Kuromanin

Kuromanin

SCHEMBL625949

Cl.OC[C@H]1O[C@@H](Oc2cc3c(O)cc(O)cc3[o+]c2-c2ccc(O)c(O)c2)[C@H](O)[C@@H](O)[C@@H]1O.[Cl-]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Kuromanin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 known ✓ P27487 2/20 0.96
GAA known ✓ P10253 4/20 0.50
ADRA2C known ✓ P18825 1/20 0.50
CA2 known ✓ P00918 1/20 0.50
MAOA known ✓ P21397 1/20 0.50
GLA known ✓ P06280 1/20 0.50
CD38 P28907 2/20 0.96
F2 P00734 2/20 0.85
SNCA P37840 1/20 0.51
GLO1 Q04760 1/20 0.51
KDM4E B2RXH2 4/20 0.50
AKR1B1 P15121 4/20 0.50
MAPT P10636 3/20 0.50
POLB P06746 2/20 0.50
P4HB P07237 2/20 0.50
EPHX2 P34913 2/20 0.50
NOX4 Q9NPH5 1/20 0.50
CA12 O43570 1/20 0.50
KDM1A O60341 1/20 0.50
SLCO2B1 O94956 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Kuromanin SCHEMBL3765133 1.00 DPP4 (0.96) DPP4CD38F2SNCAGLO1
Kuromanin SCHEMBL29762023 0.99 DPP4 (0.98) DPP4CD38F2SNCAGLO1
Kuromanin SCHEMBL440823 0.99 DPP4 (0.98) DPP4CD38F2SNCAGLO1
Kuromanin SCHEMBL29377806 0.99 DPP4 (0.98) DPP4CD38F2SNCAGLO1
Kuromanin SCHEMBL158216 0.99 DPP4 (0.98) DPP4CD38F2SNCAGLO1
Kuromanin SCHEMBL29349461 0.99 DPP4 (0.98) DPP4CD38F2SNCAGLO1
Kuromanin SCHEMBL5509009 0.99 CD38 (0.98) DPP4CD38F2SNCAGLO1
Kuromanin SCHEMBL316825 0.99 DPP4 (0.98) DPP4CD38F2SNCAGLO1
Kuromanin SCHEMBL5510421 0.98 CD38 (0.96) DPP4CD38F2SNCAGLO1
Kuromanin SCHEMBL1096430 0.98 CD38 (1.00) DPP4CD38F2SNCAGLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220313675-A1 Anti-Aging Telomere-Strengthening NAD+ Sirtuin Dietary Supplement Composition SHULTZ LARRY (US) 2022-10-06 US claimed
WO-2020263075-A1 A FORMULATION THAT REDUCES OXIDATIVE STRESS UNIVERSITI KEBANGSAAN MALAYSIA (UKM) (MY) 2020-12-30 WO claimed
US-20250114419-A1 INTESTINAL HEALTH PROMOTING COMPOSITIONS NSE PRODUCTS, INC. 2025-04-10 US disclosed
US-20240058408-A1 COMPOSITION FOR PREVENTING OR TREATING MACULAR DEGENERATION CONTAINING GINSENG BERRY EXTRACT HOLISTIC BIO CO., LTD. (KR) 2024-02-22 US disclosed
US-20230149309-A1 COMPOSITION COMPRISING ANTIMICROBIAL AGENT AND ITS USES SHARED VISION TECHNOLOGY LTD. (IE) 2023-05-18 US disclosed
CN-110636760-B Composition for promoting intestinal health NSE产品公司 2023-04-14 CN disclosed
WO-2023286950-A1 COMPOSITION CONTAINING GINSENG BERRY EXTRACT AND LUTEIN FOR PREVENTING OR TREATING MACULAR DEGENERATION 주식회사 홀리스틱바이오 2023-01-19 WO disclosed
US-20220322719-A1 INTESTINAL HEALTH PROMOTING COMPOSITIONS NSE PRODUCTS, INC. (US) 2022-10-13 US disclosed
US-20220313675-A1 Anti-Aging Telomere-Strengthening NAD+ Sirtuin Dietary Supplement Composition SHULTZ LARRY (US) 2022-10-06 US disclosed
WO-2022145813-A1 COMPOSITION FOR PREVENTING OR TREATING MACULAR DEGENERATION CONTAINING GINSENG BERRY EXTRACT 주식회사 홀리스틱바이오 2022-07-07 WO disclosed
EP-2881155-B1 Pressurised low polarity water extraction apparatus and methods of use SENSIENT NATURAL EXTRACTION INC (CA) 2022-04-06 EP disclosed
WO-2012021401-A1 COMPOSITIONS COMPRISING A POLYPEPTIDE HAVING CELLULOLYTIC ENHANCING ACTIVITY AND A BICYCLIC COMPOUND AND USES THEREOF NOVOZYMES, INC. (US) 2012-02-16 WO disclosed
US-20100316743-A1 INHIBITION OF THE FORMATION OF AGEs BASF BEAUTY CARE SOLUTIONS FRANCE S.A.S. (FR) 2010-12-16 US disclosed
US-7807422-B2 set of genes which encodes for enzymes which can convert substrates belonging to the general category of phenylpropanoids and result in the production of flavanones; without the need for chemical conversion THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 2010-10-05 US disclosed
US-20100196331-A1 COMPOSITIONS INCLUDING ANTHOCYANIN OR ANTHOCYANIDIN FOR THE PREVENTION OR TREATMENT OF ARTICULAR CARTILAGE-ASSOCIATED CONDITIONS JOHNSON LANNY L 2010-08-05 US disclosed
US-20090239272-A1 set of genes which encodes for enzymes which can convert substrates belonging to the general category of phenylpropanoids and result in the production of flavanones; without the need for chemical conversion KOFFAS MATTHEOS 2009-09-24 US disclosed
US-7338791-B2 Introducing the set of genes into a heterologous host cell, allowing growth of the cells in a suitable medium such that the expression of the genes results in production of enzymes; culturing the cell under conditions permitting the synthesis of the flavonoid by the cells; isolating s flavonoids THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 2008-03-04 US disclosed
EP-1778850-A2 PRODUCTION OF FLAVONOIDS BY RECOMBINANT MICROORGANISMS THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 2007-05-02 EP disclosed
US-20060019334-A1 Introducing the set of genes into a heterologous host cell, allowing growth of the cells in a suitable medium such that the expression of the genes results in production of enzymes; culturing the cell under conditions permitting the synthesis of the flavonoid by the cells; isolating s flavonoids NATIONAL SCIENCE FOUNDATION 2006-01-26 US disclosed
WO-2006010117-A2 PRODUCTION OF FLAVONOIDS BY RECOMBINANT MICROORGANISMS THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 2006-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100316743-A1 INHIBITION OF THE FORMATION OF AGEs AGER, GLA, S100A6 DPP4 192/4885GAA 107/4885ADRA2C 3397/4885
US-20100196331-A1 COMPOSITIONS INCLUDING ANTHOCYANIN OR ANTHOCYANIDIN FOR THE PREVENTION OR TREATMENT OF ARTICULAR CARTILAGE-ASSOCIATED CONDITIONS SLC2A1, SLC2A2, SLC2A8 DPP4 275/4885GAA 1148/4885ADRA2C 3572/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.