) 1997-09-09 US disclosed
WO-1997029757-A1 RNASE L ACTIVATORS AND ANTISENSE OLIGONUCLEOTIDES EFFECTIVE TO TREAT RSV INFECTIONS NATIONAL INSTITUTES OF HEALTH (US) 1997-08-21 WO disclosed
US-5654168-A ISOLATED NUCLEIC ACID ENCODING FUSION PROTEIN COMPRISING FIRST POLYPEPTIDE WHICH BINDS TO TET OPERATOR SEQUENCE IN PRESENCE OF TETRACYCLINE OPERATIVELY LINKED TO SECOND POLYPEPTIDE WHICH ACTIVATES TRANSCRIPTION IN EUKARYOTIC CELLS BASF AKTIENGESELLSCHAFT (DE) 1997-08-05 US disclosed
US-5650298-A Tight control of gene expression in eucaryotic cells by tetracycline-responsive promoters BASF AKTIENGESELLSCHAFT (DE) 1997-07-22 US disclosed
US-5637466-A Method of detecting bone acidic glycoprotein-75 and its 50,000 MW fragment and antibodies therefor CURATORS OF THE UNIVERSITY OF MISSOURI (US) 1997-06-10 US disclosed
US-5633449-A A DNA MOLECULE CORNELL RESEARCH FOUNDATION, INC. (US) 1997-05-27 US disclosed
US-5618927-A INCUBATION IN SOLUTION OF TRIS BOEHRINGER MANNHEIM GMBH (DE) 1997-04-08 US disclosed
WO-1997009999-A1 METHODS AND COMPOSITIONS FOR TREATMENT OF HSV-2 INFECTIONS AND CONDITIONS AVIRON (US) 1997-03-20 WO disclosed
EP-0760099-A1 METHOD AND REAGENTS USEFUL FOR IMPROVING IMMUNOASSAY SPECIFICITY ABBOTT LABORATORIES (US) 1997-03-05 EP disclosed
US-5589362-A FUSION PROTEINS, EUKARYOTIC CELLS BASF AKTIENGESELLSCHAFT (DE) 1996-12-31 US disclosed
US-5589104-A Electrophoresis separation gel and a method for preparing an electrophoresis separation gel BAMBECK GREGORY S (US) 1996-12-31 US disclosed
WO-1996040892-A1 TETRACYCLINE REGULATED TRANSCRIPTIONAL MODULATORS WITH ALTERED DNA BINDING SPECIFICITIES BASF AG (US) 1996-12-19 WO disclosed
US-5583032-A USING A CHIMERIC MOLECULE MADE UP OF AN ANTISENSE OLIGONUCLEOTIDE ATTACHED TO A 2',5'-OLIGOADENYLATE MOLECULE; ANTISENSE OLIGONUCLEOTIDE IS HYBRIDIZED TO SENSE STRAND OF RNA IN PRESENCE OF 2',5'-DEPENDENT RNASE THE CLEVELAND CLINIC FOUNDATION AND NATIONAL INSTITUTES OF HEALTH (US) 1996-12-10 US disclosed
US-5576428-A GENETIC EGINEERING THE SALK INSTITUTE BIOTECHNOLOGY/INDUSTRIAL ASSOCIATES, INC. (US) 1996-11-19 US disclosed
EP-0647277-A4 METHODS FOR USING CKS FUSION PROTEINS. ABBOTT LAB (US) 1996-10-30 EP disclosed
EP-0722492-A1 STABILISATION OF PROTEINS IN SOLUTION The University of Leeds Innovations Ltd. (GB) 1996-07-24 EP disclosed
US-5532166-A CAPILLARY ZONE ELECTROPHORESIS WITH LASER-EXCITED FLUORESCENCE DETECTION MA YINFA (US) 1996-07-02 US disclosed
US-5521215-A TREATMENT OF NERVOUS SYSTEM INJURIES RAMOT UNIVERSITY AUTHORITY FOR APPLIED RESEARCH AND INDUSTRIAL DEVELOPMENT LTD. (IL) 1996-05-28 US disclosed
EP-0705334-A1 TIGHT CONTROL OF GENE EXPRESSION IN EUCARYOTIC CELLS BY TETRACYCLINE-RESPONSIVE PROMOTERS BASF AKTIENGESELLSCHAFT (DE) 1996-04-10 EP disclosed
JP-H0849282-A TOILET OF FIRE RETARDANT RESIN TOKUYAMA CORP 1996-02-20 JP disclosed
WO-1996001313-A1 TETRACYCLINE-REGULATED TRANSCRIPTIONAL MODULATORS BUJARD HERMANN (DE) 1996-01-18 WO disclosed
WO-1995030902-A1 METHOD AND REAGENTS USEFUL FOR IMPROVING IMMUNOASSAY SPECIFICITY ABBOTT LABORATORIES (US) 1995-11-16 WO disclosed
US-5464758-A Polynucleotide molecule codes for eukarotic proteins TET SYSTEMS HOLDING GMBH & CO. KG (DE) 1995-11-07 US disclosed
EP-0673423-A1 VIRAL RESISTANCE BY PLANT TRANSFORMATION WITH A REPLICASE PORTION OF A PLANT VIRUS GENOME CORNELL RESEARCH FOUNDATION, INC. (US) 1995-09-27 EP disclosed
EP-0445423-B1 Hepatitis C assay ABBOTT LAB (US) 1995-09-20 EP disclosed
EP-0666910-A1 METHOD OF CLEAVING SPECIFIC STRANDS OF RNA THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-08-16 EP disclosed
US-5422108-A Applying lysozyme which digests cell walls of microbes under acidic conditions SMART PLANTS INTERNATIONAL INC. (US) 1995-06-06 US disclosed
EP-0612207-A4 PROTECTION OF PLANTS AGAINST PLANT PATHOGENS. SMART PLANTS INT INC (US) 1995-05-24 EP disclosed
EP-0673423-A4 VIRAL RESISTANCE BY PLANT TRANSFORMATION WITH A REPLICASE PORTION OF A PLANT VIRUS GENOME. CORNELL RES FOUNDATION INC (US) 1995-05-23 EP disclosed
EP-0649905-A1 Methods of detection of mutagens using luminescence gene KABUSHIKI KAISHA TOYOTA CHUO KENKYUSHO (JP) 1995-04-26 EP disclosed
WO-1995010605-A1 STABILISATION OF PROTEINS IN SOLUTION THE UNIVERSITY OF LEEDS INNOVATIONS LTD. (GB) 1995-04-20 WO disclosed
EP-0647277-A1 METHODS FOR USING CKS FUSION PROTEINS ABBOTT LABORATORIES (US) 1995-04-12 EP disclosed
EP-0642666-A1 HEPATITIS C ASSAY ABBOTT LABORATORIES (US) 1995-03-15 EP disclosed
EP-0600009-A4 HEPATITIS C ASSAY UTILIZING RECOMBINANT ANTIGENS TO NS1. ABBOTT LAB (US) 1995-03-01 EP disclosed
EP-0600018-A4 HEPATITIS C ASSAY UTILIZING RECOMBINANT ANTIGENS TO C-100 REGION. ABBOTT LAB (US) 1995-03-01 EP disclosed
EP-0600000-A4 HEPATITIS C ASSAY UTILIZING RECOMBINANT ANTIGENS FROM NS5 REGION. ABBOTT LAB (US) 1995-03-01 EP disclosed
WO-1994029442-A2 TIGHT CONTROL OF GENE EXPRESSION IN EUCARYOTIC CELLS BY TETRACYCLINE-RESPONSIVE PROMOTERS BASF AKTIENGESELLSCHAFT (DE) 1994-12-22 WO disclosed
EP-0642666-A4 HEPATITIS C ASSAY. ABBOTT LAB (US) 1994-11-22 EP disclosed
EP-0612207-A1 PROTECTION OF PLANTS AGAINST PLANT PATHOGENS SMART PLANTS INTERNATIONAL, INC. (US) 1994-08-31 EP disclosed
US-5330893-A Use of superoxide dismutase in specimen diluent ABBOTT LABORATORIES (US) 1994-07-19 US disclosed
EP-0568639-A4 USE OF SUPEROXIDE DISMUTASE IN SPECIMEN DILUENT ABBOTT LAB (US) 1994-06-29 EP disclosed
US-5322769-A Detecting anti-analyte antibody in test sample; kits ABBOTT LABORATORIES (US) 1994-06-21 US disclosed
EP-0600000-A1 HEPATITIS C ASSAY UTILIZING RECOMBINANT ANTIGENS FROM NS5 REGION ABBOTT LABORATORIES (US) 1994-06-08 EP disclosed
EP-0600009-A1 HEPATITIS C ASSAY UTILIZING RECOMBINANT ANTIGENS TO NS1 ABBOTT LABORATORIES (US) 1994-06-08 EP disclosed
EP-0600018-A1 HEPATITIS C ASSAY UTILIZING RECOMBINANT ANTIGENS TO C-100 REGION ABBOTT LABORATORIES (US) 1994-06-08 EP disclosed
WO-1994009129-A2 METHOD OF CLEAVING SPECIFIC STRANDS OF RNA THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1994-04-28 WO disclosed
WO-1994000594-A9 METHODS FOR USING CKS FUSION PROTEINS 1994-03-17 WO disclosed
WO-1994000594-A1 METHODS FOR USING CKS FUSION PROTEINS ABBOTT LABORATORIES (US) 1994-01-06 WO disclosed
WO-1993025068-A1 VIRAL RESISTANCE BY PLANT TRANSFORMATION WITH A REPLICASE PORTION OF A PLANT VIRUS GENOME CORNELL RESEARCH FOUNDATION, INC. (US) 1993-12-23 WO disclosed
EP-0573566-A1 NOVEL INVERTASE GENE(S) AND USES THEREOF SIBIA NEUROSCIENCES, INC. (US) 1993-12-15 EP disclosed
EP-0304151-B1 Measurement of calcium ions INSTRUMENTATION LAB SPA (IT) 1993-12-15 EP disclosed
EP-0568639-A1 USE OF SUPEROXIDE DISMUTASE IN SPECIMEN DILUENT ABBOTT LABORATORIES (US) 1993-11-10 EP disclosed
WO-1993006247-A1 HEPATITIS C ASSAY ABBOTT LABORATORIES (US) 1993-04-01 WO disclosed
WO-1993005645-A1 PROTECTION OF PLANTS AGAINST PLANT PATHOGENS SMART PLANTS INTERNATIONAL, INC. (US) 1993-04-01 WO disclosed
WO-1993004087-A1 HEPATITIS C ASSAY UTILIZING RECOMBINANT ANTIGENS TO C-100 REGION ABBOTT LABORATORIES (US) 1993-03-04 WO disclosed
WO-1993004088-A1 HEPATITIS C ASSAY UTILIZING RECOMBINANT ANTIGENS TO NS1 ABBOTT LABORATORIES (US) 1993-03-04 WO disclosed
WO-1993004089-A1 HEPATITIS C ASSAY UTILIZING RECOMBINANT ANTIGENS FROM NS5 REGION ABBOTT LABORATORIES (US) 1993-03-04 WO disclosed
US-5160739-A Moisture cream, cleanser, polyolefins, polyoxyalkylene glycol solubilizer CHESEBROUGH-POND'S USA CO., DIVISION OF CONOPCO, INC. (US) 1992-11-03 US disclosed
WO-1992014831-A1 NOVEL INVERTASE GENE(S) AND USES THEREOF THE SALK INSTITUTE BIOTECHNOLOGY/INDUSTRIAL ASSOCIATES, INC. (US) 1992-09-03 WO disclosed
WO-1992013275-A1 USE OF SUPEROXIDE DISMUTASE IN SPECIMEN DILUENT ABBOTT LABORATORIES (US) 1992-08-06 WO disclosed
US-5135748-A Quaternary ammonium functionalized phosphate ester CHESEBROUGH-POND'S USA CO., DIVISION OF CONOPCO, INC. (US) 1992-08-04 US disclosed
EP-0472207-A2 Hepatitis C assay utilizing recombinant antigens ABBOTT LABORATORIES (US) 1992-02-26 EP disclosed
US-5061336-A GEL CASTING METHOD AND APPARATUS SOANE TECHNOLOGIES, INC. (US) 1991-10-29 US disclosed
EP-0445423-A2 Hepatitis C assay ABBOTT LABORATORIES (US) 1991-09-11 EP disclosed
US-5045465-A Culturing flavobacterium, a-ketoglutaric acid, ammonium sulfate EASTMAN KODAK COMPANY (US) 1991-09-03 US disclosed
EP-0427845-A4 GEL CASTING METHOD AND APPARATUS 1991-07-10 EP disclosed
EP-0427845-A1 GEL CASTING METHOD AND APPARATUS SOANE, David S. (US) 1991-05-22 EP disclosed
US-5017489-A Antibodies MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1991-05-21 US disclosed
EP-0413285-A2 Fermentation process for creatinine iminohydrolase EASTMAN KODAK COMPANY (US) 1991-02-20 EP disclosed
WO-1990014201-A1 GEL CASTING METHOD AND APPARATUS SOANE DAVID S (US) 1990-11-29 WO disclosed
EP-0363083-A2 Pharmaceutical preparation for treatment of thrombocytopenic or platelet function-deficient disease Chugai Seiyaku Kabushiki Kaisha (JP) 1990-04-11 EP disclosed
US-4880751-A Immunoglobulin adsorption BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1989-11-14 US disclosed
US-4870024-A DILUTION WITH TRIS PHOSPHATE FISHER SCIENTIFIC COMPANY (US) 1989-09-26 US disclosed
US-4859342-A Process for industrially separating biopolymers SUNTORY LIMITED (JP) 1989-08-22 US disclosed
EP-0304151-A2 Measurement of calcium ions INSTRUMENTATION LABORATORY S.p.A. (IT) 1989-02-22 EP disclosed
EP-0254593-A2 Preparation and uses of interferon-gamma KABUSHIKI KAISHA HAYASHIBARA SEIBUTSU KAGAKU KENKYUJO (JP) 1988-01-27 EP disclosed
EP-0211756-A1 Assay for varicella-zoster virus (VZV) antibodies MERCK & CO. INC. (US) 1987-02-25 EP disclosed
US-4603108-A Method for identification of bacterial species NATIONAL RESEARCH DEVELOPMENT CORP. (GB) 1986-07-29 US disclosed
EP-0029766-B1 METHOD FOR THE RECOVERY OF CREATININE IMINOHYDROLASE EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1984-05-16 EP disclosed
US-4432877-A Organo-mercurial materials NEW ENGLAND NUCLEAR CORPORATION (US) 1984-02-21 US disclosed
US-4409275-A Decorative laminate SAMOWICH JOSEPH J 1983-10-11 US disclosed
US-4275166-A PRECIPITATING CREATINE IMINOHYDROLASE EASTMAN KODAK COMPANY (US) 1981-06-23 US disclosed
EP-0029766-A1 Method for the recovery of creatinine iminohydrolase EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1981-06-03 EP disclosed
US-4252896-A Method of stabilizing peroxidase in a serum protein based medium ABBOTT LABORATORIES (US) 1981-02-24 US disclosed
WO-1980002433-A1 THE IDENTIFICATION OF BACTERIA NAT RES DEV (GB) 1980-11-13 WO disclosed
EP-0018825-A1 A process for the identification of bacteria and a kit of reagents for use in this process NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1980-11-12 EP disclosed
US-4170614-A HYDROLYSIS OF TRIS(2,6-DIHALOPHENYL) PHOSPHATE PPG INDUSTRIES, INC. (US) 1979-10-09 US disclosed
US-4059655-A REACTING A 2,6-DIHALOPHENOL WITH PHOSPHORUS OXYHALIDE, HYDROLYSIS PPG INDUSTRIES, INC. (US) 1977-11-22 US disclosed
US-4059655-A REACTING A 2,6-DIHALOPHENOL WITH PHOSPHORUS OXYHALIDE, HYDROLYSIS PPG INDUSTRIES, INC. (US) 1977-11-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030100580-A1 Urotensin-II receptor antagonists UTS2R, TMPRSS4, PLAUR DNMT1 4879/4885MAPT 3109/4885HTT 2297/4885
US-20140113944-A1 BICYCLO (3.1.0) HEXANE-2, 6-DICARBOXYLIC ACID DERIVATIVES AS MGLU2 RECEPTOR AGONIST GRM2, GRIA2, HCAR2 DNMT1 2863/4885MAPT 1470/4885HTT 2746/4885
US-20120190699-A1 PYRIDONES USEFUL AS INHIBITORS OF KINASES MAP3K20, MAP3K6, MAP3K5 DNMT1 2390/4885MAPT 1299/4885HTT 2416/4885
US-10202325-B2 Methods for selective oxidation of alpha tocotrienol in the presence of non-alpha tocotrienols TTPA, GSTO1, TST DNMT1 1844/4885MAPT 4123/4885HTT 2651/4885
US-20140288185-A1 NICOTINIC RECEPTOR NON-COMPETITIVE MODULATORS CHRNA5, CHRNG, CHRNA2 DNMT1 4014/4885MAPT 2378/4885HTT 1416/4885
US-20040142923-A1 Pyrrolidine sulfonamides UTS2R, PRSS2, PRSS8 DNMT1 4870/4885MAPT 2548/4885HTT 1085/4885
US-10258582-B2 Nicotinic receptor non-competitive antagonists CHRNA5, CHRNA2, CHRNG DNMT1 4153/4885MAPT 2694/4885HTT 1373/4885
US-20130245273-A1 AMINOPYRIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES MAP4K5, MAP3K5, MAP3K20 DNMT1 3254/4885MAPT 1042/4885HTT 1296/4885
US-20190216753-A1 N-METHYL-D-ASPARTATE RECEPTOR ALLOSTERIC MODULATORS AND METHODS FOR THEIR USE GRIN2A, GRIN3A, GRIN1 DNMT1 412/4885MAPT 695/4885HTT 337/4885
US-12029708-B2 Alkoxy compounds for disease treatment ALDH1A2, CLN6, AGER DNMT1 4700/4885MAPT 46/4885HTT 19/4885
US-10058534-B2 Benzothiophene derivatives and compositions thereof as selective estrogen receptor degraders ESR1, CYP19A1, GPER1 DNMT1 3074/4885MAPT 2091/4885HTT 1754/4885
US-20180319730-A1 METHODS FOR SELECTIVE OXIDATION OF ALPHA TOCOTRIENOL IN THE PRESENCE OF NON-ALPHA TOCOTRIENOLS TTPA, GSTO1, TST DNMT1 1844/4885MAPT 4123/4885HTT 2651/4885
US-20130116258-A1 ANDROGEN RECEPTOR MODULATORS AND USES THEREOF AR, ESRRA, NR5A1 DNMT1 4099/4885MAPT 3119/4885HTT 4133/4885
US-20150258099-A1 METHODS AND COMPOSITIONS FOR MODULATING ESTROGEN RECEPTOR MUTANTS ESR1, ESRRG, ESR2 DNMT1 1106/4885MAPT 4151/4885HTT 3235/4885
US-12350314-B2 Liquid formulations comprising mutant FGF-21 peptide pegylated conjugates FGF1, FGFR1, FGF2 DNMT1 4844/4885MAPT 1768/4885HTT 2624/4885
US-20110046104-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS AURKC, AURKA, AURKB DNMT1 1384/4885MAPT 954/4885HTT 2296/4885
US-11596669-B2 Liquid formulations comprising mutant FGF-21 peptide pegylated conjugates FGF1, FGFR1, FGF2 DNMT1 4844/4885MAPT 1768/4885HTT 2624/4885
US-20120277425-A1 TETRAHYDROPTERIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES PRKCH, DMPK, MAP3K20 DNMT1 3043/4885MAPT 839/4885HTT 274/4885
US-20060183911-A1 Pyridones useful as inhibitors of kinases MAP3K20, MAP3K6, MAP3K5 DNMT1 2390/4885MAPT 1299/4885HTT 2416/4885
US-20090118278-A1 COMPOSITIONS USEFUL AS INHIBITORS OF GSK-3 GSK3B, GSK3A, GSKIP DNMT1 3851/4885MAPT 570/4885HTT 2902/4885
US-20120122879-A1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS MAP3K20, MAP3K6, MAP3K1 DNMT1 3556/4885MAPT 830/4885HTT 964/4885
US-20130310433-A1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES MAP3K20, MAP3K5, PACSIN2 DNMT1 3862/4885MAPT 1217/4885HTT 1109/4885
US-20040010029-A1 Indole derivatives as interleukin -4 gene expression inhibitors IL4, IL4I1, STAT4 DNMT1 3311/4885MAPT 2047/4885HTT 2627/4885
US-10961232-B2 Substituted pyrazines as ATR kinase inhibitors ATR, MAP3K5, CHEK1 DNMT1 1729/4885MAPT 3129/4885HTT 2299/4885
US-20210275557-A1 MODIFIED AMINOGLYCOSIDE COMPOUNDS AND USES THEREOF IN DISABLING BACTERIAL RIBOSOME FBL, MRPL21, NOP2 DNMT1 1788/4885MAPT 4715/4885HTT 3293/4885
US-20030022934-A1 Phenoxyphenyl alkanesulphonates SNCA, CLN6, NLN DNMT1 3981/4885MAPT 49/4885HTT 7/4885
US-20110152334-A1 MGLU2 AGONISTS GRM2, GRIA2, GRM4 DNMT1 1812/4885MAPT 1331/4885HTT 2496/4885
US-20110020376-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES PRKDC, MAP3K5, MAP3K20 DNMT1 1428/4885MAPT 1503/4885HTT 1791/4885
US-11166924-B2 N-methyl-d-aspartate receptor allosteric modulators and methods for their use GRIN2A, GRIN3A, GRIN1 DNMT1 412/4885MAPT 695/4885HTT 337/4885
US-20230338471-A1 LIQUID FORMULATIONS COMPRISING MUTANT FGF-21 PEPTIDE PEGYLATED CONJUGATES FGF1, FGFR1, FGF2 DNMT1 4844/4885MAPT 1768/4885HTT 2624/4885
US-20160008323-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS CHRNA5, CHRNA2, CHRNG DNMT1 4153/4885MAPT 2694/4885HTT 1373/4885
US-20050101650-A1 Pyrrole compositions useful as inhibitors of c-Met MET, PRKCH, DMPK DNMT1 1623/4885MAPT 1158/4885HTT 1414/4885
US-20080045570-A1 To treat autoimmune, inflammatory, proliferative, hyperproliferative,neurodegenerative or immunologically-mediated diseases; useful for the study of kinases in biological and pathological phenomena; study of intracellular signal transduction pathways mediated by such kinases, and comparative evaluation MAP3K1, MAP3K20, MAP3K2 DNMT1 2528/4885MAPT 775/4885HTT 789/4885
US-20120232275-A1 PROCESS FOR PREPARING 5-FLUORO-1H-PYRAZOLO [3,4-B] PYRIDIN-3-AMINE AND DERIVATIVES THEREOF GSK3B, GSK3A, GSKIP DNMT1 1272/4885MAPT 529/4885HTT 4662/4885
US-20100222318-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, CHEK1, MAP3K5 DNMT1 1574/4885MAPT 2916/4885HTT 2185/4885
US-20100310675-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS ABL1, PRKDC, MAP3K5 DNMT1 1376/4885MAPT 1754/4885HTT 1997/4885
US-20090281082-A1 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS MAP3K20, MAP3K6, MAP3K1 DNMT1 3556/4885MAPT 830/4885HTT 964/4885
US-20170297991-A1 METHODS FOR SELECTIVE OXIDATION OF ALPHA TOCOTRIENOL IN THE PRESENCE OF NON-ALPHA TOCOTRIENOLS TTPA, GSTO1, TST DNMT1 2139/4885MAPT 4272/4885HTT 2484/4885
US-20180271806-A1 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTS CHRNA5, CHRNA2, CHRNG DNMT1 4153/4885MAPT 2694/4885HTT 1373/4885
US-20160090378-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ESR2, ESRRG, GPER1 DNMT1 3956/4885MAPT 3601/4885HTT 4589/4885
US-20040054162-A1 Molecular detection systems utilizing reiterative oligonucleotide synthesis POLRMT, RNGTT, POLI DNMT1 91/4885MAPT 4415/4885HTT 2570/4885
US-20040152891-A1 Sulfonamides UTS2R, PRSS2, STS DNMT1 4883/4885MAPT 2260/4885HTT 1651/4885
US-20090062292-A1 Tetrahydropteridines useful as inhibitors of protein kinases PRKCH, DMPK, MAP3K20 DNMT1 3043/4885MAPT 839/4885HTT 274/4885
US-20040198979-A1 Sulfonamides UTS2R, PRSS2, STS DNMT1 4883/4885MAPT 2260/4885HTT 1651/4885
US-20040002117-A1 Specific inhibitors of NFAT activation by calcineurin and their use in treating immune-related diseases NFATC1, CHP1, PPP3R1 DNMT1 4564/4885MAPT 3702/4885HTT 2665/4885
US-20070179125-A1 Aminopyrimidines useful as kinase inhibitors ABL1, MAP3K5, MAP3K20 DNMT1 1331/4885MAPT 1628/4885HTT 1887/4885
US-20140194444-A1 AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES PRKDC, MAP3K5, MAP3K20 DNMT1 1428/4885MAPT 1503/4885HTT 1791/4885
US-20080070965-A1 Thiophene-carboxamides useful as inhibitors of protein kinases MAP3K20, MAP3K5, PACSIN2 DNMT1 3862/4885MAPT 1217/4885HTT 1109/4885
US-20100184980-A1 Process for Preparing 5-Fluoro-1H-Pyrazolo [3,4-b] Pyridin-3-amine and Derivatives Thereof GSK3B, GSK3A, GSKIP DNMT1 1272/4885MAPT 529/4885HTT 4662/4885
US-20140037754-A1 AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS AURKC, AURKA, AURKB DNMT1 1384/4885MAPT 954/4885HTT 2296/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.