Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | ALDH1A1 | P00352 | 10/20 | 0.59 |
| ▸ | CYP3A4 | P08684 | 3/20 | 0.59 |
| ▸ | TSHR | P16473 | 3/20 | 0.59 |
| ▸ | RECQL | P46063 | 1/20 | 0.59 |
| ▸ | TDP1 | Q9NUW8 | 5/20 | 0.58 |
| ▸ | ALOX15 | P16050 | 2/20 | 0.58 |
| ▸ | MAPK1 | P28482 | 1/20 | 0.55 |
| ▸ | HSD17B10 | Q99714 | 1/20 | 0.55 |
| ▸ | L3MBTL1 | Q9Y468 | 1/20 | 0.55 |
| ▸ | HTT | P42858 | 2/20 | 0.54 |
| ▸ | LMNA | P02545 | 1/20 | 0.54 |
| ▸ | GAA | P10253 | 1/20 | 0.54 |
| ▸ | TUBB4A | P04350 | 2/20 | 0.53 |
| ▸ | TUBB | P07437 | 2/20 | 0.53 |
| ▸ | TUBA3C | P0DPH7 | 2/20 | 0.53 |
| ▸ | TUBA1B | P68363 | 2/20 | 0.53 |
| ▸ | TUBA4A | P68366 | 2/20 | 0.53 |
| ▸ | TUBB4B | P68371 | 2/20 | 0.53 |
| ▸ | TUBB3 | Q13509 | 2/20 | 0.53 |
| ▸ | TUBB2A | Q13885 | 2/20 | 0.53 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL29453576 | 1.00 | ALDH1A1 (0.59) | ALDH1A1CYP3A4TSHRRECQLTDP1 | |
| Hydrochloric Acid SCHEMBL15486437 | 0.98 | ALDH1A1 (0.58) | ALDH1A1CYP3A4TSHRRECQLTDP1 | |
| SCHEMBL20906666 | 0.86 | ALDH1A1 (0.56) | ALDH1A1CYP3A4TSHRRECQLTDP1 | |
| SCHEMBL358064 | 0.85 | TDP1 (0.58) | ALDH1A1CYP3A4TSHRRECQLTDP1 | |
| SCHEMBL11295773 | 0.85 | ALDH1A1 (0.63) | ALDH1A1CYP3A4TSHRRECQLTDP1 | |
| SCHEMBL28169538 | 0.84 | ALOX15 (0.51) | ALDH1A1CYP3A4TSHRRECQLTDP1 | |
| SCHEMBL810593 | 0.84 | ALDH1A1 (0.67) | ALDH1A1CYP3A4TSHRRECQLTDP1 | |
| SCHEMBL5685016 | 0.83 | ALOX15 (0.50) | ALDH1A1TDP1ALOX15MAPK1HSD17B10 | |
| SCHEMBL13637143 | 0.83 | ALDH1A1 (0.60) | ALDH1A1CYP3A4TSHRRECQLTDP1 | |
| SCHEMBL28169000 | 0.82 | ALDH1A1 (0.44) | ALDH1A1CYP3A4TSHRRECQLTDP1 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 508 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| CN-112094405-B | Synthesis and application method of modified PEG (polyethylene glycol) ball | 安徽生源化工有限公司 | 2023-05-26 | — | — | CN | claimed |
| CN-116115777-A | Polyethylene glycol-drug conjugate and preparation method and application thereof | 成都市第三人民医院 | 2023-05-16 | — | — | CN | claimed |
| CN-113717546-A | Method for preparing organic pigment yellow and pigment orange by modifying attapulgite | 宇虹颜料股份有限公司 | 2021-11-30 | — | — | CN | claimed |
| CN-109912994-A | Compound pearlescent pigment and its preparation method and application | 福建坤彩材料科技股份有限公司 | 2019-06-21 | — | — | CN | claimed |
| CN-109486403-A | A kind of preparation method of waterproof aqueous polyurethane coating and finishing agent | 段瑶瑶 | 2019-03-19 | — | — | CN | claimed |
| CN-109181458-A | A kind of preparation method of waterproofness core-shell type aqueous acrylic resin coating and finishing agent | 段瑶瑶 | 2019-01-11 | — | — | CN | claimed |
| CN-106866449-B | A kind of method that the acetyl-anisidine of 2 amino 4 is prepared using 2,4 dinitrophenol hydrogenating reduction by-product recoveries | 九江善水科技股份有限公司 | 2018-01-05 | — | — | CN | claimed |
| CN-106866449-A | A kind of method that the acetyl-anisidine of 2 amino 4 is prepared using 2,4 dinitrophenol hydrogenating reduction by-product recoveries | 九江善水科技股份有限公司 | 2017-06-20 | — | — | CN | claimed |
| CN-103173037-B | Dye composition, dye, preparation method thereof and raw material composition of dye | YANTAI ANOKY TEXTILE MATERIAL CO LTD | 2014-07-02 | — | — | CN | claimed |
| CN-103173037-A | Dye composition, dye, preparation method thereof and raw material composition of dye | YANTAI ANOKY TEXTILE MATERIAL CO LTD | 2013-06-26 | — | — | CN | claimed |
| US-20110319257-A1 | HIGH PERFORMANCE, HIGH DURABILITY NON-PRECIOUS METAL FUEL CELL CATALYSTS | 3M INNOVATIVE PROPERTIES COMPANY | 2011-12-29 | — | — | US | claimed |
| EP-2135313-B1 | HIGH PERFORMANCE, HIGH DURABILITY NON-PRECIOUS METAL FUEL CELL CATALYSTS | 3M INNOVATIVE PROPERTIES CO (US) | 2011-09-14 | — | — | EP | claimed |
| EP-2135313-A1 | HIGH PERFORMANCE, HIGH DURABILITY NON-PRECIOUS METAL FUEL CELL CATALYSTS | 3M Innovative Properties Company (US) | 2009-12-23 | — | — | EP | claimed |
| WO-2008127828-A1 | HIGH PERFORMANCE, HIGH DURABILITY NON-PRECIOUS METAL FUEL CELL CATALYSTS | 3M INNOVATIVE PROPERTIES COMPANY (US) | 2008-10-23 | — | — | WO | claimed |
| CN-100339442-C | Method for preparing organic pigment of red benzimidazolones | UNIV HUADONG TECHNOLOGY (CN) | 2007-09-26 | — | — | CN | claimed |
| CN-1569968-A | Yellow, orange benzimidazolone like azo dye making method | UNIV EAST CHINA SCIENCE & TECH (CN) | 2005-01-26 | — | — | CN | claimed |
| CN-1563202-A | Method for preparing organic pigment of red benzimidazolones | UNIV HUADONG TECHNOLOGY (CN) | 2005-01-12 | — | — | CN | claimed |
| EP-0079303-A2 | Stabilized covering form of CI pigment yellow 74 | CIBA-GEIGY AG (CH) | 1983-05-18 | — | — | EP | claimed |
| US-3957860-A | SULFAMIC ACID | CIBA-GEIGY AG (CH) | 1976-05-18 | — | — | US | claimed |
| WO-2026086794-A1 | ANTIMICROBIAL COMPOUNDS AND METHODS OF USE THEREOF | THE CHINESE UNIVERSITY OF HONG KONG (CN) | 2026-04-30 | — | — | WO | disclosed |
| US-20260076975-A1 | TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES | SHANGHAI RAISING PHARMACEUTICAL CO LTD (CN) | 2026-03-19 | — | — | US | disclosed |
| EP-4631573-A2 | TEAD INHIBITORS | Orion Corporation (FI) | 2025-10-15 | — | — | EP | disclosed |
| EP-4628098-A1 | TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES | Shanghai Raising Pharmaceutical Co., Ltd. (CN) | 2025-10-08 | — | — | EP | disclosed |
| EP-4323338-B1 | TEAD INHIBITORS | ORION CORP (FI) | 2025-10-08 | — | — | EP | disclosed |
| US-20250154107-A1 | 3,4-Dihydroisoquinolin-1(2H)-Ones Derivatives as STING Antagonists and the Use Thereof | BEIGENE SWITZERLAND GMBH (CH) | 2025-05-15 | — | — | US | disclosed |
| WO-2025063272-A1 | NICOTINAMIDE DERIVATIVE AND AGRICULTURAL AND HORTICULTURAL PLANT DISEASE CONTROL AGENT | クミアイ化学工業株式会社 | 2025-03-27 | — | — | WO | disclosed |
| EP-4448513-A1 | 3, 4-DIHYDROISOQUINOLIN-1 (2H) -ONES DERIVATIVES AS STING ANTAGONISTS AND THE USE THEREOF | BeiGene Switzerland GmbH (CH) | 2024-10-23 | — | — | EP | disclosed |
| CN-118401514-A | 3, 4-Dihydroisoquinolin-1 (2H) -one derivatives as STING antagonists and uses thereof | 百济神州有限公司 | 2024-07-26 | — | — | CN | disclosed |
| US-20240246908-A1 | TEAD INHIBITORS | ORION CORPORATION (FI) | 2024-07-25 | — | — | US | disclosed |
| CN-118146151-A | 4-Trifluoromethyl substituted quinoline and quinazoline compound and application thereof | 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) | 2024-06-07 | — | — | CN | disclosed |
| WO-2024114781-A1 | TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES | 上海日馨医药科技股份有限公司 | 2024-06-06 | — | — | WO | disclosed |
| CN-118121699-A | TPK agonists and methods of using the same for treating neurodegenerative diseases | 上海日馨医药科技股份有限公司 | 2024-06-04 | — | — | CN | disclosed |
| CN-114716385-B | Compound of targeted focal adhesion kinase, preparation method and application | 北京师范大学 | 2024-03-12 | — | — | CN | disclosed |
| CN-111615388-B | Immunotherapeutic agent for cancer | 斯汀格瑞治疗股份有限公司 | 2023-11-14 | — | — | CN | disclosed |
| CN-114436975-B | 2-trifluoromethyl-4-aminoquinazoline compound and application thereof | 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) | 2023-10-31 | — | — | CN | disclosed |
| WO-2023193795-A1 | COMPOUND TARGETING FOCAL ADHESION KINASE AND PREPARATION METHOD FOR AND APPLICATION OF COMPOUND | 北京师范大学 | 2023-10-12 | — | — | WO | disclosed |
| US-20230310428-A1 | EGFR INHIBITOR AND PREPARATION METHOD AND USE THEREOF | Hongyun Biotech Co., Ltd. (CN) | 2023-10-05 | — | — | US | disclosed |
| CN-111704555-B | Method for synthesizing 4-methoxy-2-nitroaniline by adopting continuous flow reactor | 爱斯特(成都)生物制药股份有限公司 | 2023-08-01 | — | — | CN | disclosed |
| WO-2023109912-A1 | 3, 4-DIHYDROISOQUINOLIN-1 (2H) -ONES DERIVATIVES AS STING ANTAGONISTS AND THE USE THEREOF | BEIGENE, LTD. (KY) | 2023-06-22 | — | — | WO | disclosed |
| CN-112094405-B | Synthesis and application method of modified PEG (polyethylene glycol) ball | 安徽生源化工有限公司 | 2023-05-26 | — | — | CN | disclosed |
| CN-112094405-B | Synthesis and application method of modified PEG (polyethylene glycol) ball | 安徽生源化工有限公司 | 2023-05-26 | — | — | CN | disclosed |
| CN-116115777-A | Polyethylene glycol-drug conjugate and preparation method and application thereof | 成都市第三人民医院 | 2023-05-16 | — | — | CN | disclosed |
| CN-113717156-B | EGFR inhibitor, preparation method and application thereof | 南京红云生物科技有限公司 | 2023-05-09 | — | — | CN | disclosed |
| CN-114539269-B | Nitrogen-containing macrocyclic compound, preparation method and application thereof | 上海医药工业研究院有限公司 | 2023-04-28 | — | — | CN | disclosed |
| EP-3658138-B1 | SUBSTITUTED-3H-IMIDAZO(4,5-C)PYRIDINE AND 1H-PYRROLO(2,3-C)PYRIDINE SERIES OF NOVEL ECTONUCLEOTIDE PYROPHSPHATASE/PHOSPHODIESTRASE-1 (ENPP1) AND STIMULATOR FOR INTERFERON GENES (STING) MODULATOR AS CANCER IMMUNOTHERAPEUTICS | STINGRAY THERAPEUTICS INC (US) | 2023-04-19 | — | — | EP | disclosed |
| CN-115916759-A | Substituted quinazoline compound, preparation method, pharmaceutical composition and application thereof | 南京红云生物科技有限公司 | 2023-04-04 | — | — | CN | disclosed |
| US-11555012-B2 | ACLY inhibitors and uses thereof | Nimbus Artemis, Inc. (US) | 2023-01-17 | — | — | US | disclosed |
| CN-109983014-B | Mutant isocitrate dehydrogenase inhibitors, compositions and methods thereof | 艾科生物科技有限公司 | 2022-12-23 | — | — | CN | disclosed |
| US-20220235064-A1 | OXO-PYRIDINE FUSION RING DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME | WELLMARKER BIO CO., LTD. (KR) | 2022-07-28 | — | — | US | disclosed |
| CN-114716385-A | Compound of targeting focal adhesion kinase, preparation method and application | 北京师范大学 | 2022-07-08 | — | — | CN | disclosed |
| CN-113135983-B | Antitumor compound and preparation method thereof | 四川大学华西医院 | 2022-06-24 | — | — | CN | disclosed |
| EP-4011885-A1 | OXO-PYRIDINE FUSION RING DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME | Wellmarker Bio Co., Ltd. (KR) | 2022-06-15 | — | — | EP | disclosed |
| CN-114539269-A | Nitrogen-containing macrocyclic compound, preparation method and application thereof | 上海医药工业研究院 | 2022-05-27 | — | — | CN | disclosed |
| CN-114436975-A | 2-trifluoromethyl-4-aminoquinazoline compound and application thereof | 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) | 2022-05-06 | — | — | CN | disclosed |
| EP-3980126-A1 | BENZO[H][1,6] NAPHTHYRIDIN-2(1H)-ONES AS BMX INHIBITORS, FOR USE AGAINST CANCER | Instituto de Medicina Molecular João Lobo Antunes (PT) | 2022-04-13 | — | — | EP | disclosed |
| CN-114206867-A | Benzo [ H ] [1,6] naphthyridin-2 (1H) -ones as BMX inhibitors for combating cancer | 医学分子研究所 | 2022-03-18 | — | — | CN | disclosed |
| CN-114206883-A | Oxopyridine fused ring derivative and pharmaceutical composition comprising the same | 伟迈可生物有限公司 | 2022-03-18 | — | — | CN | disclosed |
| WO-2021254464-A1 | SUBSTITUTED QUINAZOLINE COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF | 南京红云生物科技有限公司 | 2021-12-23 | — | — | WO | disclosed |
| CN-108976172-B | 4-pyrimidinediamine micromolecule organic compound and derivative and application thereof | 华东师范大学 | 2021-12-07 | — | — | CN | disclosed |
| WO-2021238827-A1 | EGFR INHIBITOR AND PREPARATION METHOD AND USE THEREOF | 南京红云生物科技有限公司 | 2021-12-02 | — | — | WO | disclosed |
| CN-113717546-A | Method for preparing organic pigment yellow and pigment orange by modifying attapulgite | 宇虹颜料股份有限公司 | 2021-11-30 | — | — | CN | disclosed |
| CN-113717156-A | EGFR inhibitor, preparation method and application thereof | 南京红云生物科技有限公司 | 2021-11-30 | — | — | CN | disclosed |
| CN-113609442-A | Fenton oxidation high-concentration wastewater multi-factor optimization method based on response curved surface | 中冶生态环保集团有限公司 | 2021-11-05 | — | — | CN | disclosed |
| US-11142524-B2 | Substituted-3H-imidazo[4,5-c]pyridine and 1H-pyrrolo[2,3-c]pyridine series of novel Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) and stimulator for interferon genes (STING) modulators as cancer immunotherapeutics | Stingray Therapeutics, Inc. (US) | 2021-10-12 | — | — | US | disclosed |
| CN-113135983-A | Antitumor compound and preparation method thereof | 四川大学华西医院 | 2021-07-20 | — | — | CN | disclosed |
| CN-106905245-B | 2, 4-disubstituted pyrimidines | 正大天晴药业集团股份有限公司 | 2021-06-25 | — | — | CN | disclosed |
| CN-112996496-A | substituted-3H-imidazo [4,5-c ] pyridines and 1H-pyrrolo [2,3-c ] pyridines as novel ectonucleotide pyrophosphatase/phosphodiesterase-1 (ENPP1) and interferon gene Stimulator (STING) modulators for cancer immunotherapy | 斯汀格瑞治疗股份有限公司 | 2021-06-18 | — | — | CN | disclosed |
| EP-3829561-A1 | SUBSTITUTED-3H-IMIDAZO[4,5-C]PYRIDINE AND 1H PYRROLO[2,3-C]PYRIDINE SERIES OF NOVEL ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE-1 (ENPP1) AND STIMULATOR FOR INTERFERON GENES (STING) MODULATORS AS CANCER IMMUNOTHERAPEUTICS | Stingray Therapeutics, Inc. (US) | 2021-06-09 | — | — | EP | disclosed |
| US-20210101899-A1 | INHIBITORS OF MUTANT ISOCITRATE DEHYDROGENASES AND COMPOSITIONS AND METHODS THEREOF | ISOCURE BIOSCIENCES INC (US) | 2021-04-08 | — | — | US | disclosed |
| WO-2021025407-A1 | OXO-PYRIDINE FUSION RING DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME | 웰마커바이오 주식회사 | 2021-02-11 | — | — | WO | disclosed |
| CN-112094405-A | Synthesis and application method of modified PEG (polyethylene glycol) ball | 安徽生源化工有限公司 | 2020-12-18 | — | — | CN | disclosed |
| CN-112094405-A | Synthesis and application method of modified PEG (polyethylene glycol) ball | 安徽生源化工有限公司 | 2020-12-18 | — | — | CN | disclosed |
| WO-2020245430-A1 | BENZO[H][1,6] NAPHTHYRIDIN-2(1H)-ONES AS BMX INHIBITORS, FOR USE AGAINST CANCER | INSTITUTO DE MEDICINA MOLECULAR JOAO LOBO ANTUNES (PT) | 2020-12-10 | — | — | WO | disclosed |
| CN-111704555-A | Method for synthesizing 4-methoxy-2-nitroaniline by adopting continuous flow reactor | 爱斯特(成都)生物制药股份有限公司 | 2020-09-25 | — | — | CN | disclosed |
| US-10781207-B2 | Inhibitors of mutant isocitrate dehydrogenases and compositions and methods thereof | ISOCURE BIOSCIENCES INC. (US) | 2020-09-22 | — | — | US | disclosed |
| CN-111615388-A | Novel ectonucleotide pyrophosphatase/phosphodiesterase-1 (ENPP1) and interferon gene Stimulator (STING) modulators of substituted-3H-imidazo [4,5-c ] pyridines and 1H-pyrrolo [2,3-c ] pyridines series as cancer immunotherapeutic agents | 斯汀格瑞治疗股份有限公司 | 2020-09-01 | — | — | CN | disclosed |
| EP-3246328-B1 | QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR, AND PREPARATION AND APPLICATION THEREOF | BEIJING SCITECH MQ PHARMACEUTICALS LTD (CN) | 2020-07-22 | — | — | EP | disclosed |
| US-10689376-B2 | Substituted-3H-imidazo [4,5-c] pyridine and 1H-pyrrolo[2,3-c]pyridine series of novel ectonucleotide pyrophosphatase/phosphodiesterase-1 (ENPP1) and stimulator for interferon genes (STING) modulators as cancer immunotherapeutics | Stingray Therapeutics, Inc. (US) | 2020-06-23 | — | — | US | disclosed |
| CN-111247137-A | Pyrimidine compound, preparation method and medical application thereof | 恩瑞生物医药科技(上海)有限公司 | 2020-06-05 | — | — | CN | disclosed |
| US-20200148634-A1 | ACLY INHIBITORS AND USES THEREOF | Nimbus Artemis, Inc. | 2020-05-14 | — | — | US | disclosed |
| CN-106964355-B | Preparation method and application of copper-nickel oxide loaded graphene-based catalyst | 江苏金聚合金材料有限公司 | 2020-02-21 | — | — | CN | disclosed |
| WO-2020028724-A1 | SUBSTITUTED-3H-IMIDAZO[4,5-C]PYRIDINE AND 1H-PYRROLO[2,3-C]PYRIDINE SERIES OF NOVEL ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE-1 (ENPP1) AND STIMULATOR FOR INTERFERON GENES (STING) MODULATORS AS CANCER IMMUNOTHERAPEUTICS | Stingray Therapeutics, Inc. (US) | 2020-02-06 | — | — | WO | disclosed |
| US-20200039979-A1 | Substituted-3H-imidazo[4,5-c]pyridine and 1H-pyrrolo[2,3-c]pyridine series of novel Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) and Stimulator for Interferon Genes (STING) modulators as cancer immunotherapeutics | Stingray Therapeutics, Inc. | 2020-02-06 | — | — | US | disclosed |
| CN-107586278-B | 2, 4-diamino pyrimidine compound, preparation method, pharmaceutical composition and application thereof | 中国科学院上海药物研究所 | 2020-01-10 | — | — | CN | disclosed |
| EP-2844642-B1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD PHARMA INC (US) | 2019-11-13 | — | — | EP | disclosed |
| EP-2844642-B1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD PHARMA INC (US) | 2019-11-13 | — | — | EP | disclosed |
| EP-3526221-A1 | INHIBITORS OF MUTANT ISOCITRATE DEHYDROGENASES AND COMPOSITIONS AND METHODS THEREOF | Isocure Biosciences Inc. (US) | 2019-08-21 | — | — | EP | disclosed |
| US-10383831-B2 | 2,4,6-trialkoxystryl aryl sulfones, sulfonamides and carboxamides, and methods of preparation and use | Temple University—Of the Commonwealth System of Higher Education (US) | 2019-08-20 | — | — | US | disclosed |
| US-20190233414-A1 | INHIBITORS OF MUTANT ISOCITRATE DEHYDROGENASES AND COMPOSITIONS AND METHODS THEREOF | ISOCURE BIOSCIENCES INC (US) | 2019-08-01 | — | — | US | disclosed |
| CN-109912994-A | Compound pearlescent pigment and its preparation method and application | 福建坤彩材料科技股份有限公司 | 2019-06-21 | — | — | CN | disclosed |
| CN-109486403-A | A kind of preparation method of waterproof aqueous polyurethane coating and finishing agent | 段瑶瑶 | 2019-03-19 | — | — | CN | disclosed |
| US-20190031655-A1 | Substituted-3H-imidazo[4,5-c]pyridine and 1H-pyrrolo[2,3-c]pyridine series of novel Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) and Stimulator for Interferon Genes (STING) modulators as cancer immunotherapeutics | Stingray Therapeutics, Inc. | 2019-01-31 | — | — | US | disclosed |
| CN-109181458-A | A kind of preparation method of waterproofness core-shell type aqueous acrylic resin coating and finishing agent | 段瑶瑶 | 2019-01-11 | — | — | CN | disclosed |
| US-10130633-B2 | Compounds | BAYER PHARMA AKTIENGESELLSCHAFT (DE) | 2018-11-20 | — | — | US | disclosed |
| US-10106508-B2 | Quinazoline heterocyclic compound as EGFR kinase inhibitor and preparation and application thereof | BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) | 2018-10-23 | — | — | US | disclosed |
| WO-2018187812-A1 | HIGH-RATE TREATMENT OF 3-NITRO-1,2,4-TRIAZOL-5-ONE (NTO) AND OTHER MUNITIONS COMPOUNDS | ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) | 2018-10-11 | — | — | WO | disclosed |
| US-20180243239-A1 | 2,4,6-TRIALKOXYSTRYL ARYL SULFONES, SULFONAMIDES AND CARBOXAMIDES, AND METHODS OF PREPARATION AND USE | TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION | 2018-08-30 | — | — | US | disclosed |
| US-10059688-B2 | Protein tyrosine kinase modulators and methods of use | BETTA PHARMACEUTICALS CO., LTD. (CN) | 2018-08-28 | — | — | US | disclosed |
| CN-108147971-A | A kind of preparation method of adjacent nitro P-nethoxyaniline | 南京科技职业学院 | 2018-06-12 | — | — | CN | disclosed |
| WO-2018071404-A1 | INHIBITORS OF MUTANT ISOCITRATE DEHYDROGENASES AND COMPOSITIONS AND METHODS THEREOF | ISOCURE BIOSCIENCES INC. (US) | 2018-04-19 | — | — | WO | disclosed |
| CN-105669525-B | A kind of synthetic method of N ((2 (base of 1,3 dioxoisoindolin 2) propiono) 5 methoxyl groups) formamide | 苏州艾缇克药物化学有限公司 | 2018-03-09 | — | — | CN | disclosed |
| US-9902691-B2 | Intermediates and methods for synthesizing calicheamicin derivatives | PFIZER INC. (US) | 2018-02-27 | — | — | US | disclosed |
| US-20180009782-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | BETTA PHARMACEUTICALS CO., LTD. (CN) | 2018-01-11 | — | — | US | disclosed |
| US-20180009782-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | BETTA PHARMACEUTICALS CO., LTD. (CN) | 2018-01-11 | — | — | US | disclosed |
| CN-106866449-B | A kind of method that the acetyl-anisidine of 2 amino 4 is prepared using 2,4 dinitrophenol hydrogenating reduction by-product recoveries | 九江善水科技股份有限公司 | 2018-01-05 | — | — | CN | disclosed |
| US-20170355683-A1 | QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR AND PREPARATION AND APPLICATION THEREOF | BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) | 2017-12-14 | — | — | US | disclosed |
| EP-2887943-B1 | NOVEL 4,6-DISUBSTITUTED AMINOPYRIMIDINE DERIVATIVES | VIROSTATICS SRL (IT) | 2017-12-06 | — | — | EP | disclosed |
| US-9834518-B2 | Compounds for inhibiting cell proliferation in EGFR-driven cancers | ARIAD PHARMACEUTICALS, INC. (US) | 2017-12-05 | — | — | US | disclosed |
| US-9834518-B2 | Compounds for inhibiting cell proliferation in EGFR-driven cancers | ARIAD PHARMACEUTICALS, INC. (US) | 2017-12-05 | — | — | US | disclosed |
| US-9834518-B2 | Compounds for inhibiting cell proliferation in EGFR-driven cancers | ARIAD PHARMACEUTICALS, INC. (US) | 2017-12-05 | — | — | US | disclosed |
| US-9834571-B2 | Compounds for inhibiting cell proliferation in EGFR-driven cancers | ARIAD PHARMACEUTICALS, INC. (US) | 2017-12-05 | — | — | US | disclosed |
| US-9834571-B2 | Compounds for inhibiting cell proliferation in EGFR-driven cancers | ARIAD PHARMACEUTICALS, INC. (US) | 2017-12-05 | — | — | US | disclosed |
| US-9834571-B2 | Compounds for inhibiting cell proliferation in EGFR-driven cancers | ARIAD PHARMACEUTICALS, INC. (US) | 2017-12-05 | — | — | US | disclosed |
| EP-3246328-A1 | QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR, AND PREPARATION AND APPLICATION THEREOF | Beijing Scitech-MQ Pharmaceuticals Limited (CN) | 2017-11-22 | — | — | EP | disclosed |
| EP-2940000-B1 | PROCESS FOR PREPARING METHYL ACETATE | DALIAN INST CHEMICAL PHYSICS CAS (CN) | 2017-10-18 | — | — | EP | disclosed |
| US-9783524-B2 | Protein tyrosine kinase modulators and methods of use | BETTA PHARMACEUTICALS CO., LTD. (CN) | 2017-10-10 | — | — | US | disclosed |
| US-9783524-B2 | Protein tyrosine kinase modulators and methods of use | BETTA PHARMACEUTICALS CO., LTD. (CN) | 2017-10-10 | — | — | US | disclosed |
| US-9783524-B2 | Protein tyrosine kinase modulators and methods of use | BETTA PHARMACEUTICALS CO., LTD. (CN) | 2017-10-10 | — | — | US | disclosed |
| CN-107176951-A | A kind of carbamide compounds, its preparation method and its medical usage | 恩瑞生物医药科技(上海)有限公司 | 2017-09-19 | — | — | CN | disclosed |
| US-20170204084-A1 | NOVEL 4,6-DISUBSTITUTED AMINOPYRIMIDINE DERIVATIVES HAVE ANTI-HIV ACTIVITY | VIROSTATICS SRL (IT) | 2017-07-20 | — | — | US | disclosed |
| EP-2976327-B1 | 3-ACETYLAMINO-1-(PHENYL-HETEROARYL-AMINOCARBONYL OR PHENYL-HETEROARYL-CARBONYLAMINO)BENZENE DERIVATIVES FOR THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS | Bayer Pharma AG (DE) | 2017-06-21 | — | — | EP | disclosed |
| CN-106866449-A | A kind of method that the acetyl-anisidine of 2 amino 4 is prepared using 2,4 dinitrophenol hydrogenating reduction by-product recoveries | 九江善水科技股份有限公司 | 2017-06-20 | — | — | CN | disclosed |
| US-9643979-B2 | Inhibitors of DNA gyrase for the treatment of bacterial infections | VITAS PHARMA RESEARCH PRIVATE LIMITED (IN) | 2017-05-09 | — | — | US | disclosed |
| US-9617225-B2 | 4,6-disubstituted aminopyrimidine derivatives have anti-HIV activity | VIROSTATICS SRL (IT) | 2017-04-11 | — | — | US | disclosed |
| EP-3147285-A2 | PURINONE COMPOUNDS AS KINASE INHIBITORS | Pharmacyclics, Inc. (US) | 2017-03-29 | — | — | EP | disclosed |
| EP-3147285-A2 | PURINONE COMPOUNDS AS KINASE INHIBITORS | Pharmacyclics, Inc. (US) | 2017-03-29 | — | — | EP | disclosed |
| WO-2017023912-A1 | 2,4,6-TRIALKOXYSTRYL ARYL SULFONES, SULFONAMIDES AND CARBOXAMIDES, AND METHODS OF PREPARATION AND USE | TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) | 2017-02-09 | — | — | WO | disclosed |
| WO-2017023912-A1 | 2,4,6-TRIALKOXYSTRYL ARYL SULFONES, SULFONAMIDES AND CARBOXAMIDES, AND METHODS OF PREPARATION AND USE | TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) | 2017-02-09 | — | — | WO | disclosed |
| CN-106317023-A | Preparation method and application of indazole compound | 中国科学院上海药物研究所 | 2017-01-11 | — | — | CN | disclosed |
| US-20160368924-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | PHARMACYCLICS, INC. | 2016-12-22 | — | — | US | disclosed |
| US-20160368924-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | PHARMACYCLICS, INC. | 2016-12-22 | — | — | US | disclosed |
| US-20160368924-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | PHARMACYCLICS, INC. | 2016-12-22 | — | — | US | disclosed |
| US-9469642-B2 | Purinone compounds as kinase inhibitors | PHARMACYCLICS LLC (US) | 2016-10-18 | — | — | US | disclosed |
| US-9469642-B2 | Purinone compounds as kinase inhibitors | PHARMACYCLICS LLC (US) | 2016-10-18 | — | — | US | disclosed |
| US-9469642-B2 | Purinone compounds as kinase inhibitors | PHARMACYCLICS LLC (US) | 2016-10-18 | — | — | US | disclosed |
| US-9446044-B2 | DYRK1 inhibitors and uses thereof | DIAXONHIT (FR) | 2016-09-20 | — | — | US | disclosed |
| US-20160263122-A1 | NOVEL COMPOUNDS | BAYER PHARMA AKTIENGESELLSCHAFT (DE) | 2016-09-15 | — | — | US | disclosed |
| US-9440226-B2 | Method for preparing methyl acetate | DALIAN INSTITUTE OF CHEMICAL PHYSICS, CHINESE ACADEMY OF SCIENCES (CN) | 2016-09-13 | — | — | US | disclosed |
| US-20160244469-A1 | Compounds for Inhibiting Cell Proliferation in EGFR-Driven Cancers | TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) | 2016-08-25 | — | — | US | disclosed |
| US-20160244469-A1 | Compounds for Inhibiting Cell Proliferation in EGFR-Driven Cancers | TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) | 2016-08-25 | — | — | US | disclosed |
| US-20160244469-A1 | Compounds for Inhibiting Cell Proliferation in EGFR-Driven Cancers | TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) | 2016-08-25 | — | — | US | disclosed |
| CN-105669525-A | Synthetic method of N-((2-(1,3-dioxo-dihydroisoindol-2-yl)-propionyl)-5-methoxy)formamide | 苏州艾缇克药物化学有限公司 | 2016-06-15 | — | — | CN | disclosed |
| CN-105669525-A | Synthetic method of N-((2-(1,3-dioxo-dihydroisoindol-2-yl)-propionyl)-5-methoxy)formamide | 苏州艾缇克药物化学有限公司 | 2016-06-15 | — | — | CN | disclosed |
| US-20160145237-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | BETTA PHARMACEUTICALS CO., LTD (CN) | 2016-05-26 | — | — | US | disclosed |
| US-20160145237-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | BETTA PHARMACEUTICALS CO., LTD (CN) | 2016-05-26 | — | — | US | disclosed |
| US-20160145237-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | BETTA PHARMACEUTICALS CO., LTD (CN) | 2016-05-26 | — | — | US | disclosed |
| EP-3019489-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | Betta Pharmaceuticals Co., Ltd. (CN) | 2016-05-18 | — | — | EP | disclosed |
| CN-105504858-A | Single azo based pyridine ketone dye and preparation method and application thereof | HANGZHOU FULAI'ENTE FINECHEMICAL CO LTD | 2016-04-20 | — | — | CN | disclosed |
| US-9287568-B2 | High performance, high durability non-precious metal fuel cell catalysts | 3M INNOVATIVE PROPERTIES COMPANY (US) | 2016-03-15 | — | — | US | disclosed |
| US-20160052898-A1 | NOVEL COMPOUNDS | BAYER PHARMA AKTIENGESELLSCHAFT (DE) | 2016-02-25 | — | — | US | disclosed |
| EP-2976343-A2 | SUBSTITUTED N-BIPHENYL-3-ACETYLAMINO-BENZAMIDES AND N-[3-(ACETYLAMINO)PHENYL]-BIPHENYL-CARBOXAMIDES AND THEIR USE AS INHIBITORS OF THE WNT SIGNALLING PATHWAY | Bayer Pharma Aktiengesellschaft (DE) | 2016-01-27 | — | — | EP | disclosed |
| EP-2976327-A2 | 3-ACETYLAMINO-1-(PHENYL-HETEROARYL-AMINOCARBONYL OR PHENYL-HETEROARYL-CARBONYLAMINO)BENZENE DERIVATIVES FOR THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS | Bayer Pharma Aktiengesellschaft (DE) | 2016-01-27 | — | — | EP | disclosed |
| CN-103288701-B | 1,5-diaryl pyrrole derivant, preparation method and antitumor application thereof | CENTRAL SOUTH UNIVERSITY (CN) | 2016-01-27 | — | — | CN | disclosed |
| EP-2704572-B1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD PHARMA INC (US) | 2015-12-30 | — | — | EP | disclosed |
| EP-2704572-B1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD PHARMA INC (US) | 2015-12-30 | — | — | EP | disclosed |
| EP-2940000-A1 | PROCESS FOR PREPARING METHYL ACETATE | Dalian Institute Of Chemical Physics, Chinese Academy of Sciences (CN) | 2015-11-04 | — | — | EP | disclosed |
| CN-105017146-A | Synthetic method for 3,4-dihydro-7-hydroxy-2(1H)-quinolinone | ANHUI WANBANG MEDICAL TECHNOLOGY CO LTD | 2015-11-04 | — | — | CN | disclosed |
| US-20150298108-A1 | METHOD FOR PREPARING METHYL ACETATE | DALIAN INSTITUTE OF CHEMICAL PHYSICS, CHINESE ACADEMY OF SCIENCES (CN) | 2015-10-22 | — | — | US | disclosed |
| US-20150284408-A1 | INHIBITORS OF DNA GYRASE FOR THE TREATMENT OF BACTERIAL INFECTIONS | KUMAR, AJAY, DR. (GB) | 2015-10-08 | — | — | US | disclosed |
| EP-2744797-B1 | DYRK1 INHIBITORS AND USES THEREOF | DIAXONHIT (FR) | 2015-09-09 | — | — | EP | disclosed |
| CN-103554992-B | A kind of disperse dye composition for washing spandex fibre dyeing and stamp | ZHEJIANG RUNTU CO., LTD. (CN) | 2015-08-12 | — | — | CN | disclosed |
| CN-103709788-B | Dye composition, dye, preparation methods thereof and raw material composition of dye | SHANGHAI ANOKY TEXTILE CHEMICALS CO LTD | 2015-06-24 | — | — | CN | disclosed |
| US-20150166591-A1 | METHODS AND COMPOSITIONS FOR RAF KINASE MEDIATED DISEASES | ARIAD PHARMACEUTICALS, INC. | 2015-06-18 | — | — | US | disclosed |
| US-20150166591-A1 | METHODS AND COMPOSITIONS FOR RAF KINASE MEDIATED DISEASES | ARIAD PHARMACEUTICALS, INC. | 2015-06-18 | — | — | US | disclosed |
| US-20150166591-A1 | METHODS AND COMPOSITIONS FOR RAF KINASE MEDIATED DISEASES | ARIAD PHARMACEUTICALS, INC. | 2015-06-18 | — | — | US | disclosed |
| CN-104650621-A | Disperse dye composition and disperse dye as well as preparation method and application of disperse dye | ZHEJIANG RUNTU CO LTD | 2015-05-27 | — | — | CN | disclosed |
| CN-104559319-A | Disperse dye composition, disperse dye, and preparation method and application thereof | ZHEJIANG RUNTU CO LTD | 2015-04-29 | — | — | CN | disclosed |
| CN-104530752-A | Disperse dye composition, disperse dye and preparation method and use of disperse dye | ZHEJIANG RUNTU CO LTD | 2015-04-22 | — | — | CN | disclosed |
| CN-102365263-B | Polymerizable composition | BASF SE | 2015-04-01 | — | — | CN | disclosed |
| CN-104479394-A | Method for continuously preparing azo pigment in branch spiral tube | SUZHOU SUNMUN TECHNOLOGY CO LTD | 2015-04-01 | — | — | CN | disclosed |
| EP-2844642-A1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD PHARMACEUTICALS, INC. (US) | 2015-03-11 | — | — | EP | disclosed |
| CN-103449654-B | Treatment method of Omeprazole intermediate production wastewater | UNIV NANJING SCIENCE & TECH | 2015-03-11 | — | — | CN | disclosed |
| WO-2015003658-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | BETTA PHARMACEUTICALS CO., LTD (CN) | 2015-01-15 | — | — | WO | disclosed |
| WO-2015003658-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | BETTA PHARMACEUTICALS CO., LTD (CN) | 2015-01-15 | — | — | WO | disclosed |
| CN-102993068-B | Electronic transmission layer polymer for solar cell | LIYANG PRODUCTIVITY PROMOTION CT | 2015-01-07 | — | — | CN | disclosed |
| US-20140378446-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | PHARMACYCLICS, INC. (US) | 2014-12-25 | — | — | US | disclosed |
| US-20140378446-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | PHARMACYCLICS, INC. (US) | 2014-12-25 | — | — | US | disclosed |
| US-20140378446-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | PHARMACYCLICS, INC. (US) | 2014-12-25 | — | — | US | disclosed |
| CN-103554991-B | Disperse dye composition for polyester/spandex fiber dyeing and printing | ZHEJIANG RUNTU CO LTD | 2014-12-17 | — | — | CN | disclosed |
| EP-2809672-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | Pharmacyclics, Inc. (US) | 2014-12-10 | — | — | EP | disclosed |
| CN-102976986-B | Method for manufacturing polymer used as electron transfer layer of solar cell | LIYANG CITY PRODUCTIVITY PROMOTION CT | 2014-12-10 | — | — | CN | disclosed |
| CN-104151178-A | 2-amino-4-(beta-hydroxyethylamino) methoxybenzene and preparation method of 2-amino-4-(beta-hydroxyethylamino) methoxybenzene sulfate | ZHEJIANG DRAGON CHEMICAL CO LTD | 2014-11-19 | — | — | CN | disclosed |
| CN-104151178-A | 2-amino-4-(beta-hydroxyethylamino) methoxybenzene and preparation method of 2-amino-4-(beta-hydroxyethylamino) methoxybenzene sulfate | ZHEJIANG DRAGON CHEMICAL CO LTD | 2014-11-19 | — | — | CN | disclosed |
| CN-102391680-B | Disperse dye composition for dyeing and printing polyester spandex fibers | ZHEJIANG RUNTU CO LTD | 2014-11-05 | — | — | CN | disclosed |
| WO-2014147021-A2 | NOVEL COMPOUNDS | BAYER PHARMA AKTIENGESELLSCHAFT (DE) | 2014-09-25 | — | — | WO | disclosed |
| WO-2014147182-A2 | NOVEL COMPOUNDS | BAYER PHARMA AKTIENGESELLSCHAFT (DE) | 2014-09-25 | — | — | WO | disclosed |
| US-20140275064-A1 | DYRK1 INHIBITORS AND USES THEREOF | DIAXONHIT (FR) | 2014-09-18 | — | — | US | disclosed |
| CN-104003918-A | Diaryl thioether compound, preparation method and antitumor application thereof | UNIV CENTRAL SOUTH | 2014-08-27 | — | — | CN | disclosed |
| CN-102391164-B | Diaryl thioether compound, preparation method and anti-tumor application thereof | UNIV CENTRAL SOUTH | 2014-08-13 | — | — | CN | disclosed |
| EP-2435436-B1 | PYRIMIDINE INHIBITORS OF KINASE ACTIVITY | ABBVIE INC (US) | 2014-07-30 | — | — | EP | disclosed |
| CN-102702173-B | Method for preparing sulfur ether intermediates of proton pump inhibitor | TENGZHOU WUTONG PERFUME CO LTD | 2014-07-16 | — | — | CN | disclosed |
| CN-103173037-B | Dye composition, dye, preparation method thereof and raw material composition of dye | YANTAI ANOKY TEXTILE MATERIAL CO LTD | 2014-07-02 | — | — | CN | disclosed |
| EP-2744797-A1 | DYRK1 INHIBITORS AND USES THEREOF | Diaxonhit (FR) | 2014-06-25 | — | — | EP | disclosed |
| CN-103709788-A | Dye composition, dye, preparation methods thereof and raw material composition of dye | SHANGHAI ANOKY TEXTILE CHEMICALS CO LTD | 2014-04-09 | — | — | CN | disclosed |
| CN-103694733-A | Dye composition, dye, preparation method of dye composition and dye and raw material composition of dye | SHANGHAI ANOKY TEXTILE CHEMICALS CO LTD | 2014-04-02 | — | — | CN | disclosed |
| EP-2704572-A1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD Pharmaceuticals, Inc. (US) | 2014-03-12 | — | — | EP | disclosed |
| US-20140057911-A1 | NOVEL 4,6-DISUBSTITUTED AMINOPYRIMIDINE DERIVATIVES HAVING BOTH AROMATIC AND HALOGENIC SUBSTITUENTS | VIROSTATICS SRL (IT) | 2014-02-27 | — | — | US | disclosed |
| CN-103554991-A | Disperse dye composition for polyester/spandex fiber dyeing and printing | ZHEJIANG RUNTU CO LTD | 2014-02-05 | — | — | CN | disclosed |
| CN-103554992-A | Disperse dye composition for polyester/spandex fiber dyeing and printing | ZHEJIANG RUNTU CO LTD | 2014-02-05 | — | — | CN | disclosed |
| EP-2435435-B1 | PYRIMIDINE INHIBITORS OF KINASE ACTIVITY | ABBVIE INC (US) | 2014-01-29 | — | — | EP | disclosed |
| CN-103450699-A | Grinding coupling method for preparing disperse dye | HANGZHOU FULAIENTE FINE CHEMICAL CO LTD | 2013-12-18 | — | — | CN | disclosed |
| CN-103449654-A | Treatment method of Omeprazole intermediate production wastewater | UNIV NANJING SCIENCE & TECH | 2013-12-18 | — | — | CN | disclosed |
| WO-2013169401-A1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD PHARMACEUTICALS, INC. (US) | 2013-11-14 | — | — | WO | disclosed |
| WO-2013169401-A1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD PHARMACEUTICALS, INC. (US) | 2013-11-14 | — | — | WO | disclosed |
| EP-1539675-B1 | ARYL AND HETEROARYL PROPENE AMIDES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF | UNIV TEMPLE (US) | 2013-11-06 | — | — | EP | disclosed |
| EP-1539675-B1 | ARYL AND HETEROARYL PROPENE AMIDES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF | UNIV TEMPLE (US) | 2013-11-06 | — | — | EP | disclosed |
| US-8536180-B2 | Pyrimidine inhibitors of kinase activity | ABBVIE INC. (US) | 2013-09-17 | — | — | US | disclosed |
| CN-103288701-A | 1,5-diaryl pyrrole derivative as well as preparation method and anti-tumor application thereof | JIANGXI DONGBANG PHARMACEUTICAL CO LTD | 2013-09-11 | — | — | CN | disclosed |
| WO-2013116382-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | PHARMACYCLICS, INC. (US) | 2013-08-08 | — | — | WO | disclosed |
| WO-2013116382-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | PHARMACYCLICS, INC. (US) | 2013-08-08 | — | — | WO | disclosed |
| CN-103173037-A | Dye composition, dye, preparation method thereof and raw material composition of dye | YANTAI ANOKY TEXTILE MATERIAL CO LTD | 2013-06-26 | — | — | CN | disclosed |
| CN-102186931-B | Azo pigment, coloring composition, coloring method, and colored article | DAINICHISEIKA COLOR CHEM | 2013-06-12 | — | — | CN | disclosed |
| US-20130105400-A1 | COMPOSITE CONTAINING METAL COMPONENT SUPPORTED ON GRAPHENE, PREPARING METHOD OF THE SAME, AND USES OF THE SAME | Research & Business Foundation Sungkyunkwan University (KR) | 2013-05-02 | — | — | US | disclosed |
| CN-102993068-A | Electronic transmission layer polymer for solar cell | LIYANG PRODUCTIVITY PROMOTION CT | 2013-03-27 | — | — | CN | disclosed |
| CN-102976986-A | Method for manufacturing polymer used as electron transfer layer of solar cell | LIYANG CITY PRODUCTIVITY PROMOTION CT | 2013-03-20 | — | — | CN | disclosed |
| WO-2013026806-A1 | DYRK1 INHIBITORS AND USES THEREOF | EXONHIT SA (FR) | 2013-02-28 | — | — | WO | disclosed |
| US-8354422-B2 | Pyrimidine inhibitors of kinase activity | ABBOTT LABORATORIES INC. (US) | 2013-01-15 | — | — | US | disclosed |
| US-20120316135-A1 | Compounds for Inhibiting Cell Proliferation in EGFR-Driven Cancers | ARIAD PHARMACEUTICALS, INC. (US) | 2012-12-13 | — | — | US | disclosed |
| US-20120316135-A1 | Compounds for Inhibiting Cell Proliferation in EGFR-Driven Cancers | ARIAD PHARMACEUTICALS, INC. (US) | 2012-12-13 | — | — | US | disclosed |
| US-20120316135-A1 | Compounds for Inhibiting Cell Proliferation in EGFR-Driven Cancers | ARIAD PHARMACEUTICALS, INC. (US) | 2012-12-13 | — | — | US | disclosed |
| US-8324225-B2 | Pyrrolopyrimidine compounds and their uses | NOVARTIS AG (CH) | 2012-12-04 | — | — | US | disclosed |
| WO-2012151561-A1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD PHARMACEUTICALS, INC. (US) | 2012-11-08 | — | — | WO | disclosed |
| WO-2012151561-A1 | COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS | ARIAD PHARMACEUTICALS, INC. (US) | 2012-11-08 | — | — | WO | disclosed |
| CN-102702173-A | Method for preparing sulfur ether intermediates of proton pump inhibitor | TENGZHOU WUTONG PERFUME CO LTD | 2012-10-03 | — | — | CN | disclosed |
| US-20120207763-A1 | PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES | ASTEX THERAPEUTICS LIMITED (GB) | 2012-08-16 | — | — | US | disclosed |
| CN-102617536-A | Isoflavone compound, its preparation method, and its application in preparation of antiviral or antitumor drugs | SHANGHAI RUIGUANG BIOCHEMICAL SCI TECH DEV CO LTD | 2012-08-01 | — | — | CN | disclosed |
| CN-102391680-A | Disperse dye composition for dyeing and printing polyester spandex fibers | ZHEJIANG RUNTU CO LTD | 2012-03-28 | — | — | CN | disclosed |
| CN-102391164-A | Diaryl thioether compound, preparation method and anti-tumor application thereof | UNIV CENTRAL SOUTH | 2012-03-28 | — | — | CN | disclosed |
| CN-102365263-A | polymerizable composition | BASF SE | 2012-02-29 | — | — | CN | disclosed |
| US-20110319257-A1 | HIGH PERFORMANCE, HIGH DURABILITY NON-PRECIOUS METAL FUEL CELL CATALYSTS | 3M INNOVATIVE PROPERTIES COMPANY | 2011-12-29 | — | — | US | disclosed |
| EP-2135313-B1 | HIGH PERFORMANCE, HIGH DURABILITY NON-PRECIOUS METAL FUEL CELL CATALYSTS | 3M INNOVATIVE PROPERTIES CO (US) | 2011-09-14 | — | — | EP | disclosed |
| CN-102186931-A | Azo pigment, coloring composition, coloring method, and colored article | DAINICHISEIKA COLOR CHEM | 2011-09-14 | — | — | CN | disclosed |
| EP-1534284-B1 | AMINO-SUBSTITUTED SULFONANILIDES AND DERIVATIVES THEREOF FOR TREATING PROLIFERATIVE DISORDERS | UNIV TEMPLE (US) | 2011-07-27 | — | — | EP | disclosed |
| EP-2327677-A1 | Mono-nitration of aromatic compounds | F. Hoffmann-La Roche AG (CH) | 2011-06-01 | — | — | EP | disclosed |
| WO-2010138576-A1 | PYRIMIDINE INHIBITORS OF KINASE ACTIVITY | ABBOTT LABORATORIES (US) | 2010-12-02 | — | — | WO | disclosed |
| WO-2010138575-A1 | PYRIMIDINE INHIBITORS OF KINASE ACTIVITY | ABBOTT LABORATORIES (US) | 2010-12-02 | — | — | WO | disclosed |
| US-20100305118-A1 | PYRIMIDINE INHIBITORS OF KINASE ACTIVITY | ABBOTT LABORATORIES (US) | 2010-12-02 | — | — | US | disclosed |
| US-20100305126-A1 | Pyrimidine Inhibitors of Kinase Activity | ABBOTT LABORATORIES (US) | 2010-12-02 | — | — | US | disclosed |
| EP-1481679-B1 | ANTIDEPRESSANT | TAKEDA PHARMACEUTICAL (JP) | 2010-08-25 | — | — | EP | disclosed |
| CN-101070290-B | Nitro-catalytic hydrogenation method in N-(3-nitro-4-methoxyphenyl) amide | UNIV DALIAN TECH | 2010-07-07 | — | — | CN | disclosed |
| CN-101302195-B | Novel synthetic method of 7-hydroxy-3,4-dihydroquinolines | HANGZHOU GREAT FOREST BIOMEDICAL LTD | 2010-06-09 | — | — | CN | disclosed |
| CN-1926199-B | Use of pigment compositions comprising mixed crystals based on C.I. Pigment Yellow 74 | CLARIANT GMBH | 2010-04-07 | — | — | CN | disclosed |
| US-20090318441-A1 | Pyrrolopyrimidine Compounds and Their Uses | ASTEX THERAPEUTICS LTD. | 2009-12-24 | — | — | US | disclosed |
| EP-2135313-A1 | HIGH PERFORMANCE, HIGH DURABILITY NON-PRECIOUS METAL FUEL CELL CATALYSTS | 3M Innovative Properties Company (US) | 2009-12-23 | — | — | EP | disclosed |
| CN-101589019-A | Process for preparing 4-hydroxyalkylamino-2-nitrobenzyl ethers | PROCTER & GAMBLE (US) | 2009-11-25 | — | — | CN | disclosed |
| US-7482488-B2 | Aryl and heteroaryl propene amides, derivatives thereof and therapeutic uses thereof | TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) | 2009-01-27 | — | — | US | disclosed |
| US-7482488-B2 | Aryl and heteroaryl propene amides, derivatives thereof and therapeutic uses thereof | TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) | 2009-01-27 | — | — | US | disclosed |
| US-7482488-B2 | Aryl and heteroaryl propene amides, derivatives thereof and therapeutic uses thereof | TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) | 2009-01-27 | — | — | US | disclosed |
| EP-1852414-B1 | Process for the preparation of 4-Hydroxyalkylamino-2-nitro-anisoles | WELLA AG (DE) | 2008-11-26 | — | — | EP | disclosed |
| CN-101302195-A | Novel synthetic method of 7-hydroxy-3,4-dihydroquinolines | HANGZHOU GREAT FOREST BIOMEDIC (CN) | 2008-11-12 | — | — | CN | disclosed |
| WO-2008127828-A1 | HIGH PERFORMANCE, HIGH DURABILITY NON-PRECIOUS METAL FUEL CELL CATALYSTS | 3M INNOVATIVE PROPERTIES COMPANY (US) | 2008-10-23 | — | — | WO | disclosed |
| US-7429589-B2 | Mono-nitration of aromatic compounds via nitrate salts | HOFFMANN-LA ROCHE INC. (US) | 2008-09-30 | — | — | US | disclosed |
| US-7429589-B2 | Mono-nitration of aromatic compounds via nitrate salts | HOFFMANN-LA ROCHE INC. (US) | 2008-09-30 | — | — | US | disclosed |
| US-7405325-B2 | Process for the preparation of 4-hydroxalkylamino-2-nitro-anisoles | THE PROCTER & GAMBLE COMPANY (US) | 2008-07-29 | — | — | US | disclosed |
| EP-1354928-B1 | Liquid compositions for the treatment of metal surfaces | SOLVAY SOLEXIS SPA (IT) | 2008-07-23 | — | — | EP | disclosed |
| CN-101070290-A | Nitro-catalytic hydrogenation method in N-(3-nitro-4-methoxyphenyl) amide | UNIV DALIAN TECH (CN) | 2007-11-14 | — | — | CN | disclosed |
| WO-2007125034-A2 | MONO-NITRATION OF AROMATIC COMPOUNDS | F. HOFFMANN-LA ROCHE AG (CH) | 2007-11-08 | — | — | WO | disclosed |
| EP-1852414-A1 | Process for the preparation of 4-Hydroxyalkylamino-2-nitro-anisoles | Wella Aktiengesellschaft (DE) | 2007-11-07 | — | — | EP | disclosed |
| EP-1852414-A1 | Process for the preparation of 4-Hydroxyalkylamino-2-nitro-anisoles | Wella Aktiengesellschaft (DE) | 2007-11-07 | — | — | EP | disclosed |
| WO-2007122579-A2 | PROCESS FOR THE PREPARATION OF 4-HYDROXYALKYLAMINO-2-NITRO-ANISOLES | THE PROCTER & GAMBLE COMPANY (US) | 2007-11-01 | — | — | WO | disclosed |
| WO-2007122579-A2 | PROCESS FOR THE PREPARATION OF 4-HYDROXYALKYLAMINO-2-NITRO-ANISOLES | THE PROCTER & GAMBLE COMPANY (US) | 2007-11-01 | — | — | WO | disclosed |
| US-20070255057-A1 | Mono-nitration of aromatic compounds via nitrate salts | CEDILOTE MIALL | 2007-11-01 | — | — | US | disclosed |
| US-20070255057-A1 | Mono-nitration of aromatic compounds via nitrate salts | CEDILOTE MIALL | 2007-11-01 | — | — | US | disclosed |
| US-20070249868-A1 | New process for the preparation of 4-hydroxalkylamino-2-nitro-anisoles | WELLA OPERATIONS US, LLC | 2007-10-25 | — | — | US | disclosed |
| CN-100339442-C | Method for preparing organic pigment of red benzimidazolones | UNIV HUADONG TECHNOLOGY (CN) | 2007-09-26 | — | — | CN | disclosed |
| EP-1268431-B1 | 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS | WYETH CORP (US) | 2007-08-29 | — | — | EP | disclosed |
| CN-1330645-C | Benzofuran-2-ones as colorants for organic materials | CIBA SC HOLDING AG (CH) | 2007-08-08 | — | — | CN | disclosed |
| EP-1539675-A4 | ARYL AND HETEROARYL PROPENE AMIDES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF | UNIV TEMPLE (US) | 2007-07-11 | — | — | EP | disclosed |
| CN-1926199-A | Use of pigment compositions comprising mixed crystals based on C.I. Pigment Yellow 74 | CLARIANT GMBH (DE) | 2007-03-07 | — | — | CN | disclosed |
| US-7161031-B2 | Amino-substituted sulfonanilides and derivatives thereof for treating proliferative disorders | TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) | 2007-01-09 | — | — | US | disclosed |
| US-7138418-B2 | For therapy of atherosclerosis and hypercholesterolemia; 5-Pentafluorophenylsulfonamidoindazole for example; increasing LDL receptor gene expression in a cell | AMGEN, INC. (US) | 2006-11-21 | — | — | US | disclosed |
| EP-1534284-A4 | AMINO-SUBSTITUTED SULFONANILIDES AND DERIVATIVES THEREOF FOR TREATING PROLIFERATIVE DISORDERS | UNIV TEMPLE (US) | 2006-08-16 | — | — | EP | disclosed |
| CN-1268689-C | Yellow, orange benzimidazolone like azo dye making method | UNIV EAST CHINA SCIENCE & TECH (CN) | 2006-08-09 | — | — | CN | disclosed |
| US-20060167317-A1 | Aryl and heteroaryl propene amides, derivatives thereof and therapeutic uses thereof | TEMPLE UNIVERSITY- OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) | 2006-07-27 | — | — | US | disclosed |
| US-7060718-B2 | Arylsulfonanilide ureas | AMGEN INC. (US) | 2006-06-13 | — | — | US | disclosed |
| US-6962929-B2 | Pentafluorobenzenesulfonamides and analogs | TULARIK INC. (US) | 2005-11-08 | — | — | US | disclosed |
| EP-1539675-A2 | ARYL AND HETEROARYL PROPENE AMIDES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF | Temple University of the Commonwealth System of Higher Education (US) | 2005-06-15 | — | — | EP | disclosed |
| EP-1534284-A2 | AMINO-SUBSTITUTED SULFONANILIDES AND DERIVATIVES THEREOF FOR TREATING PROLIFERATIVE DISORDERS | Temple University of the Commonwealth System of Higher Education (US) | 2005-06-01 | — | — | EP | disclosed |
| US-20050096484-A1 | Amino-substituted sulfonanilides and derivatives thereof for treating proliferative disorders | ONCONOVA THERAPEUTICS, INC. | 2005-05-05 | — | — | US | disclosed |
| CN-1569968-A | Yellow, orange benzimidazolone like azo dye making method | UNIV EAST CHINA SCIENCE & TECH (CN) | 2005-01-26 | — | — | CN | disclosed |
| CN-1563202-A | Method for preparing organic pigment of red benzimidazolones | UNIV HUADONG TECHNOLOGY (CN) | 2005-01-12 | — | — | CN | disclosed |
| WO-2004092142-A1 | AN IMPROVED PROCESS FOR MANUFACTURE OF SUBSTITUTED BENZIMIDAZOLES | IPCA LABORATORIES LIMITED (IN) | 2004-10-28 | — | — | WO | disclosed |
| EP-1456188-A1 | 7-AMINO-BENZOTHIAZOLE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS | F. HOFFMANN-LA ROCHE AG (CH) | 2004-09-15 | — | — | EP | disclosed |
| US-20040176602-A1 | 3-Cyanoquinolines,3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors | WYETH | 2004-09-09 | — | — | US | disclosed |
| WO-2004037751-A2 | ARYL AND HETEROARYL PROPENE AMIDES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF | TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) | 2004-05-06 | — | — | WO | disclosed |
| US-6713499-B2 | ADENOSINE RECEPTOR AGONIST | HOFFMAN-LA ROCHE INC. | 2004-03-30 | — | — | US | disclosed |
| US-6689772-B1 | ANTINEOPLASTIC AGENTS; OSTEOPOROSIS; POLYCYSTIC KIDNEY DISEASE; ANTIVIRAL AGENTS | WYETH | 2004-02-10 | — | — | US | disclosed |
| US-6664297-B1 | Impeding formation of amyloid fibers or dissolving existing fibers in mammals | UNIVERSIDADE FEDERAL DO RIO DE JANEIRO (BR) | 2003-12-16 | — | — | US | disclosed |
| CN-1130351-C | 1,5-benzodiazepine derivatives | ZERIA PHARM CO LTD (JP) | 2003-12-10 | — | — | CN | disclosed |
| US-20030207864-A1 | Arylsulfonanilide ureas | TULARK INC. | 2003-11-06 | — | — | US | disclosed |
| US-6630513-B1 | Capable of lowering plasma cholesterol levels and inhibiting abnormal cell proliferation, such as in cervical adenocarcinoma | TULARIX INC. | 2003-10-07 | — | — | US | disclosed |
| EP-0939627-B1 | PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS | TULARIK INC (US) | 2003-09-10 | — | — | EP | disclosed |
| EP-0896533-B1 | PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS | TULARIK INC (US) | 2003-09-10 | — | — | EP | disclosed |
| WO-2003072063-A2 | AMINO-SUBSTITUTED SULFONANILIDES AND DERIVATIVES THEREOF FOR TREATING PROLIFERATIVE DISORDERS | TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) | 2003-09-04 | — | — | WO | disclosed |
| US-20030162817-A1 | Pentafluorobenzenesulfonamides and analogs | TULARIK INC. | 2003-08-28 | — | — | US | disclosed |
| EP-1054042-B1 | Process for the preparation of pigment compositions | CIBA SC HOLDING AG (CH) | 2003-08-27 | — | — | EP | disclosed |
| US-20030153566-A1 | 7-Amino-benzothiazole derivatives | F. HOFFMANN-LA ROCHE AG (CH) | 2003-08-14 | — | — | US | disclosed |
| EP-1334719-A2 | Pentafluorobenzenesulfonamides and analogs | TULARIK, INC. (US) | 2003-08-13 | — | — | EP | disclosed |
| CN-1116366-C | Pyridone-methide azo dyestuffs | BAYER AG (DE) | 2003-07-30 | — | — | CN | disclosed |
| EP-1013636-B1 | Preparation of allylic aromatic compounds | AMERSHAM HEALTH AS (NO) | 2003-07-09 | — | — | EP | disclosed |
| WO-2003053946-A1 | 7-AMINO-BENZOTHIAZOLE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS | F. HOFFMANN-LA ROCHE AG (CH) | 2003-07-03 | — | — | WO | disclosed |
| US-6583165-B2 | Anticarcinogenic, -inflammatory and -proliferative agents; viricides; bactericides; vascular restenosis, autoimmune diseases; psoriasis; anticolesterol and -lipemic agents | TULARIK INC. | 2003-06-24 | — | — | US | disclosed |
| EP-1115701-B1 | ARYLSULFONANILIDE UREAS | TULARIK INC (US) | 2003-05-21 | — | — | EP | disclosed |
| EP-1285911-A2 | Arylsulfonanilide ureas | Tularik Inc. (US) | 2003-02-26 | — | — | EP | disclosed |
| US-6521618-B2 | Antineoplastic agents, agents for treatment of osteoporosis and polycystic kidney disease | WYETH | 2003-02-18 | — | — | US | disclosed |
| EP-1268431-A1 | 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS | Wyeth (US) | 2003-01-02 | — | — | EP | disclosed |
| US-6482860-B1 | such as batabulin (2-Fluoro-1-methoxy-4-pentafluorophenylsulfonamidobenzene), use as antiproliferative agents to treat cancer | TULARIK INC. | 2002-11-19 | — | — | US | disclosed |
| CN-1377342-A | Process for preparation of tricyclic amino alcohol derivatives | ASAHI CHEMICAL IND (JP) | 2002-10-30 | — | — | CN | disclosed |
| US-20020143036-A1 | Pentafluorobenzenesulfonamides and analogs | TULARIK INC. | 2002-10-03 | — | — | US | disclosed |
| CN-1360574-A | Process for preparing tricyclic amino alcohol derivatives | ASAHI CHEMICAL IND (JP) | 2002-07-24 | — | — | CN | disclosed |
| US-6402828-B1 | MIXTURES | CIBA SPECIALTY CHEMICALS CORPORATION | 2002-06-11 | — | — | US | disclosed |
| CN-1349501-A | Novel method for mfg. tricyclic amino alcohol derivatives | ASAHI CHEMICAL IND (JP) | 2002-05-15 | — | — | CN | disclosed |
| CN-1343207-A | Benzofuran-2-ones as colorants for organic materials | CIBA SC HOLDING AG (CH) | 2002-04-03 | — | — | CN | disclosed |
| US-6361595-B1 | MIXING WATER-MISCIBLE QUATERNARY AMMONIUM COMPOUND, WATER-IMMISCIBLE ORGANIC SOLVENT AND PIGMENT; STABILIZED WITH RESPECT TO MICROBIAL CONTAMINATION AND LOSS OF COLOUR STRENGTH | CIBA SPECIALTY CHEMICALS CORPORATION | 2002-03-26 | — | — | US | disclosed |
| US-20020026052-A1 | 3-cyanoquinolines, 3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors | AMERICAN HOME PRODUCTS CORPORATION (US) | 2002-02-28 | — | — | US | disclosed |
| CN-1076034-C | Mixtures of monoazopyridone dyes | CIBA SC HOLDING AG (CH) | 2001-12-12 | — | — | CN | disclosed |
| US-6316484-B1 | FOR THERAPY OR PROPHYLAXIS OF ATHEROSCLEROSIS AND HYPERCHOLESTEROLEMIA | TULARIK INC. | 2001-11-13 | — | — | US | disclosed |
| US-20010027211-A1 | Arylsulfonanilide ureas | TULARIK INC. | 2001-10-04 | — | — | US | disclosed |
| WO-2001072711-A1 | 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS | WYETH (US) | 2001-10-04 | — | — | WO | disclosed |
| US-6284894-B1 | AROMATIC AMINE IS REACTED FIRST WITH A NITRITE AND THEN WITH AN ALLYLIC OLEFIN HAVING AN ELIMINATABLE TERMINAL SUBSTITUENT. | NYCOMED IMAGING AS (NO) | 2001-09-04 | — | — | US | disclosed |
| EP-1115701-A1 | ARYLSULFONANILIDE UREAS | Tularik Inc. (US) | 2001-07-18 | — | — | EP | disclosed |
| CN-1304306-A | Method for inhibiting MRP1 | LILLY CO ELI (US) | 2001-07-18 | — | — | CN | disclosed |
| WO-2001028546-A1 | INHIBITION OF AMYLOIDOSES BY USING AROMATIC OR HETEROAROMATIC COMPOUNDS SUBSTITUTED BY ELECTRON-WITHDRAWING GROUPS | UNIVERSIDADE FEDERAL DO RIO DE JANEIRO (BR) | 2001-04-26 | — | — | WO | disclosed |
| WO-2001025476-A1 | SIMULTANEOUS ENZYMATIC DETECTION OF TWO ANALYTES | APPLIED IMAGING CORPORATION (US) | 2001-04-12 | — | — | WO | disclosed |
| US-6214880-B1 | LOWERING PLASMA CHOLESTEROL LEVELS AND INHIBITING ABNORMAL CELL PROLIFERATION WITH SAID COMPOUND; TREATMENT OF CANCER, PSORIASIS, VASCULAR RESTENOSIS, INFECTIONS, ATHEROSCLEROSIS AND HYPERCHOLESTEROLEMIA | TULARIK INC. | 2001-04-10 | — | — | US | disclosed |
| WO-2001012593-A1 | ARYLSULFONANILIDE DERIVATIVES | TULARIK INC. (US) | 2001-02-22 | — | — | WO | disclosed |
| US-6153585-A | FOR TREATING CANCER, PSORIASIS, VASCULAR RESTENOSIS, INFECTIONS, ATHEROSCLEROSIS AND HYPERCHOLESTEROLEMIA | TULARIK INC. (US) | 2000-11-28 | — | — | US | disclosed |
| EP-1054042-A1 | Process for the preparation of pigment compositions | Ciba SC Holding AG (CH) | 2000-11-22 | — | — | EP | disclosed |
| EP-0939627-A4 | PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS | TULARIK INC (US) | 2000-10-04 | — | — | EP | disclosed |
| EP-1038925-A2 | Azo lake pigment composition | Ciba SC Holding AG (CH) | 2000-09-27 | — | — | EP | disclosed |
| US-6121304-A | SUCH AS 1-(PENTAFLUOROPHENYLSULFONYL)INDOLE; USEFUL IN TREATING ATHEROSCLEROSIS AND HYPERCHOLESTEROLERNIA | TULARIK INC (US) | 2000-09-19 | — | — | US | disclosed |
| EP-1013636-A1 | Preparation of allylic aromatic compounds | NYCOMED IMAGING AS (NO) | 2000-06-28 | — | — | EP | disclosed |
| WO-2000017159-A1 | ARYLSULFONANILIDE UREAS | TULARIK INC. (US) | 2000-03-30 | — | — | WO | disclosed |
| CN-1246850-A | 1,5-benzodiazepine derivatives | ZERIA PHARM CO LTD (JP) | 2000-03-08 | — | — | CN | disclosed |
| EP-0939627-A1 | PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS | TULARIK, INC. (US) | 1999-09-08 | — | — | EP | disclosed |
| EP-0896533-A4 | PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS | TULARIK INC (US) | 1999-04-28 | — | — | EP | disclosed |
| US-5880151-A | TREATING OR PREVENTING DISEASE CHARACTERIZED BY HIGH LEVELS OF LOW DENSITY LIPOPROTEIN PARTICLES OR CHOLESTEROL IN BLOOD | TULARIK INC. (US) | 1999-03-09 | — | — | US | disclosed |
| EP-0896533-A2 | PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS | TULARIK, INC. (US) | 1999-02-17 | — | — | EP | disclosed |
| EP-0746592-A4 | ORGANIC AZO-PIGMENT COATED LITHOPONE | SINO AMERICAN PIGMENT SYS INC (US) | 1998-09-02 | — | — | EP | disclosed |
| EP-0641764-B1 | Process for the preparation of hydroxyalkylaminonitrobenzene derivatives | CLARIANT GMBH (DE) | 1998-05-20 | — | — | EP | disclosed |
| WO-1998005315-A1 | PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS | TULARIK, INC. (US) | 1998-02-12 | — | — | WO | disclosed |
| CN-1165162-A | Mixtures of monoazopyridone dyes | CIBA GEIGY AG (CH) | 1997-11-19 | — | — | CN | disclosed |
| US-RE35654-E | Mixed coupled azo pigments | ENGELHARD CORPORATION (US) | 1997-11-11 | — | — | US | disclosed |
| CN-1159463-A | Pyridone-methide azo dyestuffs | BAYER AG (DE) | 1997-09-17 | — | — | CN | disclosed |
| EP-0524941-B1 | MONOAZO PIGMENT COMPOSITIONS | SUN CHEMICAL CORP (US) | 1997-09-03 | — | — | EP | disclosed |
| WO-1997030677-A2 | PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS | TULARIK, INC. (US) | 1997-08-28 | — | — | WO | disclosed |
| EP-0746592-A1 | ORGANIC AZO-PIGMENT COATED LITHOPONE | SINO-AMERICAN PIGMENT SYSTEMS, INC. (US) | 1996-12-11 | — | — | EP | disclosed |
| US-5508467-A | REACTING AN AMINE SUBSTITUTED BENZONITRILE WITH AN ACYLCHLORIDE IN APROTIC SOLVENT; REARRANGEMENT IN PRESENCE OF ABASE | CASSELLA AKTIENGESELLSCHAFT (DE) | 1996-04-16 | — | — | US | disclosed |
| US-5472492-A | Organic azo-pigment coated lithopone | SINO-AMERICAN PIGMENT SYSTEMS, INC., INC. (US) | 1995-12-05 | — | — | US | disclosed |
| WO-1995023191-A1 | ORGANIC AZO-PIGMENT COATED LITHOPONE | SINO-AMERICAN PIGMENT SYSTEMS, INC. (US) | 1995-08-31 | — | — | WO | disclosed |
| EP-0641764-A2 | Process for the preparation of hydroxyalkylaminonitrobenzene derivatives | HOECHST AKTIENGESELLSCHAFT (DE) | 1995-03-08 | — | — | EP | disclosed |
| EP-0595857-A1 | MIXED COUPLED AZO PIGMENTS | ENGELHARD CORPORATION (US) | 1994-05-11 | — | — | EP | disclosed |
| EP-0267491-B1 | Silver halide light-sensitive photographic material containing a novel yellow coupler | KONISHIROKU PHOTO IND (JP) | 1994-03-09 | — | — | EP | disclosed |
| US-5246494-A | MIXED COUPLED AZO PIGMENTS | ENGELHARD CORPORATION (US) | 1993-09-21 | — | — | US | disclosed |
| US-5204453-A | Process for the preparation of 1:2 metal complex azo compounds by carrying out diazotization and coupling in the presence of a metal donor | CIBA-GEIGY CORPORATION (US) | 1993-04-20 | — | — | US | disclosed |
| WO-1993002145-A1 | MIXED COUPLED AZO PIGMENTS | ENGELHARD CORPORATION (US) | 1993-02-04 | — | — | WO | disclosed |
| EP-0280156-B1 | PROCESS FOR THE PREPARATION OF ACETOACETYLARYLAMIDES-HETEROARYLAMIDES RESPECTIVELY OF DEACTIVED AROMATIC COMPOUNDS | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-11-11 | — | — | EP | disclosed |
| US-5128455-A | WATER-SOLUBLE FIBER-REACTIVE DYES, CONTAINING AN AMINO-SUBSTITUTED 5-TRIAZINE RING WITH A FIBER-REACTIVE GROUP OF THE VINYLSULFONE SERIES | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-07-07 | — | — | US | disclosed |
| US-5104416-A | Textile printing pastes; simplified preparation | HOECHT AKTIENGESELLSCHAFT (DE) | 1992-04-14 | — | — | US | disclosed |
| EP-0278910-B1 | HEAVY METAL COMPLEX DYESTUFFS, THEIR PREPARATION AND THEIR USE | CIBA-GEIGY AG (CH) | 1992-01-22 | — | — | EP | disclosed |
| EP-0184993-B1 | PROCESS FOR THE MANUFACTURE OF AZO DYE PREPARATIONS | CIBA-GEIGY AG (CH) | 1991-10-16 | — | — | EP | disclosed |
| EP-0241414-B1 | PROCESS FOR THE PREPARATION OF 1:2 METAL COMPLEX AZO DYES | CIBA-GEIGY AG (CH) | 1991-05-08 | — | — | EP | disclosed |
| EP-0168343-B1 | METAL COMPLEXES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN DYEING HIGH-MOLECULAR ORGANIC MATERIALS | CIBA-GEIGY AG (CH) | 1991-05-02 | — | — | EP | disclosed |
| US-5003049-A | Fiber-Reactive Dyes for Hydroxy Textiles | BASF AKTIENGESELLSCHAFT (DE) | 1991-03-26 | — | — | US | disclosed |
| US-5001227-A | Fibre-reactive 1:1 chromium complex azo or azomethine dyes having a bidentate chelating group and a monofunctional neutral ligand | CIBA-GEIGY CORPORATION (US) | 1991-03-19 | — | — | US | disclosed |
| EP-0271883-B1 | COLOURED WATER SOLUBLE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THEIR USE AS DYESTUFFS | HOECHST AKTIENGESELLSCHAFT (DE) | 1991-03-06 | — | — | EP | disclosed |
| US-4992360-A | Silver halide light-sensitive photographic material containing a novel yellow coupler | KONICA CORPORATION (JP) | 1991-02-12 | — | — | US | disclosed |
| US-4990598-A | Colorfastness | CIBA-GEIGY CORPORATION, A CORP. OF NEW YORK | 1991-02-05 | — | — | US | disclosed |
| US-4980459-A | Process for the manufacture of formulations of water-insoluble azo dyes | CIBA-GEIGY CORPORATION (US) | 1990-12-25 | — | — | US | disclosed |
| US-4962191-A | 1:2 chromium or cobalt complex axo dyes containing at least one 2-aryl-4-amino-6-hydroxypyrimidine radical | CIBA-GEIGY CORPORATION (US) | 1990-10-09 | — | — | US | disclosed |
| US-4960870-A | DYEING WOOL, POLYAMIDES; FIBER REACTIVE DYES | CIBA-GEIGY CORPORATION (US) | 1990-10-02 | — | — | US | disclosed |
| EP-0374911-A1 | Water-soluble, fibre-reactive dyes, methods for their preparation and their use | HOECHST AKTIENGESELLSCHAFT (DE) | 1990-06-27 | — | — | EP | disclosed |
| EP-0169167-B1 | PROCESS FOR DYEING HIGH-MOLECULAR ORGANIC MATERIALS, AND METAL COMPLEXES | CIBA-GEIGY AG (CH) | 1990-05-02 | — | — | EP | disclosed |
| EP-0361440-A1 | Water soluble fibre-reactive dyes, process for their preparation and their use | HOECHST AKTIENGESELLSCHAFT (DE) | 1990-04-04 | — | — | EP | disclosed |
| EP-0220130-B1 | METHOD FOR THE DETERMINATION OF THE CONCENTRATION OF DIAZONIUM IONS | CIBA-GEIGY AG (CH) | 1990-03-28 | — | — | EP | disclosed |
| EP-0357554-A2 | Complex metal compounds | CIBA-GEIGY AG (CH) | 1990-03-07 | — | — | EP | disclosed |
| EP-0142104-B1 | FIBRE-REACTIVE CHROMIUM COMPLEXES, THEIR PREPARATION AND THEIR USE | CIBA-GEIGY AG (CH) | 1990-01-03 | — | — | EP | disclosed |
| US-4874391-A | USING WATER SOLUBLE COPPER COMPLEX AZO DYE, LIGHT STABILIZER AND ANTIOXIDANT | CIBA-GEIGY CORPORATION (US) | 1989-10-17 | — | — | US | disclosed |
| US-4874848-A | FOR DYEING WOOL, LEATHER, POLYAMIDES BLACK OR BROWN | CIBA-GEIGY CORPORATION (US) | 1989-10-17 | — | — | US | disclosed |
| US-4874849-A | FOR DYEING WOOL, POLYAMIDES, LEATHER ORANGE OR BROWN | CIBA-GEIGY CORPORATION (US) | 1989-10-17 | — | — | US | disclosed |
| EP-0144776-B1 | FIBRE-REACTIVE CHROMIUM COMPLEXES, THEIR PREPARATION AND THEIR USE | CIBA-GEIGY AG (CH) | 1989-10-11 | — | — | EP | disclosed |
| US-4873320-A | COLORFASTNESS; FOR COTTON AND CELLULOSE FIBER MATERIALS | HOECHST AKTIENGESELLSCHAFT (DE) | 1989-10-10 | — | — | US | disclosed |
| EP-0141416-B1 | FIBRE-REACTIVE CHROMIUM COMPLEXES, THEIR PREPARATION AND THEIR USE | CIBA-GEIGY AG (CH) | 1989-08-16 | — | — | EP | disclosed |
| US-4845638-A | Method of eliminating excess nitrite in diazotisation solutions | CIBA-GEIGY CORPORATION (US) | 1989-07-04 | — | — | US | disclosed |
| EP-0212264-B1 | COLOURED WATER SOLUBLE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THEIR USE AS DYESTUFFS | HOECHST AKTIENGESELLSCHAFT (DE) | 1989-05-31 | — | — | EP | disclosed |
| EP-0136619-B1 | PROCESS FOR THE MANUFACTURE OF PREPARATIONS OF AZO DYES | CIBA-GEIGY AG (CH) | 1989-04-12 | — | — | EP | disclosed |
| US-4813972-A | USING LEVELING DYES, COLORFASTNESS | CIBA-GEIGY CORPORATION (US) | 1989-03-21 | — | — | US | disclosed |
| EP-0159962-B1 | FIBRE-REACTIVE CHROMIUM OR COBALT COMPLEXES, THEIR PREPARATION AND THEIR USE | CIBA-GEIGY AG (CH) | 1989-02-08 | — | — | EP | disclosed |
| EP-0148120-B1 | ASYMMETRICAL 1:2 CHROMIUM COMPLEX DYES | CIBA-GEIGY AG (CH) | 1988-11-23 | — | — | EP | disclosed |
| EP-0148121-B1 | ASYMMETRICAL 1:2 CHROMIUM COMPLEX DYES | CIBA-GEIGY AG (CH) | 1988-11-09 | — | — | EP | disclosed |
| EP-0150676-B1 | 1:2 CHROMIUM COMPLEX DYES | CIBA-GEIGY AG (CH) | 1988-10-12 | — | — | EP | disclosed |
| US-4775747-A | PIGMENTS FOR POLYMERS | CIBA-GEIGY CORPORATION (US) | 1988-10-04 | — | — | US | disclosed |
| EP-0185611-B1 | PROCESS FOR THE PHOTOCHEMICAL STABILISATION OF SYNTHETIC FIBROUS MATERIALS CONTAINING POLYAMIDE FIBRES | CIBA-GEIGY AG (CH) | 1988-09-21 | — | — | EP | disclosed |
| EP-0280156-A2 | Process for the preparation of acetoacetylarylamides-heteroarylamides respectively of deactived aromatic compounds | HOECHST AKTIENGESELLSCHAFT (DE) | 1988-08-31 | — | — | EP | disclosed |
| EP-0278910-A2 | Heavy metal complex dyestuffs, their preparation and their use | CIBA-GEIGY AG (CH) | 1988-08-17 | — | — | EP | disclosed |
| EP-0271883-A2 | Coloured water soluble compounds, process for their preparation and their use as dyestuffs | HOECHST AKTIENGESELLSCHAFT (DE) | 1988-06-22 | — | — | EP | disclosed |
| EP-0267491-A2 | Silver halide light-sensitive photographic material containing a novel yellow coupler | KONICA CORPORATION (JP) | 1988-05-18 | — | — | EP | disclosed |
| US-4730037-A | Process for the application of IR spectroscopy for modulation and monitoring of diazonium ion concentration | CIBA-GEIGY CORPORATION (US) | 1988-03-08 | — | — | US | disclosed |
| EP-0255481-A1 | Process for the photochemical stabilisation of a fibrous polyamide material and its mixtures with other fibres | CIBA-GEIGY AG (CH) | 1988-02-03 | — | — | EP | disclosed |
| US-4723001-A | Fibre-reactive chromium complexes and their preparation and use | CIBA-GEIGY CORPORATION (US) | 1988-02-02 | — | — | US | disclosed |
| US-4719053-A | FOR DYES | HOECHST AKTIENGESELLSCHAFT (DE) | 1988-01-12 | — | — | US | disclosed |
| US-4704133-A | FIBER-REACTIVE | CIBA-GEIGY CORPORATION (US) | 1987-11-03 | — | — | US | disclosed |
| EP-0241414-A2 | Process for the preparation of 1:2 metal complex azo dyes | CIBA-GEIGY AG (CH) | 1987-10-14 | — | — | EP | disclosed |
| EP-0151369-B1 | ASYMMETRICAL 1:2 CHROME COMPLEXES CONTAINING AN AZO COMPOUND AND AN AZOMETHINE COMPOUND | CIBA-GEIGY AG (CH) | 1987-09-09 | — | — | EP | disclosed |
| US-4680385-A | Metal dye complexes containing an azo or azomethine dye and a colorless ligand with the C═N--N═C group | CIBA-GEIGY CORPORATION (US) | 1987-07-14 | — | — | US | disclosed |
| US-4678851-A | FIBER-RACTIVE | CIBA-GEIGY CORPORATION (US) | 1987-07-07 | — | — | US | disclosed |
| US-4677199-A | Reactive dyes containing substituted 4-fluoropyridaz-6-one radicals | BASF AKTIENGESELLSCHAFT (DE) | 1987-06-30 | — | — | US | disclosed |
| US-4670486-A | Polymer composition pigmented with copper or nickel complexes of ligands containing a semicarbazone moiety | CIBA-GEIGY CORPORATION (US) | 1987-06-02 | — | — | US | disclosed |
| US-4661587-A | Bis 1:2 chromium complexes of disazo and azo or azomethine dyes | CIBA-GEIGY CORPORATION (US) | 1987-04-28 | — | — | US | disclosed |
| EP-0110825-B1 | ASYMMETRICAL 1:2 CHROMIUM COMPLEX DYESTUFFS CONTAINING ONE AZO AND ONE AZOMETHINE COMPOUND | CIBA-GEIGY AG (CH) | 1987-04-08 | — | — | EP | disclosed |
| US-4652631-A | LEATHER, WOOL, POLYAMIDES | CIBA-GEIGY CORPORATION (US) | 1987-03-24 | — | — | US | disclosed |
| US-4650859-A | WOOL,POLYAMIDES, LEATHER | CIBA-GEIGY CORPORATION (US) | 1987-03-17 | — | — | US | disclosed |
| EP-0212264-A1 | Coloured water soluble compounds, process for their preparation and their use as dyestuffs | HOECHST AKTIENGESELLSCHAFT (DE) | 1987-03-04 | — | — | EP | disclosed |
| EP-0119441-B1 | REACTIVE DYES WITH SUBSTITUTED 4-FLUOROPYRIDAZ-6-ONE GROUPS | BASF Aktiengesellschaft (DE) | 1987-02-25 | — | — | EP | disclosed |
| US-4639477-A | AZO DYES | CIBA-GEIGY CORPORATION (US) | 1987-01-27 | — | — | US | disclosed |
| EP-0209492-A2 | Process to eliminate the nitrite excess in diazotization solutions | CIBA-GEIGY AG (CH) | 1987-01-21 | — | — | EP | disclosed |
| US-4625017-A | LEATHER, COLORFASTNESS | CIBA-GEIGY CORPORATION (US) | 1986-11-25 | — | — | US | disclosed |
| US-4617382-A | PRINTING; DYEING; SILK, LEATHER, WOOL AND POLYAMIDES | CIBA-GEIGY CORPORATION (US) | 1986-10-14 | — | — | US | disclosed |
| EP-0190586-A1 | Triazine dyes, their preparation and their use | BAYER AG (DE) | 1986-08-13 | — | — | EP | disclosed |
| EP-0099857-B1 | METAL COMPLEXES OF AZO DYESTUFFS | CIBA-GEIGY AG (CH) | 1986-08-06 | — | — | EP | disclosed |
| EP-0185611-A1 | Process for the photochemical stabilisation of synthetic fibrous materials containing polyamide fibres | CIBA-GEIGY AG (CH) | 1986-06-25 | — | — | EP | disclosed |
| EP-0184993-A2 | Process for the manufacture of azo dye preparations | CIBA-GEIGY AG (CH) | 1986-06-18 | — | — | EP | disclosed |
| US-4582896-A | 1:2-metal complex dyes containing one atom of chromium or cobalt and two azo dyes each formed by coupling two diazo compounds to resorcinol | CIBA-GEIGY CORPORATION (US) | 1986-04-15 | — | — | US | disclosed |
| EP-0055218-B1 | MANUFACTURE OF AZOIC COMPOUNDS | CIBA-GEIGY AG (CH) | 1986-03-26 | — | — | EP | disclosed |
| EP-0169167-A2 | Process for dyeing high-molecular organic materials, and metal complexes | CIBA-GEIGY AG (CH) | 1986-01-22 | — | — | EP | disclosed |
| EP-0168343-A2 | Metal complexes, process for their preparation and their use in dyeing high-molecular organic materials | CIBA-GEIGY AG (CH) | 1986-01-15 | — | — | EP | disclosed |
| EP-0100297-B1 | BIS-1:2-CHROMIUM COMPLEXES OF DISAZO DYESTUFFS, THEIR PREPARATION AND THEIR USE | CIBA-GEIGY AG (CH) | 1986-01-08 | — | — | EP | disclosed |
| US-4563193-A | WOOL, POLYAMIDES, LEATHER | CIBA GEIGY CORPORATION (US) | 1986-01-07 | — | — | US | disclosed |
| EP-0054513-B1 | PROCESS FOR THE PRODUCTION OF PHOTOGRAPHIC COLOUR IMAGES ACCORDING TO THE SILVER DYE BLEACHING PROCESS, AND PHOTOGRAPHIC MATERIAL USED IN THIS PROCESS | CIBA-GEIGY AG (CH) | 1985-10-30 | — | — | EP | disclosed |
| EP-0159962-A2 | Fibre-reactive chromium or cobalt complexes, their preparation and their use | CIBA-GEIGY AG (CH) | 1985-10-30 | — | — | EP | disclosed |
| US-4537955-A | Unsymmetrical 1:2 chromium complex of a monoazo dyestuff and a disazo dyestuff which is non-fiber reactive and contains no sulfonamido or amino groups | BASF AKTIENGESELLSCHAFT (DE) | 1985-08-27 | — | — | US | disclosed |
| EP-0151369-A2 | Asymmetrical 1:2 chrome complexes containing an azo compound and an azomethine compound | CIBA-GEIGY AG (CH) | 1985-08-14 | — | — | EP | disclosed |
| EP-0087715-B1 | COMPLEX METAL DYESTUFFS FREE FROM SULPHON AMIDE AND AMINO GROUPS | BASF Aktiengesellschaft (DE) | 1985-08-07 | — | — | EP | disclosed |
| EP-0150676-A2 | 1:2 Chromium complex dyes | CIBA-GEIGY AG (CH) | 1985-08-07 | — | — | EP | disclosed |
| EP-0148120-A2 | Asymmetrical 1:2 chromium complex dyes | CIBA-GEIGY AG (CH) | 1985-07-10 | — | — | EP | disclosed |
| EP-0148121-A2 | Asymmetrical 1:2 chromium complex dyes | CIBA-GEIGY AG (CH) | 1985-07-10 | — | — | EP | disclosed |
| EP-0147938-A2 | Disperse dyestuffs | IMPERIAL CHEMICAL INDUSTRIES PLC (GB) | 1985-07-10 | — | — | EP | disclosed |
| EP-0045488-B1 | WATER-SOLUBLE FIBRE-REACTIVE COMPOUNDS AND THEIR USE IN FINISHING TEXTILES, AS WELL AS THE BETA-CHLOROETHYL-SULFONYL-METHYL-BENZOIC-ACID HALOGENIDES, AND THEIR USE AS A FIBRE-REACTIVE ANCHOR | HOECHST AKTIENGESELLSCHAFT (DE) | 1985-06-19 | — | — | EP | disclosed |
| EP-0144776-A2 | Fibre-reactive chromium complexes, their preparation and their use | CIBA-GEIGY AG (CH) | 1985-06-19 | — | — | EP | disclosed |
| EP-0062824-B1 | CATIONIC AZO DYESTUFFS CONTAINING SULFONIC-ACID GROUPS, THEIR PREPARATION AND THEIR USE | BAYER AG (DE) | 1985-06-05 | — | — | EP | disclosed |
| EP-0142104-A2 | Fibre-reactive chromium complexes, their preparation and their use | CIBA-GEIGY AG (CH) | 1985-05-22 | — | — | EP | disclosed |
| EP-0141416-A2 | Fibre-reactive chromium complexes, their preparation and their use | CIBA-GEIGY AG (CH) | 1985-05-15 | — | — | EP | disclosed |
| US-4517357-A | COLORING PAPER | BAYER AKTIENGESELLSCHAFT (DE) | 1985-05-14 | — | — | US | disclosed |
| EP-0082117-B1 | CHROMIUM COMPLEXES OF POLYAZO DYESTUFFS | CIBA-GEIGY AG (CH) | 1985-04-10 | — | — | EP | disclosed |
| EP-0136619-A2 | Process for the manufacture of preparations of azo dyes | CIBA-GEIGY AG (CH) | 1985-04-10 | — | — | EP | disclosed |
| US-4502860-A | WOOL, POLYAMIDES, LEATHER | CIBA-GEIGY CORPORATION (US) | 1985-03-05 | — | — | US | disclosed |
| EP-0133270-A1 | Reactive dyes | BASF Aktiengesellschaft (DE) | 1985-02-20 | — | — | EP | disclosed |
| US-4496481-A | REACTING AMINE, COUPLING COMPONENT AND NITRITE;PIGMENTS AND DISPERSE DYES | CIBA-GEIGY CORPORATION (US) | 1985-01-29 | — | — | US | disclosed |
| EP-0074589-B1 | TRIAZINE DYES, THEIR PREPARATION AND THEIR USE | BAYER AG (DE) | 1984-12-05 | — | — | EP | disclosed |
| US-4486348-A | YELLOW COLOR ON PAPER | BAYER AKTIENGESELLSCHAFT (DE) | 1984-12-04 | — | — | US | disclosed |
| EP-0051559-B1 | BASIC AND/OR CATIONIC AZO COMPOUNDS FREE FROM SULFONIC-ACID GROUPS | SANDOZ AG (CH) | 1984-11-07 | — | — | EP | disclosed |
| EP-0123300-A2 | Complexing of biologically active or functional compounds and methods of preparing and utilizing same | ENZO BIOCHEM, INC. (US) | 1984-10-31 | — | — | EP | disclosed |
| EP-0119441-A2 | Reactive dyes with substituted 4-fluoropyridaz-6-one groups | BASF Aktiengesellschaft (DE) | 1984-09-26 | — | — | EP | disclosed |
| US-4473498-A | Water-soluble, fiber-reactive organic dyestuffs containing a β-chloro-ethylsulfonyl-methyl-benzoic acid amide group | HOECHST AKTIENGESELLSCHAFT (DE) | 1984-09-25 | — | — | US | disclosed |
| US-4465627-A | FOR CELLULOSE AND LEATHER | SANDOZ LTD. (CH) | 1984-08-14 | — | — | US | disclosed |
| US-4465763-A | OIL SOLUBLE TRIAZINE COMPOUND AND A PHENYL AMINE COUPLER | CIBA GEIGY AG (CH) | 1984-08-14 | — | — | US | disclosed |
| EP-0037377-B1 | METAL-COMPLEX DYESTUFFS, THEIR PREPARATION AND USE | CIBA-GEIGY AG (CH) | 1984-08-01 | — | — | EP | disclosed |
| EP-0110825-A1 | Asymmetrical 1:2 chromium complex dyestuffs containing one azo and one azomethine compound | CIBA-GEIGY AG (CH) | 1984-06-13 | — | — | EP | disclosed |
| EP-0057245-B1 | CATIONIC TRIAZINE DYESTUFFS, THEIR PREPARATION AND THEIR USE | BAYER AG (DE) | 1984-05-30 | — | — | EP | disclosed |
| EP-0057418-B1 | NITRO-ANILINE PREPARATIONS | HOECHST AKTIENGESELLSCHAFT (DE) | 1984-05-02 | — | — | EP | disclosed |
| EP-0100297-A1 | Bis-1:2-chromium complexes of disazo dyestuffs, their preparation and their use | CIBA-GEIGY AG (CH) | 1984-02-08 | — | — | EP | disclosed |
| EP-0054616-B1 | CATIONIC TRIAZINE DYESTUFFS, THEIR PREPARATION AND PROCESS OF DYING | BAYER AG (DE) | 1984-02-08 | — | — | EP | disclosed |
| EP-0099857-A2 | Metal complexes of azo dyestuffs | CIBA-GEIGY AG (CH) | 1984-02-01 | — | — | EP | disclosed |
| EP-0039312-B1 | COLOUR PHOTOPGRAPHIC MATERIAL FOR THE SILVER-DYE BLEACHING PROCESS, PROCESS FOR THE PRODUCTION OF THIS MATERIAL AND ITS USE IN THE PRODUCTION OF PHOTOGRAPHIC IMAGES | CIBA-GEIGY AG (CH) | 1983-12-28 | — | — | EP | disclosed |
| US-4404273-A | Process for the production of photographic color images by the silver dye bleach process | CIBA-GEIGY AG (CH) | 1983-09-13 | — | — | US | disclosed |
| EP-0087715-A1 | Complex metal dyestuffs free from sulphon amide and amino groups | BASF Aktiengesellschaft (DE) | 1983-09-07 | — | — | EP | disclosed |
| EP-0082117-A1 | Chromium complexes of polyazo dyestuffs | CIBA-GEIGY AG (CH) | 1983-06-22 | — | — | EP | disclosed |
| EP-0012969-B1 | WATER-SOLUBLE FIBRE-REACTIVE COMPOUNDS AND THEIR USE IN FIBRE FINISHING,ESPECIALLY AS DYESTUFFS,AND DIHALOGENO-PYRIDAZONYL-CARBOXYLIC AND SULFONIC ACID HALIDES AND THEIR USE AS FIBRE-REACTIVE ANCHORS,AS WELL AS PROCESS FOR THE PREPARATION OF THESE COMPOUND | HOECHST AKTIENGESELLSCHAFT (DE) | 1983-06-08 | — | — | EP | disclosed |
| EP-0079858-A1 | Azo dyestuffs, metal complexes thereof, their preparation and use | CIBA-GEIGY AG (CH) | 1983-05-25 | — | — | EP | disclosed |
| EP-0019851-B1 | 1:2 CHROMIUM COMPLEX DYESTUFFS OF THE AZOMETHINE AND/OR AZO SERIES, THEIR PREPARATION AND USE IN DYEING AND PRINTING POLYAMIDE OR CELLULOSE MATERIALS | CIBA-GEIGY AG (CH) | 1983-05-11 | — | — | EP | disclosed |
| US-4379819-A | OIL SOLUBLE MONOAZO DYE | CIBA-GEIGY AG (CH) | 1983-04-12 | — | — | US | disclosed |
| EP-0074589-A2 | Triazine dyes, their preparation and their use | BAYER AG (DE) | 1983-03-23 | — | — | EP | disclosed |
| US-4368054-A | Compositions of nitro-anilines for producing azo dyes on fibers | HOECHST AKTIENGESELLSCHAFT (DE) | 1983-01-11 | — | — | US | disclosed |
| US-4367172-A | DYEING PAPER, CELLULOSE, OR LEATHER | SANDOZ LTD. (CH) | 1983-01-04 | — | — | US | disclosed |
| US-4363761-A | DYEING CELLULOSE AND LEATHER; TEXTILES; PAPERMAKING | SANDOZ LTD. (CH) | 1982-12-14 | — | — | US | disclosed |
| EP-0062824-A2 | Cationic azo dyestuffs containing sulfonic-acid groups, their preparation and their use | BAYER AG (DE) | 1982-10-20 | — | — | EP | disclosed |
| EP-0057245-A2 | Cationic triazine dyestuffs, their preparation and their use | BAYER AG (DE) | 1982-08-11 | — | — | EP | disclosed |
| EP-0057418-A1 | Nitro-aniline preparations | HOECHST AKTIENGESELLSCHAFT (DE) | 1982-08-11 | — | — | EP | disclosed |
| US-4340536-A | Chrome-complex dyes and the production and use thereof | CIBA-GEIGY CORPORATION (US) | 1982-07-20 | — | — | US | disclosed |
| EP-0054616-A2 | Cationic triazine dyestuffs, their preparation and process of dying | BAYER AG (DE) | 1982-06-30 | — | — | EP | disclosed |
| EP-0055218-A2 | Manufacture of azoic compounds | CIBA-GEIGY AG (CH) | 1982-06-30 | — | — | EP | disclosed |
| EP-0054513-A1 | Process for the production of photographic colour images according to the silver dye bleaching process, and photographic material used in this process | CIBA-GEIGY AG (CH) | 1982-06-23 | — | — | EP | disclosed |
| US-4331596-A | Arylazoarylazo-substituted azo, azomethine 1:2 chromium complex dyes | CIBA-GEIGY CORPORATION (US) | 1982-05-25 | — | — | US | disclosed |
| EP-0051559-A1 | Basic and/or cationic azo compounds free from sulfonic-acid groups | SANDOZ AG (CH) | 1982-05-12 | — | — | EP | disclosed |
| EP-0045488-A2 | Water-soluble fibre-reactive compounds and their use in finishing textiles, as well as the beta-chloroethyl-sulfonyl-methyl-benzoic-acid halogenides, and their use as a fibre-reactive anchor | HOECHST AKTIENGESELLSCHAFT (DE) | 1982-02-10 | — | — | EP | disclosed |
| EP-0005207-B1 | BIS-1:2 CHROME-DISAZO-BISAZO METHINE DYESTUFFS, THEIR PREPARATION AND USE FOR DYEING OF LEATHER | CIBA-GEIGY AG (CH) | 1981-12-09 | — | — | EP | disclosed |
| EP-0039312-A1 | Colour photopgraphic material for the silver-dye bleaching process, process for the production of this material and its use in the production of photographic images | CIBA-GEIGY AG (CH) | 1981-11-04 | — | — | EP | disclosed |
| EP-0008472-B1 | LIGHT SENSITIVE BENZENEDIAZONIUM SALTS AND DIAZOTYPE MATERIAL USING SAME | Aerni-Leuch Ag (CH) | 1981-10-21 | — | — | EP | disclosed |
| EP-0037377-A1 | Metal-complex dyestuffs, their preparation and use | CIBA-GEIGY AG (CH) | 1981-10-07 | — | — | EP | disclosed |
| US-4293566-A | FUNGICIDES, BACTERICIDES, INSECTICIDES | BAYER AKTIENGESELLSCHAFT (DE) | 1981-10-06 | — | — | US | disclosed |
| US-4273707-A | Monoazo and disazo dyes containing at least one sulfo group and at least two basic or cationic groups | SANDOZ LTD. (CH) | 1981-06-16 | — | — | US | disclosed |
| US-4267249-A | Benzene diazonium salts and diazotype material utilizing same | AERNI-LEUCH AG (CH) | 1981-05-12 | — | — | US | disclosed |
| US-4256633-A | AZO DYES; AZOMETHINE DYES; WOOL, POLYAMIDES, AND LEATHER | CIBA-GEIGY CORPORATION (US) | 1981-03-17 | — | — | US | disclosed |
| EP-0019851-A1 | 1:2 Chromium complex dyestuffs of the azomethine and/or azo series, their preparation and use in dyeing and printing polyamide or cellulose materials | CIBA-GEIGY AG (CH) | 1980-12-10 | — | — | EP | disclosed |
| EP-0012969-A2 | Water-soluble fibre-reactive compounds and their use in fibre finishing,especially as dyestuffs,and dihalogeno-pyridazonyl-carboxylic and sulfonic acid halides and their use as fibre-reactive anchors,as well as process for the preparation of these compound | HOECHST AKTIENGESELLSCHAFT (DE) | 1980-07-09 | — | — | EP | disclosed |
| EP-0008472-A2 | Light sensitive benzenediazonium salts and diazotype material using same | Aerni-Leuch Ag (CH) | 1980-03-05 | — | — | EP | disclosed |
| US-4183949-A | Pesticidally active 1-arylamino-2,4-dinitronaphthalenes | BAYER AKTIENGESELLSCHAFT (DE) | 1980-01-15 | — | — | US | disclosed |
| EP-0005207-A2 | Bis-1:2 chrome-disazo-bisazo methine dyestuffs, their preparation and use for dyeing of leather | CIBA-GEIGY AG (CH) | 1979-11-14 | — | — | EP | disclosed |
| US-4118384-A | DIAZOTIZATION | BAYER AKTIENGESELLSCHAFT (DE) | 1978-10-03 | — | — | US | disclosed |
| US-4116952-A | POLYAMIDES | CIBA-GEIGY CORPORATION (US) | 1978-09-26 | — | — | US | disclosed |
| US-4110337-A | ANALGESIC, ANTIINFLAMMATORY | LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) | 1978-08-29 | — | — | US | disclosed |
| US-4092307-A | COPPER, NICKEL, COBALT OR CHROMIUM | CIBA-GEIGY CORPORATION (US) | 1978-05-30 | — | — | US | disclosed |
| US-4035350-A | Process for the preparation of water-soluble azo dyestuffs by reacting an aromatic amine and a coupling component with alkali metal nitrite or alkyl nitrite in the absence of acid | HOECHST AKTIENGESELLSCHAFT (DT) | 1977-07-12 | — | — | US | disclosed |
| US-4033942-A | Chromium complex dye, including azo and azo methine dye compounds | CIBA-GEIGY AG (CH) | 1977-07-05 | — | — | US | disclosed |
| US-3978037-A | POLYAMIDES | CIBA-GEIGY CORPORATION (US) | 1976-08-31 | — | — | US | disclosed |
| US-3978038-A | POLYAMIDES, POLYESTERS, POLYURETHANES | CIBA-GEIGY CORPORATION (US) | 1976-08-31 | — | — | US | disclosed |
| US-3957860-A | SULFAMIC ACID | CIBA-GEIGY AG (CH) | 1976-05-18 | — | — | US | disclosed |
| US-3947434-A | 9-(P-phenylazoanilino)-7-methyl-1H-imidazo[4,5-f]quinolines | MORTON-NORWICH PRODUCTS, INC. (US) | 1976-03-30 | — | — | US | disclosed |
| US-3947434-A | 9-(P-phenylazoanilino)-7-methyl-1H-imidazo[4,5-f]quinolines | MORTON-NORWICH PRODUCTS, INC. (US) | 1976-03-30 | — | — | US | disclosed |
Patent text — is the patent's own abstract consistent with the prediction?
For each of this compound's patents that has machine-readable text (49 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.
| Patent | Title | Text reads most about | Predicted target · text-rank |
|---|---|---|---|
| US-20040176602-A1 | 3-Cyanoquinolines,3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors | PKD1, PKD2, CSNK1A1 | ALDH1A1 4705/4885CYP3A4 4137/4885TSHR 1863/4885 |
| US-20200039979-A1 | Substituted-3H-imidazo[4,5-c]pyridine and 1H-pyrrolo[2,3-c]pyridine series of novel Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) and Stimulator for Interferon Genes (STING) modulators as cancer immunotherapeutics | STING1, ENPP1, CGAS | ALDH1A1 3527/4885CYP3A4 2995/4885TSHR 3344/4885 |
| US-20160263122-A1 | NOVEL COMPOUNDS | NAT1, AADAC, CBR3 | ALDH1A1 264/4885CYP3A4 131/4885TSHR 1816/4885 |
| US-20210101899-A1 | INHIBITORS OF MUTANT ISOCITRATE DEHYDROGENASES AND COMPOSITIONS AND METHODS THEREOF | IDH1, IDH2, IDH3A | ALDH1A1 198/4885CYP3A4 1151/4885TSHR 4834/4885 |
| US-20160145237-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | ALK, EGFR, ERBB2 | ALDH1A1 2546/4885CYP3A4 3760/4885TSHR 2149/4885 |
| US-20150166591-A1 | METHODS AND COMPOSITIONS FOR RAF KINASE MEDIATED DISEASES | BRAF, RAF1, EGFR | ALDH1A1 2855/4885CYP3A4 3015/4885TSHR 2717/4885 |
| US-20150298108-A1 | METHOD FOR PREPARING METHYL ACETATE | EHMT2, EHMT1, DNMT1 | ALDH1A1 1863/4885CYP3A4 173/4885TSHR 3004/4885 |
| US-20060167317-A1 | Aryl and heteroaryl propene amides, derivatives thereof and therapeutic uses thereof | BCL2A1, NFE2L2, BCL2 | ALDH1A1 389/4885CYP3A4 2777/4885TSHR 1304/4885 |
| US-20090318441-A1 | Pyrrolopyrimidine Compounds and Their Uses | PRKDC, TK2, PNKP | ALDH1A1 1780/4885CYP3A4 3277/4885TSHR 4367/4885 |
| US-20120316135-A1 | Compounds for Inhibiting Cell Proliferation in EGFR-Driven Cancers | EGFR, MKI67, ERBB2 | ALDH1A1 1376/4885CYP3A4 2447/4885TSHR 2573/4885 |
| US-20230310428-A1 | EGFR INHIBITOR AND PREPARATION METHOD AND USE THEREOF | EGFR, ERBB2, ERBB4 | ALDH1A1 3822/4885CYP3A4 1058/4885TSHR 1374/4885 |
| US-20100305126-A1 | Pyrimidine Inhibitors of Kinase Activity | IGF1R, CDK2, TK1 | ALDH1A1 1481/4885CYP3A4 3650/4885TSHR 724/4885 |
| US-20220235064-A1 | OXO-PYRIDINE FUSION RING DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME | ROS1, ROR1, RET | ALDH1A1 3759/4885CYP3A4 2385/4885TSHR 546/4885 |
| US-10383831-B2 | 2,4,6-trialkoxystryl aryl sulfones, sulfonamides and carboxamides, and methods of preparation and use | CCNY, STS, ARSA | ALDH1A1 1603/4885CYP3A4 762/4885TSHR 297/4885 |
| US-20030207864-A1 | Arylsulfonanilide ureas | UTS2R, UACA, UMPS | ALDH1A1 4087/4885CYP3A4 1298/4885TSHR 1927/4885 |
| US-20030162817-A1 | Pentafluorobenzenesulfonamides and analogs | FGFR1, FPR1, FGF1 | ALDH1A1 1192/4885CYP3A4 2141/4885TSHR 1857/4885 |
| US-20190031655-A1 | Substituted-3H-imidazo[4,5-c]pyridine and 1H-pyrrolo[2,3-c]pyridine series of novel Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) and Stimulator for Interferon Genes (STING) modulators as cancer immunotherapeutics | STING1, ENPP1, CGAS | ALDH1A1 3527/4885CYP3A4 2995/4885TSHR 3344/4885 |
| US-20100305118-A1 | PYRIMIDINE INHIBITORS OF KINASE ACTIVITY | IGF1R, TK1, CDK2 | ALDH1A1 982/4885CYP3A4 3939/4885TSHR 625/4885 |
| US-20070249868-A1 | New process for the preparation of 4-hydroxalkylamino-2-nitro-anisoles | HAO2, HCN2, NISCH | ALDH1A1 1176/4885CYP3A4 163/4885TSHR 4279/4885 |
| US-20160368924-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | BTK, LCK, BCL9 | ALDH1A1 3729/4885CYP3A4 3543/4885TSHR 3511/4885 |
| US-20240246908-A1 | TEAD INHIBITORS | TEAD3, TEAD1, TEAD2 | ALDH1A1 630/4885CYP3A4 1748/4885TSHR 628/4885 |
| US-20170355683-A1 | QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR AND PREPARATION AND APPLICATION THEREOF | EGFR, ERBB2, ERBB4 | ALDH1A1 2176/4885CYP3A4 2142/4885TSHR 1524/4885 |
| US-20200148634-A1 | ACLY INHIBITORS AND USES THEREOF | ACLY, ATP5ME, ATP5MG | ALDH1A1 1455/4885CYP3A4 2849/4885TSHR 4803/4885 |
| US-20120207763-A1 | PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES | PRKDC, TK2, PNKP | ALDH1A1 1780/4885CYP3A4 3277/4885TSHR 4367/4885 |
| US-20010027211-A1 | Arylsulfonanilide ureas | UTS2R, UACA, UMPS | ALDH1A1 4087/4885CYP3A4 1298/4885TSHR 1927/4885 |
| US-10781207-B2 | Inhibitors of mutant isocitrate dehydrogenases and compositions and methods thereof | IDH1, IDH2, IDH3A | ALDH1A1 198/4885CYP3A4 1151/4885TSHR 4834/4885 |
| US-11555012-B2 | ACLY inhibitors and uses thereof | ACLY, ATP5ME, ATP5MG | ALDH1A1 1455/4885CYP3A4 2849/4885TSHR 4803/4885 |
| US-20140057911-A1 | NOVEL 4,6-DISUBSTITUTED AMINOPYRIMIDINE DERIVATIVES HAVING BOTH AROMATIC AND HALOGENIC SUBSTITUENTS | DPYD, ABL1, BRD4 | ALDH1A1 507/4885CYP3A4 43/4885TSHR 1627/4885 |
| US-20160052898-A1 | NOVEL COMPOUNDS | AADAC, NAT1, CCNA1 | ALDH1A1 325/4885CYP3A4 1384/4885TSHR 3456/4885 |
| US-20150284408-A1 | INHIBITORS OF DNA GYRASE FOR THE TREATMENT OF BACTERIAL INFECTIONS | TOP1, TOP2A, DNASE1 | ALDH1A1 3693/4885CYP3A4 1533/4885TSHR 4565/4885 |
| US-10059688-B2 | Protein tyrosine kinase modulators and methods of use | ALK, EGFR, ERBB2 | ALDH1A1 2546/4885CYP3A4 3760/4885TSHR 2149/4885 |
| US-10106508-B2 | Quinazoline heterocyclic compound as EGFR kinase inhibitor and preparation and application thereof | EGFR, ERBB2, ERBB4 | ALDH1A1 2176/4885CYP3A4 2142/4885TSHR 1524/4885 |
| US-20140378446-A1 | PURINONE COMPOUNDS AS KINASE INHIBITORS | BTK, LCK, BCL9 | ALDH1A1 3729/4885CYP3A4 3543/4885TSHR 3511/4885 |
| US-20260076975-A1 | TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES | PDXK, NADK, HYPK | ALDH1A1 1101/4885CYP3A4 1454/4885TSHR 753/4885 |
| US-10130633-B2 | Compounds | AADAC, NAT1, CBR3 | ALDH1A1 277/4885CYP3A4 113/4885TSHR 2036/4885 |
| US-20160244469-A1 | Compounds for Inhibiting Cell Proliferation in EGFR-Driven Cancers | EGFR, MKI67, ERBB2 | ALDH1A1 1376/4885CYP3A4 2447/4885TSHR 2573/4885 |
| US-11142524-B2 | Substituted-3H-imidazo[4,5-c]pyridine and 1H-pyrrolo[2,3-c]pyridine series of novel Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) and stimulator for interferon genes (STING) modulators as cancer immunotherapeutics | STING1, ENPP1, CGAS | ALDH1A1 3527/4885CYP3A4 2995/4885TSHR 3344/4885 |
| US-20140275064-A1 | DYRK1 INHIBITORS AND USES THEREOF | DYRK1A, DYRK1B, DYRK2 | ALDH1A1 4162/4885CYP3A4 4620/4885TSHR 1871/4885 |
| US-20020143036-A1 | Pentafluorobenzenesulfonamides and analogs | FFAR1, PCSK9, PFAS | ALDH1A1 1403/4885CYP3A4 877/4885TSHR 1540/4885 |
| US-20050096484-A1 | Amino-substituted sulfonanilides and derivatives thereof for treating proliferative disorders | ARSA, MKI67, CCNA1 | ALDH1A1 1651/4885CYP3A4 3950/4885TSHR 795/4885 |
| US-20190233414-A1 | INHIBITORS OF MUTANT ISOCITRATE DEHYDROGENASES AND COMPOSITIONS AND METHODS THEREOF | IDH1, IDH2, IDH3A | ALDH1A1 198/4885CYP3A4 1151/4885TSHR 4834/4885 |
| US-20180009782-A1 | PROTEIN TYROSINE KINASE MODULATORS AND METHODS OF USE | ALK, EGFR, ERBB2 | ALDH1A1 2546/4885CYP3A4 3760/4885TSHR 2149/4885 |
| US-20180243239-A1 | 2,4,6-TRIALKOXYSTRYL ARYL SULFONES, SULFONAMIDES AND CARBOXAMIDES, AND METHODS OF PREPARATION AND USE | CCNY, STS, ARSA | ALDH1A1 1603/4885CYP3A4 762/4885TSHR 297/4885 |
| US-20170204084-A1 | NOVEL 4,6-DISUBSTITUTED AMINOPYRIMIDINE DERIVATIVES HAVE ANTI-HIV ACTIVITY | UMPS, DPYD, DUT | ALDH1A1 942/4885CYP3A4 101/4885TSHR 4853/4885 |
| US-20030153566-A1 | 7-Amino-benzothiazole derivatives | ADORA1, ADORA2A, ADORA3 | ALDH1A1 308/4885CYP3A4 954/4885TSHR 208/4885 |
| US-20070255057-A1 | Mono-nitration of aromatic compounds via nitrate salts | NOS2, NOS3, NOS1 | ALDH1A1 722/4885CYP3A4 41/4885TSHR 4662/4885 |
| US-20020026052-A1 | 3-cyanoquinolines, 3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors | PKD1, PKD2, CSNK1A1 | ALDH1A1 4705/4885CYP3A4 4137/4885TSHR 1863/4885 |
| US-20250154107-A1 | 3,4-Dihydroisoquinolin-1(2H)-Ones Derivatives as STING Antagonists and the Use Thereof | STING1, IRF3, MAVS | ALDH1A1 4770/4885CYP3A4 4459/4885TSHR 3730/4885 |
| US-10689376-B2 | Substituted-3H-imidazo [4,5-c] pyridine and 1H-pyrrolo[2,3-c]pyridine series of novel ectonucleotide pyrophosphatase/phosphodiesterase-1 (ENPP1) and stimulator for interferon genes (STING) modulators as cancer immunotherapeutics | STING1, ENPP1, CGAS | ALDH1A1 3527/4885CYP3A4 2995/4885TSHR 3344/4885 |
“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.