4-Guanidino-Benzoic Acid

4-Guanidino-Benzoic Acid

SCHEMBL273175

Cl.N=C(N)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of 4-Guanidino-Benzoic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 known ✓ P00918 1/20 0.47
F2 P00734 1/20 0.55
PRSS1 P07477 1/20 0.55
PRSS2 P07478 1/20 0.55
PRSS3 P35030 1/20 0.55
TMPRSS6 Q8IU80 1/20 0.55
ST14 Q9Y5Y6 1/20 0.55
ALDH1A1 P00352 1/20 0.52
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
MITF O75030 1/20 0.50
FFAR1 O14842 1/20 0.49
TP53 P04637 1/20 0.48
TSHR P16473 1/20 0.48
CA1 P00915 1/20 0.47
PTPN11 Q06124 1/20 0.47
EPHX2 P34913 1/20 0.47
NR1H4 Q96RI1 1/20 0.47
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
4-Guanidino-Benzoic Acid SCHEMBL10674543 1.00 F2 (0.55) F2PRSS1PRSS2PRSS3TMPRSS6
4-Guanidino-Benzoic Acid SCHEMBL28796971 0.98 F2 (0.53) F2PRSS1PRSS2PRSS3TMPRSS6
4-Guanidino-Benzoic Acid SCHEMBL211005 0.98 F2 (0.57) F2PRSS1PRSS2PRSS3TMPRSS6
4-Guanidino-Benzoic Acid SCHEMBL22127093 0.96 F2 (0.55) F2PRSS1PRSS2PRSS3TMPRSS6
4-Guanidino-Benzoic Acid SCHEMBL11123754 0.96 F2 (0.55) F2PRSS1PRSS2PRSS3TMPRSS6
4-Guanidino-Benzoic Acid SCHEMBL22127091 0.94 F2 (0.58) F2PRSS1PRSS2PRSS3TMPRSS6
4-Guanidino-Benzoic Acid SCHEMBL7563601 0.89 CA2 (0.50) F2PRSS1PRSS2PRSS3TMPRSS6
4-Guanidino-Benzoic Acid SCHEMBL19205978 0.89 CA2 (0.50) F2PRSS1PRSS2PRSS3TMPRSS6
4-Guanidino-Benzoic Acid SCHEMBL9303333 0.88 F2 (0.61) F2PRSS1PRSS2PRSS3TMPRSS6
Hydrochloric Acid SCHEMBL11226180 0.86 F2 (0.57) F2PRSS1PRSS2PRSS3TMPRSS6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 234 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119212415-A Perovskite solar cell and preparation method thereof 国网甘肃省电力公司电力科学研究院 2024-12-27 CN claimed
CN-115915788-A Perovskite solar cell and preparation method thereof 无锡极电光能科技有限公司 2023-04-04 CN claimed
CN-114805141-A 4-guanidinobenzoic acid aryl ester compound and application thereof in resisting SARS-CoV-2 virus 中国科学院上海药物研究所 2022-07-29 CN claimed
CN-114315651-A Preparation method of p-guanidinobenzoic acid hydrochloride 安徽昊帆生物有限公司 2022-04-12 CN claimed
CN-112827368-A Anti-pollution reverse osmosis membrane and preparation method thereof 中化(宁波)润沃膜科技有限公司 2021-05-25 CN claimed
CN-109792996-B Avermectin nano-powder and preparation and use method thereof 中国农业科学院农业环境与可持续发展研究所 2021-04-09 CN claimed
CN-111574409-A Recrystallization process method of nafamostat mesylate 河北省医疗器械与药品包装材料检验研究院(河北省医疗器械技术审评中心) 2020-08-25 CN claimed
CN-109792996-A A kind of Avermectins nano powder and its preparation and application method 中国农业科学院农业环境与可持续发展研究所 2019-05-24 CN claimed
US-20160296449-A1 Semi-Permanent Hair Straightening Composition And Method LUBRIZOL ADVANCED MATERIALS, INC. 2016-10-13 US claimed
EP-3065831-A1 SEMI-PERMANENT HAIR STRAIGHTENING COMPOSITION AND METHOD Lubrizol Advanced Materials, Inc. (US) 2016-09-14 EP claimed
CN-103641749-B A kind of preparation method of nafamostat mesylate SHANDONG YONGTAI CHEMICAL Co.,Ltd. (CN) 2016-02-10 CN claimed
WO-2015069823-A1 SEMI-PERMANENT HAIR STRAIGHTENING COMPOSITION AND METHOD LUBRIZOL ADVANCED MATERIALS, INC. (US) 2015-05-14 WO claimed
CN-103641749-A Preparation method of nafamostat mesylate SHANDONG YONGTAI CHEMICAL CO 2014-03-19 CN claimed
US-12610734-B2 Organic-inorganic hybrid perovskites CITY UNIVERSITY OF HONG KONG (CN) 2026-04-21 US disclosed
US-12408548-B2 Perovskite layer, fabrication method and use the same CITY UNIVERSITY OF HONG KONG (HK) 2025-09-02 US disclosed
US-20250188022-A1 PROCESS FOR THE PREPARATION OF NAFAMOSTAT, CAMOSTAT AND THEIR DERIVATIVES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2025-06-12 US disclosed
EP-0048433-A2 Novel amidine compounds, process for producing same and anti-complement agent comprising them TORII & CO., LTD. (JP) 1982-03-31 EP disclosed
US-4179511-A Antibacterial 3-(5-tetrazolyl) penam compounds PFIZER INC. (US) 1979-12-18 US disclosed
US-4143039-A ANTIBACTERIAL 3-(5-TETRAZOLYL)PENAM COMPOUNDS PFIZER INC. (US) 1979-03-06 US disclosed
US-4115385-A PENICILLINS PFIZER INC. (US) 1978-09-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250188022-A1 PROCESS FOR THE PREPARATION OF NAFAMOSTAT, CAMOSTAT AND THEIR DERIVATIVES TPMT, ADH1C, ADH1A CA2 588/4885F2 1213/4885PRSS1 1209/4885
US-12408548-B2 Perovskite layer, fabrication method and use the same KCNQ1, KCNQ2, SCNN1B CA2 895/4885F2 4794/4885PRSS1 2304/4885
US-20160296449-A1 Semi-Permanent Hair Straightening Composition And Method KRT18, PRKDC, DNMT1 CA2 3006/4885F2 1386/4885PRSS1 3492/4885
US-12610734-B2 Organic-inorganic hybrid perovskites CHN2, AR, H1-2 CA2 55/4885F2 4229/4885PRSS1 4631/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.