Apigenin

Apigenin

SCHEMBL31168790

Cl.O=c1cc(-c2ccc(O)cc2)oc2cc(O)cc(O)c12

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Apigenin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA known ✓ P21397 4/20 0.97
MAOB known ✓ P27338 4/20 0.97
FLT3 known ✓ P36888 4/20 0.97
HDAC6 known ✓ Q9UBN7 4/20 0.97
CYP19A1 known ✓ P11511 3/20 0.97
GABRP known ✓ O00591 3/20 0.97
GABRD known ✓ O14764 3/20 0.97
GABRA1 known ✓ P14867 3/20 0.97
GABRB1 known ✓ P18505 3/20 0.97
GABRG2 known ✓ P18507 3/20 0.97
GABRB3 known ✓ P28472 3/20 0.97
GABRA5 known ✓ P31644 3/20 0.97
GABRA3 known ✓ P34903 3/20 0.97
GABRA2 known ✓ P47869 3/20 0.97
GABRB2 known ✓ P47870 3/20 0.97
GABRA4 known ✓ P48169 3/20 0.97
GABRE known ✓ P78334 3/20 0.97
GABRA6 known ✓ Q16445 3/20 0.97
GABRG1 known ✓ Q8N1C3 3/20 0.97
GABRG3 known ✓ Q99928 3/20 0.97

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Apigenin SCHEMBL19428 0.98 KMT2A (1.00) KMT2ACYP1B1ABCB1MEN1CYP3A4
Apigenin SCHEMBL5083245 0.98 KMT2A (1.00) KMT2ACYP1B1ABCB1MEN1CYP3A4
Apigenin SCHEMBL29351464 0.98 KMT2A (1.00) KMT2ACYP1B1ABCB1MEN1CYP3A4
Apigenin SCHEMBL29968480 0.97 KMT2A (0.97) KMT2ACYP1B1ABCB1MEN1CYP3A4
Apigenin SCHEMBL29458838 0.97 KMT2A (0.97) KMT2ACYP1B1ABCB1MEN1CYP3A4
Apigenin SCHEMBL1658882 0.97 KMT2A (0.97) KMT2ACYP1B1ABCB1MEN1CYP3A4
Apigenin SCHEMBL30544810 0.97 KMT2A (0.97) KMT2ACYP1B1ABCB1MEN1CYP3A4
Apigenin SCHEMBL31477961 0.97 KMT2A (0.97) KMT2ACYP1B1ABCB1MEN1CYP3A4
Apigenin SCHEMBL29448148 0.97 KMT2A (0.97) KMT2ACYP1B1ABCB1MEN1CYP3A4
Apigenin SCHEMBL29872582 0.97 KMT2A (0.97) KMT2ACYP1B1ABCB1MEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119792270-A Application of apigenin chloride in preparation of medicines for preventing and treating respiratory syncytial virus infection 暨南大学 2025-04-11 CN claimed
CN-118914413-B Ultra-high performance liquid chromatography-tandem mass spectrometry method for simultaneously detecting 39 kinds of anthocyanin in litchi 海南省农业科学院三亚研究院(海南省实验动物研究中心) 2024-12-03 CN claimed
CN-119013022-A Combination therapy for cancer 来凯有限公司 2024-11-22 CN claimed
CN-118914413-A Ultra-high performance liquid chromatography-tandem mass spectrometry method for simultaneously detecting 39 kinds of anthocyanin in litchi 海南省农业科学院三亚研究院(海南省实验动物研究中心) 2024-11-08 CN claimed
CN-119792270-A Application of apigenin chloride in preparation of medicines for preventing and treating respiratory syncytial virus infection 暨南大学 2025-04-11 CN disclosed
CN-119792270-A Application of apigenin chloride in preparation of medicines for preventing and treating respiratory syncytial virus infection 暨南大学 2025-04-11 CN disclosed
CN-119792270-A Application of apigenin chloride in preparation of medicines for preventing and treating respiratory syncytial virus infection 暨南大学 2025-04-11 CN disclosed
CN-118914413-B Ultra-high performance liquid chromatography-tandem mass spectrometry method for simultaneously detecting 39 kinds of anthocyanin in litchi 海南省农业科学院三亚研究院(海南省实验动物研究中心) 2024-12-03 CN disclosed
CN-111787945-B Engineered nanovesicles as checkpoint blockers for cancer immunotherapy 北卡罗莱纳州立大学 2024-11-29 CN disclosed
CN-118914413-A Ultra-high performance liquid chromatography-tandem mass spectrometry method for simultaneously detecting 39 kinds of anthocyanin in litchi 海南省农业科学院三亚研究院(海南省实验动物研究中心) 2024-11-08 CN disclosed