Hydrochloric Acid

Hydrochloric Acid

SCHEMBL548656

Cl.O=C(O)c1ccc2nccnc2c1

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Hydrochloric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP known ✓ O00591 1/20 0.52
GABRD known ✓ O14764 1/20 0.52
GABRA1 known ✓ P14867 1/20 0.52
GABRB1 known ✓ P18505 1/20 0.52
GABRG2 known ✓ P18507 1/20 0.52
GABRB3 known ✓ P28472 1/20 0.52
GABRA5 known ✓ P31644 1/20 0.52
GABRA3 known ✓ P34903 1/20 0.52
GABRA2 known ✓ P47869 1/20 0.52
GABRB2 known ✓ P47870 1/20 0.52
GABRA4 known ✓ P48169 1/20 0.52
GABRE known ✓ P78334 1/20 0.52
GABRA6 known ✓ Q16445 1/20 0.52
GABRG1 known ✓ Q8N1C3 1/20 0.52
GABRG3 known ✓ Q99928 1/20 0.52
GABRQ known ✓ Q9UN88 1/20 0.52
GAA known ✓ P10253 2/20 0.51
ESR2 known ✓ Q92731 1/20 0.49
HDAC3 known ✓ O15379 1/20 0.47
HDAC4 known ✓ P56524 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30390410 0.98 MAPT (0.59) MAPTALDH1A1TDP1HPGDGABRP
SCHEMBL193423 0.98 MAPT (0.59) MAPTALDH1A1TDP1HPGDGABRP
Lithium Ion SCHEMBL31133341 0.96 MAPT (0.57) MAPTALDH1A1TDP1HPGDGABRP
SCHEMBL28612277 0.96 MAPT (0.57) MAPTALDH1A1TDP1HPGDGABRP
Pyridine SCHEMBL18550491 0.89 MAPT (0.55) MAPTALDH1A1TDP1HPGDGABRP
SCHEMBL1892689 0.86 GABRP (0.51) MAPTALDH1A1TDP1HPGDGABRP
SCHEMBL21819460 0.85 MAPT (0.47) MAPTALDH1A1TDP1HPGDGABRP
SCHEMBL27293915 0.83 MAPT (0.56) MAPTALDH1A1TDP1HPGDNPC1
Hydrochloric Acid SCHEMBL3596374 0.82 HTT (0.53) MAPTALDH1A1TDP1HPGDNPC1
SCHEMBL31175233 0.82 TDP1 (0.52) MAPTALDH1A1TDP1HPGDGABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240300931-A1 Composition and Methods for Treating Attention Deficit Disorders LIPPA ARNOLD STAN (US) 2024-09-12 US disclosed
US-20240100023-A1 Compositions and Methods For Treating Spinal Cord Injuries LIPPA ARNOLD S (US) 2024-03-28 US disclosed
US-20230373982-A1 Compositions And Methods For Treating Attention Deficit Disorders LIPPA ARNOLD STAN (US) 2023-11-23 US disclosed
US-20230129330-A1 Compositions And Methods For Treating Attention Deficit Disorders LIPPA ARNOLD STAN (US) 2023-04-27 US disclosed
US-20210340130-A1 Compositions and methods for treating attention deficit disorders LIPPA ARNOLD STAN (US) 2021-11-04 US disclosed
US-20190112300-A1 Compositions And Methods For Treating Attention Deficit Disorders LIPPA ARNOLD STAN (US) 2019-04-18 US disclosed
EP-3436021-A1 COMPOSITIONS AND METHODS FOR TREATING ATTENTION DEFICIT DISORDERS RespireRx Pharmaceuticals Inc. (US) 2019-02-06 EP disclosed
WO-2018009256-A1 COMPOSITIONS AND METHODS FOR TREATING ATTENTION DEFICIT DISORDERS RESPIRERX PHARMACEUTICALS, INC. (US) 2018-01-11 WO disclosed
US-9492440-B2 Bicyclic amides for enhancing glutamatergic synaptic responses RESPIRERX PHARMACEUTICALS INC (US) 2016-11-15 US disclosed
EP-2187888-B1 BICYCLIC AMIDES FOR ENHANCING GLUTAMATERGIC SYNAPTIC RESPONSES CORTEX PHARMA INC (US) 2015-10-21 EP disclosed
EP-2314295-A1 Pharmaceutical compositions for the prevention and treatment of complex diseases and their delivery by insertable medical devices Resverlogix, Inc (CA) 2011-04-27 EP disclosed
US-20110003835-A1 Methods for the treatment of respiratory depression CORTEX PHARMACEUTICALS, INC. (US) 2011-01-06 US disclosed
CN-101896183-A Bicyclic amides for enhancing glutamatergic synaptic responses CORTEX PHARMA INC 2010-11-24 CN disclosed
US-20100286177-A1 BICYCLIC AMIDES FOR THE TREATMENT OF RESPIRATORY DEPRESSION CORTEX PHARMACEUTICALS, INC. (US) 2010-11-11 US disclosed
CN-101862330-A Bicyclic amide is used for the treatment of application in the medicament of respiration inhibition in preparation CORTEX PHARMA INC 2010-10-20 CN disclosed
EP-2233140-A1 Bicyclic amides for enhancing glutamatergic synaptic responses Biovail Laboratories International SRL (BB) 2010-09-29 EP disclosed
EP-2187888-A2 BICYCLIC AMIDES FOR ENHANCING GLUTAMATERGIC SYNAPTIC RESPONSES CORTEX PHARMACEUTICALS, INC. (US) 2010-05-26 EP disclosed
WO-2009023126-A2 BICYCLIC AMIDES FOR ENHANCING GLUTAMATERGIC SYNAPTIC RESPONSES CORTEX PHARMACEUTICALS, INC. (US) 2009-02-19 WO disclosed
CN-101365446-A Pharmaceutical compositions for the prevention and treatment of complex diseases and their delivery via implantable medical devices RESVERLOGIX CORP (CA) 2009-02-11 CN disclosed
US-20090029987-A1 Pharmaceutical Compositions for the Prevention and Treatment of Complex Diseases and Their Delivery by Insertable Medical Devices RESVERLOGIX CORP. (CA) 2009-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210340130-A1 Compositions and methods for treating attention deficit disorders GRIN2A, GRIN2C, GRM2 GABRP 101/4885GABRD 119/4885GABRA1 148/4885
US-20240100023-A1 Compositions and Methods For Treating Spinal Cord Injuries CHAT, NTRK2, GMFG GABRP 206/4885GABRD 340/4885GABRA1 293/4885
US-20110003835-A1 Methods for the treatment of respiratory depression BDNF, CHRNA10, CHRNA3 GABRP 129/4885GABRD 174/4885GABRA1 104/4885
US-20230129330-A1 Compositions And Methods For Treating Attention Deficit Disorders GRIN2A, GRIN2C, GRM2 GABRP 101/4885GABRD 119/4885GABRA1 148/4885
US-20100286177-A1 BICYCLIC AMIDES FOR THE TREATMENT OF RESPIRATORY DEPRESSION BDNF, HCRTR2, CHRNA10 GABRP 102/4885GABRD 162/4885GABRA1 127/4885
US-20090029987-A1 Pharmaceutical Compositions for the Prevention and Treatment of Complex Diseases and Their Delivery by Insertable Medical Devices VCAM1, ICAM1, TGFB1 GABRP 3587/4885GABRD 3876/4885GABRA1 3737/4885
US-20230373982-A1 Compositions And Methods For Treating Attention Deficit Disorders GRIN2A, GRIN2C, GRM2 GABRP 101/4885GABRD 119/4885GABRA1 148/4885
US-20240300931-A1 Composition and Methods for Treating Attention Deficit Disorders GRIN2A, GRIN2C, NTRK2 GABRP 107/4885GABRD 130/4885GABRA1 159/4885
US-20190112300-A1 Compositions And Methods For Treating Attention Deficit Disorders GRIN2A, GRIN2C, GRM2 GABRP 101/4885GABRD 119/4885GABRA1 148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.