SCHEMBL13299549

SCHEMBL13299549

Cc1ccc(-c2ccccc2)nc1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.58
RAB9A P51151 4/20 0.52
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
KDM4E B2RXH2 6/20 0.47
MAPT P10636 4/20 0.47
PKM P14618 2/20 0.47
POLB P06746 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.44
NPC1 O15118 2/20 0.44
PDGFRB P09619 1/20 0.44
KDR P35968 1/20 0.44
FLT3 P36888 1/20 0.44
ASIC3 Q9UHC3 1/20 0.43
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
HPGD P15428 4/20 0.42
L3MBTL1 Q9Y468 4/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL28686928 0.98 ALDH1A1 (0.56) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL8989162 0.82 SMN1; SMN2 (0.56) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL10205828 0.80 ALDH1A1 (0.60) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL2189712 0.80 ALDH1A1 (0.56) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL3071714 0.80 NOS3 (0.55) ALDH1A1KDM4EMAPTSMN1; SMN2NOS3
SCHEMBL13299577 0.79 KMO (0.47) ALDH1A1RAB9AKDM4ESMN1; SMN2NPC1
SCHEMBL24250307 0.78 MEN1 (0.48) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL28173781 0.78 MEN1 (0.48) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL14975395 0.78 RAB9A (0.48) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL28247990 0.78 ASIC3 (0.50) ALDH1A1RAB9AMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240074301-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2024-02-29 US disclosed
US-20230348508-A1 METAL COMPLEX, ORGANIC ELECTROLUMINESCENT ELEMENT COMPRISING SAME, AND CONSUMER PRODUCT BEIJING BAYI SPACE LIQUID CRYSTAL TECHNOLOGY CO. LTD. (CN) 2023-11-02 US disclosed
US-20230345811-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-10-26 US disclosed
US-20230345812-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-10-26 US disclosed
US-11785839-B2 Organic light-emitting materials containing cyano-substituted ligand Beijing Summer Sprout Technology Co., Ltd. (CN) 2023-10-10 US disclosed
US-20230312627-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND DEVICE THEREOF Beijing Summer Sprout Technology Co., Ltd. (CN) 2023-10-05 US disclosed
US-20230320188-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-10-05 US disclosed
US-20230309375-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND DEVICE THEREOF Beijing Summer Sprout Technology Co., Ltd. (CN) 2023-09-28 US disclosed
US-20230303601-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-09-28 US disclosed
US-20230287011-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-09-14 US disclosed
US-20210376261-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2021-12-02 US disclosed
US-20210280802-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND DEVICE BEIJING SUMMER SPROUT TECHNOLOGY CO., LTD (CN) 2021-09-09 US disclosed
US-20210094978-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2021-04-01 US disclosed
US-9828360-B2 Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors ARRAY BIOPHARMA INC. (US) 2017-11-28 US disclosed
US-20160297796-A1 PYRROLIDINYL UREA, THIOUREA, GUANIDINE AND CYANOGUANIDINE COMPOUNDS AS TRKA KINASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2016-10-13 US disclosed
US-8367223-B2 Heteroleptic phosphorescent emitters UNIVERSAL DISPLAY CORPORATION (US) 2013-02-05 US disclosed
US-8367223-B2 Heteroleptic phosphorescent emitters UNIVERSAL DISPLAY CORPORATION (US) 2013-02-05 US disclosed
US-20100141127-A1 PHOSPHORESCENT EMITTERS UNIVERSAL DISPLAY CORPORATION (US) 2010-06-10 US disclosed
US-20100141127-A1 PHOSPHORESCENT EMITTERS UNIVERSAL DISPLAY CORPORATION (US) 2010-06-10 US disclosed
WO-2010056669-A1 PHOSPHORESCENT EMITTERS UNIVERSAL DISPLAY CORPORATION (US) 2010-05-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (15 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160297796-A1 PYRROLIDINYL UREA, THIOUREA, GUANIDINE AND CYANOGUANIDINE COMPOUNDS AS TRKA KINASE INHIBITORS TK1, UACA, TYMP ALDH1A1 3113/4885RAB9A 984/4885MEN1 3667/4885
US-20230309375-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND DEVICE THEREOF LEF1, L1CAM, PIEZO1 ALDH1A1 395/4885RAB9A 2516/4885MEN1 620/4885
US-20230303601-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES MGLL, SELENOI, APOL1 ALDH1A1 1729/4885RAB9A 2676/4885MEN1 4040/4885
US-20230312627-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND DEVICE THEREOF LEF1, CTCF, DNMT1 ALDH1A1 698/4885RAB9A 528/4885MEN1 2740/4885
US-20100141127-A1 PHOSPHORESCENT EMITTERS PAICS, TYMP, NUDT1 ALDH1A1 695/4885RAB9A 2958/4885MEN1 2832/4885
US-20230345812-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD1, OPRD1, OCIAD2 ALDH1A1 987/4885RAB9A 799/4885MEN1 2847/4885
US-20230320188-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD1, OCIAD2, MLX ALDH1A1 1799/4885RAB9A 1713/4885MEN1 2650/4885
US-20230287011-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD2, OXGR1, OCIAD1 ALDH1A1 983/4885RAB9A 1311/4885MEN1 3516/4885
US-11785839-B2 Organic light-emitting materials containing cyano-substituted ligand L1CAM, CYBA, ICOSLG ALDH1A1 1974/4885RAB9A 3060/4885MEN1 2531/4885
US-20240074301-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES ICOSLG, OCIAD2, OSBP ALDH1A1 658/4885RAB9A 1853/4885MEN1 4145/4885
US-20210376261-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD2, OCIAD1, TPO ALDH1A1 721/4885RAB9A 3415/4885MEN1 2992/4885
US-20210280802-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND DEVICE MLX, L1CAM, MCOLN1 ALDH1A1 1283/4885RAB9A 2551/4885MEN1 856/4885
US-20230348508-A1 METAL COMPLEX, ORGANIC ELECTROLUMINESCENT ELEMENT COMPRISING SAME, AND CONSUMER PRODUCT TRPM5, TRPM6, TRPM2 ALDH1A1 1357/4885RAB9A 2374/4885MEN1 641/4885
US-20210094978-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES L1CAM, EPCAM, LEF1 ALDH1A1 187/4885RAB9A 2535/4885MEN1 984/4885
US-20230345811-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OPRD1, L1CAM, OPRM1 ALDH1A1 2748/4885RAB9A 1045/4885MEN1 1446/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.