SCHEMBL882501

SCHEMBL882501

CCC[C@H](NC(=O)/C(C#N)=C/c1cccc(Br)n1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP9X Q93008 11/20 1.00
UCHL1 P09936 1/20 1.00
USP5 P45974 1/20 1.00
STAT3 P40763 1/20 0.72
USP24 Q9UPU5 1/20 0.41
TACR3 P29371 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KDM4E B2RXH2 2/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
RGS12 O14924 1/20 0.40
GMNN O75496 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1317674 1.00 USP9X (1.00) USP9XUCHL1USP5STAT3USP24
SCHEMBL1317671 1.00 USP9X (1.00) USP9XUCHL1USP5STAT3USP24
SCHEMBL1317669 1.00 USP9X (1.00) USP9XUCHL1USP5STAT3USP24
SCHEMBL21592386 0.92 USP9X (0.85) USP9XUCHL1USP5STAT3USP24
SCHEMBL864886 0.92 USP9X (0.85) USP9XUCHL1USP5STAT3USP24
SCHEMBL864885 0.92 USP9X (0.85) USP9XUCHL1USP5STAT3USP24
SCHEMBL1315701 0.92 USP9X (0.85) USP9XUCHL1USP5STAT3ALDH1A1
SCHEMBL1315698 0.92 USP9X (0.85) USP9XUCHL1USP5STAT3ALDH1A1
SCHEMBL1315700 0.92 USP9X (0.85) USP9XUCHL1USP5STAT3ALDH1A1
SCHEMBL1315703 0.92 USP9X (0.85) USP9XUCHL1USP5STAT3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 220 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250262167-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2025-08-21 US claimed
CN-119909183-A Application of USP9X inhibitor in preparing ovarian cancer treatment drug and combined drug for improving ovarian cancer chemotherapeutic drug effect 天津康巢生物医药股份有限公司 2025-05-02 CN claimed
US-20250129430-A1 HIGH ATP-AFFINITY PROTEIN AS THERAPEUTIC TARGET FOR INTRACTABLE CANCER MOLECULAR SUBTYPES AND INHIBITOR THEREOF VeraVerse Co., Ltd. (KR) 2025-04-24 US claimed
EP-4442840-A1 HIGH ATP-AFFINITY PROTEIN AS THERAPEUTIC TARGET FOR INTRACTABLE CANCER MOLECULAR SUBTYPES AND INHIBITOR THEREOF Veraverse Co., Ltd. (KR) 2024-10-09 EP claimed
CN-118525105-A High ATP affinity proteins and inhibitors thereof as targets for treatment of refractory molecular subtype cancers 维拉沃斯公司 2024-08-20 CN claimed
CN-118203576-A Application of combination of USP5 inhibitor and PD-1 antibody in preparation of antitumor drugs 重庆医科大学附属第二医院 2024-06-18 CN claimed
US-20240118266-A1 CELL DEATH BIOMARKER UCL BUSINESS PLC (GB) 2024-04-11 US claimed
CN-113786409-B Compositions comprising phosphoinositide 3-kinase inhibitors and a second antiproliferative agent 甫康(上海)健康科技有限责任公司 2024-04-02 CN claimed
WO-2023204640-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF GASTRIC MUCOSAL DAMAGE-RELATED DISEASES CAUSED BY HELICOBACTER PYLORI AND PLATFORM FOR SCREENING FOR ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF HELICOBACTER PYLORI INFECTION 한국생명공학연구원 2023-10-26 WO claimed
EP-4213901-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION Massachusetts Institute of Technology (US) 2023-07-26 EP claimed
CN-116368384-A Compounds, targets and pathways for macrophage modulation 麻省理工学院 2023-06-30 CN claimed
WO-2023085716-A1 HIGH ATP-AFFINITY PROTEIN AS THERAPEUTIC TARGET FOR INTRACTABLE CANCER MOLECULAR SUBTYPES AND INHIBITOR THEREOF 연세대학교 산학협력단 2023-05-19 WO claimed
US-20230123585-A1 COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING CANCER USING DEUBIQUITINASE INHIBITORS UNIV CHICAGO (US) 2023-04-20 US claimed
EP-3337477-B1 COMPOSITIONS COMPRISING PHOSPHOINOSITIDE 3-KINASE INHIBITORS AND A SECOND ANTIPROLIFERATIVE AGENT CONVALIFE SHANGHAI CO LTD (CN) 2023-02-01 EP claimed
EP-3674300-B1 NOVEL BICYCLIC BROMODOMAIN INHIBITORS ZENITH EPIGENETICS LTD (CA) 2022-10-12 EP claimed
US-11446306-B2 Bicyclic bromodomain inhibitors ZENITH EPIGENETICS LTD. (CA) 2022-09-20 US claimed
US-20220111019-A1 BRCA1 MODULATING COMPOUNDS, FORMULATIONS THEREOF, AND USES THEREOF VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. 2022-04-14 US claimed
US-20220087950-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-03-24 US claimed
WO-2022060466-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2022-03-24 WO claimed
US-20260128175-A1 Methods and Systems for Analysis of Gene Expression Data AMPEL BIOSOLUTIONS LLC (US) 2026-05-07 US disclosed
US-20260125760-A1 METHODS OF TREATMENT AND DIAGNOSIS HUDSON INST OF MEDICAL RESEARCH (AU) 2026-05-07 US disclosed
US-20260109694-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF KUMQUAT BIOSCIENCES INC (US) 2026-04-23 US disclosed
US-12599592-B2 Therapeutic small molecules for treatment of pulmonary hypertension UNIVERSITY OF PITTSBURGH-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2026-04-14 US disclosed
US-20260097224-A1 METHODS FOR MODULATING NEUROPLASTICITY AMPA INC (US) 2026-04-09 US disclosed
EP-4720059-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Kumquat Biosciences Inc. (US) 2026-04-08 EP disclosed
US-12551555-B2 Compositions and methods for potentiating immune activity KUMQUAT BIOSCIENCES INC. (US) 2026-02-17 US disclosed
US-12548678-B2 Methods and systems for machine learning analysis of single nucleotide polymorphisms in lupus AMPEL BIOSOLUTIONS, LLC (US) 2026-02-10 US disclosed
US-20260024617-A1 METHODS AND SYSTEMS FOR PERSONALIZED THERAPIES SCIPHER MEDICINE CORP (US) 2026-01-22 US disclosed
US-12503464-B2 1,2,5-thiadiazolidin-3-one 1,1-dioxide containing compounds and uses thereof KUMQUAT BIOSCIENCES INC. (US) 2025-12-23 US disclosed
US-12475972-B2 Prediction system for identifying key heterogeneous molecules driving tumor metastasis NANJING HANWEI PUBLIC HEALTH TECHNOLOGY CO., LTD. (CN) 2025-11-18 US disclosed
EP-4443437-B1 PREDICTION SYSTEM FOR IDENTIFYING KEY HETEROGENEOUS MOLECULES THAT DRIVE TUMOR METASTASIS NANJING HANWEI PUBLIC HEALTH TECH CO LTD (CN) 2025-11-05 EP disclosed
CN-120789060-A Use of Degrasyn (WP 1130) as PTBP1 degrading agent in preparation of DMD therapeutic drug 中国药科大学 2025-10-17 CN disclosed
CN-120789060-A Use of Degrasyn (WP 1130) as PTBP1 degrading agent in preparation of DMD therapeutic drug 中国药科大学 2025-10-17 CN disclosed
US-20250304570-A1 BENZO-FUSED N-HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC (US) 2025-10-02 US disclosed
US-20250295659-A1 METHODS FOR TREATING TRAUMATIC BRAIN INJURY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-09-25 US disclosed
US-20250296927-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF KUMQUAT BIOSCIENCES INC. 2025-09-25 US disclosed
CN-120678923-A Application of USP9X as target in preparation of medicament for treating psoriasis 中国人民解放军空军军医大学 2025-09-23 CN disclosed
US-12419891-B2 Compositions for the treatment of pathogenic- and/or chemical-induced lung injury and for the treatment of cancer and methods of using same DUKE UNIVERSITY (US) 2025-09-23 US disclosed
US-20250288572-A1 COMPOSITIONS AND METHODS FOR TREATING PULMONARY VASCULAR DISEASE UNIVERSITY OF PITTSBURGH-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2025-09-18 US disclosed
EP-4615869-A1 COMBINATION THERAPY COMPRISING BISPECIFIC ANTIBODIES COMPRISING AN NRP1 BINDING DOMAIN Pinetree Therapeutics, Inc. (US) 2025-09-17 EP disclosed
US-20250262167-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2025-08-21 US disclosed
US-20250223580-A1 PROGRAMMABLE NUCLEASE-PEPTIDASE COMPOSITIONS THE BROAD INSTITUTE, INC. 2025-07-10 US disclosed
EP-3515559-B1 COMPOSITIONS AND METHODS FOR IDENTIFICATION, ASSESSMENT, PREVENTION, AND TREATMENT OF AML USING USP10 BIOMARKERS AND MODULATORS DANA FARBER CANCER INST INC (US) 2025-05-21 EP disclosed
US-12295955-B2 TTP phosphorylation for the identification of personalized medicines KING FAISAL SPECIALIST HOSPITAL & RESEARCH CENTRE (SA) 2025-05-13 US disclosed
US-20250145635-A1 COMPOUND CONTAINING BIS(AZANYLYLIDENE) SULFONYL STRUCTURE AND USE THEREOF IN MEDICINE SCINNOHUB PHARMACEUTICAL CO., LTD. (CN) 2025-05-08 US disclosed
CN-119909183-A Application of USP9X inhibitor in preparing ovarian cancer treatment drug and combined drug for improving ovarian cancer chemotherapeutic drug effect 天津康巢生物医药股份有限公司 2025-05-02 CN disclosed
US-20250129430-A1 HIGH ATP-AFFINITY PROTEIN AS THERAPEUTIC TARGET FOR INTRACTABLE CANCER MOLECULAR SUBTYPES AND INHIBITOR THEREOF VeraVerse Co., Ltd. (KR) 2025-04-24 US disclosed
US-12281301-B2 Sequencing-based proteomics THE BROAD INSTITUTE, INC. (US) 2025-04-22 US disclosed
US-12257254-B2 Compositions comprising phosphoinositide 3-kinase inhibitors and a second antiproliferative agent CONVALIFE (SHANGHAI) CO. LIMITED (CN) 2025-03-25 US disclosed
WO-2025053670-A1 VANILLIC ACID DERIVATIVE COMPOUND, THERAPEUTIC AGENT COMPOSITION FOR ALZHEIMER'S DISEASE COMPRISING SAME, AND THERAPEUTIC AGENT COMPOSITION FOR NEUROINFLAMMATION 주식회사 테라노큐어 2025-03-13 WO disclosed
US-12195490-B2 STRAD-binding agents and uses thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-01-14 US disclosed
US-12168640-B2 USP9X inhibitors ProDeg, LLC (US) 2024-12-17 US disclosed
US-20240398828-A1 HETERO-ATOM CONTAINING COMPOUNDS AND USES THEREOF KUMQUAT BIOSCIENCES INC. 2024-12-05 US disclosed
US-20240390406-A1 PHOSPHORYLATED TRISTETRAPROLIN AS A BIOMARKER AND THERAPEUTIC TARGET FOR ANTIAGING DRUGS KING FAISAL SPECIALIST HOSPITAL & RESEARCH CENTRE (SA) 2024-11-28 US disclosed
WO-2024243441-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF KUMQUAT BIOSCIENCES INC. (US) 2024-11-28 WO disclosed
US-20240390370-A1 Compositions for the Treatment of Pathogenic- And/Or Chemical-Induced Lung Injury and for the Treatment of Cancer and Methods of Using Same DUKE UNIVERSITY 2024-11-28 US disclosed
EP-4467978-A1 PHOSPHORYLATED TRISTETRAPROLIN AS A BIOMARKER AND THERAPEUTIC TARGET FOR ANTI-AGING DRUGS King Faisal Specialist Hospital & Research Centre (SA) 2024-11-27 EP disclosed
EP-4455136-A1 COMPOUND CONTAINING BIS(AZANYLYLIDENE) SULFONYL STRUCTURE AND USE THEREOF IN MEDICINE Scinnohub Pharmaceutical Co., Ltd. (CN) 2024-10-30 EP disclosed
EP-4442840-A1 HIGH ATP-AFFINITY PROTEIN AS THERAPEUTIC TARGET FOR INTRACTABLE CANCER MOLECULAR SUBTYPES AND INHIBITOR THEREOF Veraverse Co., Ltd. (KR) 2024-10-09 EP disclosed
EP-4443437-A1 PREDICTION SYSTEM FOR IDENTIFYING KEY HETEROGENEOUS MOLECULES THAT DRIVE TUMOR METASTASIS Nanjing Hanwei Public Health Technology Co., Ltd. (CN) 2024-10-09 EP disclosed
EP-4436967-A1 HETERO-ATOM CONTAINING COMPOUNDS AND USES THEREOF Kumquat Biosciences Inc. (US) 2024-10-02 EP disclosed
EP-4433462-A1 USP9X INHIBITORS Prodeg, LLC (US) 2024-09-25 EP disclosed
WO-2024189607-A1 METHODS AND BIOAVAILABLE HIGHLY PERMEABLE COMPOUNDS FOR DISEASES TREATMENT DIDENKO KIRILL (MX) 2024-09-19 WO disclosed
US-20240294467-A1 USP9X Inhibitors ProDeg, LLC 2024-09-05 US disclosed
CN-118556056-A Heteroatom-containing compounds and uses thereof 金橘生物科技公司 2024-08-27 CN disclosed
US-20240282453-A1 METHODS AND SYSTEMS FOR MACHINE LEARNING ANALYSIS OF SINGLE NUCLEOTIDE POLYMORPHISMS IN LUPUS AMPEL BIOSOLUTIONS, LLC 2024-08-22 US disclosed
CN-118525105-A High ATP affinity proteins and inhibitors thereof as targets for treatment of refractory molecular subtype cancers 维拉沃斯公司 2024-08-20 CN disclosed
CN-118510768-A Diazasulfinyl structure-containing compounds and their use in medicine 赛诺哈勃药业(成都)有限公司 2024-08-16 CN disclosed
CN-112794878-B Deubiquitinase activity probe and preparation and application thereof 中国科学院上海有机化学研究所 2024-08-16 CN disclosed
US-20240221867-A1 PREDICTION SYSTEM FOR IDENTIFYING KEY HETEROGENEOUS MOLECULES DRIVING TUMOR METASTASIS NANJING HANWEI PUBLIC HEALTH TECHNOLOGY CO., LTD. (CN) 2024-07-04 US disclosed
US-20240203555-A1 METHODS AND SYSTEMS FOR THERAPY MONITORING AND TRIAL DESIGN SCIPHER MEDICINE CORP (US) 2024-06-20 US disclosed
CN-118203576-A Application of combination of USP5 inhibitor and PD-1 antibody in preparation of antitumor drugs 重庆医科大学附属第二医院 2024-06-18 CN disclosed
CN-118203576-A Application of combination of USP5 inhibitor and PD-1 antibody in preparation of antitumor drugs 重庆医科大学附属第二医院 2024-06-18 CN disclosed
US-11993775-B2 Ubiquitin-specific peptidase 24 inhibitor, medicinal composition and method of delaying or reversing multidrug resistance in cancers using the same NATIONAL CHENG KUNG UNIVERSITY (TW) 2024-05-28 US disclosed
US-20240166641-A1 HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC. 2024-05-23 US disclosed
WO-2024102187-A1 COMBINATION THERAPY COMPRISING BISPECIFIC ANTIBODIES COMPRISING AN NRP1 BINDING DOMAIN PINETREE THERAPEUTICS, INC. (US) 2024-05-16 WO disclosed
US-20240153580-A1 METHODS AND SYSTEMS FOR PERSONALIZED THERAPIES Scipher Medicine Corporation 2024-05-09 US disclosed
US-11971402-B2 Methods and reagents for determination and treatment of organotropic metastasis CORNELL UNIVERSITY (US) 2024-04-30 US disclosed
US-20240118266-A1 CELL DEATH BIOMARKER UCL BUSINESS PLC (GB) 2024-04-11 US disclosed
US-11946094-B2 Combination therapies and methods of use thereof AUGUSTA UNIVERSITY RESEARCH INSTITUTE, INC. (US) 2024-04-02 US disclosed
WO-2024059041-A1 BENZO-FUSED N-HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES, INC. (US) 2024-03-21 WO disclosed
US-11925654-B2 Esters of 2-deoxy-monosaccharides with anti proliferative activity BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-03-12 US disclosed
CN-117542442-A Screening and anti-myeloma application of targeted c-Maf small molecule inhibitor 徐州医科大学 2024-02-09 CN disclosed
US-11883401-B2 Compositions for the treatment of pathogenic- and/or chemical-induced lung injury and for the treatment of cancer and methods of using same DUKE UNIVERSITY (US) 2024-01-30 US disclosed
EP-4305030-A1 HETEROCYCLES AND USES THEREOF Kumquat Biosciences Inc. (US) 2024-01-17 EP disclosed
US-11859014-B2 Peptidomimetics for the treatment of Norovirus infection EMORY UNIVERSITY (US) 2024-01-02 US disclosed
US-11859014-B2 Peptidomimetics for the treatment of Norovirus infection EMORY UNIVERSITY (US) 2024-01-02 US disclosed
US-11859014-B2 Peptidomimetics for the treatment of Norovirus infection EMORY UNIVERSITY (US) 2024-01-02 US disclosed
US-20230414590-A1 THERAPEUTIC SMALL MOLECULES FOR TREATMENT OF PULMONARY HYPERTENSION THE TEXAS A&M UNIVERSITY SYSTEM 2023-12-28 US disclosed
US-11827611-B2 Ubiquitin-specific peptidase 24 inhibitor, medicinal composition including the same and method of delaying or reversing multidrug resistance in cancers using the same NATIONAL CHENG KUNG UNIVERSITY (TW) 2023-11-28 US disclosed
US-20230364061-A1 THIAZOLIDINE DERIVATIVES FOR INHIBITING CAV3.2-USP5 INTERACTIONS ZYMEDYNE THERAPEUTICS INC. (CA) 2023-11-16 US disclosed
US-20230364243-A1 CANCER-SELECTIVE TARGET DEGRADATION BY TARGETING GROUP CAGED PROTACS BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2023-11-16 US disclosed
WO-2023204640-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF GASTRIC MUCOSAL DAMAGE-RELATED DISEASES CAUSED BY HELICOBACTER PYLORI AND PLATFORM FOR SCREENING FOR ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF HELICOBACTER PYLORI INFECTION 한국생명공학연구원 2023-10-26 WO disclosed
US-11789012-B2 Cell death biomarker UCL BUSINESS LTD (GB) 2023-10-17 US disclosed
US-20230310437-A1 TTP PHOSPHORYLATION FOR THE IDENTIFICATION OF PERSONALIZED MEDICINES KING FAISAL SPECIALIST HOSPITAL & RESEARCH CENTRE (SA) 2023-10-05 US disclosed
EP-3434788-B1 CLASSIFICATION AND ACTIONABILITY INDICES FOR LUNG CANCER LIFE TECHNOLOGIES CORP (US) 2023-08-23 EP disclosed
WO-2023150147-A1 METHOD OF PREVENTING HEARING LOSS THE JOHNS HOPKINS UNIVERSITY (US) 2023-08-10 WO disclosed
EP-4213901-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION Massachusetts Institute of Technology (US) 2023-07-26 EP disclosed
US-20230227418-A1 USP9X INHIBITORS ProDeg, LLC 2023-07-20 US disclosed
US-11691945-B2 USP9X inhibitors ProDeg, LLC (US) 2023-07-04 US disclosed
CN-116368384-A Compounds, targets and pathways for macrophage modulation 麻省理工学院 2023-06-30 CN disclosed
WO-2023116774-A1 COMPOUND CONTAINING BIS(AZANYLYLIDENE) SULFONYL STRUCTURE AND USE THEREOF IN MEDICINE 赛诺哈勃药业(成都)有限公司 2023-06-29 WO disclosed
WO-2023097927-A1 PREDICTION SYSTEM FOR IDENTIFYING KEY HETEROGENEOUS MOLECULES THAT DRIVE TUMOR METASTASIS 周建伟 2023-06-08 WO disclosed
WO-2023096928-A1 HETERO-ATOM CONTAINING COMPOUNDS AND USES THEREOF KUMQUAT BIOSCIENCES INC. (US) 2023-06-01 WO disclosed
US-20230160878-A1 METHOD OF SCREENING A THERAPY FOR INDUCTION OF FERROPTOSIS ARPEGGIO BIOSCIENCES, INC. 2023-05-25 US disclosed
WO-2023089601-A2 USP9X INHIBITORS ProDeg, LLC (US) 2023-05-25 WO disclosed
US-20230159916-A1 METHODS OF FUNCTIONAL LINKAGE OF CHROMOSOMAL POSITIONS ARPEGGIO BIOSCIENCES, INC. 2023-05-25 US disclosed
WO-2023091464-A1 USP9X INHIBITORS ProDeg, LLC (US) 2023-05-25 WO disclosed
WO-2023085716-A1 HIGH ATP-AFFINITY PROTEIN AS THERAPEUTIC TARGET FOR INTRACTABLE CANCER MOLECULAR SUBTYPES AND INHIBITOR THEREOF 연세대학교 산학협력단 2023-05-19 WO disclosed
US-20230150925-A1 USP9X INHIBITORS ProDeg, LLC 2023-05-18 US disclosed
US-11648251-B2 TTP phosphorylation as a biomarker in targeted therapy KING FAISAL SPECIALIST HOSPITAL & RESEARCH CENTRE (SA) 2023-05-16 US disclosed
US-20230142981-A1 METHOD FOR IDENTIFING A MARKER FOR A BIOLOGICAL INTERACTION ARPEGGIO BIOSCIENCES, INC. 2023-05-11 US disclosed
US-20230123585-A1 COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING CANCER USING DEUBIQUITINASE INHIBITORS UNIV CHICAGO (US) 2023-04-20 US disclosed
US-20230087443-A1 ENHANCEMENT OF CD47 BLOCKADE THERAPY BY PROTEASOME INHIBITORS PF ARGENTUM IP HOLDINGS LLC (US) 2023-03-23 US disclosed
US-20230092294-A1 COMPOSITIONS AND METHODS FOR POTENTIATING IMMUNE RESPONSE KUMQUAT BIOSCIENCES INC. 2023-03-23 US disclosed
EP-4150623-A2 METHODS AND SYSTEMS FOR MACHINE LEARNING ANALYSIS OF SINGLE NUCLEOTIDE POLYMORPHISMS IN LUPUS Ampel Biosolutions, LLC (US) 2023-03-22 EP disclosed
US-20230066999-A1 COMPOSITIONS COMPRISING PHOSPHOINOSITIDE 3-KINASE INHIBITORS AND A SECOND ANTIPROLIFERATIVE AGENT KARUS THERAPEUTICS LIMITED (GB) 2023-03-02 US disclosed
US-20230044323-A1 COMPOSITIONS AND METHODS FOR POTENTIATING IMMUNE ACTIVITY KUMQUAT BIOSCIENCES INC. 2023-02-09 US disclosed
EP-3337477-B1 COMPOSITIONS COMPRISING PHOSPHOINOSITIDE 3-KINASE INHIBITORS AND A SECOND ANTIPROLIFERATIVE AGENT CONVALIFE SHANGHAI CO LTD (CN) 2023-02-01 EP disclosed
WO-2022165185-A9 CANCER-SELECTIVE TARGET DEGRADATION BY TARGETING GROUP CAGED PROTACS BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2022-12-01 WO disclosed
CN-112206323-B Application of USP9x inhibitor in preparation of medicine for treating osteosarcoma 上海交通大学医学院 2022-11-25 CN disclosed
US-11491206-B1 Compositions and methods for the treatment of trail-resistant cancer DUKE UNIVERSITY (US) 2022-11-08 US disclosed
EP-4073242-A1 COMPOSITIONS AND METHODS FOR POTENTIATING IMMUNE ACTIVITY Kumquat Biosciences Inc. (US) 2022-10-19 EP disclosed
EP-3674300-B1 NOVEL BICYCLIC BROMODOMAIN INHIBITORS ZENITH EPIGENETICS LTD (CA) 2022-10-12 EP disclosed
CN-115103907-A Compositions and methods for enhancing immune activity 金橘生物科技公司 2022-09-23 CN disclosed
US-11446315-B2 Enhancement of CD47 blockade therapy by proteasome inhibitors PF ARGENTUM IP HOLDINGS LLC (US) 2022-09-20 US disclosed
US-11446306-B2 Bicyclic bromodomain inhibitors ZENITH EPIGENETICS LTD. (CA) 2022-09-20 US disclosed
WO-2022192598-A1 HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC. (US) 2022-09-15 WO disclosed
US-20220288207-A1 PHOTO INDUCED CONTROL OF PROTEIN DESTRUCTION BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2022-09-15 US disclosed
US-20220244263-A1 METHODS FOR TREATING SMALL CELL NEUROENDOCRINE AND RELATED CANCERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-08-04 US disclosed
WO-2022165185-A1 CANCER-SELECTIVE TARGET DEGRADATION BY TARGETING GROUP CAGED PROTACS BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2022-08-04 WO disclosed
CN-114652837-A Use of USP14 inhibitor for treating sepsis 南京医科大学 2022-06-24 CN disclosed
CN-114652837-A Use of USP14 inhibitor for treating sepsis 南京医科大学 2022-06-24 CN disclosed
WO-2022103706-A1 THERAPEUTIC SMALL MOLECULES FOR TREATMENT OF PULMONARY HYPERTENSION UNIVERSITY OF PITTSBURGH-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2022-05-19 WO disclosed
US-11324827-B2 Multifunctionalized polyethylene glycol derivative and preparation method therefor XIAMEN SINOPEG BIOTECH CO., LTD. (CN) 2022-05-10 US disclosed
US-20220111019-A1 BRCA1 MODULATING COMPOUNDS, FORMULATIONS THEREOF, AND USES THEREOF VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. 2022-04-14 US disclosed
US-11291669-B2 Compositions comprising phosphoinositide 3-kinase inhibitors and a second antiproliferative agent KARUS THERAPEUTICS LIMITED (GB) 2022-04-05 US disclosed
WO-2022061460-A1 THIAZOLIDINE DERIVATIVES FOR INHIBITING CAV3.2-USP5 INTERACTIONS ZYMEDYNE THERAPEUTICS INC. (CA) 2022-03-31 WO disclosed
US-20220087950-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-03-24 US disclosed
WO-2022060466-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2022-03-24 WO disclosed
US-20220041597-A1 INHIBITING UBIQUITIN SPECIFIC PEPTIDASE 9X FORMA THERAPEUTICS, INC. 2022-02-10 US disclosed
US-20210395300-A1 PEPTIDOMIMETICS FOR THE TREATMENT OF NOROVIRUS INFECTION UNIV EMORY (US) 2021-12-23 US disclosed
US-20210283139-A1 BIFUNCTIONAL MOLECULES FOR TARGETING UCHL5 AMPHISTA THERAPEUTICS LIMITED (GB) 2021-09-16 US disclosed
US-11021513-B2 Peptidomimetics for the treatment of norovirus infection EMORY UNIVERSITY (US) 2021-06-01 US disclosed
EP-3166604-B1 SUBSTANCES FOR THE TREATMENT OF RETROVIRAL INFECTIOUS DISEASES IMMUNOLOGIK GMBH (DE) 2020-11-18 EP disclosed
US-20200325130-A1 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same UNIV YALE (US) 2020-10-15 US disclosed
US-20200325130-A1 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same UNIV YALE (US) 2020-10-15 US disclosed
EP-3199181-B1 ANTI-INFLUENZA VIRUS AGENT, AND SCREENING METHOD FOR ANTI-INFLUENZA VIRUS AGENT JAPAN SCIENCE & TECH AGENCY (JP) 2020-05-06 EP disclosed
US-10588896-B2 Agents for the treatment of retroviral infectious diseases IMMUNOLOGIK GMBH (DE) 2020-03-17 US disclosed
US-20200071354-A1 PEPTIDOMIMETICS FOR THE TREATMENT OF NOROVIRUS INFECTION EMORY UNIVERSITY (US) 2020-03-05 US disclosed
US-20190105341-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies THE BOARD OF TRUSTEE OF THE LELAND STANFORD JUNIOR UNIVERSITY 2019-04-11 US disclosed
US-20190105341-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies THE BOARD OF TRUSTEE OF THE LELAND STANFORD JUNIOR UNIVERSITY 2019-04-11 US disclosed
US-20180360819-A1 ANTI-INFLUENZA VIRUS AGENT AND SCREENING METHOD FOR ANTI-INFLUENZA VIRUS AGENT JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2018-12-20 US disclosed
US-10149860-B2 Compositions and methods for treating alzheimer's disease and other tauopathies Board of Trustees of the Leland Stanford Junior University, Stanford University Office of Technology Licensing (US) 2018-12-11 US disclosed
EP-3370715-A1 PROTEOLYSIS TARGETING CHIMERA COMPOUNDS AND METHODS OF PREPARING AND USING SAME Yale University (US) 2018-09-12 EP disclosed
US-20180186785-A1 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same UNIV YALE (US) 2018-07-05 US disclosed
US-20180186785-A1 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same UNIV YALE (US) 2018-07-05 US disclosed
EP-2619184-B1 DEUBIQUITINASE INHIBITORS AND METHODS FOR USE OF THE SAME UNIV MICHIGAN REGENTS (US) 2018-05-23 EP disclosed
US-9938264-B2 Proteolysis targeting chimera compounds and methods of preparing and using same YALE UNIVERSITY (US) 2018-04-10 US disclosed
US-9938264-B2 Proteolysis targeting chimera compounds and methods of preparing and using same YALE UNIVERSITY (US) 2018-04-10 US disclosed
US-20170290821-A1 ANTI-INFLUENZA VIRUS AGENT AND SCREENING METHOD FOR ANTI-INFLUENZA VIRUS AGENT JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2017-10-12 US disclosed
EP-3199181-A1 ANTI-INFLUENZA VIRUS AGENT, AND SCREENING METHOD FOR ANTI-INFLUENZA VIRUS AGENT Japan Science and Technology Agency (JP) 2017-08-02 EP disclosed
US-20170202814-A1 AGENTS FOR THE TREATMENT OF RETROVIRAL INFECTIOUS DISEASES IMMUNOLOGIK GMBH (DE) 2017-07-20 US disclosed
WO-2017079267-A1 PROTEOLYSIS TARGETING CHIMERA COMPOUNDS AND METHODS OF PREPARING AND USING SAME YALE UNIVERSITY (US) 2017-05-11 WO disclosed
US-20170121321-A1 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same YALE UNIVERSITY 2017-05-04 US disclosed
US-20170121321-A1 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same YALE UNIVERSITY 2017-05-04 US disclosed
US-20170095457-A1 COMPOSITIONS AND METHODS OF DELIVERY OF DEUBIQUITINASE INHIBITORS PHARMAKEA, INC. 2017-04-06 US disclosed
US-20170095457-A1 COMPOSITIONS AND METHODS OF DELIVERY OF DEUBIQUITINASE INHIBITORS PHARMAKEA, INC. 2017-04-06 US disclosed
US-20170095457-A1 COMPOSITIONS AND METHODS OF DELIVERY OF DEUBIQUITINASE INHIBITORS PHARMAKEA, INC. 2017-04-06 US disclosed
US-20160151407-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2016-06-02 US disclosed
US-20160151407-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2016-06-02 US disclosed
US-20160151407-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2016-06-02 US disclosed
US-9289448-B2 Compositions and methods for treating alzheimer's disease and other tauopathies BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2016-03-22 US disclosed
US-9289448-B2 Compositions and methods for treating alzheimer's disease and other tauopathies BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2016-03-22 US disclosed
US-9289448-B2 Compositions and methods for treating alzheimer's disease and other tauopathies BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2016-03-22 US disclosed
WO-2016004915-A1 SUBSTANCES FOR THE TREATMENT OF RETROVIRAL INFECTIOUS DISEASES IMMUNOLOGIK GMBH (DE) 2016-01-14 WO disclosed
WO-2015183987-A1 COMPOSITIONS AND METHODS OF DELIVERY OF DEUBIQUITINASE INHIBITORS PHARMAKEA, INC. (US) 2015-12-03 WO disclosed
US-9096499-B2 Compounds for treatment of cell proliferative diseases BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-08-04 US disclosed
US-9096499-B2 Compounds for treatment of cell proliferative diseases BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-08-04 US disclosed
US-20150174150-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2015-06-25 US disclosed
US-20150174150-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2015-06-25 US disclosed
US-20150174150-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2015-06-25 US disclosed
US-20140357673-A1 Deubiquitinase Inhibitors and Methods for Use of the Same UNIV MICHIGAN (US) 2014-12-04 US disclosed
US-20140357673-A1 Deubiquitinase Inhibitors and Methods for Use of the Same UNIV MICHIGAN (US) 2014-12-04 US disclosed
US-20140329901-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-11-06 US disclosed
US-20140329901-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-11-06 US disclosed
US-8809377-B2 Deubiquitinase inhibitors and methods for use of the same THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2014-08-19 US disclosed
US-8809377-B2 Deubiquitinase inhibitors and methods for use of the same THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2014-08-19 US disclosed
US-8648102-B2 Compounds for treatment of cell proliferative diseases BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-02-11 US disclosed
US-8648102-B2 Compounds for treatment of cell proliferative diseases BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-02-11 US disclosed
US-20130244986-A1 METHODS OF TREATING SKIN DISORDERS WITH CAFFEIC ACID ANALOGS MOLECULIN LLC (US) 2013-09-19 US disclosed
US-20130244986-A1 METHODS OF TREATING SKIN DISORDERS WITH CAFFEIC ACID ANALOGS MOLECULIN LLC (US) 2013-09-19 US disclosed
US-8450337-B2 Methods of treating skin disorders with caffeic acid analogs MOLECULIN, LLC (US) 2013-05-28 US disclosed
US-8450337-B2 Methods of treating skin disorders with caffeic acid analogs MOLECULIN, LLC (US) 2013-05-28 US disclosed
US-20130129675-A1 INTERFERON THERAPIES IN COMBINATION WITH BLOCKADE OF STAT3 ACTIVATION BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-05-23 US disclosed
US-20130129675-A1 INTERFERON THERAPIES IN COMBINATION WITH BLOCKADE OF STAT3 ACTIVATION BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-05-23 US disclosed
US-20130129675-A1 INTERFERON THERAPIES IN COMBINATION WITH BLOCKADE OF STAT3 ACTIVATION BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-05-23 US disclosed
US-20120214850-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES PRIEBE WALDEMAR (US) 2012-08-23 US disclosed
US-20120214850-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES PRIEBE WALDEMAR (US) 2012-08-23 US disclosed
EP-2487156-A1 Compounds for treatment of cell proliferative diseases BOARD OF REGENTS THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-08-15 EP disclosed
EP-1701941-B1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES UNIV TEXAS (US) 2012-05-30 EP disclosed
US-20120077806-A1 Deubiquitinase Inhibitors and Methods for Use of the Same THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2012-03-29 US disclosed
WO-2012040527-A2 DEUBIQUITINASE INHIBITORS AND METHODS FOR USE OF THE SAME THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2012-03-29 WO disclosed
US-20120077806-A1 Deubiquitinase Inhibitors and Methods for Use of the Same THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2012-03-29 US disclosed
US-8119827-B2 Compounds for treatment of cell proliferative diseases BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-02-21 US disclosed
US-8119827-B2 Compounds for treatment of cell proliferative diseases BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-02-21 US disclosed
US-20110275577-A1 METHODS OF TREATING DERMATOLOGIC, GYNECOLOGIC, AND GENITAL DISORDERS WITH CAFFEIC ACID ANALOGS MOLECULIN, LLC (US) 2011-11-10 US disclosed
US-20110275577-A1 METHODS OF TREATING DERMATOLOGIC, GYNECOLOGIC, AND GENITAL DISORDERS WITH CAFFEIC ACID ANALOGS MOLECULIN, LLC (US) 2011-11-10 US disclosed
US-20110275577-A1 METHODS OF TREATING DERMATOLOGIC, GYNECOLOGIC, AND GENITAL DISORDERS WITH CAFFEIC ACID ANALOGS MOLECULIN, LLC (US) 2011-11-10 US disclosed
WO-2011069141-A2 INTERFERON THERAPIES IN COMBINATION WITH BLOCKADE OF STAT3 ACTIVATION BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2011-06-09 WO disclosed
US-20110021805-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2011-01-27 US disclosed
US-20110021805-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2011-01-27 US disclosed
US-20100292229-A1 TRYPHOSTIN-ANALOGS FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-11-18 US disclosed
US-20100292229-A1 TRYPHOSTIN-ANALOGS FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-11-18 US disclosed
US-7745468-B2 tyrphostin-like compounds that display a significant potency as kinase inhibitors, cause the downregulation of c-myc proto-oncogene and inhibit the growth and survival of cancerous cell lines; antiproliferative agents Board of Regents, University of Texas Systems The (US) 2010-06-29 US disclosed
US-7745468-B2 tyrphostin-like compounds that display a significant potency as kinase inhibitors, cause the downregulation of c-myc proto-oncogene and inhibit the growth and survival of cancerous cell lines; antiproliferative agents Board of Regents, University of Texas Systems The (US) 2010-06-29 US disclosed
US-20100152143-A1 Methods of Treating Skin Disorders with Caffeic Acid Analogs MOLECULIN, LLC (US) 2010-06-17 US disclosed
US-20100152143-A1 Methods of Treating Skin Disorders with Caffeic Acid Analogs MOLECULIN, LLC (US) 2010-06-17 US disclosed
WO-2008005954-A2 TRYPHOSTIN-ANALOGS FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2008-01-10 WO disclosed
WO-2005058829-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2005-06-30 WO disclosed
WO-2005058829-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2005-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11883401-B2 Compositions for the treatment of pathogenic- and/or chemical-induced lung injury and for the treatment of cancer and methods of using same DDIT3, MCL1, MYD88 USP9X 2668/4885UCHL1 1320/4885USP5 2054/4885
US-20100292229-A1 TRYPHOSTIN-ANALOGS FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES MYC, STAT3, MYCBP USP9X 4451/4885UCHL1 4077/4885USP5 3468/4885
US-20250295659-A1 METHODS FOR TREATING TRAUMATIC BRAIN INJURY CTTN, SRC, FYN USP9X 2210/4885UCHL1 238/4885USP5 1329/4885
US-10149860-B2 Compositions and methods for treating alzheimer's disease and other tauopathies USP9X, PSEN1, PSEN2 USP9X 1/4885UCHL1 24/4885USP5 25/4885
US-20230092294-A1 COMPOSITIONS AND METHODS FOR POTENTIATING IMMUNE RESPONSE MYD88, NFATC1, ICOS USP9X 1522/4885UCHL1 4026/4885USP5 2306/4885
US-20260109694-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF CCR10, SLC11A2, MSR1 USP9X 4466/4885UCHL1 4491/4885USP5 4866/4885
US-20100152143-A1 Methods of Treating Skin Disorders with Caffeic Acid Analogs CUTA, TYR, PPARA USP9X 4553/4885UCHL1 3330/4885USP5 3332/4885
US-11021513-B2 Peptidomimetics for the treatment of norovirus infection VIP, HAVCR2, NGLY1 USP9X 1168/4885UCHL1 1223/4885USP5 902/4885
US-11691945-B2 USP9X inhibitors USP9X, USP19, USP39 USP9X 1/4885UCHL1 54/4885USP5 7/4885
US-11925654-B2 Esters of 2-deoxy-monosaccharides with anti proliferative activity SLC2A2, SLC2A1, SLC2A4 USP9X 4139/4885UCHL1 3059/4885USP5 3988/4885
US-20110275577-A1 METHODS OF TREATING DERMATOLOGIC, GYNECOLOGIC, AND GENITAL DISORDERS WITH CAFFEIC ACID ANALOGS VHL, PRKDC, POLR1C USP9X 3737/4885UCHL1 3312/4885USP5 3130/4885
US-20200325130-A1 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same NEDD4, MDM2, CBL USP9X 203/4885UCHL1 9/4885USP5 31/4885
US-20250145635-A1 COMPOUND CONTAINING BIS(AZANYLYLIDENE) SULFONYL STRUCTURE AND USE THEREOF IN MEDICINE BCL9, USP9X, BCL9L USP9X 2/4885UCHL1 420/4885USP5 170/4885
US-20260125760-A1 METHODS OF TREATMENT AND DIAGNOSIS MCL1, BCL2L1, BCL2L11 USP9X 909/4885UCHL1 37/4885USP5 652/4885
US-20250288572-A1 COMPOSITIONS AND METHODS FOR TREATING PULMONARY VASCULAR DISEASE GLUL, GGT1, GLS USP9X 1946/4885UCHL1 638/4885USP5 1115/4885
US-20110021805-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES MYC, MKI67, MYCBP USP9X 3371/4885UCHL1 3672/4885USP5 3228/4885
US-20170121321-A1 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same NEDD4, MDM2, CBL USP9X 203/4885UCHL1 9/4885USP5 31/4885
US-20210283139-A1 BIFUNCTIONAL MOLECULES FOR TARGETING UCHL5 UCHL5, UCHL3, UCHL1 USP9X 99/4885UCHL1 3/4885USP5 4/4885
US-11993775-B2 Ubiquitin-specific peptidase 24 inhibitor, medicinal composition and method of delaying or reversing multidrug resistance in cancers using the same USP24, USP36, USP47 USP9X 56/4885UCHL1 154/4885USP5 52/4885
US-20160151407-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies USP9X, PSEN1, PSEN2 USP9X 1/4885UCHL1 24/4885USP5 25/4885
US-11859014-B2 Peptidomimetics for the treatment of Norovirus infection VIP, HAVCR2, NGLY1 USP9X 1168/4885UCHL1 1223/4885USP5 902/4885
US-12551555-B2 Compositions and methods for potentiating immune activity PTPRCAP, PTPN2, PTPRC USP9X 2195/4885UCHL1 2577/4885USP5 2560/4885
US-20240294467-A1 USP9X Inhibitors USP9X, USP19, USP39 USP9X 1/4885UCHL1 54/4885USP5 7/4885
US-20240390370-A1 Compositions for the Treatment of Pathogenic- And/Or Chemical-Induced Lung Injury and for the Treatment of Cancer and Methods of Using Same DDIT3, MCL1, MYD88 USP9X 2668/4885UCHL1 1320/4885USP5 2054/4885
US-20230364061-A1 THIAZOLIDINE DERIVATIVES FOR INHIBITING CAV3.2-USP5 INTERACTIONS USP3, USP5, CACNA1I USP9X 158/4885UCHL1 178/4885USP5 2/4885
US-11446306-B2 Bicyclic bromodomain inhibitors BRD4, BRD3, BRD2 USP9X 2268/4885UCHL1 4043/4885USP5 2272/4885
US-11446315-B2 Enhancement of CD47 blockade therapy by proteasome inhibitors CD47, PSMC1, PSMA5 USP9X 2246/4885UCHL1 3658/4885USP5 663/4885
US-20230087443-A1 ENHANCEMENT OF CD47 BLOCKADE THERAPY BY PROTEASOME INHIBITORS CD47, PSMC1, PSMA5 USP9X 2261/4885UCHL1 3656/4885USP5 633/4885
US-20180186785-A1 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same NEDD4, MDM2, CBL USP9X 203/4885UCHL1 9/4885USP5 31/4885
US-12599592-B2 Therapeutic small molecules for treatment of pulmonary hypertension GSTP1, GSTK1, GSTM1 USP9X 2208/4885UCHL1 924/4885USP5 1959/4885
US-20230044323-A1 COMPOSITIONS AND METHODS FOR POTENTIATING IMMUNE ACTIVITY NFATC1, MYD88, ICOS USP9X 1725/4885UCHL1 3700/4885USP5 2634/4885
US-20230364243-A1 CANCER-SELECTIVE TARGET DEGRADATION BY TARGETING GROUP CAGED PROTACS ADRM1, MYC, SKP2 USP9X 167/4885UCHL1 535/4885USP5 547/4885
US-20130244986-A1 METHODS OF TREATING SKIN DISORDERS WITH CAFFEIC ACID ANALOGS CUTA, TYR, PPARA USP9X 4553/4885UCHL1 3330/4885USP5 3332/4885
US-12503464-B2 1,2,5-thiadiazolidin-3-one 1,1-dioxide containing compounds and uses thereof BRCA1, STING1, IFNG USP9X 2788/4885UCHL1 4487/4885USP5 2148/4885
US-20190105341-A1 Compositions and Methods for Treating Alzheimer's Disease and Other Tauopathies USP9X, PSEN1, PSEN2 USP9X 1/4885UCHL1 24/4885USP5 25/4885
US-20220288207-A1 PHOTO INDUCED CONTROL OF PROTEIN DESTRUCTION UBE3C, PSMC1, UBE3A USP9X 173/4885UCHL1 141/4885USP5 127/4885
US-11291669-B2 Compositions comprising phosphoinositide 3-kinase inhibitors and a second antiproliferative agent MCL1, MYC, XIAP USP9X 2427/4885UCHL1 3419/4885USP5 2941/4885
US-20140357673-A1 Deubiquitinase Inhibitors and Methods for Use of the Same UCHL1, USP2, USP1 USP9X 33/4885UCHL1 1/4885USP5 19/4885
US-20240398828-A1 HETERO-ATOM CONTAINING COMPOUNDS AND USES THEREOF CD74, HLA-DRB1, CD47 USP9X 2444/4885UCHL1 2612/4885USP5 3358/4885
US-20120214850-A1 COMPOUNDS FOR TREATMENT OF CELL PROLIFERATIVE DISEASES MYC, MKI67, MYCBP USP9X 3371/4885UCHL1 3672/4885USP5 3228/4885
US-20230150925-A1 USP9X INHIBITORS USP9X, USP19, USP39 USP9X 1/4885UCHL1 54/4885USP5 7/4885
US-20230414590-A1 THERAPEUTIC SMALL MOLECULES FOR TREATMENT OF PULMONARY HYPERTENSION GSTP1, GSTK1, GSTM1 USP9X 1336/4885UCHL1 536/4885USP5 1909/4885
US-20260128175-A1 Methods and Systems for Analysis of Gene Expression Data IRAK4, TLR4, TLR2 USP9X 1716/4885UCHL1 2572/4885USP5 1923/4885
US-20120077806-A1 Deubiquitinase Inhibitors and Methods for Use of the Same UCHL1, USP2, USP1 USP9X 33/4885UCHL1 1/4885USP5 19/4885
US-20260024617-A1 METHODS AND SYSTEMS FOR PERSONALIZED THERAPIES SET, SSB, CNKSR1 USP9X 731/4885UCHL1 1561/4885USP5 1058/4885
US-11827611-B2 Ubiquitin-specific peptidase 24 inhibitor, medicinal composition including the same and method of delaying or reversing multidrug resistance in cancers using the same USP24, USP47, USP39 USP9X 62/4885UCHL1 118/4885USP5 51/4885
US-20200071354-A1 PEPTIDOMIMETICS FOR THE TREATMENT OF NOROVIRUS INFECTION VIP, HAVCR2, NGLY1 USP9X 1168/4885UCHL1 1223/4885USP5 902/4885
US-20260097224-A1 METHODS FOR MODULATING NEUROPLASTICITY GABRE, BDNF, GRIN2A USP9X 4260/4885UCHL1 2347/4885USP5 4159/4885
US-20130129675-A1 INTERFERON THERAPIES IN COMBINATION WITH BLOCKADE OF STAT3 ACTIVATION STAT3, STAT1, STAT5B USP9X 3930/4885UCHL1 4553/4885USP5 4112/4885
US-20210395300-A1 PEPTIDOMIMETICS FOR THE TREATMENT OF NOROVIRUS INFECTION VIP, HAVCR2, NGLY1 USP9X 1168/4885UCHL1 1223/4885USP5 902/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.