3-Hydroxybenzylhydrazine Dihydrochloride

3-Hydroxybenzylhydrazine Dihydrochloride

SCHEMBL473713

Cl.NNCc1cccc(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of 3-Hydroxybenzylhydrazine Dihydrochloride. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 1/20 0.53
DRD1 known ✓ P21728 1/20 0.53
CHRM2 known ✓ P08172 1/20 0.44
CHRM1 known ✓ P11229 1/20 0.44
CHRM3 known ✓ P20309 1/20 0.44
CA2 known ✓ P00918 1/20 0.44
OPRK1 known ✓ P41145 1/20 0.44
MAPT P10636 2/20 1.00
KDM4E B2RXH2 2/20 1.00
LMNA P02545 2/20 1.00
KMT2A Q03164 1/20 1.00
BLM P54132 1/20 1.00
PMP22 Q01453 1/20 1.00
CYP3A4 P08684 3/20 0.96
CYP1A2 P05177 1/20 0.96
PKM P14618 1/20 0.96
ALOX15 P16050 1/20 0.96
NFKB1 P19838 1/20 0.96
MAPK1 P28482 1/20 0.96
ENPP2 Q13822 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
3-Hydroxybenzylhydrazine Dihydrochloride SCHEMBL31298984 1.00 MAPT (1.00) MAPTKDM4ELMNAKMT2ABLM
3-Hydroxybenzylhydrazine Dihydrochloride SCHEMBL1309761 1.00 MAPT (1.00) MAPTKDM4ELMNAKMT2ABLM
3-Hydroxybenzylhydrazine Dihydrochloride SCHEMBL31298981 1.00 MAPT (1.00) MAPTKDM4ELMNAKMT2ABLM
3-Hydroxybenzylhydrazine Dihydrochloride SCHEMBL160617 0.98 CYP3A4 (1.00) MAPTKDM4ELMNAKMT2ABLM
3-Hydroxybenzylhydrazine Dihydrochloride SCHEMBL29594115 0.98 CYP3A4 (1.00) MAPTKDM4ELMNAKMT2ABLM
3-Hydroxybenzylhydrazine Dihydrochloride SCHEMBL23645200 0.89 CYP3A4 (0.82) MAPTKDM4ELMNAKMT2ABLM
SCHEMBL28584924 0.82 CYP3A4 (0.71) MAPTKDM4ELMNAKMT2ABLM
SCHEMBL14923237 0.82 CYP3A4 (0.71) MAPTKDM4ELMNAKMT2ABLM
SCHEMBL9416529 0.80 SLC2A4 (0.75) MAPTKDM4ELMNAKMT2ABLM
SCHEMBL6898308 0.78 CYP3A4 (0.67) MAPTKDM4ELMNAKMT2ABLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 329 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3274004-B1 CONTROLLED RELEASE MATRIX BARRIER STRUCTURE FOR SUBCUTANEOUS MEDICAL DEVICES SURMODICS INC (US) 2023-12-06 EP disclosed
US-11052177-B2 Antimicrobial polymer layers THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2021-07-06 US disclosed
EP-2611868-B1 BIODEGRADABLE TERPOLYMERS AND TERPOLYMER BLENDS AS PRESSURE-SENSITIVE ADHESIVES SURMODICS PHARMACEUTICALS INC (US) 2020-01-08 EP disclosed
US-10322209-B2 Polyurethanes for osteoimplants WARSAW ORTHOPEDIC, INC. (US) 2019-06-18 US disclosed
US-10308943-B2 Compositions with improved intravitreal half-life and uses thereof VITRISA THERAPEUTICS, INC. (US) 2019-06-04 US disclosed
US-20180340179-A1 COMPOSITIONS WITH IMPROVED INTRAVITREAL HALF-LIFE AND USES THEREOF SILICON VALLEY BANK 2018-11-29 US disclosed
US-10117974-B2 Non-fouling, anti-microbial, anti-thrombogenic graft-from compositions ARROW INTERNATIONAL, INC. (US) 2018-11-06 US disclosed
US-20180263919-A1 THERAPEUTIC ELECTROSPUN FIBER COMPOSITIONS UNIV JOHNS HOPKINS (US) 2018-09-20 US disclosed
US-20180250442-A1 POLYURETHANES FOR OSTEOIMPLANTS WARSAW ORTHOPEDIC INC (US) 2018-09-06 US disclosed
EP-1434608-B1 IMPROVED BONE GRAFT WARSAW ORTHOPEDIC INC (US) 2018-08-22 EP disclosed
EP-0064964-B1 THERAPEUTICALLY USEFUL 1-ALKYL-2-AMINOTETRALIN DERIVATIVES Astra Läkemedel Aktiebolag (SE) 1984-08-08 EP disclosed
US-4426386-A CNS DISORDERS ASTRA LAKEMEDEL AKTIEBOLAG (SE) 1984-01-17 US disclosed
EP-0097628-A2 Piperidine derivatives, processes for their preparation and pharmaceutical preparation containing them Carlsson, Per Arvid Emil (SE) 1984-01-04 EP disclosed
EP-0091437-A1 THERAPEUTICALLY USEFUL TETRALIN DERIVATIVES III, PROCESSES FOR PREPARATION AND PHARMACEUTICAL PREPARATIONS FOR SUCH COMPOUNDS Arvidsson, Folke Lars-Erik (SE) 1983-10-19 EP disclosed
EP-0084920-A2 New compounds useful as intermediates or starting materials for preparation of therapeutically useful phenyl-azacycloalkanes Carlsson, Per Arvid Emil (SE) 1983-08-03 EP disclosed
WO-1982004042-A1 THERAPEUTICALLY USEFUL TETRALIN DERIVATIVES III,PROCESSES FOR PREPARATION AND PHARMACEUTICAL PREPARATIONS FOR SUCH COMPOUNDS ARVIDSSON FOLKE LARS ERIK 1982-11-25 WO disclosed
EP-0064964-A1 Therapeutically useful 1-alkyl-2-aminotetralin derivatives Astra Läkemedel Aktiebolag (SE) 1982-11-17 EP disclosed
WO-1981003491-A1 THERAPEUTICALLY USEFUL TETRALIN DERIVATIVES ASTRA LAEKEMEDEL AB (SE) 1981-12-10 WO disclosed
EP-0041488-A1 Therapeutically useful tetralin derivatives Arvidsson, Folke Lars-Erik (SE) 1981-12-09 EP disclosed
EP-0030526-A1 New phenyl-azacycloalkanes, processes for preparation and pharmaceutical preparations for such compounds Astra Läkemedel Aktiebolag (SE) 1981-06-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180263919-A1 THERAPEUTIC ELECTROSPUN FIBER COMPOSITIONS NGF, BDNF, NTRK2 DRD2 4751/4885DRD1 4830/4885CHRM2 4096/4885
US-20180340179-A1 COMPOSITIONS WITH IMPROVED INTRAVITREAL HALF-LIFE AND USES THEREOF UACA, CRYAA, CRYAB DRD2 3814/4885DRD1 3637/4885CHRM2 3642/4885
US-10308943-B2 Compositions with improved intravitreal half-life and uses thereof UACA, CRYAA, CRYAB DRD2 3814/4885DRD1 3637/4885CHRM2 3642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.